DOI: 10.1055/s-00000084

Synthesis

eFirst

Publication Date: 05 June 2020

Publication Date: 04 June 2020

special topic

Kolympadi Marković, Maria; Marković, Dean; Laclef, Sylvain: Amide Synthesis by Transamidation of Primary Carboxamides
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0202_ga_10-1055_s-0040-1707133.gif

Publication Date: 03 June 2020

review

Publication Date: 02 June 2020

Publication Date: 27 May 2020

psp

Steinebach, Christian; Voell, Sabine Anna; Vu, Lan Phuong; Bricelj, Aleša; Sosič, Izidor; Schnakenburg, Gregor; Gütschow, Michael: A Facile Synthesis of Ligands for the von Hippel–Lindau E3 Ligase
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0128_ga_10-1055_s-0040-1707400.gif

psp

Zisopoulou, Stavroula A.; Pafili, Anastasia E.; Gkizis, Petros; Andreou, Thanos; Koftis, Theoharis V.; Lithadioti, Alexandra; Neokosmidis, Efstratios; Gallos, John K.: Environmentally Benign Large-Scale Synthesis of a Precursor to Vortioxetine
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0176_ga_10-1055_s-0040-1707823.gif

Publication Date: 26 May 2020

review

Christodoulou, Michael S.; Beccalli, Egle M.; Foschi, Francesca; Giofrè, Sabrina: Pd-Catalyzed Domino Reactions Involving Alkenes To Access Substituted Indole Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0125_ga_10-1055_s-0040-1707123.gif

Publication Date: 25 May 2020

paper

Baranov, Vladimir V.; Galochkin, Anton A.; Nelyubina, Yulia V.; Kravchenko, Angelina N.; Makhova, Nina N.: Synthesis and Structure of 1-Substituted Semithioglycolurils
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0161_ga_10-1055_s-0040-1707391.gif

psp

Cavarischia, Claudia; Comely, Alex; Écija, Marta; Iacoangeli, Tommaso; Pastó, Mireia; Silvestri, Lavinia; Furlotti, Guido: A Convenient, Scalable Process for the Preparation and Purification of Calcium Acamprosate
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0163_ga_10-1055_s-0040-1707399.gif

special topic

Verma, Saumya; Kumar, Puneet; Khatana, Anil K.; Chandra, Dinesh; Yadav, Ajay K.; Tiwari, Bhoopendra; Jat, Jawahar L.: Zinc(II)-Catalyzed Synthesis of Secondary Amides from Ketones via Beckmann Rearrangement Using Hydroxylamine-O-sulfonic Acid in Aqueous Media
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0225_ga_10-1055_s-0040-1707809.gif

Publication Date: 20 May 2020

Publication Date: 19 May 2020

Publication Date: 18 May 2020

short review

Publication Date: 15 May 2020

Publication Date: 14 May 2020

paper

Zhou, Hongyan; Duan, Jiaokui; Xie, Dongtai; Yang, Jingya; Ma, Ben; Wang, Ganggang; Wu, Chengqi; Wang, Xi-Cun: Electrochemical Synthesis of Sulfinic Esters via Aerobic Oxidative Esterification of Thiophenols with Alcohols
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0043_ga_10-1055_s-0040-1707966.gif

short review

Liu, Xue; Wu, Xiangmei; Zhang, Ling; Lin, Xiaoyan; Huang, Dayun: Recent Advances in Triarylmethane Synthesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0156_ga_10-1055_s-0040-1707115.gif

Publication Date: 13 May 2020

special topic

Spiliopoulou, Nikoleta; Constantinou, Constantinos T.; Triandafillidi, Ierasia; Kokotos, Christoforos G.: Synthetic Approaches to Acyl Hydrazides and Their Use as Synthons in Organic Synthesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0186_ga_10-1055_s-0040-1707394.gif

Publication Date: 12 May 2020

paper

Camargo, Adriano F.; Marangoni, Mário A.; de Moraes, Paulo A.; Nogara, Pablo A.; Afolabi, Blessing A.; Bencke, Carlos E.; Rocha, João B. T.; Bonacorso, Helio G.; Martins, Marcos A. P.; Zanatta, Nilo: Regioselective Synthesis of Pyrazolyl-pyrimidine Hybrids of Pharmacological Interest
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0114_ga_10-1055_s-0040-1707948.gif

paper

Cocoletzi-Xochitiotzi, Ana Patricia; Hernández-Hernández, Miguel; Medina-Mercado, Ignacio; Jiménez-Martínez, Williams de Jesús; Mastranzo, Virginia Maricela; Porcel, Susana: Gold-Catalyzed Partial Hydrogenation of Activated Alkynes Mediated by Triphenylphosphine
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0020_ga_10-1055_s-0040-1707395.gif

Publication Date: 05 May 2020

Publication Date: 28 April 2020

Publication Date: 27 April 2020

paper

Saraiva Rosa, Nathalie; Glachet, Thomas; Ibert, Quentin; Lohier, Jean-François; Franck, Xavier; Reboul, Vincent: A Straightforward Synthesis of N-Substituted Ureas from Primary Amides
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0087_ga_10-1055_s-0040-1707103.gif

paper

Sekino, Tomoyuki; Sato, Shunta; Kuwabara, Kazuki; Takizawa, Koji; Yoshino, Tatsuhiko; Kojima, Masahiro; Matsunaga, Shigeki: Allyl 4-Chlorophenyl Sulfone as a Versatile 1,1-Synthon for Sequential α-Alkylation/Cobalt-Catalyzed Allylic Substitution
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0137_ga_10-1055_s-0040-1707524.gif

Publication Date: 22 April 2020

paper

Gusarova, Nina K.; Ivanova, Nina I.; Khrapova, Kseniya O.; Volkov, Pavel A.; Telezhkin, Anton A.; Larina, Lyudmila I.; Afonin, Andrei V.; Pavlov, Dmitry V.; Trofimov, Boris A.: Catalyst- and Solvent-Free Hydrophosphorylation of Ketones with Secondary Phosphine Oxides: Green Synthesis of Tertiary α-Hydroxyphosphine Oxides
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0088_ga_10-1055_s-0040-1707945.gif

Publication Date: 21 April 2020

Publication Date: 20 April 2020

paper

Ichikawa, Yoshiyasu; Hasegawa, Tomoyuki; Minami, Takahiro; Sato, Hiroshi; Morishita, Yukinori; Ochi, Rika; Masuda, Toshiya: Further Development of the Tin-Catalyzed Transcarbamoylation Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0143_ga_10-1055_s-0040-1708020.gif

paper

Kafle, Arjun; Bhattarai, Shrijiana; Handy, Scott T.: An Unusual Triazole Synthesis from Aurones
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0018_ga_10-1055_s-0040-1708019.gif

Publication Date: 16 April 2020

paper

Obydennov, Dmitrii L.; Viktorova, Viktoria V.; Chernyshova, Elena V.; Shirinkin, Alexander S.; Usachev, Sergey A.; Sosnovskikh, Vyacheslav Y.: Direct Synthesis of 5-Acyl-3-oxy-4-pyrones Based On Acid-­Catalyzed Acylation of Enaminodiones with Acylbenzotriazoles via Soft Enolization
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0122_ga_10-1055_s-0040-1707471.gif

Publication Date: 14 April 2020

paper

short review

Danilkina, Natalia A.; Govdi, Anastasia I.; Balova, Irina A.: 5-Iodo-1H-1,2,3-triazoles as Versatile Building Blocks
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0696_ga_10-1055_s-0039-1690858.gif

short review

Mittersteiner, Mateus; Bonacorso, Helio G.; Martins, Marcos A. P.; Zanatta, Nilo: Brominated β-Alkoxyvinyl Trihalomethyl Ketones as Promising Synthons in Heterocyclic Synthesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0082_ga_10-1055_s-0039-1690890.gif

short review

Smolobochkin, Andrey V.; Gazizov, Almir S.; Turmanov, Rakhymzhan A.; Abdullaeva, Dinara S.; Burilov, Alexander R.; Pudovik, Michail A.: N-Phosphorylated Pyrrolidines: An Overview of Synthetic Approaches
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0098_ga_10-1055_s-0039-1690889.gif

Publication Date: 09 April 2020

review

Publication Date: 07 April 2020

paper

Vetica, Fabrizio; Bailey, Stephen J.; Kumar, Mukesh; Mahajan, Suruchi; von Essen, Carolina; Rissanen, Kari; Enders, Dieter: Palladium-Catalyzed [3+2] Cycloaddition of Vinylaziridine and Indane-1,3-diones: Diastereo- and Enantioselective Access to Spiro-Pyrrolidines
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0014_ga_10-1055_s-0040-1707472.gif

Publication Date: 06 April 2020

paper

Lan, Jin; Jiang, Guofang; Yang, Jiangnan; Zhu, Haibo; Le, Zhanggao; Xie, Zongbo: α-Chymotrypsin-Induced Acetalization of Aldehydes and Ketones with Alcohols
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0067_ga_10-1055_s-0039-1690883.gif

Publication Date: 02 April 2020

Publication Date: 30 March 2020

Publication Date: 27 March 2020

paper

Sharathna, Puthiyaparambath; Meenu, Murugan Thulasi; Dhanya, Bhandara Purayil; Gopalan, Greeshma; Sasikumar, Parameswaran; Krishnan, Radhakrishnan Syam; Radhakrishnan, Kokkuvayil Vasu: Accessing Polycyclic Terpenoids from Zerumbone via Lewis Acid Catalyzed Synthetic Strategies
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0695_ga_10-1055_s-0039-1690840.gif

Publication Date: 26 March 2020

Publication Date: 24 March 2020

paper

Soeiro, Pedro F.; Serrano, João L.; Paixão, José A.; Boto, Renato E. F.; Silvestre, Samuel; Almeida, Paulo: The Synthesis of 2-Spiroindolin-3-one-(thio)barbiturates from 2,1-Benzisoxazoles: A Rearrangement Promoted by Thermal Conditions
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0050_ga_10-1055_s-0039-1690865.gif

Publication Date: 18 March 2020

paper

Dennis, Francesca M.; Robertson, Craig C.; Partridge, Benjamin M.: Nickel-Catalysed Allylboration of Aldehydes
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0028_ga_10-1055_s-0039-1690091.gif

Publication Date: 16 March 2020

special topic

Maligres, Peter E.; Song, Zhiguo Jake; Strotman, Neil A.; Yin, Jinquin; Pei, Tao; Strotman, Hallena R.; Itoh, Tetsuji; Sherer, Edward C.; Humphrey, Guy R.: Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0045_ga_10-1055_s-0040-1707994.gif

Publication Date: 12 March 2020

paper

Nadirova, Maryana A.; Laba, Yevhen-Oleh V.; Zaytsev, Vladimir P.; Sokolova, Julya S.; Pokazeev, Kuzma M.; Anokhina, Victoria A.; Khrustalev, Victor N.; Horak, Yuriy I.; Lytvyn, Roman Z.; Siczek, Miłosz; Kinzhybalo, Vasyl; Zubavichus, Yan V.; Kuznetsov, Maxim L.; Obushak, Mykola D.; Zubkov, Fedor I.: Application of the Intramolecular Diels–Alder Vinylarenе (IMDAV) Approach for the Synthesis of Thieno[2,3-f]isoindoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0672_ga_10-1055_s-0039-1690833.jpg

paper

Stepaniuk, Oleksandr O.; Rudenko, Tymofii V.; Vashchenko, Bohdan V.; Matvienko, Vitalii O.; Kondratov, Ivan S.; Tolmachev, Andrey A.; Grygorenko, Oleksandr O.: Synthesis of Fused Pyridine Carboxylates by Reaction of β-Alkoxyvinyl Glyoxylates with Amino Heterocycles
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0064_ga_10-1055_s-0039-1707987.gif

Publication Date: 05 March 2020

paper

Egashira, Gen; Kajimoto, Chihiro; Kataoka, Takuto; Yamada, Shigeyuki; Konno, Tsutomu: Synthesis and Application of Tetrafluoroethylene (CF2CF2)-Containing Acetylene Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0009_ga_10-1055_s-0039-1691744.gif

Publication Date: 03 March 2020

Publication Date: 20 February 2020

paper