DOI: 10.1055/s-00000131

Synfacts

Issue 07 · Volume 2010 · July 2010 DOI: 10.1055/s-002-21135

Synform

A56
Zanda, Matteo: SYNFORM ISSUE 2010/07

Synthesis of Natural Products and Potential Drugs

z735
All PDFs of this category
0735
Hanessian, S.; Guesné, S.; Chénard, E.: Synthesis of Aliskiren
0736
Hsu, D.-S.; Chou, Y.-Y.; Tung, Y.-S.; Liao, C.-C.: Synthesis of (±)-Δ-Capnellene
0737
Carr, J. L.; Offermann, D. A.; Holdom, M. D.; Dusart, P.; White, A. J. P.; Beavil, A. J.; Leatherbarrow, R. J.; Lindell, S. D.; Sutton, B. J.; Spivey, A. C.: Synthesis of (±)-Aspercyclide A
0738
Hayakawa, I.; Takemura, T.; Fukasawa, E.; Ebihara, Y.; Sato, N.; Nakamura, T.; Suenaga, K.; Kigoshi, H.: Synthesis of Auripyrones A and B
0739
Pitsinos, E.; Athinaios, N.; Xu, Z.; Wang, G.; Negishi, E.-i.: Synthesis of (+)-Scyphostatin
0740
Kakinuma, H.: Synthesis of TS-071
0741
Liu, P.; Seo, J. H.; Weinreb, S. M.: Total Synthesis of (±)-Communesin F
0742
McCauley, J. A.: Synthesis of Vaniprevir (MK-7009)
0743
Black, F. J.; Kocienski, P. J.: Synthesis of Phalluside-1 and Sch II
0744
Candy, M.; Audran, G.; Bienaymé, H.; Bressy, C.; Pons, J.-M.: Synthesis of (+)-Crocacin C
0745
Chernyak, N.; Gevorgyan, V.: Synthesis of Zolpidem
0746
Venukadasula, P. K. M.; Chegondi, R.; Maitra, S.; Hanson, P. R.: Synthesis of (-)-Tetrahydrolipstatin
0747
Krumlinde, P.; Bogár, K.; Bäckvall, J.-E.: Synthesis of Sertraline

Synthesis of Heterocycles

z749
All PDFs of this category
0749
Reddy, U. C.; Saikia, A. K.: Multicomponent Prins-Friedel-Crafts Synthesis of 4-Aryl-5,6-Dihydropyrans
0750
Zhou, H.; Zhu, D.; Xie, Y.; Huang, H.; Wang, K.: Gallium-Catalyzed Synthesis of 1,3-Dihydrobenzo[c]thiophenes
0751
Yang, X.; Fu, H.; Qiao, R.; Jiang, Y.; Zhao, Y.: α-Arylation-Heteroannulation Route to 2-Amino-1H-indole-3-carboxylates
0752
Zhang, X.; Lu, Z.; Fu, C.; Ma, S.: Synthesis of Polysubstituted Furans by a Sonogashira-Cyclization Route
0753
Chernyak, D.; Chernyak, N.; Gevorgyan, V.: Copper-Catalyzed Three-Component Coupling Synthesis of 3-Aminoindol(in)es
0754
Lu, Y.; Wang, D.-H.; Engle, K. M.; Yu, J.-Q.: Synthesis of Isochromans by Palladium-Catalyzed C-H Olefination
0755
Coy B., E. D.; Jovanovic, L.; Sefkow, M.: trans-Dihydrobenzofurans via Diazotization-Palladium-Catalyzed Oxyarylation
0756
Xing, C.-H.; Liao, Y.-X.; He, P.; Hu, Q.-S.: Rhodium-Catalyzed Synthesis of Chiral 3-Substituted Phthalides
0757
Mohanan, K.; Martin, A. R.; Toupet, L.; Smietana, M.; Vasseur, J.-J.: Regioselective Synthesis of Phosphonyl Pyrazoles
0758
Fuwa, H.; Matsukida, S.; Sasaki, M.: Dihydropyranone Synthesis Using a Sonogashira Coupling
0759
Shen, G.; Bao, W.: Copper(I)-Catalyzed Synthesis of Benzoxazoles and Benzimidazoles
0760
Xin, Y.; Zhao, J.; Han, J.; Zhu, S.: 1,3-Dipolar Cycloaddition Synthesis of 3-Trifluoroacetyl Pyrroles
0761
Yu, X.; Du, B.; Wang, K.; Zhang, J.: Synthesis of 2,3-Dihydroisoxazoles from Enynes and Hydroxylamines
0762
Lefebvre, V.; Cailly, T.; Fabis, F.; Rault, S.: Hydrazone C-N Coupling Route to 3-Aminoindazoles

Synthesis of Materials and Unnatural Products

z763
All PDFs of this category
0763
Behof, W. J.; Wang, D.; Niu, W.; Gorman, C. B.: Domino Aromatizing Cyclization
0764
Wagner, K.; Crowe, L. L.; Wagner, P.; Gambhir, S.; Partridge, A. C.; Earles, J. C.; Clarke, T. M.; Gordon, K. C.; Officer, D. L.: Intermolecular Charge Transfer in a Novel Polythiophene
0765
Frank, B. B.; Kivala, M.; Blanco, B. C.; Breiten, B.; Schweizer, W. B.; Laporta, P. R.; Biaggio, I.; Jahnke, E.; Tykwinski, R. R.; Boudon, C.; Gisselbrecht, J. P.; Diederich, F.: Chirality Induction in the Backbone of a Charge-Transfer Oligomer
0766
Yu, H.; Li, J.; Kou, Z.; Du, X.; Wei, Y.; Fun, H.-K.; Xu, J.; Zhang, Y.: Azapolycycles through Photo-Tandem Reactions
0767
Lélias-Vanderperre, A.; Aubert, E.; Chambron, J.-C.; Espinosa, E.: Substituent Effect on Molecular Shape of a Macrotricyclic Receptor
0768
Durola, F.; Rebek, Jr., J.: A Self-Associating Cavitand
0769
Davis, N. K. S.; Thompson, A. L.; Anderson, H. L.: Extending the Aromatic Core of Porphyrins
0770
Banert, K.; Joo, Y.-H.; Rüffer, T.; Walfort, B.; Lang, H.: Azidochloro- and Azidobromomethane
0771
Morimoto, K.; Hirano, H.; Satoh, T.; Miura, M.: Chromophores from Air Oxidation
0772
Yuan, Z.; Xiao, Y.; Qian, X.: Fusing Together Perylene Bisimides with Arene Cores
0773
Gryko, D. T.; Rogacki, M. K.; Klajn, J.; Gałęzowski, M.; Stępień, D. K.; Cyrański, M. K.: Cycloaddition and Rearrangement
0774
Norris, B. C.; Bielawski, C. W.: Reversible Conjugated Polymer Synthesis
0775
Xu, Y.; Smith, M. D.; Geer, M. F.; Pellechia, P. J.; Brown, J. C.; Wibowo, A. C.; Shimizu, L. S.: Zipping Up Diacetylene Macrocycles
0776
Song, J.; Aratani, N.; Kim, P.; Kim, D.; Shinokubo, H.; Osuka, A.: Fused Porphyrin Rings
0777
Kanda, K.; Endo, K.; Shibata, T.: Chiral Cyclophanes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z779
All PDFs of this category
0779
Lou, S.; Fu, G. C.: Enantioselective Cross-Coupling of Activated Secondary Alkyl Electrophiles
0780
Zhao, D.; Mao, L.; Wang, Y.; Yang, D.; Zhang, Q.; Wang, R.: Zinc-Catalyzed Phospha-Michael Reaction of Phosphine Oxides
0781
Dutta, B.; Gilboa, N.; Marek, I.: Homoallylic Alcohols from Simple Terminal Alkynes
0782
Miklášová, N.; Julínek, O.; Mešková, M.; Setnička, V.; Urbanová, M.; Putala, M.: New Binol-Based Phosphoramidites for Asymmetric Conjugate Addition
0783
Mazuela, J.; Paptchikhine, A.; Pàmies, O.; Andersson, P. G.; Diéguez, M.: New Ligands for Asymmetric Iridium-Catalyzed Hydrogenation of Alkenes
0784
Seiser, T.; Cramer, N.: Rhodium Catalysts Cleave Cyclobutanol to Asymmetric Methyl Quaternary Centers
0785
Shintani, R.; Isobe, S.; Takeda, M.; Hayashi, T.: Rhodium-Catalyzed Asymmetric Synthesis of Spirocarbocycles
0786
Yasutomi, Y.; Suematsu, H.; Katsuki, T.: Ir(Salen)-Catalyzed Enantioselective Si-H Bond Insertion
0787
Yanagisawa, A.; Takeshita, S.; Izumi, Y.; Yoshida, K.: Asymmetric QuinoxP*˙Silver(I)-Catalyzed Nitroso Aldol Reaction
0788
Bugarin, A.; Connell, B. T.: MgI2-Accelerated Enantioselective ;Morita-Baylis-Hillman Reactions
0789
Zhu, M.-K.; Zhao, J.-F.; Loh, T.-P.: Palladium-Catalyzed Dioxygenation of Alkenes
0790
Chen, J.; Lang, F.; Zhang, X.; Cun, L.; Zhu, J.; Deng, J.; Liao, J.: Chiral Rhodium Bis-Sulfoxide Complex Catalyzed 1,4-Addition
0791
Kawato, Y.; Takahashi, N.; Kumagai, N.; Shibasaki, M.: Quaternary Stereocenters Generated by Conjugate Addition of α-Cyano Ketones
0792
Nguyen, N. N. M.; Leclère, M.; Stogaitis, N.; Fallis, A. G.: Diastereoselective Domino Synthesis of Triquinanes
0793
Zhang, X.; Cao, B.; Yu, S.: Rhodium-Catalyzed Asymmetric Hydroformylation of N-Allyl Amides
0794
Zheng, B.-H.; Ding, C.-H.; Hou, X.-L.; Dai, L.-X.: Synthesis of β-Substituted Tryptophans from Sulfonylindoles
0795
Lee, J. C. H.; Hall, D. G.: Asymmetric Conjugate Additions of 3-Boronyl Unsaturated Esters
0796
Luo, Y.; Carnell, A. J.: Electronically Tunable Chiral Ligands for Rhodium-Catalyzed Conjugate Addition
0797
Shintani, R.; Takeda, M.; Nishimura, T.; Hayashi, T.: Asymmetric 1,4-Addition of Arylboroxines to β,β-Disubstituted α,β-Unsaturated Ketones
0798
Xie, M.; Chen, X.; Zhu, Y.; Gao, B.; Lin, L.; Liu, X.; Feng, X.: Tetrahydroquinolines by Inverse Electron-Demand Aza-Diels-Alder Reaction
0799
Sonawane, M. R.; CÍsaŘovÁ, I.; Lyapkalo, I. M.: Diastereoselective Aldol Reaction of ;N-Trimethylsilyloxyenamines
0800
Shibatomi, K.; Futatsugi, K.; Kobayashi, F.; Iwasa, S.; Yamamoto, H.: Halogenated Quaternary Centers via Asymmetric Diels-Alder Reaction
0801
Zhang, Y. J.; Yang, J. H.; Kim, S. H.; Krische, M. J.: Iridium-Catalyzed Enantioselective Carbonyl (Hydroxymethyl)allylation
0802
Shirakura, M.; Suginome, M.: Nickel-Catalyzed Asymmetric Hydroalkynylation of 1,3-Dienes
0803
Trost, B. M.; Chan, V. S.; Yamamoto, D.: Asymmetric Addition of 1,3-Diynes to Aldehydes
0804
Xie, J.-B.; Xie, J.-H.; Liu, X.-Y.; Kong, W.-L.; Li, S.; Zhou, Q.-L.: Iridium-Catalyzed Asymmetric Hydrogenation of α-Arylmethylene Cycloalkanones
0805
Mundal, D. A.; Avetta, C. T.; Thomson, R. J.: Acid-Catalyzed Stevens Sigmatropic Rearrangement of N-Allylhydrazones
0806
Chen, X.; Liu, Q.; Sun, H.-B.; Yu, X.-Q.; Pu, L.: A Novel Catalyst for Tandem Oxidation and Alkylation
0807
Yamaoka, Y.; Yamamoto, H.: Super Silyl Directing Groups: Highly Diastereoselective Aldol Reactions
0808
Guo, S.; Xie, Y.; Hu, X.; Xia, C.; Huang, H.: Highly Selective Copper-Catalyzed Tandem Michael Addition/Mannich Reaction

Metal-Mediated Synthesis

z809
All PDFs of this category
0809
Williamson, K. S.; Yoon, T. P.: Iron-Catalyzed Aminohydroxylation of Olefins
0810
Hilt, G.; Paul, A.; Treutwein, J.: Cobalt-Catalyzed Alder-Ene Reaction and [2+2] Cycloaddition
0811
Zhao, X.; Yeung, C. S.; Dong, V. M.: Palladium-Catalyzed Oxidative Arylation of ortho-Phenylcarbamates with Arenes
0812
Yang, W.; Liu, C.; Qiu, J.: In situ Formation of a N,O-Bidentate Ligand for Efficient Suzuki Reactions
0813
Hatcher, J. M.; Coltart, D. M.: Copper-Catalyzed Addition of Grignard Reagents to N-Sulfonyl Azoalkenes
0814
Gruit, M.; Michalik, D.; Krüger, K.; Spannenberg, A.; Tillack, A.; Pews-Davtyan, A.; Beller, M.: Platinum- and Gold-Catalyzed Cyclizations of Alkynes
0815
Sperotto, E.; van Klink, G. P. M.; de Vries, J. G.; van Koten, G.: C-N Coupling of Nitrogen Nucleophiles with Aryl and Heteroaryl Bromides
0816
Bonin, H.; Delbrayelle, D.; Demonchaux, P.; Gras, E.: Base-Free Aryl Coupling of Diazonium Compounds and Boronic Esters
0817
Cronin, L.; Manoni, F.; O’Connor, C. J.; Connon, S. J.: Bromomagnesium Thiolate Catalyzed Tishchenko Reaction
0818
Shimasaki, T.; Tobisu, M.; Chatani, N.: Nickel-Catalyzed Amination of Aryl Pivalates via C-O Cleavage
0819
Hatano, M.; Ito, O.; Suzuki, S.; Ishihara, K.: Zinc(II)-Catalyzed Grignard Additions to Ketones with RMgBr and RMgI
0820
Yoshikai, N.; Mieczkowski, A.; Matsumoto, A.; Ilies, L.; Nakamura, E.: Iron-Catalyzed C-C Bond Formation via 1,5-Hydrogen Transfer
0821
Hatakeyama, T.; Yoshimoto, Y.; Ghorai, S. K.; Nakamura, M.: Transition-Metal-Free Amination of Aryl Grignard Reagents
0822
Xiao, K.-J.; Lua, J.-M.; Ye, K.-Y.; Wang, Y.; Huang, P.-Q.: One-Pot Reductive Alkylation of Lactams and Amides with Grignard Reagents
0823
Ye, S.; Yang, X.; Wu, J.: Palladium-Catalyzed Tandem Reactions of Dibromovinylalkynylbenzenes

Organo- and Biocatalysis

z825
All PDFs of this category
0825
Peschiulli, A.; Procuranti, B.; O’Connor, C. J.; Connon, S. J.: Kinetic Resolution of Thiols
0826
Yao, W.; Pan, L.; Wu, Y.; Ma, C.: An Organocatalytic Approach to ;Spiro-3,4-dihydropyrans
0827
North, M.; Villuendas, P.: The Influence of Chiral Solvents in Proline Catalysis
0828
Gu, Q.; Rong, Z.-Q.; Zheng, C.; You, S.-L.: Chiral Phosphoric Acid Catalyzed Intramolecular Oxo-Michael Reactions
0829
Wakchaure, V. N.; List, B.: Novel Bifunctional Chiral Brønsted Acid/Base Organocatalysis
0830
Gutierrez, E. G.; Moorhead, E. J.; Smith, E. H.; Lin, V.; Ackerman, L. K. G.; Knezevic, ;C. E.; Sun, V.; Grant, S.; Wenzel, A. G.: New Backbones for Brønsted Acid Catalysts
0831
Hu, S.; Li, J.; Xiang, J.; Pan, J.; Luo, S.; Cheng, J.-P.: Cyclodextrin-Supported Primary Amine Catalyzed Aldol Reaction
0832
Nair, V.; Varghese, V.; Paul, R. R.; Jose, A.; Sinu, C. R.; Menon, R. S.: NHC-Catalyzed Oxidation of Aromatic Aldehydes to Acids with CO2
0833
Bradshaw, B.; Etxebarria-Jardí, G.; Bonjoch, J.: Total Synthesis of (-)-Anominine with an Organocatalytic Key Step
0834
Hatano, M.; Moriyama, K.; Maki, T.; Ishihara, K.: Acid or Salt? New Insights into ‘Phosphoric Acid Catalysis’
0835
Misaki, T.; Takimoto, G.; Sugimura, T.: Chiral Guanidine Catalyzed Direct Aldol Reaction

Polymer-Supported Synthesis

z837
All PDFs of this category
0837
Ma, J.; Ng, S.; Yong, Y.; Luo, X.-Z.; Wang, X.; Liu, X.-W.: Alkylation of Indoles with a Sulfonated Carbon-Based Solid Acid
0838
Soh, C. H.; Lam, Y.: Synthesis of Imidazo[1,2-a]pyrimidin-5-ones on a Polymer Support
0839
Akagawa, K.; Fujiwara, T.; Sakamoto, S.; Kudo, K.: Supported Peptide for Asymmetric α-Oxyamination of Aldehydes
0840
Chari, M. A.; Karthikeyan, G.; Pandurangan, A.; Naidu, T. S.; Sathyaseelan, B.; Zaidi, S. M. J.; Vinu, A.: Synthesis of Indazole-1,3,8-triones Using an Aluminosilicate Catalyst
0841
Balakrishnan, U.; Ananthi, N.; Selvan, S. T.; Pal, R.; Ariga, K.; Velmathi, S.; Vinu, A.: Asymmetric Reduction by SBA-15-Supported Chiral Oxazaborolidine
0842
Veisi, H.: Paal-Knorr Pyrrole Synthesis Catalyzed by Silica Sulfuric Acid
0843
Turner, R. A.; Weber, R. J.; Lokey, R. S.: Direct Conversion of Resin-Bound Peptides into C-Terminal Esters
0844
Kitamura, Y.; Sako, S.; Tsutsui, A.; Monguchi, Y.; Maegawa, T.; Kitade, Y.; Sajiki, H.: Hetero-Suzuki-Miyaura Cross-Coupling Using Palladium on Carbon
0845
Lee, J.-M.; Kim, J.; Shin, Y.; Yeom, C.-E.; Lee, J. E.; Hyeon, T.; Kim, B. M.: Asymmetric Henry Reaction with an M-HMMS-Supported Copper Complex
0846
Afonso, A.; Rosés, C.; Planas, M.; Feliu, L: Synthesis of Biaryl Peptides via Solid-Phase Borylation and Cross-Coupling
0847
Miura, H.; Wada, K.; Hosokawa, S.; Inoue, M.: Direct Arylation of Aromatic C-H Bonds with 3Ph3P-Ru/CeO2
0848
Pellegrino, G.; Leonetti, F.; Carotti, A.; Nicolotti, O.; Pisani, L.; Stefanachi, A.; Catto, M.: Solid-Phase Synthesis of Pyrimidines, Pyrazoles, and Isoxazoles
0849
Liu, P.; Zhou, C.-Y.; Xiang, S.; Che, C.-M.: Oxidative C-C Coupling with an SBA-Supported Iron Complex