DOI: 10.1055/s-00000131

Synfacts

Issue 03 · Volume 2011 · March 2011 DOI: 10.1055/s-002-21701

Synform

A20
Zanda, Matteo: SYNFORM ISSUE 2011/03

Synthesis of Natural Products and Potential Drugs

z237
All PDFs of this category
0237
Stuart, D. R.; Alsabeh, P.; Kuhn, M.; Fagnou, K.: Synthesis of Paullone
0238
Nilson, M. G.; Funk, R. L.: Synthesis of (-)-Nakadomarin
0239
Gong, J.; Lin, G.; Sun, W.; Li, C.-C.; Yang, Z.: Total Synthesis of (±)-Maoecrystal V
0240
Campeau, L.-C.; O’Shea, P. D.: Synthesis of an HCV RNA Polymerase Inhibitor
0241
Crimmins, M. T.; Mans, M. C.; Rodríguez, A. D.: Synthesis of the Proposed Structure of Briarellin J
0242
Sawant, P.; Maier, M. E.: Synthesis of Atorvastatin Lactone
0243
Schindler, C. S.; Bertschi, L.; Carreira, E. M.: Synthesis of Nominal Banyaside B
0244
Haag, B. A.; Zhang, Z.-G.; Li, J.-S.; Knochel, P.: Synthesis of Indomethacin and Iprindole
0245
Reiter, M.; Torssell, S.; Lee, S.; MacMillan, D. W. C.: Synthesis of (+)-Frondosin B
0246
Pronin, S. V.; Kozmin, S. A.: Synthesis of Streptolydigin
0247
Wu, H.; Xue, F.; Xiao, X.; Qin, Y.: Synthesis of (+)-Perophoramidine
0248
Webster, R.; Boyer, A.; Fleming, M. J.; Lautens, M.: Synthesis of Rotigotine and (S)-8-OH-DPAT

Synthesis of Heterocycles

z249
All PDFs of this category
0249
Too, P. C.; Wang, Y.-F.; Chiba, S.: Rhodium(III)-Catalyzed Heteroannulation Route to Isoquinolines
0250
Zhang, X.; Teo, W. T.; Chan, P. W. H.: Ytterbium(III)-Catalyzed Synthesis of 2-Aryloxazoles
0251
Shafi, S.; Kędziorek, M.; Grela, K.: Cross-Metathesis Strategy for Pyrrole Synthesis
0252
Nayak, M.; Batra, S.: Copper-Catalyzed Synthesis of Heterofused Benzoxazepines and -diazepines
0253
Maestri, G.; Larraufie, M.-H.; Derat, E.; Ollivier, C.; Fensterbank, L.; Lacôte, E.; Malacria, M.: Synthesis of Phenanthridines via Palladium/Norbornene Catalysis
0254
Siry, S. A.; Timoshenko, V. M.: Synthesis and Reactivity of 2-Polyfluoroalkyl Thiopyrylium Salts
0255
Halland, N.; Nazaré, M.; Alonso, J.; R’kyek, O.; Lindenschmidt, A.: Domino Approach to 1-Aminoindoles from 2-Halophenylacetylenes
0256
Alonso, J.; Halland, N.; Nazaré, M.; R’kyek, O.; Urmann, M.; Lindenschmidt, A.: Pd-Catalyzed Heteroannulative Synthesis of Benzimidazoles and Imidazopyridines
0257
Bartrum, H. E.; Blakemore, D. C.; Moody, C. J.; Hayes, C. J.: In-Flow Approach to β-Keto Esters and Use in the Synthesis of Pyrimidines
0258
Kazmaier, U.; Persch, A.: Synthesis of 5-Substituted Thiazolyl Peptides via the Thio-Ugi Reaction
0259
Chen, K.-P.; Chen, Y.-J.; Chuang, C.-P.: α-Nitrocinnamate Esters for the Synthesis of Highly Functionalized Isoxazoles
0260
Majumdar, K. C.; Ponra, S.; Ghosh, D.; Taher, A.: Multicomponent Aza-Diels-Alder Synthesis of Phenanthrolines and Pyranoquinolines
0261
Cao, H.; Vieira, T. O.; Alper, H.: Palladium-Catalyzed Heteroannulation Route to Benzazepinones
0262
Hu, H.; Shi, K.; Hou, R.; Zhang, Z.; Zhu, Y.; Zhoua, J.: One-Pot Synthesis of Indolizines from Pyridines, Benzyl Halides, and Alkenes
0263
Ouyang, H.-C.; Tang, R.-Y.; Zhong, P.; Zhang, X.-G.; Li, J.-H.: CuI/I2-Mediated Synthesis of Iodoisoquinoline-Fused Benzimidazoles

Synthesis of Materials and Unnatural Products

z265
All PDFs of this category
0265
Jarre, G.; Liang, Y.; Betz, P.; Lang, D.; Krueger, A.: ‘Hard-Core’ Diels-Alder
0266
Johnson, J. A.; Lu, Y. Y.; Burts, A. O.; Xia, Y.; Durrell, A. C.; Tirrell, D. A.; Grubbs, R. H.: Drug-Loaded, Bivalent-Bottle-Brush Polymers by Graft-through ROMP
0267
Omachi, H.; Matsuura, S.; Segawa, Y.; Itami, K.: Odd- and Even-Numbered Cyclopara-phenylenes
0268
Haddadin, M. J.; El-Nachef, C.; Kisserwani, H.; Chaaban, Y.; Kurth, M. J.; Fettinger, J. C.: A New Route to Thieno[3,2-b]quinolines via an Original Heterocycle
0269
Senkovskyy, V.; Sommer, M.; Tkachov, R.; Komber, H.; Huck, W. T. S.; Kiriy, A.: Nickel Initiators for Kumada Poly-condensation
0270
Pastor-Pérez, L.; Kemmer-Jonas, U.; Wurm, F.; Stiriba, S.-E.; Pérez-Prieto, J.; Frey, H.: Core Values
0271
Lalevée, J.; Blanchard, N.; Tehfe, M.-A.; Morlet-Savary, F.; Fouassier, J. P.: Round and Round We Go
0272
Reddy, V. P.; Kumar, A. V.; Rao, K. R.: Serendipitous Synthesis of Diaryl Selenides
0273
Jiang, W.; Zhou, Y.; Geng, H.; Jiang, S.; Yan, S.; Hu, W.; Wang, Z.; Shuai, Z.; Pei, J.: Dithioperylene Transistors
0274
Ishida, N.; Moriya, T.; Goya, T.; Murakami, M.: A Facile Route to Pyridine-Borane Complexes
0275
Lou, K.; Prior, A. M.; Wiredu, B.; Desper, J.; Hua, D. H.: The First Cycloiptycene
0276
Hergué, N.; Frère, P.; Roncali, J.: Rigid Thienothiophene Blocks for Electropolymerization

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z277
All PDFs of this category
0277
Seiser, T.; Cramer, N.: 1,4-Rhodium-Silicon Shift in an Enantioselective Synthesis of Indanols
0278
Zhang, C.; Yu, S.-B.; Hu, X.-P.; Wang, D.-Y.; Zheng, Z.: Novel Ligands for Asymmetric [3+2] Cycloaddition of Enones
0279
Bao, H.; Wu, J.; Li, H.; Wang, Z.; You, T.; Ding, K.: Asymmetric Opening of meso-Epoxides with Aromatic and Aliphatic Amines
0280
Aikawa, K.; Hioki, Y.; Mikami, K.: Asymmetric Construction of α-Trifluoro-methyl-Substituted Tertiary Alcohols
0281
Xu, H.; Wolf, C.: Asymmetric Synthesis of Tertiary Trifluoromethyl Alcohols
0282
Chen, C.; Voss, T.; Fröhlich, R.; Kehr, G.; Erker, G.: 1,1-Carboboration of 1-Alkynes
0283
Chang, M.; Li, W.; Hou, G.; Zhang, X.: Asymmetric Hydrogenation of Cyclic Imines
0284
Hesp, K. D.; Stradiotto, M.: Gold-Catalyzed Hydroamination of Internal Alkynes
0285
Cui, L.; Li, C.; Zhang, L.: Stereoselective Synthesis of Substituted Piperidin-4-ols
0286
Wang, Y.; Hu, X.; Du, H.: Acyclic Chiral Diene Ligands for Rhodium(I)-Catalyzed Conjugated Additions
0287
Chen, C.-T.; Kao, J.-Q.; Salunke, S. B.; Lin, Y.-H.: Oxidovanadium(V)-Catalyzed Kinetic Resolution of α-Hydroxy Ketones
0288
Ogasawara, M.; Okada, A.; Subbarayan, V.; Sörgel, S.; Takahashi, T.: Palladium-Catalyzed Asymmetric Synthesis of Allenylsilanes
0289
Duan, Z.-C.; Hu, X.-P.; Zhang, C.; Zheng, Z.: Rhodium-Catalyzed Asymmetric Hydrogenation of Phosphonobutenoates
0290
Yang, H.-Y.; Xu, M.-H.: Asymmetric Addition of Arylboronic Acids to 3-Indolylimines
0291
Watkins, A. L.; Landis, C. R.: Rhodium-Catalyzed Asymmetric Hydroformylation of 1,3-Dienes
0292
Usanov, D. L.; Yamamoto, H.: Chromium-Catalyzed Enantioselective Alkynylation of Aldehydes
0293
Shibata, I.; Tsunoi, S.; Sakabe, K.; Miyamoto, S.; Kato, H.; Nakajima, H.; Yasuda, M.; Baba, A.: Halogenotin Hydride Catalyzed Diastereoselective Reductive Aldol Reaction
0294
Thamapipol, S.; Bernardinelli, G.; Besnard, C.; Kündig, E. P.: Asymmetric Intramolecular Diels-Alder Reactions Catalyzed by Ruthenium
0295
Aikawa, K.; Kojima, M.; Mikami, K.: Synergistic Catalysis of Chiral Gold Complexes and Chiral Anions
0296
Huang, K.; Zhang, X.; Emge, T. J.; Hou, G.; Cao, B.: Design of a New Bisphosphine Ligand for Asymmetric Hydrogenation
0297
Bandini, M.; Monari, M.; Romaniello, A.; Tragni, M.: Gold-Catalyzed Synthesis of Functionalized Morpholines
0298
Nakagawa, Y.; Muramatsu, Y.; Harada, T.: Catalytic Enantioselective Synthesis of Diarylmethanols
0299
Hayashi, R.; Walton, M. C.; Hsung, R. P.; Schwab, J. H.; Yu, X.: Stereoselective 6π-Electron Electrocyclic Ring Closures
0300
Inagaki, T.; Ito, A.; Ito, J.-i.; Nishiyama, H.: Effect of Zinc Metal on the Stereocontrol of Iron-Catalyzed Hydrosilane Reduction
0301
Ito, S.; Itoh, T.; Nakamura, M.: Iron-Promoted Carbometalation of Bicyclic Alkenes
0302
Padilla, S.; Tejero, R.; Adrio, J.; Carretero, J. C.: Copper(I)-Catalyzed Asymmetric [3+2] Cycloaddition
0303
Uehara, M.; Suematsu, H.; Yasutomi, Y.; Katsuki, T.: Iridium-Catalyzed Enantioselective Cyclopropenation
0304
Xu, X.; Qian, Y.; Yang, L.; Hu, W.: Enantioselective Mannich-Type Three-Component Reaction
0305
Paley, R. S.; Laupheimer, M. C.; Erskine, N. A. K.; Rablen, P. R.; Pike, R. D.; Jones, J. S.: Selective Spiroketalization of Iron Diene Complexes

Metal-Mediated Synthesis

z307
All PDFs of this category
0307
Kalek, M.; Johansson, T.; Jezowska, M.; Stawinski, J.: Palladium-Catalyzed Propargylic Substitution with Phosphorus Nucleophiles
0308
Painter, R. M.; Pearson, D. M.; Waymouth, R. M.: Selective Palladium-Catalyzed Oxidation of Glycerol to Dihydroxyacetone
0309
Burton, P. M.; Morris, J. A.: Palladium-Catalyzed Benzylic Arylation
0310
Ho, C.-Y.; He, L.: Nickel-Catalyzed Tail-to-Tail Hydro-alkenylation of Styrenes with α-Olefins
0311
Feng, C.; Loh, T.-P.: Palladium-Catalyzed Bisolefination of C-C Triple Bonds to Yield Naphthalene Derivatives
0312
Kim, J. Y.; Cho, S. H.; Joseph, J.; Chang, S.: Cobalt- and Manganese-Catalyzed Direct Amination of Azoles
0313
Molander, G. A.; Trice, S. L. J.; Dreher, S. D.: Palladium-Catalyzed Boronic Acid and Trifluoroborate Synthesis from Aryl Chlorides
0314
Takada, Y.; Nomura, K.; Matsubara, S.: Highly Stereoselective Preparation of Cycloheptane-1,3-diones
0315
Nelson, J. M.; Vedejs, E.: Palladium-Catalyzed Cross-Coupling of Metalated Aziridines
0316
Taniguchi, T.; Sugiura, Y.; Zaimoku, H.; Ishibashi, H.: Iron-Catalyzed Oxidative Addition of Alkoxycarbonyl Radicals
0317
Henderson, J. L.; McDermott, S. M.; Buchwald, S. L.: Palladium-Catalyzed Amination of Unprotected Halo-7-azaindoles
0318
Huang, L.; Jiang, H.; Qi, C.; Liu, X.: Copper-Catalyzed Intermolecular Oxidative [3+2] Cycloaddition
0319
Álvarez-Bercedo, P.; Martín, R.: Nickel-Catalyzed Reductive Cleavage of Aryl Ethers
0320
Panteleev, J.; Geyer, K.; Aguilar-Aguilar, A.; Wang, L.; Lautens, M.: One-Pot Synthesis of 1,2,3-Triazoles by Copper and Palladium Catalysis
0321
Naber, J. R.; Buchwald, S. L.: Palladium-Catalyzed Packed-Bed Continuous-Flow C-N Cross-Coupling

Organo- and Biocatalysis

z323
All PDFs of this category
0323
Siegel, J. B.; Zanghellini, A.; Lovick, H. M.; Kiss, G.; Lambert, A. R.; St.Clair, J. L.; Gallaher, J. L.; Hilvert, D.; Gelb, M. H.; Stoddard, B. L.; Houk, K. N.; Michael, F. E.; Baker, D.: A Biocatalytic Diels-Alder Reaction Using a Designed Enzyme
0324
Ohmatsu, K.; Kiyokawa, M.; Ooi, T.: Asymmetric Alkylation of Oxindoles Catalyzed by 1,2,3-Triazolium Salts
0325
Kobayashi, S.; Kiyohara, H.; Yamaguchi, M.: Silicon-Catalyzed Mannich Reaction of Unactivated Amides
0326
Lu, G.; Birman, V. B.: Phosphoric Acid Catalyzed Dynamic Kinetic Resolution of Azlactones
0327
Monge, D.; Jensen, K. L.; Marín, I.; Jørgensen, K. A.: Base-Catalyzed Synthesis of 1,2,4-Triazolines
0328
Capitta, F.; Frongia, A.; Ollivier, J.; Piras, P. P.; Secci, F.: Organocatalytic Asymmetric Ring Expansion of Cyclobutanones
0329
Cheng, Y.; An, J.; Lu, L.-Q.; Luo, L.; Wang, Z.-Y.; Chen, J.-R.; Xiao, W.-J.: Asymmetric Cyclopropanation Catalyzed by C2-Symmetric Ureas
0330
Terada, M.; Nii, H.: Formal [4+2] Cycloaddition of Azlactones to β,γ-Unsaturated α-Keto Esters
0331
Dickmeiss, G.; Jensen, K. L.; Worgull, D.; Franke, P. T.; Jørgensen, K. A.: Catalytic Asymmetric Synthesis of Octahydroacridines
0332
Li, X.-m.; Wang, B.; Zhang, J.-m.; Yan, M.: Synthesis of Cyclohexanones via Double-Conjugate Addition of Dienones
0333
Applegate, G. A.; Cheloha, R. W.; Nelson, D. L.; Berkowitz, D. B.: Highly Efficient Biocatalytic Reduction of Keto Esters

Polymer-Supported Synthesis

z335
All PDFs of this category
0335
Méndez, L.; Mata, E. G.: Synthesis of β-Lactam Derivatives from a Resin-Supported Ketene
0336
Wang, L.; Yi, W.-b.; Cai, C.: Arylation of Indoles with Supported Palladium Nanoparticles
0337
Choi, J.; Yang, H. Y.; Kim, H. J.; Son, S. U.: Self-Supported NHC-Palladium Catalyst for the Strecker Synthesis
0338
Li, J.; Wang, L.; Liu, S.; Li, X.; Shi, F.; Deng, Y.: An MCM-41 Grafted Quaternary Ammonium Salt as a Catalyst
0339
Bhadra, S.; Adak, L.; Samanta, S.; Islam, A. K. M. M.; Mukherjee, M.; Ranu, B. C.: Synthesis of Oxazines and Dioxanes from Aziridines and Epoxides
0340
Chen, W.; Li, P.; Wang, L.: Suzuki-Miyaura Reaction with a Silica- Supported Palladium Complex
0341
Yoon, H.-J.; Choi, J.-W.; Kang, H.; Kang, T.; Lee, S.-M.; Jun, B.-H.; Lee, Y.-S.: Immobilized NHC-Ni for C-S Coupling of Aryl Halides with Thiols
0342
Ni, J.; He, L.; Liu, Y.-M.; Cao, Y.; He, H.-Y.; Fan, K.-N.: Deoxygenation of Epoxides with Supported Gold Nanoparticles
0343
He, J.; Yamaguchi, K.; Mizuno, N.: Selective Synthesis of Secondary Amines with Cu(OH)x/Al2O3
0344
Maltsev, O. V.; Kucherenko, A. S.; Chimishkyan, A. L.; Zlotin, S. G.: Domino Reaction with Ionic Liquid Immobilized Prolinol Derivatives
0345
Cohrt, A. E.; Jensen, J. F.; Nielsen, T. E.: Traceless Solid-Phase Click Synthesis of NH-1,2,3-Triazoles
0346
He, L.; Lou, X.-B.; Ni, J.; Liu, Y.-M.; Cao, Y.; He, H.-Y.; Fan, K.-N.: One-Pot N-Alkylation of Amine with Alcohols Using Au/TiO2-VS
0347
Das, R. N.; Sarma, K.; Pathak, M. G.; Goswami, A.: Silica Gel Supported KHSO4 for Hydroalkoxylation of Styrenes

Addenda and Errata

0348
Taming the Silicon Tetraazide Beast
0348
Coupling of Aryl Halides and Diaryl Diselenides with CuS/Fe