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Issue Accepted Manuscripts

Issue 04/2025

  • Song, Xizhong; Yin, Wei; Zeng, Xiaowen; Zhang, Wenping; Fu, Wenyan; Qian, Limei; Jin, Yi; Yang, Ming:

    PIFA-Mediated Ring-Opening/Coupling Reaction of Benzoxazoles: Access to 2-Hydroxy Diarylureas

    Image for article: PIFA-Mediated Ring-Opening/Coupling Reaction of Benzoxazoles: Access to 2-Hydroxy Diarylureas
  • Issue 01/2025

  • Shehta, Wael; Alsaiari, Norah A.; Farag, Basant; Abdel-Aziz, Marwa M.; Youssif, Shaker; Elfeky, Sherin M; El-Kalyoubi, Samar; Osman, Nermine A.:

    Synthesis, In Vitro and In Silico Molecular Docking Studies of Novel Phthalimide–Pyrimidine Hybrid Analogues to Thalidomide as Potent Antitubercular Agents

    Image for article: Synthesis, <i>In Vitro</i> and <i>In Silico</i> Molecular Docking Studies of Novel Phthalimide–Pyrimidine Hybrid Analogues to Thalidomide as Potent Antitubercular Agents
  • Nakao, Michiyasu; Okamoto, Marie; Isetani, Satoshi; Imai, Ayato; Kitaike, Syuji; Sano, Shigeki:

    Development of a Novel Horner–Wadsworth–Emmons Reagent for the Facile Preparation of Mixed Phosphonoacetates

    Image for article: Development of a Novel Horner–Wadsworth–Emmons Reagent for the Facile Preparation of Mixed Phosphonoacetates
  • Issue 04/2024

    Issue 03/2024

    Issue 02/2024

  • Lipson, Victoria V.; Yaremenko, Fedyr G.; Vakula, Volodymyr M.; Kovalenko, Svitlana V.; Kyrychenko, Alexander V.; Desenko, Sergiy M.; Borysko, Petro О.; Zozulya, Sergiy O.:

    Discovery of Novel N-Acylhydrazone Derivatives as Potent Inhibitors of Sirtuin-1

    Image for article: Discovery of Novel <i>N</i>-Acylhydrazone Derivatives as Potent Inhibitors of Sirtuin-1
  • Issue 01/2024

  • Pitchai, Manivel; Kaspady, Mahammed; Indasi, Gopikumar; Krishnan, Rajesh; Maheswarappa, Gururaju Sannakki; Vetrichelvan, Muthalagu; Mathur, Arvind; Gupta, Anuradha:

    Regioselective C3-Formylation of 2H-Indazoles Using Selectfluor under Microwave-Assisted Conditions

    Image for article: Regioselective C3-Formylation of 2<i>H</i>-Indazoles Using Selectfluor under Microwave-Assisted Conditions
  • Issue 04/2023

  • Vetrichelvan, Muthalagu; Lanke, Veeranjaneyulu; Chandu, Bellam; Mathur, Arvind; Gupta, Anuradha:

    Cost-Effective and Scalable Synthesis of 4-Bromo-1,2-dimethyl-1H-imidazole: A Key Building Block for Bioactive Molecules

    Image for article: Cost-Effective and Scalable Synthesis of 4-Bromo-1,2-dimethyl-1<i>H</i>-imidazole: A Key Building Block for Bioactive Molecules
  • Yang, Qi-Liang; Lei, Ping-Ping; Hao, Er-Jun; Zhang, Bei-Ning; Zhou, Hong-Hao; Li, Wan-Wan; Guo, Hai-Ming:

    Oxidative C–H Sulfonylation of Hydrazones Enabled by Electrochemistry

    Image for article: Oxidative C–H Sulfonylation of Hydrazones Enabled by Electrochemistry
  • Lipson, Victoria; Zhikol, Oleg; Shishkina, Svetlana; Semenenko, Alexander; Kulyk, Karina; Mateychenko, Pavel; Musatov, Vladimir; Mazepa, Alexander; Vakula, Vladimir; Borisov, Alexander; Kyrychenko, Alexander:

    Low Molecular Weight Supramolecular Allobetuline-, Cyclohexanol-, or Undecanol-Appended 1,2,3-Triazole-Based Gelators: Synthesis and Molecular Dynamics Simulation Study

    Image for article: Low Molecular Weight Supramolecular Allobetuline-, Cyclohexanol-, or Undecanol-Appended 1,2,3-Triazole-Based Gelators: Synthesis and Molecular Dynamics Simulation Study
  • Issue 03/2023

    Issue 02/2023

  • Sakhno, Yana; Radchenko, Oleksandr; Saraev, Vyacheslav; Shliapkina, Yuliia; Kaidash, Mariia; Shyshkina, Mariia; Shishkina, Svitlana; Musatov, Vladimir; Desenko, Sergey; Chebanov, Valentyn:

    Temperature-Controlled Diastereoselective Doebner/Ugi Tandem Reaction

    Image for article: Temperature-Controlled Diastereoselective Doebner/Ugi Tandem Reaction
  • Issue 01/2023

  • Mitra, Trisha; Joardar, Soumen; Chakravorty, Santanu; Majumdar, Manoj; Kundu, Mrinalkanti; Roy, Brindaban:

    Palladium-Mediated Reductive Heck Cyclization for the Synthesis of Fused Retinoid Derivatives

    Image for article: Palladium-Mediated Reductive Heck Cyclization for the Synthesis of Fused Retinoid Derivatives
  • Burke, Adam; Spiccio, Silvia; Di Filippo, Mara; Baumann, Marcus:

    Photochemical Synthesis of Pyrazolines from Tetrazoles in Flow

    Image for article: Photochemical Synthesis of Pyrazolines from Tetrazoles in Flow
  • Mallesham, Poosa; Raghavulu, Karri; Miriyala, Venkatesh; Doddipalla, Raju; Yennam, Satyanarayana; Sanasi, Paul Douglas; Behera, Manoranjan:

    Synthesis of Acidiphilamide A–C: Secondary Metabolites from the Genus Streptacidiphilus

    Image for article: Synthesis of Acidiphilamide A–C: Secondary Metabolites from the Genus <i>Streptacidiphilus</i>
  • Issue 04/2022

  • Noble, Jeffrey M.; Chang, Le; Chen, Dan; Wang, Binglin; Dominey, Raymond N.; Cook, Daniel W.; Burns, Justina M.; Stringham, Rodger W.; Cardoso, Flavio S. P.; Snead, David R.:

    A Practical and Economical Route to (S)-Glycidyl Pivalate

    Image for article: A Practical and Economical Route to (<i>S</i>)-Glycidyl Pivalate
  • Biradar, D. O.; Mane, Y. D.; Sarnikar, Y. P.; Kulkarni, S. G.; Reddy, B. V. Subba; Narsaiah, A. Venkat:

    Zn/ZnBr2 Catalysed Reaction of Aldehydes with Allylbromide: Synthesis of 2,6-Disubstituted 4-Bromotetrahydropyrans

    Image for article: Zn/ZnBr<sub>2</sub> Catalysed Reaction of Aldehydes with Allylbromide: Synthesis of 2,6-Disubstituted 4-Bromotetrahydropyrans
  • Issue 03/2022

    Issue 02/2022

    Issue 01/2022

    Issue 04/2021

    Issue 03/2021

    Issue 02/2021

    Issue 01/2021

    Issue 04/2020

  • Guirado, Antonio; Vera, María; Martiz, Bruno; Ródenas, Francisco; Sandoval, José A.; Alarcón, Enrique; Bautista, Delia:

    Synthesis and Crystal Structures of 4,5-Dihydroimidazo[1,5-b]pyrazol-6-ones

    Image for article: Synthesis and Crystal Structures of 4,5-Dihydroimidazo[1,5-<i>b</i>]pyrazol-6-ones
  • Avula, Satya Kumar; Das, Biswanath; Csuk, Rene; Al-Rawahi, Ahmed; Al-Harrasi, Ahmed:

    Total Synthesis of Surinamensinols A and B

    Image for article: Total Synthesis of Surinamensinols A and B
  • Nariki, Haruna; Miyamura, Takuya; Matsui, Daiki; Sonoda, Motohiro; Tanimori, Shinji:

    Iodine-Mediated Facile One-Pot Access to N-Aryl-2-benzoxazolamines

    Image for article: Iodine-Mediated Facile One-Pot Access to <i>N</i>-Aryl-2-benzoxazolamines
  • Faverio, Chiara; Boselli, Monica Fiorenza; Raimondi, Laura; Benaglia, Maurizio:

    Ammonia–Borane-Mediated Reduction of Nitroalkenes

    Image for article: Ammonia–Borane-Mediated Reduction of Nitroalkenes
  • Rickertsen, Dillon R. L.; Ma, Longle; Paul, Anirudra; Abboud, Khalil A.; Seidel, Daniel:

    Traceless Redox-Annulations of Alicyclic Amines

    Image for article: Traceless Redox-Annulations of Alicyclic Amines
  • Issue 03/2020

  • Raghunadh, Akula; Tadiparthi, Krishnaji; Meruva, Suresh Babu; Murthy, V. Narayana; Rao, L. Vaikunta; Kumar, U. K. Syam:

    Synthesis of Quinoxalin-2(1H)-ones and Hexahydroquinoxalin-2(1H)-ones via Oxidative Amidation–Heterocycloannulation

    Image for article: Synthesis of Quinoxalin-2(1<i>H</i>)-ones and Hexahydroquinoxalin-2(1<i>H</i>)-ones via Oxidative Amidation–Heterocycloannulation
  • Issue 02/2020

    Issue 04/2019

    Issue 02/2019

  • Sharada, Ambati; Kundeti, Lakshmi Srinivasa Rao; Ramakrishna, Kallaganti V. S.; Nagaiah, Kommu:

    First Stereoselective Total Synthesis of Ciryneol C

    Image for article: First Stereoselective Total Synthesis of Ciryneol C
  • Issue 01/2019

  • Kawtharani, Ranin.; Elmasri, Mirvat; Cherry, Khalil; Jacquemin, Johan; Abarbri, Mohamed:

    Highly Regio- and Stereoselective Hydrogermylation of Fluorinated Alkyl Propiolate

    Image for article: Highly Regio- and Stereoselective Hydrogermylation of Fluorinated Alkyl Propiolate
  • Kitagawa, Saori; Mori, Hiromitsu; Odagiri, Tatsuya; Suzuki, Katsuya; Kikkawa, You; Osugi, Rie; Takizawa, Shinobu; Kimura, Yoshikazu; Kirihara, Masayuki:

    A Concise, Catalyst-Free Synthesis of Davis’ Oxaziridines using Sodium Hypochlorite

    Image for article: A Concise, Catalyst-Free Synthesis of Davis’ Oxaziridines using Sodium Hypochlorite
  • Issue 04/2018

    Issue 03/2018

    Issue 02/2018

  • Ahsan, Mohamed J.; Kumawat, Bhawani S.; Kumawat, Sonu; Sharma, Piush; Bakht, Mohammad A.; Hassan, Mohd Z.; Hussain, Afzal; Saraswat, Pankaj; Khalilullah, Habibullah:

    Synthesis and Cytotoxic Evaluation of 3-(4-Fluorophenyl)-4,5-dihydro-5-(3,4,5-trimethoxy/4-nitrophenyl)-N-(substituted-phenyl)pyrazole-1-carboxamide Analogues

    Image for article: Synthesis and Cytotoxic Evaluation of 3-(4-Fluorophenyl)-4,5-dihydro-5-(3,4,5-trimethoxy/4-nitrophenyl)-<i>N</i>-(substituted-phenyl)pyrazole-1-carboxamide Analogues
  • Gujjarappa, Raghuram; Vodnala, Nagaraju; Kabi, Arup K.; Kaldhi, Dhananjaya; Kumar, Mohan; Beifuss, Uwe; Malakar, Chandi C.:

    Efficient Syntheses of Diverse N-Heterocycles: The Molybdenum(VI)-Catalyzed Reductive Cyclization of Nitroarenes using Pinacol as a Deoxygenating­ Agent

    Image for article: Efficient Syntheses of Diverse N-Heterocycles: The Molybdenum(VI)-Catalyzed Reductive Cyclization of Nitroarenes using Pinacol as a Deoxygenating­ Agent
  • Rana, Anil; Kumar, Varun; Tiwari, Lata; Thakur, Anamika; Meena, Chhuttan Lal; Mahajan, Dinesh:

    Triflic Anhydride Promoted Synthesis of Primary Amides and their Conversion into Nitriles

    Image for article: Triflic Anhydride Promoted Synthesis of Primary Amides and their Conversion into Nitriles
  • Rahman, Masood ur; Ayoob, Iram; Rehman, Shakeel u; Bhat, Khursheed A.; Ara, Tabassum:

    Microwave-Assisted Synthesis of Andrographolide Analogues as Potent β-Glycosidase Inhibitors

    Image for article: Microwave-Assisted Synthesis of Andrographolide Analogues as Potent β-Glycosidase Inhibitors
  • Choudhary, Rakhee; Bai, Rekha; Singh, Pratibha; Sharma, Mahesh C.; Badsara, Satpal Singh:

    Room Temperature, Open-Flask C–P Bond-Formation on Water under Catalyst-Free Conditions

    Image for article: Room Temperature, Open-Flask C–P Bond-Formation on Water under Catalyst-Free Conditions
  • Issue 01/2018

  • Songsichan, T.; Katrun, P.; Khaikate, O.; Soorukram, D.; Pohmakotr, M.; Reutrakul, V.; Kuhakarn, C.:

    Thiocyanation of Pyrazoles Using KSCN/K2S2O8 Combination

    Image for article: Thiocyanation of Pyrazoles Using KSCN/K<sub>2</sub>S<sub>2</sub>O<sub>8</sub> Combination
  • Kummari, Bhaskar; Ramesh, Perla; Polkam, Naveen; Malthum, Shankaraiah; Vishnuvardhan, M. V. P. S.; Anireddy, Jaya Shree:

    Design, Synthesis, and Cytotoxic Evaluation of Etodolac-1,3,4-oxadiazole-1,2,3-triazole Molecules

    Image for article: Design, Synthesis, and Cytotoxic Evaluation of Etodolac-1,3,4-oxadiazole-1,2,3-triazole Molecules
  • Caillé, Julien; Setzer, Paul; Boeda, Fabien; Pearson-Long, Morwenna S. M.; Bertus, Philippe:

    Asymmetric Titanium-Catalyzed Cyclopropanation of Nitriles with Grignard Reagents

    Image for article: Asymmetric Titanium-Catalyzed Cyclopropanation of Nitriles with Grignard Reagents
  • Nakao, Michiyasu; Nishikiori, Nanako; Nakamura, Akihito; Miyagi, Murasaki; Shibata, Nao; Kitaike, Syuji; Fukui, Makoto; Ito, Hiro-O; Sano, Shigeki:

    Synthesis of Sterically Protected Isoindoles from ortho-Phthalaldehyde

    Image for article: Synthesis of Sterically Protected Isoindoles from <i>ortho</i>-Phthalaldehyde
  • Issue 01/2017

  • Ghosal, Nirnita Chakraborty; Mahato, Sachinta; Chatterjee, Rana; Santra, Sougata; Zyryanov, Grigory V.; Majee, Adinath:

    A Mild and Efficient Method for the Syntheses and Regioselective Ring-Opening of Aziridines

    Image for article: A Mild and Efficient Method for the Syntheses and Regioselective Ring-Opening of Aziridines
  • Panda, Siva S.; Asiri, Abdullah M.; Elagawany, Mohamed; Buchanan, Devan D.; Torkian, Behrad; Bathala, Keerthana; Thomas, Sean J.; Capito, Jason E.; Arshad, Muhammad N.; Al-Romaizan, Abeer N.:

    Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates

    Image for article: Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates
  • Nosik, Pavel S.; Artamonov, Oleksiy S.; Ryabukhin, Sergey V.; Grygorenko, Oleksandr O.:

    An Approach to 1,1-Disubstituted Pyrazolylcyclopropane Building Blocks

    Image for article: An Approach to 1,1-Disubstituted Pyrazolylcyclopropane Building Blocks
  • Majeed, Anju; Nagabhushanam, Kalyanam; Majeed, Muhammed; Thomas, Samuel Manoharan; Thajuddin, Nooruddin:

    An Expeditious, Green and Protecting-Group-Free Synthesis of a Potent Secondary Metabolite Calebin-A and Its Analogues

    Image for article: An Expeditious, Green and Protecting-Group-Free Synthesis of a Potent Secondary Metabolite Calebin-A and Its Analogues
  • Yang, Yi-Qiu; Ke, Long-Zhi; Wang, Gui-Fei; Song, Shu-Yong; Qiu, Ming-Ning; Liu, Jian-Jun; Huang, Yun-Sheng:

    Synthesis of N-Pyridin-2-ylmethyl and N-Quinolin-2-ylmethyl ­Substituted Ethane-1,2-diamines

    Image for article: Synthesis of <i>N</i>-Pyridin-2-ylmethyl and <i>N</i>-Quinolin-2-ylmethyl ­Substituted Ethane-1,2-diamines
  • Barcia, Jose C.; Cruces, Jacobo; Salas, Cristian O.; Estévez, Juan C.; Cuellar, Mauricio A.; Tapia, Ricardo A.; Estévez, Ramón J.:

    A New Approach to the Synthesis of Benzo[b]naphtho[2,3-b]furan-6,11-diones and 2-Benzyl-3-hydroxynaphthalene-1,4-diones

    Image for article: A New Approach to the Synthesis of Benzo[<i>b</i>]naphtho[2,3-<i>b</i>]furan-6,11-diones and 2-Benzyl-3-hydroxynaphthalene-1,4-diones