Synthesis

Publication Date: 23 February 2021

special topic > Special Issue dedicated to Prof. Sarah Reisman, recipient of the 2019 Dr. Margaret Faul Women in Chemistry Award

Lam, Heather; Abel-Snape, Xavier; Köllen, Martin F.; Lautens, Mark: Recent Advances in Transition-Metal-Free (4+3)-Annulations

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Publication Date: 22 February 2021

paper

Schädel, Nicole; Icik, Esra; Martini, Maike; Altevogt, Luca; Ramming, Isabell; Greulich, Andreas; Baro, Angelika; Bilitewski, Ursula; Laschat, Sabine: Synthesis of Imidazole and Histidine-Derived Cross-Linkers as Analogues of GOLD and Desmosine

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Watanabe, Hikaru; Nakajima, Kazuki; Ekuni, Kento; Edagawa, Ryota; Akagi, Yuta; Okuda, Yasuhiro; Wakamatsu, Kan; Orita, Akihiro: Custom-Made Pyrene Photocatalyst-Promoted Desulfonylation of Arylethenyl Sulfones Using Green-Light-Emitting Diodes

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Publication Date: 18 February 2021

feature

Li, Fusheng; Lin, Shuangjie; Li, Xiyu; Shi, Lei: Photocatalytic Generation of π-Allyltitanium Complexes from Butadiene via a Radical Strategy

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feature

Shaaban, Saad; Li, Houhua; Merten, Christian; Antonchick, Andrey P.; Waldmann, Herbert: Rhodium(III)-Catalyzed Enantioselective Benzamidation of Cyclopropenes

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Publication Date: 15 February 2021

paper

Zhang, Wenjie; Liu, Xueyan; Tian, Zhenfeng; Li, Hongji: Rh(III)-Catalyzed Olefination and Alkylation of Arenes with Maleimides: A Tunable Strategy for C(sp²)–H Functionalization

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Supporting Information CIF File

Publication Date: 10 February 2021

feature

Sirvent, Ana; Hernández-Ibáñez, Sandra; Yus, Miguel; Foubelo, Francisco: Pyrrolidine and Indolizidine Alkaloids from Chiral N-tert-Butanesulfinyl Imines Derived from 4-Halobutanal

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paper

Saravanan, Velu; Mohanakrishnan, Arasambattu K.: Synthesis of Annulated Carbazoles via FeCl₃/SnCl₄‑Mediated Domino Reaction of Vinyl Ketone Tethered Bromomethylindoles with Arenes and Heteroarenes

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Publication Date: 09 February 2021

paper

Schefzig, Luise; Kurzawa, Timon; Rancan, Giaime; Linder, Igor; Leisering, Stefan; Bera, Mrinal K.; Gart, Max; Zimmer, Reinhold; Reissig, Hans-Ulrich: Access to Highly Substituted Pyrimidine N-Oxides and 4-Acetoxymethyl-Substituted Pyrimidines via the LANCA Three-Component Reaction–Cyclocondensation Sequence

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Publication Date: 08 February 2021

paper

Avila-Melo, José Luis; Benavides, Adriana; Fuentes-Gutiérrez, Alfredo; Tamariz, Joaquín; Jiménez-Vázquez, Hugo A.: Total Synthesis of the Natural Carbazoles O-Demethylmurrayanine and Murrastanine A, and of a C4,C4′ Symmetric Murrastanine A Dimer from N-Phenyl-4,5-dimethylene-1,3-oxazolidin-2-one

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paper

Yadav, Mamta; Jat, Ram Singh; Sarma, Bibek; Bhanuchandra, M.: 2-Pyridyl Sulfoxide Directed Pd(II)-Catalyzed C–H Olefination of Arenes with Molecular Oxygen as the Sole Oxidant

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Publication Date: 01 February 2021

paper

Kuwabara, Motoi; Matsuo, Ami; Kamo, Shogo; Matsuzawa, Akinobu; Sugita, Kazuyuki: Stereoselective Convergent Synthesis of Carbon Skeleton of Cotylenin A Aglycone

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review

Badart, Michael P.; Hawkins, Bill C.: Synthetic Strategies to Access Heteroatomic Spirocentres Embedded in Natural Products

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Publication Date: 28 January 2021

short review

Walther, Melanie; Kipke, Waldemar; Schultzke, Sven; Ghosh, Souvik; Staubitz, Anne: Modification of Azobenzenes by Cross-Coupling Reactions

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Publication Date: 27 January 2021

paper

Peng, Jing; Hu, Ludan; Chen, Mu-Wang; Deng, Zhihong; Peng, Yiyuan: Synthesis of Difluoromethyl-Substituted Quinazolines through Selective Difluoromethylation

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Fukumoto, Yoshiya; Shiratani, Motohiro; Noguchi, Hikaru; Chatani, Naoto: Iridium-Catalyzed Direct Amidation of Imidazoles at the C-2 Position with Isocyanates in the Presence of Hydrosilanes Leading to Imidazole-2-Carboxamides

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Publication Date: 26 January 2021

paper

He, Chang; Wang, Zijuan; Chen, Yitong; Zhang, Guolin; Yu, Yongping: Palladium(II)-Catalyzed C(sp)–C(sp²) Coupling: A Direct Approach to Multi-Substituted Pyrrolo[1,2-a]pyrazines

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Publication Date: 25 January 2021

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Steinke, Tim; Wonner, Patrick; Engelage, Elric; Huber, Stefan M.: Catalytic Activation of a Carbon–Chloride Bond by Dicationic Tellurium-Based Chalcogen Bond Donors

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paper

Khalili Foumeshi, Maryam; Ziyaei Halimehjani, Azim; Alaei, Ali; Klepetářová, Blanka; Beier, Petr: Tandem Alkylation/Michael Addition Reaction of Dithiocarbamic Acids with Alkyl γ-Bromocrotonates: Access to Functionalized 1,3-Thiazolidine-2-thiones

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paper

Zhu, Xiao-Rui; Deng, Chen-Liang: Nickel-Catalyzed Intramolecular Nucleophilic Addition of Aryl Halides to Aryl Ketones for the Synthesis of Benzofuran Derivatives

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short review

Yu, Jingxun; Luan, Xinjun: Hydroxylamines as One-Atom Nitrogen Sources for Metal-Catalyzed Cycloadditions

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short review

Zu, Bing; Guo, Yonghong; Ke, Jie; He, Chuan: Transient- and Native-Directing-Group-Enabled Enantioselective C–H Functionalization

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Publication Date: 22 January 2021

paper

Yavari, Issa; Sheikhi, Sara; Sheykhahmadi, Jamil; Taheri, Zohreh; Halvagar, Mohammad Reza: Ultrasound-Promoted Synthesis of Spirocyclopropanes from Switchable Starting Materials via Azomethine Ylide [3+2]-Cycloaddition

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short review

Neri, Raul; Bossmann, Stefan H.: Isoselenocyanates: Synthesis and Their Use for Preparing Selenium-Based Heterocycles

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Publication Date: 21 January 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Yamamoto, Sonoka; Shibuya, Yushin; Suzuki, Toyoko; Okano, Kentaro; Horie, Masaki; Mori, Atsunori: One-Shot Deprotonative Metalation/Transmetalation/Polymerization of Halothiophenes Catalyzed by Nickel Complex for Polythiophene Synthesis

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Publication Date: 20 January 2021

paper

Majeed, Kashif; Liu, Bangjie; Zhou, Fengtao; Zhang, Qiuyu: Synthesis of 1,2,3-Triazole-Fused Indole Derivatives via Copper-Catalyzed Cascade Reaction

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Publication Date: 19 January 2021

paper

Chen, Jyun-Siao; Ke, Yi-Fan; Lin, Heng-Yan; Lin, Wesley; Yen, Wei-Chung; Wu, Hsin-Ru; Luo, Shun-Yuan: Development of a Novel Method for Trimethylsilylation of Saccharides­

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paper

Nazarian, Zohreh; Forsyth, Craig M.: A Cascade Process of Hydroxamates Renders 1,6-Dioxa-3,9-diazaspiro[4.4]nonane-2,8-diones

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Publication Date: 18 January 2021

errata

Srinivasulu, Vunnam; Al-Marzooq, Farah; Hamad, Mohamad; Khanfar, Monther A.; Ramanathan, Mani; Soares, Nelson C.; Al-Tel, Taleb H.: Sequencing Groebke–Blackburn–Bienaymé and Aza-Michael Addition Reactions: A Modular Strategy for Accessing a Diverse Collection of Constrained Benzoxazepine and Imidazopyrazine Systems

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paper

Gairola, Deepti; Peddinti, Rama Krishna: Methanesulfonic Acid Catalyzed Friedel–Crafts Reaction of Electron-Rich Arenes with N-Arylmaleimides: A Highly Efficient Metal-Free Route To Access 3-Arylsuccinimides

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paper

Mityuk, Andrey P.; Hrebonkin, Andrii; Lebed, Pavlo S.; Grabchuk, Galyna P.; Volochnyuk, Dmitriy M.; Ryabukhin, Sergey V.: Efficient Route for the Synthesis of Diverse Heteroannelated 5-Cyanopyridines

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Supporting Information CIF File

paper

Sun, Zheng; Shao, Yu; Zhang, Shuwei; Zhang, Yuxian; Yuan, Yu; Jia, Xiaodong: Oxidative Desymmetrization of Isoindolines Realized by tert-Butyl Nitrite (TBN) Initiated Radical sp³ C–H Activation Relay (CHAR)

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paper

Wang, Siqi; Filatov, Alexander S.; Lozovskiy, Stanislav V.; Shmakov, Stanislav V.; Khoroshilova, Olesya V.; Larina, Anna G.; Selivanov, Stanislav I.; Boitsov, Vitali M.; Stepakov, Alexander V.: Construction of Spiro[3-azabicyclo[3.1.0]hexanes] via 1,3-Dipolar Cycloaddition of 1,2-Diphenylcyclopropenes to Ninhydrin-Derived Azomethine Ylides

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short review

Ashikari, Yosuke; Nagaki, Aiichiro: Homogeneous Catalyzed Aryl–Aryl Cross-Couplings in Flow

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Publication Date: 15 January 2021

paper

Zheng, Qiang; Boltjes, André; Dömling, Alexander: An Ugi Reaction/Intramolecular Cyclization/Oxidation Cascade towards Tetrazole-Linked Dibenzoxazepines

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Publication Date: 14 January 2021

errata

Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)

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review

Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)

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Publication Date: 13 January 2021

paper

You, Shengyong; Zhang, Rongli; Cai, Mingzhong: A Magnetically Recyclable Palladium-Catalyzed Formylation of Aryl Iodides with Formic Acid as CO Source: A Practical Access to Aromatic Aldehydes

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Publication Date: 11 January 2021

feature

Pruteanu, Elena; Tappin, Nicholas D. C.; Gîrbu, Vladilena; Morarescu, Olga; Dénès, Fabrice; Kulciţki, Veaceslav; Renaud, Philippe: Forskolin Editing via Radical Iodo- and Hydroalkylation

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paper

Dziuba, Kamil; Frynas, Sławomir; Szwaczko, Katarzyna: Knoevenagel Condensation of Phosphinoylacetic Acids with Aldehydes: An Efficient One-Pot Strategy for the Synthesis of P-Functionalized Alkenyl Compounds

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paper

Lisovenko, Natalya Yu.; Nasibullina, Ekaterina R.; Kharitonova, Svetlana S.; Myshkina, Olga A.: Simple Synthesis of Substituted 3-Hydroxyfuran-2(5H)-ones

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paper

Yassine, Hasna; Bouali, Jamila; Oumessaoud, Asmaa; Ourhzif, El Mahdi; Hamri, Salha; Hafid, Abderrafia; Khouili, Mostafa; Pujol, Maria Dolors: Synthesis of New Dialkyl 2,2′-[Carbonylbis(azanediyl)]dibenzoates via Curtius Rearrangement

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paper

Yu, Haifeng; Wang, Kehua; Zhang, Xue; Wang, Wenju: Complementary and Regioselective Synthesis of Isomeric 3-[Isoxazol-3(or 5)-yl]indoles from β-Ethylthio-β-indolyl-α,β-unsaturated Ketones

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short review

Mazumdar, Wrickban; Driver, Tom G.: Recent Advances in the Development of Catalytic Methods that Construct Medium-Ring Lactams, Partially Saturated Benzazepines and Their Derivatives

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short review

Zhao, Xuchen; Rainier, Jon D.: The Synthesis of Conjugated Bis-Aryl Vinyl Substrates and Their Photoelectrocyclization Reactions towards Phenanthrene Derivatives

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Publication Date: 08 January 2021

paper

Borisov, Denis D.; Chermashentsev, Grigorii R.; Novikov, Roman A.; Tomilov, Yury V.: Synthesis of Substituted β-Styrylmalonates by Sequential Isomerization of 2-Arylcyclopropane-1,1-dicarboxylates and (2-Arylethylidene)malonates

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paper

Budeev, Anton V.; Kantin, Grigory; Dar’in, Dmitry; Krasavin, Mikhail: Continued Exploration of Trifunctional Alkyl 4-Chloro-2-diazo-3-oxobutanoates: Streamlined Entry into [1,2,3]Triazolo[5,1-c][1,4]benzoxazines and [1,2,3]Triazolo[5,1-c][1,4]benzoxazepines

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paper

Kotha, Sambasivarao; Pulletikurti, Sunil; Fatma, Ambareen; Dhangar, Gopal; Naidu, Gonna Somu: Synthesis of Polycycles and Oxacycles via Tandem Metathesis of endo-Norbornene Derivatives

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review

Pellissier, Hélène: Enantioselective Indium-Catalyzed Transformations

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Publication Date: 07 January 2021

paper

Glas, Carina; Wirawan, Ricky; Bracher, Franz: A Short Approach to N-Aryl-1,2,3,4-tetrahydroisoquinolines from N-(2-Bromobenzyl)anilines via a Reductive Amination/Palladium-Catalyzed Ethoxyvinylation/Reductive N-Alkylation Sequence

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paper

Srinivasulu, Vunnam; Al-Marzooq, Farah; Hamad, Mohamad; Khanfar, Monther A.; Ramanathan, Mani; Soares, Nelson C.; Al-Tel, Taleb H.: Sequencing Groebke–Blackburn–Bienaymé and Aza-Michael Addition Reactions: A Modular Strategy for Accessing a Diverse Collection of Constrained Benzoxazepine and Imidazopyrazine Systems

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Supporting Information

Publication Date: 04 January 2021

paper

Chu, Xianglong; Niu, Yadi; Wang, Xiaodong; Lin, Yunliang; Li, Fuwei; Ma, Chen: Regioselective Oxidative Cross-Coupling Reaction: Synthesis of Imidazo[1,2-a]pyridine Fluorophores

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short review

Singh, Pushpinder; Batra, Aanchal; Singh, Kamal Nain; Mritunjay, Mritunjay: Transition-Metal-Free Strategies for the Synthesis of C-1 Aryl-Substituted Tetrahydroisoquinolines

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Publication Date: 30 December 2020

paper

Xia, Yanping; Ouyang, Lu; Liao, Jianhua; Yang, Xiao; Luo, Renshi: Construction of α-Alkylated Amines by Iridium Complex-Catalyzed One-Step Transfer Hydrogenation of C=C and C=N Bonds

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short review

Li, Yanjun; Ye, Ziqi; Cai, Jiaxin; Gong, Lei: Visible-Light-Promoted Asymmetric Catalysis by Chiral Complexes of First-Row Transition Metals

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short review

Zheng, Songlin; Hu, Yuanyuan; Yuan, Weiming: Recent Advances in C(sp³)–C(sp³) Cross-Coupling via Metalla­photoredox Strategies

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Publication Date: 29 December 2020

paper

Klochkova, Anastasiia; Bubyrev, Andrey; Dar’in, Dmitry; Bakulina, Olga; Krasavin, Mikhail; Sokolov, Viktor: Straightforward Route to γ-Sultams via Novel Tandem S_N/Michael Addition

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Publication Date: 28 December 2020

feature

Ikari, Yuta; Kaihara, Takahito; Goto, Shimpei; Bovenkerk, Marcel; Grenz, David C.; Esser, Birgit; Ferreira, Marli; Stachelek, Patrycja; Data, Przemyslaw; Yoshida, Takumu; Ikai, Tomoyuki; Tohnai, Norimitsu; Minakata, Satoshi; Takeda, Youhei: Peripherally Donor-Installed 7,8-Diaza[5]helicenes as a Platform for Helical Luminophores

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Supporting Information CIF File

paper

Gao, Yanhui; Li, Laiqiang; Liu, Jie; Wang, Lei; Wang, Min: C2-gem-Aryldifluoromethylation of Quinoline N-Oxides with Potassium 2,2-Difluoro-2-arylacetates under Transition-Metal-Free Conditions

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paper

Lapcinska, Sindija; Arsenyan, Pavel: Straightforward Functionalization of Sulfur-Containing Peptides via 5- and 6-endo-dig Cyclization Reactions

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short review

Zhao, Jia-Jia; Zhang, Hong-Hao; Yu, Shouyun: Enantioselective Radical Functionalization of Imines and Iminium Intermediates via Visible-Light Photoredox Catalysis

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Publication Date: 21 December 2020

feature

Ponce, Marian Blanco; Parpart, Silvio; Villinger, Alexander; Rodríguez, Eugenio Torres; Ehlers, Peter; Langer, Peter: Synthesis of Pyrrolo[1,2-a][1,6]- and [1,8]naphthyridines by Alkyne-Carbonyl Metathesis

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paper

Im, Jeong Kyun; Jeong, Ilju; Yang, ByeongDo; Moon, Hyeon; Choi, Jun-Ho; Chung, Won-jin: N-Chlorinative Ring Contraction of 1,4-Dimethoxyphthalazines via a Bicyclization/Ring-Opening Mechanism

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paper

Jurkowski, Kellsie; Bauer, Eike B.: Ferrocenium Ions as Catalysts: Decomposition Studies and Counteranion Influence on Catalytic Activity

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Publication Date: 18 December 2020

short review

Bartoccini, Francesca; Piersanti, Giovanni: Synthesis and Reactivity of Uhle’s Ketone and Its Derivatives

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Publication Date: 17 December 2020

short review

Yu, Hsien-Cheng; Mankad, Neal P.: Catalytic Reactions by Heterobimetallic Carbonyl Complexes with Polar Metal–Metal Interactions

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Publication Date: 15 December 2020

paper

Gurbanov, Rustam; Sokolov, Andriy; Golovach, Sergey; Melnykov, Kostiantyn; Dobrydnev, Alexey V.; Grygorenko, Oleksandr O.: Synthesis of sp³-Enriched β-Fluoro Sulfonyl Chlorides

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paper

He, Ze-Ying; Jang, Ho-Chol; Teng, Le-Sheng; Wei, Zhong-Lin; Liao, Wei-Wei: Controllable Lewis Base Catalyzed Michael Addition of α-Amino­nitriles to Activated Alkenes: Facile Synthesis of Functionalized γ-Amino Acid Esters and γ-Lactams

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paper

Li, Ruoling; Li, Chenchen; Yang, Wen; Zhao, Wanxiang: Homogeneous Palladium-Catalyzed Selective Reduction of 2,2′-Biphenols Using HCO₂H as Hydrogen Source

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Kawakami, Haruka; Nohira, Itsuki; Chatani, Naoto: Nickel-Catalyzed C–F/N–H Annulation of 2-(2-Fluoroaryl) N-Heteroaromatic Compounds with Alkynes: Activation of C–F Bonds

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Supporting Information CIF File

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Xu, Wengang; Wu, Mingbo; Yoshikai, Naohiko: Iron-Catalyzed Remote C–H Alkylation of 8-Amidoquinolines with Cycloalkanes

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Publication Date: 14 December 2020

feature

Bubyrev, Andrey; Kantin, Grigory; Dar’in, Dmitry; Krasavin, Mikhail: CH-Diazomethane Sulfonamides Generated in Situ for Intramolecular [3+2] Cycloaddition of Alkynes: An Entry into Novel Pyrazole-Fused Five-Membered Sultams

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paper

Zhou, Xiao-Yu; Chen, Xia: Oxidative C–H Acyloxylation of Acetone with Carboxylic Acids under Iodine Catalysis

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review

Nguyen, Thanh T.; Wipf, Peter: Intramolecular Diels–Alder Reactions of Oxazoles, Imidazoles, and Thiazoles

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Publication Date: 10 December 2020

paper

Kitamura, Kei; Kanagawa, Hinano; Ozakai, Chiharu; Nishimura, Taichi; Tokuda, Hayato; Tsunoda, Tetsuto; Kaku, Hiroto: Synthesis of the Common Monomeric Unit of Uroleuconaphins and Viridaphins via Hauser–Kraus Annulation

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paper

Sole, Roberto; Agostinis, Lodovico; Conca, Silvia; Gatto, Vanessa; Bardella, Noemi; Morandini, Andrea; Buranello, Chiara; Beghetto, Valentina: Synthesis of Amidation Agents and Their Reactivity in Condensation Reactions

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Publication Date: 08 December 2020

paper

Han, Wei; Inoue, Chika; Onizawa, Tsunaki; Oriyama, Takeshi: Synthesis of N-Aryl-4-arylhexahydroquinoline Derivatives by Reaction of Cyclic Enaminones with Arylidenemalononitriles in DMSO

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Publication Date: 07 December 2020

paper

Ji, Jiu-Jian; Zhu, Zhi-Qiang; Xie, Zong-Bo; Tang, Juan; Yuan, En; Le, Zhang-Gao: Highly Efficient Copper-Catalyzed Dehydrogenative Cross-Coupling of Azoles with α-Amino Carbonyl Compounds

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paper

Talavera-Alemán, Armando; Marrot, Jérome; Dagousset, Guillaume; Thomassigny, Christine: Synthesis of Nitrogen- and Oxygen-Containing Heterocycles by Prins Cyclization in Continuous Flow

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Publication Date: 03 December 2020

paper

Shen, Peng; Guo, Yeting; Wei, Jian; Zhao, Hua; Zhai, Hongbin; Zhao, Yufen: Straightforward Synthesis of Succinimide-Fused Pyrrolizidines by A Three-Component Reaction of α-Diketone, Amino Acid, and Maleimide

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Takahashi, Hiroto; Honjo, Yusaku; Shibata, Yu; Nagashima, Yuki; Tanaka, Ken: Dienylation of Unfunctionalized Arenes with 1,6-Diynes via Rhodium-Catalyzed Directing-Group-Free C–H Bond Activation

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Publication Date: 02 December 2020

paper

Chaubey, Narendra R.; Kapdi, Anant R.; Maity, Biswanath: Organophotoredox-Catalyzed C–H Alkylation of Imidazoheterocycles with Malonates: Total Synthesis of Zolpidem

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paper

Suzuki, Hiroyuki; Yamaguchi, Eiji; Itoh, Akichika: Nickel-Catalyzed Reductive Allylation of Aldehydes with Allyl Acetates

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Publication Date: 30 November 2020

paper

Kianmehr, Ebrahim; Afaridoun, Hadi: Nickel(II)- and Silver(I)-Catalyzed C–H Bond Halogenation of Anilides and Carbamates

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short review

Su, Shixia; Wang, Chuan: Catalytic Asymmetric Osmium-Free Dihydroxylation of Alkenes

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Publication Date: 26 November 2020

paper

Siera, Hannah; Semleit, Nina; Kreuzahler, Mathis; Wölper, Christoph; Haberhauer, Gebhard: Gold Catalysis of Non-Conjugated Haloacetylenes

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Publication Date: 23 November 2020

paper

Smoleń, Sabina; Wincenciuk, Aleksandra; Drapała, Olga; Gryko, Dorota: Vitamin B₁₂-Catalyzed Dicarbofunctionalization of Bromoalkenes Under Visible Light Irradiation

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Publication Date: 19 November 2020

paper

García-Ramírez, Jazmín; Miranda, Luis D.: Peroxide-Mediated Oxidative Radical Cyclization to the Quinazolinone System: Efficient Syntheses of Deoxyvasicinone, Mackinazolinone and (±)-Leucomidine C

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paper

Prasad, Sure Siva; Joshi, Dirgha Raj; Kim, Ikyon: Facile Access to 3,4-Disubstituted 2H-Chromenes via Domino [4+2] Annulation

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paper

Zhao, Qing-he; Yu, Guang-hao; Meng, Ye-chen; Sui, Feng; Yang, Mi-yi; Liu, Li; Li, Hui-jie; Li, Feng; Ma, Hai: An Efficient Substrate-Induced Method for the Synthesis of CF₃-Substituted Cyclopropanes by Metal-Free Reaction of Trifluoromethyl Styrylisoxazoles with Nitromethane

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Publication Date: 17 November 2020

paper

Gan, Zhenjie; Li, Ke; Zhang, Hui; Li, Er-Qing: Copper/GanPhos-Catalyzed 1,3-Dipolar Cycloaddition of Azo­methine Ylides: An Efficient Access to Chiral Pyrrolidine Spirocycles

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Publication Date: 12 November 2020

paper

Jeminejs, Andris; Goliškina, Svetlana M.; Novosjolova, Irina; Stepanovs, Dmitrijs; Bizdēna, Ērika; Turks, Māris: Application of Azide-Tetrazole Tautomerism and Arylsulfanyl Group Dance in the Synthesis of Thiosubstituted Tetrazoloquinazolines

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Publication Date: 11 November 2020

paper

Cheng, Dongping; Pu, Yueqi; Wang, Mingliang; Shen, Yinqiang; Shen, Jing; Xu, Xiaoliang; Yan, Jizhong: 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone (DDQ)-Mediated Tandem Oxidative-Coupling/Annulation of o-Hydroxyaryl Enaminones with Cycloheptatriene

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Publication Date: 10 November 2020

paper

Sun, Mei; Zhao, Long; Yu, Yan-Ling; Ding, Ming-Wu: DEAD-Mediated Oxidative Ugi/Aza-Wittig Reaction for the Synthesis of 5-(1,2,3,4-Tetrahydroisoquinolin-1-yl)-1,3,4-oxadi­­azoles Starting from (N-Isocyanimine)triphenylphosphorane

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Publication Date: 05 November 2020

paper

Chupakhin, Evgeny; Gecht, Martha; Ivanov, Alexander; Kantin, Grigory; Dar’in, Dmitry; Krasavin, Mikhail: (E)-3-Arylidene-4-diazopyrrolidine-2,5-diones: Preparation and Use in Rh^II-Catalyzed X–H Insertion Reactions towards Novel, Medicinally Important Michael Acceptors

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Publication Date: 04 November 2020

paper

Collin, Diego E.; Jackman, Edward H.; Jouandon, Nicolas; Sun, Wei; Light, Mark E.; Harrowven, David C.; Linclau, Bruno: Decagram Synthesis of Dimethyl 1,4-Cubanedicarboxylate Using Continuous-Flow Photochemistry

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paper

Zhao, Xinxin; Guo, Lin; Yang, Chao; Xia, Wujiong: Photoinduced [3+2] Annulation of Alkene with o-Iodoanilines: An Expedient Approach to Indolines

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Publication Date: 02 November 2020

paper

Ji, Haojie; He, Chonglong; Gao, Hongjie; Fu, Weijun; Xu, Jianfeng: DBU-Promoted Formal [4+2] Annulation Reactions of o-Chloromethyl Anilines with Azlactones

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Publication Date: 29 October 2020

paper

Ivanov, Konstantin L.; Melnikov, Mikhail Ya.; Budynina, Ekaterina M.: Reductive Knoevenagel Condensation with the Zn–AcOH System

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Publication Date: 28 October 2020

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Ishida, Naoyoshi; Iwamoto, Hiroaki; Sunagawa, Denise Eimi; Ohashi, Masato; Ogoshi, Sensuke: CsF-Catalyzed Fluoroacylation of Tetrafluoroethylene Using Acyl Fluorides for the Synthesis of Pentafluoroethyl Ketones

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Publication Date: 26 October 2020

paper

Bouarfa, Salima; Bentabed-Ababsa, Ghenia; Erb, William; Picot, Laurent; Thiéry, Valérie; Roisnel, Thierry; Dorcet, Vincent; Mongin, Florence: Iodothiophenes and Related Compounds as Coupling Partners in Copper-Mediated N-Arylation of Anilines

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Publication Date: 22 October 2020

paper

dos Santos, Beatriz F.; da Silva, Beatriz A. L.; de Oliveira, Aline R.; Sarragiotto, Maria H.; Rinaldi, Andrelson W.; Domingues, Nelson Luís C.: Palladium Nanoparticles Anchored on Magnesium Organosilicate: An Effective and Selective Catalyst for the Heck Reaction

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Publication Date: 19 October 2020

paper

Wang, Zijuan; Chen, Wenteng; He, Chang; Zhang, Guolin; Yu, Yongping: Palladium(II)-Catalyzed Three-Component Tandem Cyclization Reaction for the One-Pot Assembly of 4-Arylquinazolines

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Publication Date: 15 October 2020

paper

Guerrero, Sergio Andrés; Ramírez, Juan E.; Sanabria, Carlos M.; Acosta, Lina M.; Cobo, Justo; Nogueras, Manuel; Palma, Alirio: Easy Access to Novel Tetrahydro-1-benzazepine-2-carboxylic Acids and Tetrahydro-1-benzazepines Carrying [a]-Fused Heterocyclic Units from 2-(Allylaryl)glycinates

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