DOI: 10.1055/s-00000084

Synthesis

eFirst

Publication Date: 20 July 2017

paper

Denisova, Alexandra O.; Tokunova, Yulia A.; Fateev, Ilja V.; Breslav, Alexandra A.; Leonov, Vladimir N.; Dorofeeva, Elena V.; Lutonina, Olga I.; Muzyka, Inessa S.; Esipov, Roman S.; Kayushin, Alexey L.; Konstantinova, Irina D.; Miroshnikov, Anatoly I.; Stepchenko, Vladimir A.; Mikhailopulo, Igor A.: The Chemoenzymatic Synthesis of 2-Chloro- and 2-Fluorocordycepins
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0220_ga_10-1055_s-0036-1590804.gif
Supporting Information

paper

Doan, Bao Nguyen Do; Tan, Xin Yi; Ang, Chin May; Bates, Roderick W.: Synthesis of (±)-γ-Lycorane by Using an Intramolecular Friedel–Crafts Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0284_ga_10-1055_s-0036-1589067.gif
Supporting Information

paper

Kadikova, Rita N.; Ramazanov, Ilfir R.; Vyatkin, Alexey V.; Dzhemilev, Usein M.: Zirconium-Catalyzed Alkyne Carbo- and Cycloalumination Reactions in Stereoselective Preparation of 1-Alkenyl Selenides
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0189_ga_10-1055_s-0036-1589062.gif
Supporting Information

paper

Kaneko, Yuki; Wakamori, Shinnosuke; Ikeuchi, Kazutada; Ohara, Kenya; Tanaka, Takashi; Yamada, Hidetoshi: Total Synthesis of Lagerstannin C: Follow-up of the Khanbabaee’s Synthesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0296_ga_10-1055_s-0036-1588477.gif
Supporting Information

special topic

Paul, Kartick; Jalal, Swapnadeep; Kundal, Sandip; Chakraborty, Baitan; Jana, Umasish: Iron-Catalyzed Intramolecular Alkyne–Carbonyl Metathesis: A New Cyclization Strategy for the Synthesis of Benzocarbazole and Azepino[1,2-a]indole Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0250_ga_10-1055_s-0036-1588472.gif
Supporting Information

Publication Date: 19 July 2017

paper

Amara, Rim; Bentabed-Ababsa, Ghenia; Hedidi, Madani; Khoury, Joseph; Awad, Haçan; Nassar, Ekhlass; Roisnel, Thierry; Dorcet, Vincent; Chevallier, Floris; Fajloun, Ziad; Mongin, Florence: Synthesis of N-Aryl and N-Heteroaryl γ-, δ-, and ε-Lactams Using Deprotometalation–Iodination and N-Arylation, and Properties Thereof
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0343_ga_10-1055_s-0036-1590798.gif
Supporting Information CIF File

paper

Bhagat, Ujjawal Kumar; Kamaluddin; Peddinti, Rama Krishna: Base-Mediated Ring Opening of meso-Epoxides with 4-Aryl-NH-1,2,3-triazoles: Synthesis of trans-2-(Aryltriazolyl)cycloalkanols
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0098_ga_10-1055_s-0036-1589045.gif
Supporting Information

paper

Wang, Deqiang; Sun, Peng; Jia, Peiyun; Peng, Jinsong; Yue, Yixia; Chen, Chunxia: Transition-Metal-Free One-Pot Tandem Synthesis of 4-Quinolone and 4H-Thiochromen-4-one Derivatives Through Sequential Nucleophilic Addition–Elimination–SNAr Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0221_ga_10-1055_s-0036-1588466.gif
Supporting Information

paper

Wang, Chun-Meng; Yang, Sheng-Wei; Tang, Kai-Xiang; Gao, Tian-Hong; Pang, Bo; Chen, Yu-Ting; Wu, Jing; Liu, Jia; Shi, Yu-Fan; Sun, Li-Ping: Convenient Synthesis of Oxazolo[5,4-h]pyrrolo[4,3,2-de]quino­lones via Hypervalent Iodine Mediated Intramolecular Oxidative Cyclization
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0177_ga_10-1055_s-0036-1588498.gif
Supporting Information

special topic

Li, Jie; Xiao, Jun-An; Zhao, Shu-Juan; Xiang, Hao-Yue; Yang, Hua: Facile Construction of Pyrrolo[1,2-a]indolenine Scaffold via Dia­stereoselective [3+2] Annulation of Donor–Acceptor Cyclopropane with Indolenine
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0244_ga_10-1055_s-0036-1588876.gif
Supporting Information

Publication Date: 11 July 2017

feature

An, Yu; He, Huan; Liu, Tiantian; Zhang, Yong; Lu, Xiaoyun; Cai, Qian: Diversified Synthesis of 2-(4-Oxo[1,2,3]triazolo[1,5-a]quinoxalin-5(4H)-yl)acetamide Derivatives through Ugi-4-CR and Copper-Catalyzed Tandem Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_e0272_ga_10-1055_s-0036-1590791.gif
Supporting Information

paper

Li, Runrun; Wei, Qiang; Wang, Xin; Ge, Zemei; Li, Runtao: An Efficient Cascade Synthesis of Ethyl 3-Amino-5-oxoisoxazolidine-4-carboxylate Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0218_ga_10-1055_s-0036-1590803.gif
Supporting Information

paper

Sobenina, Lyubov N.; Sagitova, Elena F.; Ushakov, Igor A.; Trofimov, Boris A.: Transition-Metal-Free Synthesis of Pyrrolo[1,2-a]pyrazines via Intramolecular Cyclization of N-Propargyl(pyrrolyl)enaminones
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0230_ga_10-1055_s-0036-1588454.gif
Supporting Information

special topic

Midya, Siba P.; Mondal, Akash; Begum, Ayesha; Balaraman, Ekambaram: A Simple Cobalt(II) Chloride Catalyzed N-Alkylation of Amines with Alcohols
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0248_ga_10-1055_s-0036-1589064.gif
Supporting Information

Publication Date: 05 July 2017

paper

Hernández-Benitez, R. Israel; Zárate-Zárate, Daniel; Delgado, Francisco; Tamariz, Joaquín: Palladium-Catalyzed Synthesis of Diarylamines and 1- and 2-Oxygenated Carbazoles: Total Syntheses of Natural Alkaloids Clauraila A, Clausenal, Clausine P, and 7-Methoxy-O-methylmukonal
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0232_ga_10-1055_s-0036-1588467.gif
Supporting Information

paper

Porwal, Digvijay; Oestreich, Martin: B(C6F5)3-Catalyzed Reduction of Sulfoxides and Sulfones to Sulfides with Hydrosilanes
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0361_ga_10-1055_s-0036-1588476.gif
Supporting Information

special topic

Yu, Zhao; Bo, Tang; Aiying, Guan; Weiwei, Wang; Zhenhua, Zhang; Mingan, Wang: Synthesis and Fungicidal Activity of (E)-5-[1-(4-Phenyl-2-oxo-1-oxaspiro[4.5]dec-3-en-3-yl)ethylidene]-2-aminoimidazolin-4-one Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0247_ga_10-1055_s-0036-1588463.gif

Publication Date: 04 July 2017

feature

Sato, Yuki; Kawaguchi, Shin-ichi; Nomoto, Akihiro; Ogawa, Akiya: Photoinduced Coupling Reaction of Diphenyl(2,4,6-trimethylbenzoyl)phosphine Oxide with Interelement Compounds: Application to the Synthesis of Thio- or Selenophosphinates
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0251_ga_10-1055_s-0036-1588867.gif
Supporting Information

psp

Weiberth, Franz J.; Bourque, Andre J.; Elenbaas, Steven; Hanna, Reda; Powers, Matthew R.; Siegel, Craig S.; Zhao, Jin: Scalable Syntheses of Chirally Pure Mono-protected and Orthogonally Di-protected cis-3,4-Diaminotetrahydrofurans
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0298_ga_10-1055_s-0036-1588459.gif
Supporting Information

Publication Date: 03 July 2017

paper

Zhang, Chuancheng; Yue, Qiang; Xiao, Zhen; Wang, Xianglan; Zhang, Qian; Li, Dong: Synthesis of O-Aroyl-N,N-dimethylhydroxylamines through Hypervalent Iodine-Mediated Amination of Carboxylic Acids with N,N-Dimethylformamide
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0201_ga_10-1055_s-0036-1588460.gif
Supporting Information

special topic

Li, Dianjun; Li, Ying; Yu, Wei: tert-Butyl Hypochlorite Induced Cyclization of Ethyl 2-(N-Aryl­carbamoyl)-2-iminoacetates
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0243_ga_10-1055_s-0036-1588462.gif
Supporting Information

Publication Date: 29 June 2017

special topic

Li, Xue-Fei; Lin, Jin-Shun; Liu, Xin-Yuan: Catalytic Radical Intramolecular Aminoperfluoroalkylation and Aminodifluoromethylation of Unactivated Alkenes with Fluoro­alkylsulfonyl Chlorides
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0255_ga_10-1055_s-0036-1589044.gif
Supporting Information

Publication Date: 28 June 2017

special topic

Sumida, Yuto; Sumida, Tomoe; Hosoya, Takamitsu: Nickel-Catalyzed Reductive Cross-Coupling of Aryl Triflates and Nonaflates with Alkyl Iodides
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0215_ga_10-1055_s-0036-1588464.gif
Supporting Information

Publication Date: 27 June 2017

paper

Cívicos, José F.; Coimbra, Juliana S. M.; Costa, Paulo R. R.: Solvent-Free Synthesis of Salen Ligands and Pd(II)– and Cu(II)–Salen Complexes: Their Use in the Oxidation of α-Tetralones to α-Naphthols
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0200_ga_10-1055_s-0036-1588446.gif
Supporting Information

special topic

Barday, Manuel; Janot, Christopher; Clare, Daniel; Carr-Knox, Caitlin; Higginson, Bradley; Ho, Kelvin Y. T.; Aïssa, Christophe: On the Regioselectivity of the Nickel-Catalyzed Insertion of Alkynes into the Carbon–Carbon Bond of Oxetan-3-one
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0213_ga_10-1055_s-0036-1589052.gif
Supporting Information

special topic

Shang, Xiao-Jie; Liu, Zhong-Quan: A Catalyzed Aerobic Intramolecular C–O Bond Formation: Facile Access to Ring-Fused Dihydrobenzoxazine Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0242_ga_10-1055_s-0036-1588465.gif
Supporting Information

Publication Date: 26 June 2017

paper

Gracheva, Iuliia A.; Svirshchevskaya, Elena V.; Zaburdaeva, Elena A.; Fedorov, Alexey Yu.: Synthesis of Bifunctional Furano-Allocolchicinoids
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0234_ga_10-1055_s-0036-1589060.gif
Supporting Information

short review

Arava, Shlomy; Diesendruck, Charles E.: Strategies for the Synthesis of N-Arylammonium Salts
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0238_ga_10-1055_s-0036-1588868.gif

special topic

Skonieczny, Kamil; Jaźwiński, Jarosław; Gryko, Daniel T.: The Synthesis of Imidazo[1,2-f]phenanthridines, Phenanthro-[9,10-d]imidazoles, and Phenanthro[9′,10′:4,5]imidazo[1,2-f]-phenanthridines via Intramolecular Oxidative Aromatic Coupling
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0239_ga_10-1055_s-0036-1589053.gif
Supporting Information

Publication Date: 20 June 2017

feature

Muraca, Ana Carolina A.; Perecim, Givago P.; Rodrigues, Alessandro; Raminelli, Cristiano: Convergent Total Synthesis of (±)-Apomorphine via Benzyne Chemistry: Insights into the Mechanisms Involved in the Key Step
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0172_ga_10-1055_s-0036-1588855.gif
Supporting Information

paper

Ai, Bai-Ru; Chen, Xu-Ling; Dong, Yu; Tang, Lei; Wang, Ji-Yu: Tetrabutylammonium Iodide Catalyzed Epoxidation of Naphthoquinone Derivatives with tert-Butyl Hydroperoxide as an Oxidant
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0174_ga_10-1055_s0036-1589035.gif
Supporting Information

paper

Ban, Jaeyoung; Shabbir, Saira; Lim, Minkyung; Lee, Byunghoon; Rhee, Hakjune: Synthesis of l-Ribose from d-Ribose by a Stereoconversion through Sequential Lactonization as the Key Transformation
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0254_ga_10-1055_s-0036-1588857.gif
Supporting Information

paper

Liu, Ge; Li, Yan; Sheng, Jie; Wang, Xi-Sheng: Oxidative Cleavage of Enamides with Hypervalent Iodine(III)/TMSN3 under an Air Atmosphere
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0205_ga_10-1055_s-0036-1589041.gif
Supporting Information

paper

Luo, A-Yun; Bao, Yan; Cheng, Xiu-Fen; Wang, Xi-Sheng: A Neutral Metal-Free System for Head-to-Tail Dimerization of Electron-Rich Alkenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0208_ga_10-1055_s-0036-1589039.gif
Supporting Information

paper

Perez, Vincent; Fadel, Antoine; Rabasso, Nicolas: Synthesis of N-Sulfonyl Ynamido-Phosphonates: Valuable Partners for Cycloadditions
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0190_ga_10-1055_s-0036-1589042.gif
Supporting Information

paper

Shen, Yang; Zhu, Zi-Qi; Liu, Jin-Xi; Yu, Lei; Du, Bai-Xiang; Mei, Guang-Jian; Shi, Feng: Brønsted Acid Catalyzed C3-Alkylation of 2-Indolylmethanols with Azlactones via an Umpolung Strategy
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0204_ga_10-1055_s-0036-1589036.gif
Supporting Information CIF File

paper

Tang, Wu-Bang; Cao, Kou-Sen; Meng, Shan-Shui; Zheng, Wen-Hua: Boronic Acid Catalysis for Aza-Piancatelli Rearrangement
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0261_ga_10-1055_s-0036-1589040.gif
Supporting Information

special topic

Sabat, Nazarii; Smoleń, Sabina; Nauš, Petr; Perlíková, Pavla; Cebová, Magdaléna; Poštová Slavětínská, Lenka; Hocek, Michal: Synthesis of 2,6-Substituted 7-(Het)aryl-7-deazapurine Nucleobases (2,4-Disubstituted 5-(Het)aryl-pyrrolo[2,3-d]pyrimidines)
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0206_ga_10-1055_s-0036-1588443.gif
Supporting Information

Publication Date: 13 June 2017

paper

Honraedt, Aurélien; Méndez, Lucía Reyes; Campagne, Jean-Marc; Leclerc, Eric: A Three-Component Reaction for the One-Pot Preparation of β-Amino-α,α-Difluoroketones from Trimethyl(trifluoromethyl)silane (CF3TMS), Acylsilanes and Imines
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0246_ga_10-1055_s-0036-1588447.gif
Supporting Information

special topic

Joshi, Hemant; Ghosh, Subrata K.; Gladysz, John A.: Enantioselective Additions of Stabilized Carbanions to Imines Generated from α-Amido Sulfones By Using Lipophilic Salts of Chiral Tris(1,2-diphenylethylenediamine) Cobalt(III) Trications as Hydrogen Bond Donor Catalysts
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0236_ga_10-1055_s-0036-1590502.gif
Supporting Information

special topic

Nagamoto, Midori; Nishimura, Takahiro; Yorimitsu, Hideki: Iridium-Catalyzed Intramolecular Oxidative Cyclization of Alkenyl Amides and Alkenoic Acids
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0211_ga_10-1055_s-0036-1588435.gif
Supporting Information

special topic

Shi, Shicheng; Szostak, Michal: Nickel-Catalyzed Negishi Cross-Coupling of N-Acylsuccinimides: Stable, Amide-Based, Twist-Controlled Acyl-Transfer Reagents via N–C Activation
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0192_ga_10-1055_s-0036-1588845.jpg
Supporting Information

Publication Date: 12 June 2017

special topic

Couly, Florence; Dubouilh-Benard, Carole; Besson, Thierry; Fruit, Corinne: Late-Stage C–H Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one Backbone: Synthesis of an Array of Potential Kinase Inhibitors
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0132_ga_10-1055_s-0036-1588434.gif
Supporting Information

special topic

Nayak, Sanatan; Prabagar, B.; Ghosh, Nayan; Mallick, Rajendra K.; Sahoo, Akhila K.: Ag(I)-Catalyzed Cycloisomerization and Cyclization of Ketene Aminals: Construction of Azepine and 1,2-Dihydropyridine Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0185_ga_10-1055_s-0036-1588841.gif
CIF File Supporting Information

special topic

Watabe, Yota; Kanazawa, Kohei; Fujita, Takeshi; Ichikawa, Junji: Nickel-Catalyzed Hydroalkenylation of Alkynes through C–F Bond Activation: Synthesis of 2-Fluoro-1,3-dienes
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0187_ga_10-1055_s-0036-1588842.gif
Supporting Information

Publication Date: 07 June 2017

paper

Bessi, Matteo; Monini, Marco; Calamante, Massimo; Mordini, Alessandro; Sinicropi, Adalgisa; Basosi, Riccardo; Di Donato, Mariangela; Foggi, Paolo; Iagatti, Alessandro; Zani, Lorenzo; Reginato, Gianna: Synthesis of Silatrane-Containing Organic Sensitizers as Precursors for the Silyloxyl Anchoring Group in Dye-Sensitized Solar Cells
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0163_ga_10-1055_s-0036-1588836.jpg
Supporting Information

paper

Desyatkin, Victor G.; Beletskaya, Irina P.: Asymmetric Friedel–Crafts/Michael Reaction of Indoles and Pyrroles with Coumarin-3-carbonylates
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0198_ga_10-1055_s-0036-1589024.gif
Supporting Information

paper

Kulakov, Ivan V.; Shatsauskas, Anton L.; Matsukevich, Mariya V.; Palamarchuk, Irina V.; Seilkhanov, Tulegen M.; Gatilov, Yuriy V.; Fisyuk, Alexander S.: A New Approach to the Synthesis of Benzo[c][1,7]naphthyridin-4(3H)-ones
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0120_ga_10-1055_s-0036-1590470.gif
Supporting Information

paper

Law, Robert P.; Ukuser, Sabri; Tape, Daniel T.; Talbot, Eric P. A.: Regioselective Synthesis of 3-Aminoimidazo[1,2-a]pyrimidines with Triflic Anhydride
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0145_ga_10-1055_s-0036-1588425.gif
Supporting Information

paper

Xu, Wenke; Yang, Hui; Liu, Yingju; Hua, Yingchun; He, Bin; Ning, Xin; Qin, Zhiyan; Liu, Hong-Min; Liu, Feng-Wu: Facile Approaches to 2-Deoxy-d-glucose and 2-Deoxy-α-d-glucopyranonucleosides from d-Glucal
https://www.thieme-connect.de/media/synthesis/EFirst/i_h1887_ga_10-1055_s-0036-1589501.gif
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special topic

Abe, Takumi; Haruyama, Tomohiro; Yamada, Koji: C4 Pictet–Spengler Reactions for the Synthesis of Core Structures in Hyrtiazepine Alkaloids
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0153_ga_10-1055_s-0036-1588438.gif
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special topic

Opsomer, Tomas; Thomas, Joice; Dehaen, Wim: Chemoselectivity in the Synthesis of 1,2,3-Triazoles from Enolizable Ketones, Primary Alkylamines, and 4-Nitrophenyl Azide
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0209_ga_10-1055_s-0036-1588856.gif
Supporting Information

Publication Date: 06 June 2017

paper

Hu, Yixin; Zhou, Lihong; Lu, Wenjun: Transition-Metal- and Halogen-Free Oxidation of Benzylic sp3 C–H Bonds to Carbonyl Groups Using Potassium Persulfate
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0168_ga_10-1055_s-0036-1588429.gif
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Publication Date: 30 May 2017

paper

Nowacki, Michał; Wojciechowski, Krzysztof: Synthesis of [1]Benzothieno[2,3-b]quinolines via Transition-Metal-Free [3+3] Annulation of Nitroarenes and Benzo[b]thiophen-3-ylacetonitrile or 3-(Phenylsulfonylmethyl)benzo[b]thiophene Carbanions
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0150_ga_10-1055_s-0036-1588426.gif
Supporting Information

Publication Date: 29 May 2017

paper

Singh, Pallavi; Peddinti, Rama Krishna: Waste-Free Swift Synthesis of Symmetrical and Unsymmetrical Diarylmethyl Thioethers from Diaryl Carbinols
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0061_ga_10-1055_s-0036-1589022.gif
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special topic

Hammann, Jeffrey M.; Hofmayer, Maximilian S.; Lutter, Ferdinand H.; Thomas, Lucie; Knochel, Paul: Recent Advances in Cobalt-Catalyzed Csp2 and Csp3 Cross-Couplings
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0069_ga_10-1055_s-0036-1588430.gif

special topic

Pinet, Sandra; Liautard, Virginie; Debiais, Mégane; Pucheault, Mathieu: Radical Metal-Free Borylation of Aryl Iodides
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0180_ga_10-1055_s-0036-1588431.gif
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special topic

Saito, Hayate; Nogi, Keisuke; Yorimitsu, Hideki: Palladium-Catalyzed Double Borylation of Diaryl Sulfoxides with Diboron
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0217_ga_10-1055_s-0036-1588848.gif
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special topic

Xu, Kun; Tan, Zhoumei; Zhang, Haonan; Zhang, Sheng: Cobalt-Catalyzed Monoselective ortho-C–H Ethylation of Carboxamides with Triethylaluminum
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0095_ga_10-1055_s-0036-1589010.gif
Supporting Information

Publication Date: 24 May 2017

paper

Hassan, Alaa A.; Mohamed, Nasr K.; El-Shaieb, Kamal M. A.; Tawfeek, Hendawy N.; Bräse, Stefan; Nieger, Martin: Eschenmoser Coupling Reaction and Reactivity of Hydrazinecarbo­thioamides in the Synthesis of Benzindazole and Naphthothiazole Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0149_ga_10-1055_s-0036-1588179.gif
Supporting Information CIF File

special topic

Fujita, Shoji; Shibuya, Masatoshi; Yamamoto, Yoshihiko: Intramolecular Hydroalkoxylation/Reduction and Hydroamination/Reduction of Unactivated Alkynes Using a Silane–Iodine Catalytic System
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0212_ga_10-1055_s-0036-1588436.gif
Supporting Information

Publication Date: 18 May 2017

paper

Bouattour, Ali; Fakhfakh, Mehdi; Abid, Souhir; Paquin, Ludovic; Ammar, Houcine; Bazureau, Jean-Pierre: An Efficient and Concise Synthesis of N-3-Substituted 9-Methoxy-4H-[1]-benzopyrano[2,3-d]pyrimidine-4(5H)-imines and Form­amidine Derivatives from Methyl N-(3-Cyano-8-methoxy-4H-[1]-benzopyran-2-yl)methanimidate
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0036_ga_10-1055_s-0036-1588825.gif
Supporting Information

paper

Nakao, Michiyasu; Tanaka, Kazue; Kitaike, Syuji; Sano, Shigeki: Synthesis of Fluorine-Containing Analogues of 1-Lysoglycerophospholipids via Horner–Wadsworth–Emmons Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0142_ga_10-1055_s-0036-1588826.gif
Supporting Information

paper

Rappenglück, Sebastian; Niessen, Karin V.; Seeger, Thomas; Worek, Franz; Thiermann, Horst; Wanner, Klaus T.: Regioselective and Transition-Metal-Free Addition of tert-Butyl Magnesium Reagents to Pyridine Derivatives: A Convenient Method for the Synthesis of 3-Substituted 4-tert-Butylpyridine Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0199_ga_10-1055_s0036-1589025.gif
Supporting Information

paper

Zheng, Weiping; Li, Yuming; Zhang, Jiayong; Du, Siyi; Miao, Zhiwei: Highly Regio- and Diastereoselective [3+2]-Annulation Reaction of Morita–Baylis–Hillman Carbonates with Pyrazolones Catalyzed by Tertiary Phosphines
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0852_ga_10-1055_s-0036-1589030.gif
Supporting Information

paper

Zhou, Xiao-Yu; Chen, Xia; Wang, Liang-Guang; Yang, Dan; Li, Zhi: Palladium-Catalyzed Oxidation-Hydroxylation and Oxidation-Methoxylation­ of N-Boc Indoles for the Synthesis of 3-Oxoindolines
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0109_ga_10-1055_s-0036-1589032.gif
Supporting Information

Publication Date: 15 May 2017

paper

Úr, Györgyi; Fekete, Gergely Gulyás; Jekő, József; Hideg, Kálmán; Kálai, Tamás: Palladium- and/or Copper-Catalyzed Cross-Coupling Reactions of Paramagnetic Vinyl Bromides and Iodides
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0058_ga_10-1055_s-0036-1589034.gif
Supporting Information

special topic

Takenouchi, Yuta; Ito, Hajime: Copper(I)-Catalyzed Boryl Substitution of Allyl Aminals: Selective Synthesis of Linear γ-Aminoallylboronates
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0078_ga_10-1055_s-0036-1588802.gif
Supporting Information

special topic

Zheng, Min; Chen, Kai; Zhu, Shifa: One-Pot Synthesis of Indole Derivatives from the Reaction of Nitroalkynes and Alkynes via a Mercury-Carbene Intermediate
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0170_ga_10-1055_s-0036-1588416.gif
Supporting Information CIF File

Publication Date: 11 May 2017

paper

Deng, Xu; Guan, Yu-Qing; Huo, Ning-Ning; Wang, Ya-Jing; Lv, Hui; Zhang, Xu-Mu: An Efficient and Modular Route to C3*-TunePhos-Type Ligands
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0115_ga_10-1055_s-0036-1588421.gif
Supporting Information

special topic

Kalsi, Deepti; Barsu, Nagaraju; Dahiya, Pardeep; Sundararaju, Basker: C–H and N–H Bond Annulation of Benzamides with Isonitriles Catalyzed by Cobalt(III)
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0137_ga_10-1055_s-0036-1589011.gif
Supporting Information

Publication Date: 09 May 2017

paper

Kasapidou, Paraskevi M.; Zarganes-Tzitzikas, Tryfon; Tsoleridis, Constantinos A.; Stephanidou-Stephanatou, Julia; Neochoritis, Constantinos G.: Manipulating a Multicomponent Reaction: A Straightforward Approach to Chromenopyrazole Hybrid Scaffolds
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0057_ga_10-1055_s-0036-1589013.gif
Supporting Information

paper

Zhao, Yulei; Yuan, Yang; Kong, Lingkai; Zhang, Fangfang; Li, Yanzhong: Synthesis of 1-Alkyl-3-(2-oxo-2-aryl/alkyl-ethyl)indolin-2-ones through Gold/Brønsted Acid Relay Actions: Observation of Selective C=C Bond Cleavage of Enaminones
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0157_ga_10-1055_s-0036-1588820.gif
Supporting Information

special topic

Pertschi, Romain; Miaskiewicz, Solène; Weibel, Jean-Marc; Pale, Patrick; Blanc, Aurélien: Gold(I)-Catalyzed Cascade: Synthesis of 2,5-Disubstituted Pyrroles from N-Sulfonyl-2-(1-ethoxypropargyl)azetidines through Cyclization/Nucleophilic Substitution/Elimination
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0158_ga_10-1055_s-0036-1589017.gif
Supporting Information

special topic

Shimizu, Maki; Hayama, Noboru; Kimachi, Tetsutaro; Inamoto, Kiyofumi: Copper-Catalyzed Intramolecular C–H Amination: A New Entry to Substituted Xanthine Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0173_ga_10-1055_s-0036-1588821.gif
Supporting Information

Publication Date: 08 May 2017

feature

Eastabrook, Andrew S.; Sperry, Jonathan: Synthetic Access to 3,5,7-Trisubstituted Indoles Enabled by Iridium­-Catalyzed C–H Borylation
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0155_ga_10-1055_s-0036-1589018.gif
Supporting Information

paper

Jiang, Jie; Wu, Mingshu; Zhu, Zhongxiang; Kong, Dulin: Catalyst-Free Intramolecular 1,3-Dipolar Cycloaddition of Ethyl (2-Formylphenyl) Vinylphosphonates: A Highly Stereoselective Access to Phosphadihydrocoumarin-Fused Pyrrolizidines/Pyrrolidines
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0825_ga_10-1055_s-0036-1588818.gif
Supporting Information CIF File

special topic

Jamieson, Megan L.; Brant, Nicola Z.; Brimble, Margaret A.; Furkert, Daniel P.: Remarkable Influence of Cobalt Catalysis on Epoxide Ring-Opening with Sulfoxonium Ylides
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0181_ga_10-1055_s-0036-1588814.gif

Publication Date: 05 May 2017

paper

Zaytsev, Vladimir P.; Revutskaya, Ekaterina L.; Nikanorova, Tatiana V.; Nikitina, Eugeniya V.; Dorovatovskii, Pavel V.; Khrustalev, Victor N.; Yagafarov, Niyaz Z.; Zubkov, Fedor I.; Varlamov, Alexey V.: An Intramolecular Diels–Alder Furan (IMDAF) Approach towards the Synthesis of Isoindolo[2,1-a]quinazolines and Isoindolo[1,2-b]quinazolines
https://www.thieme-connect.de/media/synthesis/EFirst/i_n1752_ga_10-1055_s-0036-1588812.gif
Supporting Information

Publication Date: 04 May 2017

paper

Zhang, Zhen; Shao, Xuebei; Zhang, Gang; Li, Qinghan; Li, Xinying: Highly Efficient Synthesis of Multi-Substituted Allenes from Propargyl­ Acetates and Organoaluminum Reagents Mediated by Palladium
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0101_ga_10-1055_s-0036-1588177.gif
Supporting Information

special topic

Xiao, Jian; Wang, Ya-Wen; Peng, Yu: Nickel-Promoted Reductive Cyclization Cascade: A Short Synthesis of a New Aromatic Strigolactone Analogue
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0156_ga_10-1055_s-0036-1588804.gif
Supporting Information

Publication Date: 03 May 2017

special topic

Jang, Won Jun; Han, Jung Tae; Yun, Jaesook: NHC-Copper-Catalyzed Tandem Hydrocupration and Allylation of Alkenyl Boronates
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0138_ga_10-1055_s-0036-1588811.gif
Supporting Information

special topic

Zhang, Xiaojuan; Han, Xiuling; Hu, Zhiyong; Lu, Xiyan: Synthesis of Substituted Piperidines via Cationic Palladium(II)-Catalyzed Reductive Coupling of N-Tosyl-Tethered Alkynones
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0141_ga_10-1055_s-0036-1588803.gif
Supporting Information

Publication Date: 28 April 2017

special topic

Cacchi, Sandro; Fabrizi, Giancarlo; Goggiamani, Antonella; Iazzetti, Antonia; Verdiglione, Rosanna: 2-(Aminomethyl)-3-arylindoles from 3-(o-Trifluoroacetamidoaryl)-1-propargylic Alcohols, Aryl Halides, and Amines: A Domino Palladium-Catalyzed Three-Component Approach
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0159_ga_10-1055_s-0036-1589016.gif
Supporting Information

Publication Date: 27 April 2017

special topic

Cabré, Albert; Verdaguer, Xavier; Riera, Antoni: Ethylene Glycol Assisted Intermolecular Pauson–Khand Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0165_ga_10-1055_s-0036-1588813.gif
Supporting Information

Publication Date: 20 April 2017

special topic

Triandafillidi, Ierasia; Sideri, Ioanna K.; Tzaras, Dimitrios Ioannis; Spiliopoulou, Nikoleta; Kokotos, Christoforos G.: Green Organocatalytic Synthesis of Dihydrobenzofurans by Oxidation–Cyclization of Allylphenols
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0154_ga_10-1055_s-0036-1588998.gif
Supporting Information

Publication Date: 18 April 2017

paper

Belov, Dmitry S.; Ivanov, Vladimir N.; Curreli, Francesca; Kurkin, Alexander V.; Altieri, Andrea; Debnath, Asim K.: Synthesis of 5-Arylpyrrole-2-carboxylic Acids as Key Intermediates for NBD Series HIV-1 Entry Inhibitors
https://www.thieme-connect.de/media/synthesis/EFirst/i_m1861_ga_10-1055_s-0036-1588780.gif
Supporting Information

paper

Demidov, Oleg P.; Amangasieva, Gulminat A.; Avakyan, Elena K.; Borovlev, Ivan V.: Nucleophilic Addition of Amides to 10-Alkylacridinium Cations: A Case of Double N-Nucleophilicity of Some Monoamides
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0146_ga_10-1055_s-0036-1588786.gif
Supporting Information

special topic

Hofmayer, Maximilian S.; Hammann, Jeffrey M.; Lutter, Ferdinand H.; Knochel, Paul: Large-Scale Cobalt-Catalyzed Cross-Couplings of Functionalized Bench-Stable Arylzinc Pivalates with (Hetero)Aryl and Alkenyl Halides­
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0090_ga_10-1055_s-0036-1588986.gif
Supporting Information

Publication Date: 06 April 2017

special topic

Ferrand, Laura; Lyu, Ye; Rivera-Hernández, Alejandro; Fallon, Brendan J.; Amatore, Muriel; Aubert, Corinne; Petit, Marc: Hydroboration and Diboration of Internal Alkynes Catalyzed by a Well-Defined Low-Valent Cobalt Catalyst
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0089_ga_10-1055_s-0036-1588996.gif
Supporting Information

Publication Date: 29 March 2017

special topic

Suo, Jian-Feng; Zhao, Xue-Mei; Zhang, Kai-Xin; Zhou, Sheng-Li; Niu, Jun-Long; Song, Mao-Ping: Cobalt-Catalyzed Perfluoroalkylation of Quinoline Amides at the C5 Position
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0033_ga_10-1055_s-0036-1588160.gif
Supporting Information

Publication Date: 14 March 2017

special topic

Lee, Sang Eun; Lee, Seong Jong; Cheon, Cheol-Hong: Concise Total Syntheses of Paullone and Kenpaullone via Cyanide-Catalyzed Intramolecular Imino-Stetter Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0063_ga_10-1055_s-0036-1588749.gif
Supporting Information

Publication Date: 02 March 2017

special topic

Miura, Wataru; Hirano, Koji; Miura, Masahiro: Iridium-Catalyzed Site-Selective C–H Borylation of 2-Pyridones
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0044_ga_10-1055_s-0036-1588735.gif
Supporting Information