DOI: 10.1055/s-00000084

Synthesis

eFirst

Publication Date: 08 August 2022

paper

Han, Qiang; Li, Shichen; Cai, Zepeng; Ding, Chengcheng; Feng, Lei; Ma, Chen: One-Pot Synthesis of 2-Arylquinolines via in situ Acid Catalysis
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0253_ga_10-1055_a-1889-9354.gif

paper

Kushwaha, Ambuj Kumar; Maury, Suresh Kumar; Kumari, Savita; Kamal, Arsala; Singh, Himanshu Kumar; Kumar, Dhirendra; Singh, Sundaram: Visible-Light-Initiated Oxidative Coupling of Indole and Active Methylene Compounds Using Eosin Y as a Photocatalyst
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0098_ga_10-1055_a-1894-8303.gif

review

Germer, Philipp; Andexer, Jennifer N.; Müller, Michael: Biocatalytic One-Carbon Transfer – A Review
https://www.thieme-connect.de/media/synthesis/EFirst/i_r0538_ga_10-1055_s-0040-1719884.jpg

Publication Date: 03 August 2022

short review > Special Issue dedicated to Prof. Alain Krief

Publication Date: 02 August 2022

paper

He, Yong; Chen, Shiyun; Gao, Yonghao; Gui, Shuangying; Feng, Yisi: A Novel and Practical Synthesis of Tryptanthrin
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0210_ga_10-1055_a-1878-8448.gif

Publication Date: 01 August 2022

paper

Boujdi, Khalid; El Brahmi, Nabil; Collet, Sylvain; Dubreuil, Didier; Mathé-Allainmat, Monique; Akssira, Mohamed; Guillaumet, Gérald; Lebreton, Jacques; El Kazzouli, Saïd: Solvent/Ligand-Controlled Switchable C3 or C7 C–H Arylations of 1-Methyl-4-nitro-1H-indazole
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0218_ga_10-1055_a-1891-0797.gif

paper

Publication Date: 27 July 2022

paper

Fu, Xuegang; Guo, Dongyang; Yan, Yuting; Marselo, Timotius; Zhang, Mingyu; Zhang, Zhenghan; Li, Siying; Huang, Jianhui: Carbon Chain Rupture: Base-Induced Radical C–C Bond Cleavage of Alkylbenzimidazoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_b0179_ga_10-1055_a-1883-1357.gif

review

Entgelmeier, Lukas-M.; Mancheño, Olga García: Activation Modes in Asymmetric Anion-Binding Catalysis
https://www.thieme-connect.de/media/synthesis/EFirst/i_r0181_ga_10-1055_a-1846-6139.gif

Publication Date: 26 July 2022

Publication Date: 21 July 2022

short review

Reyes, Efraim; Prieto, Liher; Carrillo, Luisa; Uria, Uxue; Vicario, Jose L.: Recent Developments in Transannular Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_r0156_ga_10-1055_a-1843-1954.gif

Publication Date: 20 July 2022

paper

special topic > Special Issue dedicated to Prof. Cristina Nevado, recipient of the 2021 Dr. Margaret Faul Women in Chemistry Award

Publication Date: 12 July 2022

feature

Pal, Parul; Fragis, Meghan; Dharavath, Srinivas; Johnson, Jarrod W.; Magolan, Jakob: Use of Vinyl Sulfides in Fischer Indole Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0196_ga_10-1055_a-1868-4148.gif

paper > Special Issue dedicated to Prof. Alain Krief

special topic > Aryne Chemistry in Synthesis

Publication Date: 08 July 2022

Publication Date: 05 July 2022

paper

Wang, Liqin; Song, Guangjun; Wu, Qiufang; Qin, Jiaxin; Yu, Xinhong; Chen, Niangen; Li, Cuiqing: Palladium/Norbornene-Cocatalyzed Three-Component Synthesis of ortho-Acylated Benzonitriles
https://www.thieme-connect.de/media/synthesis/EFirst/i_b0164_ga_10-1055_a-1866-7737.gif

special topic > Aryne Chemistry in Synthesis

Publication Date: 30 June 2022

short review

Publication Date: 28 June 2022

paper

Wang, Cai-Xia; Sheng, Fei-Fei; Liu, Kai-Hui; Gu, Jian-Guo; Shen, Kang; Sun, Zheng-Yi; Hong, Kunlun; Zhang, Hong-Hai: Bromide as the Directing Group for β-Arylation of Thiophenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0058_ga_10-1055_a-1838-8958.gif

Publication Date: 23 June 2022

Publication Date: 21 June 2022

Publication Date: 20 June 2022

special topic > Aryne Chemistry in Synthesis

Agudelo, Brian Castro; Rigoulet, Florian; Giorgi, Michel; Sayah, Babak; Rodriguez, Jean; Coquerel, Yoann: Synthesis of Axially Chiral Cationic Benzo[c]phenanthridinium Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0170_ga_10-1055_a-1845-3128.gif

special topic > Aryne Chemistry in Synthesis

special topic > Aryne Chemistry in Synthesis

Rai, Shweta; Samatha, Polasani; Addipilli, Ramunaidu; Mainkar, Prathama S.; Sripadi, Prabhakar; Adepu, Raju; Chandrasekhar, Srivari: Poly(ethylene glycol) Dimethyl Ethers (PEGDME): Efficient and Recyclable Solvents for Aryne-Involved Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0147_ga_10-1055_a-1846-5598.gif

Publication Date: 14 June 2022

feature

Mouthaan, Marc L. M. C.; Pouwer, Kees; Borst, Mark L. G.; Witte, Martin D.; Minnaard, Adriaan J.: α-C–H Photoalkylation of a Glucose Derivative in Continuous Flow
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0141_ga_10-1055_a-1840-5483.gif

Publication Date: 09 June 2022

feature

Guan, Yong; Buivydas, Tadas; Lalisse, Remy F.; Ali, Rameez; Hadad, Christopher M.; Mattson, Anita E.: Enantioselective Dearomative Alkynylation of Chromanones: Opportunities and Obstacles
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0778_ga_10-1055_a-1811-8075.gif

paper > Special Issue dedicated to Prof. Alain Krief

Osi, Arnaud; Tumanov, Nikolay; Wouters, Johan; Chardon, Aurélien; Berionni, Guillaume: A Selenenium-Bridged 10-Boratriptycene Lewis Acid
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0143_ga_10-1055_a-1840-5680.gif

special topic > Aryne Chemistry in Synthesis

Nagai, Akira; Kobayashi, Akihiro; Sakata, Yuki; Minami, Yasunori; Uchida, Keisuke; Hosoya, Takamitsu; Yoshida, Suguru: Synthesis of Multisubstituted Benzenes from Phenols via Multisubstituted Benzynes
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0139_ga_10-1055_a-1834-2927.gif

Publication Date: 08 June 2022

paper > SYNTHESIS Conference Special Issue ISySyCat21

Carreiro, Elisabete P.; Gastalho, Carlos M.; Ernesto, Sofia; Costa, Ana R.; Antunes, Célia M.; Burke, Anthony J.: Synthesis and Antiproliferative Activity of Novel Quercetin-1,2,3-Triazole Hybrids using the 1,3-Dipolar Cycloaddition (Click) Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0074_ga_10-1055_s-0040-1719928.gif

paper

Maegawa, Tomohiro; Oishi, Ryohei; Maekawa, Ayumi; Segi, Kazutoshi; Hamamoto, Hiromi; Nakamura, Akira; Miki, Yasuyoshi: The Reaction of Ketoximes with Hypervalent Iodine Reagents: Beckmann Rearrangement and Hydrolysis to Ketones
https://www.thieme-connect.de/media/synthesis/EFirst/i_b0128_ga_10-1055_a-1835-2188.gif

Publication Date: 07 June 2022

special topic > Aryne Chemistry in Synthesis

Publication Date: 02 June 2022

Publication Date: 31 May 2022

paper

Balaraman, Kaluvu; Kyriazakos, Samantha; Palmer, Rachel; Thanzeel, F. Yushra; Wolf, Christian: Selective Csp3–F Bond Functionalization with Lithium Iodide
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0057_ga_10-1055_s-0041-1738383.gif

paper

Kirihara, Masayuki; Yamahara, Sho; Okada, Tomohide; Matsumuro, Hiroaki; Kinoshita, Yukari; Kitajima, Atsuhito; Takamura, Yuya; Odagiri, Tatsuya; Asawa, Tomotake; Sugiyama, Yukihiro; Kimura, Yoshikazu: Synthesis of Sulfonyl Halides from Disulfides or Thiols Using Sodium Hypochlorite Pentahydrate (NaOCl·5H2O) Crystals
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0140_ga_10-1055_a-1823-3604.gif

short review > Aryne Chemistry in Synthesis

Yang, Yun; Jones, Christopher R.: The Aryne Ene Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0171_ga_10-1055_a-1827-2987.gif

special topic > Aryne Chemistry in Synthesis

Publication Date: 30 May 2022

Publication Date: 23 May 2022

Publication Date: 19 May 2022

special topic > Asymmetric C–H Functionalization

Yang, Zhenjie; Cheng, Hong-Gang; Chen, Ruiming; Cao, Liming; Wei, Qiang; Wang, Qingqing; Zhou, Qianghui: Eight-Step Asymmetric Synthesis of (–)-Berkelic Acid
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0085_ga_10-1055_a-1799-0459.gif

Publication Date: 17 May 2022

Publication Date: 12 May 2022

special topic > Asymmetric C–H Functionalization

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Remete, Attila M.; Nonn, Melinda; Volk, Balázs; Kiss, Loránd: Developments in the Alkynyltrifluoromethylations of Alkenes and Alkynes
https://www.thieme-connect.de/media/synthesis/EFirst/i_r0123_ga_10-1055_a-1811-8679.gif

special topic > Asymmetric C–H Functionalization

Publication Date: 10 May 2022

special topic > Special Issue dedicated to Prof. Alain Krief

Publication Date: 04 May 2022

Publication Date: 03 May 2022

feature

Publication Date: 28 April 2022

Publication Date: 25 April 2022

Publication Date: 20 April 2022

special topic > Asymmetric C–H Functionalization

Publication Date: 07 April 2022

Publication Date: 06 April 2022

short review > Special Issue dedicated to Prof. Alain Krief

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Cserép, Gergely B.; Németh, Krisztina; Szatmári, Ágnes; Horváth, Flóra; Imre, Tímea; Németh, Krisztina; Kele, Péter: Beyond the Bioorthogonal Inverse-Electron-Demand Diels–Alder Reactions of Tetrazines: 2-Pyrone-Functionalized Fluorogenic Probes
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0622_ga_10-1055_a-1761-4672.jpg

Publication Date: 05 April 2022

special topic > Aryne Chemistry in Synthesis

Publication Date: 28 March 2022

short review > SYNTHESIS Conference Special Issue ISySyCat21

Publication Date: 24 March 2022

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Publication Date: 23 March 2022

paper > Special Issue dedicated to Prof. Cristina Nevado, recipient of the 2021 Dr. Margaret Faul Women in Chemistry Award

Morgenstern, Martin; Mayer, Camilla; Pöthig, Alexander; Bach, Thorsten: Synthetic Studies towards Pyrido[1,2-a]azepine Stemona Alkaloids
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0025_ga_10-1055_a-1777-2477.gif

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Raji, Mounir; Le, Tam Minh; Csámpai, Antal; Nagy, Viktória; Zupkó, István; Szakonyi, Zsolt: Stereoselective Synthesis and Applications of Pinane-Based Chiral 1,4-Amino Alcohol Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0668_ga_10-1055_s-0040-1719887.gif

Publication Date: 16 March 2022

special topic > SYNTHESIS Conference Special Issue ISySyCat21

Kachkovskyi, Georgii; Cieślak, Marcin; Graczyk, Piotr; Zawadzki, Przemysław; Kalinowska-Tłuścik, Justyna; Werłos, Mateusz: Photocatalytic Approach to α,α-Difluoroalkyl Alcohols
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0729_ga_10-1055_s-0041-1737546.gif

Publication Date: 07 March 2022

short review > SYNTHESIS Conference Special Issue ISySyCat21

Publication Date: 03 March 2022

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Publication Date: 01 March 2022

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Fichez, Jeanne; Dupommier, Dorian; Besset, Tatiana: Direct Synthesis of Disubstituted Trifluoromethylthiolated Alkenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_r0707_ga_10-1055_s-0040-1719891.gif

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Salamon-Krokosz, Katarzyna; Gołdyn, Mateusz; Siodła, Tomasz; Bartoszak-Adamska, Elżbieta; Koroniak, Henryk; Koroniak-Szejn, Katarzyna: Fluorinated Olefinic Lactams: The Case of Amino Acids – Preparation and Mechanistic Studies
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0658_ga_10-1055_s-0041-1737346.jpg

Publication Date: 24 February 2022

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Takao, Go; Hakozaki, Tomohiro; Miura, Keisuke; Urushibara, Yusuke; Fuchibe, Kohei; Ichikawa, Junji: Construction of Substituted [4]Acene Frameworks Based on Double Cationic Cyclizations of Fluoroalkenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0693_ga_10-1055_s-0037-1610791.gif

Publication Date: 21 February 2022

short review > SYNTHESIS Conference Special Issue ISySyCat21

Nori, Valeria; Sinibaldi, Arianna; Pesciaioli, Fabio; Carlone, Armando: Impact of Design of Experiments in the Optimisation of Catalytic Reactions in Academia
https://www.thieme-connect.de/media/synthesis/EFirst/i_r0735_ga_10-1055_a-1736-6703.gif

Publication Date: 16 February 2022

paper > SYNTHESIS Conference Special Issue ISySyCat21

Marques, Carolina S.; López, Óscar; Leitzbach, Luisa; Fernández-Bolaños, José G.; Stark, Holger; Burke, Anthony J.: Survey of New, Small-Molecule Isatin-Based Oxindole Hybrids as Multi-Targeted Drugs for the Treatment of Alzheimer’s Disease
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0728_ga_10-1055_s-0041-1737343.gif

Publication Date: 15 February 2022

paper

Filimonchuk, Sergiy L.; Nazarenko, Kostiantyn; Shvydenko, Tetiana; Shvydenko, Kostiantyn; Rusanov, Eduard B.; Kostyuk, Aleksandr: Convenient Approach to Bicyclic Sultams
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0740_ga_10-1055_s-0040-1719894.gif

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Szabó, Tímea; Görür, Funda Lidya; Horváth, Simon; Volk, Balázs; Milen, Mátyás: Synthesis of Racemic and Enantiopure Forms of β-Carboline Alkaloid Brevicolline
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0720_ga_10-1055_s-0041-1737830.gif

Publication Date: 09 February 2022

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Dargó, Gyula; Nagy, Sándor; Kis, Dávid; Bagi, Péter; Mátravölgyi, Béla; Tóth, Blanka; Huszthy, Péter; Drahos, László; Kupai, József: Application of Proline-Derived (Thio)squaramide Organocatalysts in Asymmetric Diels–Alder and Conjugate Addition Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0619_ga_10-1055_s-0040-1719886.gif

Publication Date: 07 February 2022

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Publication Date: 04 February 2022

Publication Date: 26 January 2022

Publication Date: 12 January 2022

special topic > Special Issue dedicated to Prof. Alain Krief

Zhao, Ziyang; Lv, Qingwei; Geng, Jialin; Liu, Yang; Hu, Chao; Du, Yuguo; Liu, Jun: Stereoselective Total Synthesis of (+)-Brevipolide H from d-Galactal
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0642_ga_10-1055_a-1700-3520.gif

Publication Date: 11 January 2022

paper > SYNTHESIS Conference Special Issue ISySyCat21

Publication Date: 05 January 2022

special topic > Special Issue dedicated to Prof. Alain Krief

Publication Date: 14 December 2021

special topic > Asymmetric C–H Functionalization

special topic > Asymmetric C–H Functionalization

Publication Date: 07 December 2021

special topic > Special Issue dedicated to Prof. Ferenc Fülöp

Publication Date: 01 December 2021

Publication Date: 22 November 2021

special topic > Asymmetric C–H Functionalization

special topic > Asymmetric C–H Functionalization

Publication Date: 11 November 2021

special topic > Aryne Chemistry in Synthesis

Heinz, Benjamin; Djukanovic, Dimitrije; Siemens, Fiona; Idriess, Mohamed; Martin, Benjamin; Knochel, Paul: Regioselective Amination or Alkoxylation of Halogenated Amino-, Thio- or Alkoxypyridines via Pyridyne Intermediates
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0548_ga_10-1055_s-0037-1610786.gif

Publication Date: 10 November 2021

special topic > Special Issue in memory of Prof. Ferenc Fülöp

Publication Date: 14 October 2021

special topic > Asymmetric C–H Functionalization

Publication Date: 13 October 2021

paper > Special Issue dedicated to Prof. Alain Krief

Everaert, Jonas; Debruyne, Maarten; Vanden Bussche, Flore; Van Hecke, Kristof; Heugebaert, Thomas S. A.; Van Der Voort, Pascal; Van Speybroeck, Veronique; Stevens, Christian V.: Synthesis of Nitrile-Functionalized Polydentate N-Heterocycles as Building Blocks for Covalent Triazine Frameworks
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0406_ga_10-1055_a-1626-5749.jpg

Publication Date: 11 October 2021

special topic > Asymmetric C–H Functionalization

Huang, Long-Tao; Hirata, Yuki; Kato, Yoshimi; Lin, Luqing; Kojima, Masahiro; Yoshino, Tatsuhiko; Matsunaga, Shigeki: Ruthenium(II)/Chiral Carboxylic Acid Catalyzed Enantioselective C–H Functionalization of Sulfoximines
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0414_ga_10-1055_a-1588-0072.gif

Publication Date: 14 June 2021

special topic > Special Issue dedicated to Prof. Alain Krief

Publication Date: 09 June 2021

special topic > Special Issue dedicated to Prof. Ferenc Fülöp

Publication Date: 02 June 2021

special topic > Special Issue dedicated to Prof. Alain Krief