DOI: 10.1055/s-00000131

Synfacts

Issue 12 · Volume 2011 · December 2011 DOI: 10.1055/s-002-22456

Synform

  • A109

    SYNFORM ISSUE 2011/12

    • Synthesis of Natural Products and Potential Drugs

  • z1265

    All PDFs of this category

  • 1265

    Synthesis of (+)-Ophiobolin A

  • 1266

    Synthesis of MK-3281

  • 1267

    Synthesis of PF-03463275

  • 1268

    Synthesis of (+)-Gliocladin C

  • 1269

    Synthesis of Fesoterodine

  • 1270

    Synthesis of the Bismurrayaquinone A

  • 1271

    Synthesis of (-)-Maoecrystal Z

  • 1272

    Synthesis of (-)-Hodgkinsine B

  • 1273

    Synthesis of BIRT2584

  • 1274

    Synthesis of Crizotinib (PF-02341066)

  • 1275

    Synthesis of PF-04191834

  • 1276

    Synthesis of MK-8245

  • 1277

    Synthesis of a Renin Inhibitor

  • 1278

    Synthesis of (+)-Grandisine D

  • 1279

    Synthesis of a TRPV1 Antagonist

  • 1280

    Synthesis of TAK-475

  • 1281

    Synthesis of (-)-N-Methylwelwitindolinone C Isothiocyanate

    • Synthesis of Heterocycles

  • z1283

    All PDFs of this category

  • 1283

    Pd-Catalyzed Synthesis of Phenanthridinones by Double C-H Activation

  • 1284

    Palladium-Catalyzed Enantioselective Synthesis of Silacyles

  • 1285

    Ethers via Catalytic Asymmetric Thiofunctionalization of Alkenyl Alcohols

  • 1286

    Synthesis of Pyrimidines via N-Vinyl Tertiary Enamides

  • 1287

    Pd-Catalyzed Enantioselective Synthesis of 2-Methyl Indolines

  • 1288

    Metal-Free Synthesis of 2-Trifluoromethyl Furans

  • 1289

    Synthesis of Chromones from 2,3-Allenoic Acids and Benzynes

  • 1290

    Iron-Catalyzed Synthesis of Aminoindolizines and Quinolines

  • 1291

    Metal-Free Synthesis of Pyrroles From Morita-Baylis-Hillman Acetates

  • 1292

    Copper-Catalyzed One-Pot Synthesis of 5-Sulfonamidopyrazoles

  • 1293

    Two-Step Heck-Mediated Synthesis of Pyrroles from Sulfonamides and Bromoacetylenes

  • 1294

    Cycloaddition Approach to Substituted Thiophenes

  • 1295

    Heteroannulation Route to Benzothiophenes from 2-Bromo Alkynylbenzenes

  • 1296

    A Multicatalytic Domino Heteroannulation Approach to Dihydroquinolines

  • 1297

    Pd-Catalyzed C-H Activation Route to Dibenzophosphole Oxides

    • Synthesis of Materials and Unnatural Products

  • z1299

    All PDFs of this category

  • 1299

    Nickel-Catalyzed Synthesis of Strained Phenacenes

  • 1300

    One Step to Polyenes

  • 1301

    An All-Organic Porphyrin and its Properties

  • 1302

    Polymerization of Diisocyanobenzenes Bearing Alkoxy Side Chains

  • 1303

    A One-Pot Approach to ‘Shutting the Lights Off’ in the Presence of Mercury Ion

  • 1304

    Delocalized Radicals

  • 1305

    Synthesis of a New exo-Heterocyclic Diene

  • 1306

    High-Yielding One-Pot Synthesis of Oxazine Photochromes

  • 1307

    Anion-Templated Yin Yang: Janus [2]Rotaxanes

  • 1308

    Putting a B in Polymer

  • 1309

    The Smaller the Redder

  • 1310

    A One-Pot Route to 3-Vinyl Coumarins

  • 1311

    Route to Functionalized Sumanenes

    • Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

  • z1313

    All PDFs of this category

  • 1313

    Asymmetric α-Allylation of Aldehydes with Simple Allylic Alcohols

  • 1314

    Copper-Catalyzed Asymmetric α-Arylation of N-Acyloxazolidinones

  • 1315

    Cu-Catalyzed Asymmetric α-Arylation of Carbonyls

  • 1316

    Palladium-Catalyzed Enantioselective Fluorination of Allylic Halides

  • 1317

    Enantioselective Fluorination of Epoxides via Cooperative Catalysis

  • 1318

    Enantioselective Rhodium-Catalyzed Conjugate Addition

  • 1319

    A Simplified Catalytic System for Direct Asymmetric Aldol Reaction of Thioamides

  • 1320

    Hydroamination of Dienes by Gold(I)/Menthol Cooperative Catalysis

  • 1321

    Silver-Catalyzed Enantioselective [3+2] Cycloadditions

  • 1322

    Helical Macromolecular Ligand for Asymmetric Suzuki Coupling

  • 1323

    Pd-Catalyzed Asymmetric Allylic Amination

  • 1324

    Palladium-Catalyzed Enantioselective α-Arylation

  • 1325

    Readily Accessible Diene Ligands for Enantioselective Conjugate Additions

  • 1326

    Enantioselective Intramolecular Benzylic C-H Bond Amination

  • 1327

    Asymmetric Epoxidation Catalyzed by Titanium(salalen) Complex

  • 1328

    Titanium-Catalyzed Enantioselective Oxidation of Aryl Sulfides

  • 1329

    Diastereo- and Enantioselective Direct Aldol Reactions Mediated by CoCl2/l-Proline

  • 1330

    Niobium-Catalyzed Asymmetric Aldol-Type Reactions

  • 1331

    Rh-Catalyzed Enantioselective Addition of Arylboronic Acids to Enones

  • 1332

    Cu-Catalyzed Asymmetric Tandem Dual Michael Reaction of Dialkylzinc to Enones

  • 1333

    Cu(I)/BINAP-Catalyzed Synthesis of Pyro-glutamates

  • 1334

    Copper-Catalyzed Asymmetric Henry Reaction

  • 1335

    Stereoselective Rhodium-Catalyzed Amination of Alkenes

  • 1336

    Catalyst-Controlled Diastereo- and Enantioselective Hydrogenation

  • 1337

    Manganese-Catalyzed Enantioselective cis-Dihydroxylation

  • 1338

    Copper-Catalyzed Tandem 1,4-Addition-Fluorination Sequence

  • 1339

    Pd-Catalyzed Intramolecular Asymmetric Allylic Amination

  • 1340

    Ir(I)-Catalyzed C-H Bond Activation of 2-(Alkylamino)pyridines with Alkenes

  • 1341

    Synthesis of Optically Pure Bulky Carbinols via Kinetic Resolution

  • 1342

    Stereocontrol of the Combined C-H Functionalization/Cope Rearrangement

    • Metal-Mediated Synthesis

  • z1343

    All PDFs of this category

  • 1343

    Catalytic Enantioselective γ-Alkylation of Carbonyl Compounds

  • 1344

    Synthesis of Trifluoroethyl-Substituted Ketones

  • 1345

    Takai-Analogous One-Step Preparation of (E)-Vinylsilanes

  • 1346

    Direct Conversion of Carboxylic Acids into Ketones

  • 1347

    Bridgehead Radicals for Coupling of Oxygenated Carbocycles

  • 1348

    Copper-Catalyzed Intramolecular Oxidative Cyclization

  • 1349

    An Organocatalyzed Michael Addition-Cyclization Sequence to Spirolactones

  • 1350

    One-Pot Synthesis of 2,4-Dienols from Cycloalkenones

  • 1351

    Improved Conversion of Aryl and Vinyl Triflates into Bromides and Chlorides

  • 1352

    Cu-Mediated Cyanation of Aryl Halides

  • 1353

    Ti-Mediated Tandem Ethylation and Functionalization of Allylic Alcohols

  • 1354

    New Insights into Anion Relay Chemistry

  • 1355

    Difluoromethylation of Carbonyls and Imines with TMSCF2H

  • 1356

    Mukaiyama Cross-Aldol Reaction to Yield anti-β-Siloxy-α-haloaldehydes

  • 1357

    Nickel-Catalyzed Formation of Cyclo-pentenones via Cycloaddition

    • Organo- and Biocatalysis

  • z1359

    All PDFs of this category

  • 1359

    Friedel-Crafts Alkylation, Internal Redox Reaction, and Umpolung Cascade

  • 1360

    Asymmetric Reduction of Unprotected Indoles

  • 1361

    Enantiopure RNA Precursors from Nearly Racemic Starting Materials

  • 1362

    Morpholine-Catalyzed C3 Alkenylation of Indoles with Enals

  • 1363

    Phosphine-Catalyzed Heine Reaction

  • 1364

    Asymmetric Reduction of Ketones

  • 1365

    Dual-Catalytic Asymmetric Reactions

  • 1366

    Organocatalytic Pictet-Spengler Reaction in Natural Product Synthesis

  • 1367

    Organo-Click Synthesis of 1,2,3-Triazoles from Unactivated Ketones

  • 1368

    Phosphoric Acid Catalyzed Enantioselective Friedländer Condensations

  • 1369

    Synthesis of Piperidines through Intramolecular Aza-Michael Addition

  • 1370

    Catalytic Cycloetherification Using Bifunctional Thiourea Catalysts

    • Polymer-Supported Synthesis

  • z1371

    All PDFs of this category

  • 1371

    Reduction of Nitroarenes with N2H4˙H2O Using Fe-Phen/C

  • 1372

    Oxidative Amidation of Alcohols with Amines Catalyzed by Au/DNA

  • 1373

    Suzuki-Miyaura Reaction with NHC-Cu-Pd MOF Catalysts

  • 1374

    Pd/C-Catalyzed Hiyama Cross-Coupling

  • 1375

    Solid-Supported Prolinol Ether Catalysts

  • 1376

    Ullmann Reaction of Aryl Iodides with Au@PMO

  • 1377

    Suzuki-Miyaura Coupling in Water with Pd@SBA-15©

  • 1378

    Oxidation with SiO2-Supported Iodoarene-RuCl3 Bifunctional Catalysts

  • 1379

    Microwave-Assisted Thionation of Amides Using a Solid-Supported P2S5

  • 1380

    A Poly(Imidazole-Palladium) Catalyst for Allylic Arylation/Alkenylation

  • 1381

    CuO on Alumina for C-O Coupling of Halides with Alcohols

  • 1382

    Disulfide Bond Formation with Polymer-Supported Reagent

  • 1383

    Suzuki Coupling of Alkynyl Bromides with Boronic Acids by Pd-SiO2@Fe3O4

  • 1384

    C-N and C-S Bond-Forming Cross-Coupling in Water with PS-PEG-Pd

    • Addenda and Errata

  • 1385

    Trienamines in Organocatalysis

  • 1385

    exo-Selective Diels-Alder Reaction of 2,4-Dienals and Nitroalkenes