DOI: 10.1055/s-00000131

Synfacts

Issue 12 · Volume 2010 · December 2010 DOI: 10.1055/s-002-21480

Synform

  • A94

    SYNFORM ISSUE 2010/11

    • Synthesis of Natural Products and Potential Drugs

  • z1327

    All PDFs of this category

  • 1327

    Synthesis of (R)-Ofloxacin

  • 1328

    Synthesis of (S)-(-)-Ropivacaine

  • 1329

    Synthesis of endo-6-Aryl-8-oxabicyclo-[3.2.1]oct-3-en-2-one

  • 1330

    Synthesis of (+)-Peloruside A

  • 1331

    Synthesis of (+)-Peloruside A

  • 1332

    Synthesis of BMS-764459

  • 1333

    Total Synthesis of Chloptosin

  • 1334

    Synthesis of (±)-Pseudotabersonine

  • 1335

    Synthesis of (+)-Barekoxide and (-)-Barekol

  • 1336

    Synthesis of an LFA-1 Inhibitor

  • 1337

    Synthesis of Telcagepant

  • 1338

    Synthesis of Trilobacin

  • 1339

    Formal Synthesis of (±)-Cortistatin A

  • 1340

    Synthesis of Tenofovir Disoproxil Fumarate

    • Synthesis of Heterocycles

  • z1341

    All PDFs of this category

  • 1341

    Synthesis of Chiral Aziridines from Imines and Diazoacetamides

  • 1342

    Direct C2 Indole Trifluoromethylation Using Togni’s Reagent

  • 1343

    Synthesis of Pyridopyrrolopyrimidines. Total Synthesis of Varioline B and Deoxyvariolin B

  • 1344

    Synthesis of Quinoxalines via Ru/C Benzoin Oxidation and Diamine Condensation

  • 1345

    Facile Acid-Catalyzed Route to Thiazoles from Propargylic Alcohols and Thioamides

  • 1346

    Synthesis of Indoles from 2-Azidoacrylate and ortho-Silyl Aryltriflates

  • 1347

    Synthesis of Tetrasubstituted Furans by Michael Addition to β-Nitroacrylates

  • 1348

    Palladium-Catalyzed Synthesis of 3,3-Disubstituted Oxindoles

  • 1349

    Copper(I)-Catalyzed Annulation Route to Indolizines

  • 1350

    Synthesis of N-Arylindazoles and Benz-imidazoles from ortho-Aminobenzoximes

  • 1351

    Copper-Mediated Synthesis of Indolequinones from Bromoquinones

  • 1352

    Palladium-Catalyzed Cyclocarbonylative Synthesis of Dibenzoxazepinones

  • 1353

    Enantioselective Synthesis of Dihydro-isochromanones Using Hypervalent Iodine

  • 1354

    Synthesis of 1,5-Diaryl-1,2,3-triazoles Under Transition-Metal-Free Conditions

  • 1355

    Rhodium(II)-Catalyzed Synthesis of Polyether Macrocyles

    • Synthesis of Materials and Unnatural Products

  • z1357

    All PDFs of this category

  • 1357

    Soluble and Stable Zethrenebis(carboximide) and Its Quinone

  • 1358

    Alternating Copolymers of Anthracene via Novel Radical ROP

  • 1359

    Unsubstituted Polyphenylenes via a ‘Shaving’ Approach

  • 1360

    Highly Selective Synthesis of Dibenzo[a,c]cyclooctatetraenes

  • 1361

    A New Functionalization Method of SWCNTs through Cycloaddition

  • 1362

    Scale Up, Spice Up

  • 1363

    Efficient Bipolar Transport Material for OLEDs

  • 1364

    Annulated Fullerenes

  • 1365

    Hosting Hydrogel Formation

  • 1366

    One Scaffold, Different Motifs

  • 1367

    Light-Emitting Platinum-Containing Polymers

  • 1368

    A New Route to Diaminoacetylenes

  • 1369

    Phenylene-Bridged Boron-Nitrogen Containing Dendrimers

  • 1370

    Alkyne ROMP: ‘It’s Alive!!!’

    • Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

  • z1371

    All PDFs of this category

  • 1371

    Cooperative Ruthenium and Organocatalysis

  • 1372

    Iridium-Catalyzed Asymmetric Hydrogenation of Unprotected β-Enamine Esters

  • 1373

    Asymmetric Cyclopropanation Using Dimethyl Diazomalonate

  • 1374

    Stereoselective Synthesis of (E)-α,β-Diarylacrylates

  • 1375

    Solvent-Free Magnesium-Catalyzed Enantioselective Ketone-Ene Reactions

  • 1376

    Nickel-Catalyzed Aldol Reaction Between α-Isothiocyanato Imide and Aldehydes

  • 1377

    Catalytic Asymmetric Michael Addition to 4-Oxo-4-arylbutenoates

  • 1378

    New Chiral Bidentate Secondary Phosphine Oxide Ligands for Hydrogenation

  • 1379

    Enantioselective Synthesis of Spirooxindoles Inspired by Natural Products

  • 1380

    Synthesis of 1,3-syn and -anti-Tetrahydro-pyrimidinones

  • 1381

    Asymmetric Ru-Phebox Catalyzed Alkynylation

  • 1382

    Cobalt(II)-Catalyzed Stereoselective Cyclopropanation of Alkenes

  • 1383

    Gold(I)-Catalyzed Diastereoselective Pyrrolidine Synthesis

  • 1384

    Rhodium-Catalyzed Asymmetric 1,6-Addition of Enynamides

  • 1385

    A Lewis Acid Catalyzed Asymmetric Photocycloaddition

  • 1386

    Indium-Mediated Enantioselective Allylation

  • 1387

    Asymmetric Arylation of N-Tosyl Ketimines

  • 1388

    Reductive Enolization in Aldol Addition to Enolizable Aldehydes

  • 1389

    Copper-Catalyzed Addition of Grignards to Allylic α-Haloacetates

  • 1390

    Rhodium-Catalyzed Asymmetric Hydro-formylation

  • 1391

    C1-Symmetric Dicyclopentadienes in Rh-Catalyzed Arylation of N-Tosylarylimines

  • 1392

    Chiral N-Heterocycles via Asymmetric Allylic Methylation-Ring-Closing Metathesis

  • 1393

    Regio- and Stereospecific Aziridinzation of Unsymmetric Conjugated Dienes

  • 1394

    Asymmetric Allylic Alkylation with Phosphaalkene-Oxazoline Ligands

  • 1395

    Atropselective Biaryl Coupling in the Synthesis of (+)-Korupensamine B

  • 1396

    Ruthenium-Catalyzed Asymmetric Monohydrogenation of meso-Cyclic Imides

  • 1397

    Combined Acid System for Asymmetric Addition of Boronates to Chromene Acetals

  • 1398

    Conjugate Addition of Aryl Alanes to Form Quaternary Stereocenters

  • 1399

    Ruthenium-Catalyzed Asymmetric Reduction of α-Keto Acids

  • 1400

    Synthesis of Enantiopure Allyl Phenyl Sulfides

    • Metal-Mediated Synthesis

  • z1401

    All PDFs of this category

  • 1401

    Metal-Free Coupling of Aryl and Alkynyl Grignard Reagents Mediated by TEMPO

  • 1402

    Alkenylative Cross-Coupling between Alkyl Sulfides and Grignard Reagents

  • 1403

    Stereospecific Suzuki Coupling with Inversion of Stereoconfiguration

  • 1404

    Csp³-Csp³ Suzuki Cross-Coupling Using Unactivated Secondary Alkyl Chlorides

  • 1405

    Nickel-Catalyzed C-O Activation of Phenol Derivatives

  • 1406

    Allylation of Nitrosobenzene with Pinacol Allylboronates

  • 1407

    ZnCl2-Enhanced Negishi Coupling of Secondary Benzyl Trifluoroacetates

  • 1408

    Zinc Alkoxide Catalyzed Allylations of Ketones with Allyl Pinacol Boronates

  • 1409

    Palladium-Catalyzed β-Arylation of Carboxylic Esters

  • 1410

    Cobalt-Catalyzed Hydroarylation of Alkynes Through C-H Bond Activation

  • 1411

    Radical Addition of Arylboronic Acids to Olefins

  • 1412

    Nucleophilic Addition to N-Methoxyamides via N-Oxyiminium Ions

  • 1413

    C-H Arylation of N-Heterocycles with Arylboronic Acids

  • 1414

    Catalytic Magnesium in Direct Coupling of Benzylic Halides with Pinacolborane

  • 1415

    Cross-Coupling of Aryltrimethylammonium Triflates with Aryl Grignard Reagents

    • Organo- and Biocatalysis

  • z1417

    All PDFs of this category

  • 1417

    Brønsted Acid Catalyzed Pictet-Spengler Cyclization of Keto Acids

  • 1418

    Organocatalytic Corey-Chaykovsky Reaction of Ketones

  • 1419

    Organophotoredox Catalysis

  • 1420

    One-Pot Synthesis of Chiral Piperidines Using Diphenylprolinol Silyl Ether

  • 1421

    Sulfa-Michael Reaction Cascade for the Synthesis of Chromans

  • 1422

    Asymmetric Morita-Baylis-Hillman Reactions of Acrolein

  • 1423

    Highly Efficient Desymmetrization of Glutaric Anhydrides

  • 1424

    Formal [3+2] Cycloaddition of Ketenes and Oxaziridines

  • 1425

    Practical Enantioselective One-Pot Syntheses of β-Hydroxy and β-Amino Esters

  • 1426

    Asymmetric Anion Binding DMAP Catalysis in the Kinetic Resolution of Propargylic Amines

  • 1427

    Hypervalent Iodine(III) Organocatalysts

  • 1428

    Intramolecular Aza-Michael Addition of Indoles

  • 1429

    A Bifunctional Enzyme for a Michael Addition-Oxidation Sequence

    • Polymer-Supported Synthesis

  • z1431

    All PDFs of this category

  • 1431

    A Flow Reaction System Using Catalytic Magnetic Particles

  • 1432

    Perfluoroalkylated Polymer-Supported Palladium Catalyst

  • 1433

    Palladium Nanoparticles in Silica Hollow Spheres with Mesoporous Walls

  • 1434

    Cross-Dehydrogenative Coupling with Fe3O4 Nanoparticles

  • 1435

    Modification of a Vitamin D Analogue Using a Supported Selenium Reagent

  • 1436

    Asymmetric Cyanosilylation with Supported Cu(II) Salen Complexes

  • 1437

    ortho-Borylation of Phenols with Silica-SMAP-Ir

  • 1438

    Asymmetric Aldol Reaction in Water Catalyzed by Chitosan Aerogel

  • 1439

    Suzuki-Miyaura Couplings with Palladium Membrane Installed Microreactors

  • 1440

    An Iron Metal-Organic Framework Catalyst for Thiol Oxidation

  • 1441

    Deoxygenation of Epoxides with Hydrotalcite-Supported Silver Nanoparticles

  • 1442

    Asymmetric C-H Insertion with a Polymer-Supported Rhodium Complex

  • 1443

    Enantioselective Hydrolysis of Soluble Polymer-Supported Carboxylates