DOI: 10.1055/s-00000084

Synthesis

eFirst

Publication Date: 05 September 2019

paper

Agafonova, Anastasiya V.; Smetanin, Ilia A.; Rostovskii, Nikolai V.; Khlebnikov, Alexander F.; Novikov, Mikhail S.: Easy Access to 2-Fluoro- and 2-Iodo-2H-azirines via the Halex Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0403_ga_10-1055_s-0039-1690200.gif
Supporting Information

paper

Bhilare, Shatrughn; Shah, Jagrut; Gaikwad, Vinayak; Gupta, Gaurav; Sanghvi, Yogesh S.; Bhanage, Bhalchandra M.; Kapdi, Anant R.: Pd/PTABS: An Efficient Catalytic System for the Aminocarbonylation of a Sugar-Protected Nucleoside
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0370_ga_10-1055_s-0039-1690190.gif
Supporting Information

paper

Mangaonkar, Saeesh R.; Singh, Fateh V.: Hypervalent Iodine(III)-Catalyzed Epoxidation of β-Cyanostyrenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0347_ga_10-1055_s-0039-1690621.gif
Supporting Information

paper

Rudy, Heinrich-Karl A.; Wanner, Klaus T.: Accessing Tricyclic Imines Comprising a 2-Azabicyclo[2.2.2]octane Scaffold by Intramolecular Hetero-Diels–Alder Reaction of 4-Alkenyl-Substituted N-Silyl-1,4-dihydropyridines
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0378_ga_10-1055_s-0039-1690619.gif
Supporting Information

Publication Date: 03 September 2019

paper

Bannwart, Linda M.; Rieder, Pascal S.; Mayor, Marcel: 2-(3-Cyanopropyldimethylsilyl)ethyl as a Polar Sulfur Protecting Group
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0337_ga_10-1055_s-0039-1690184.gif
Supporting Information Primary Data

paper

Heinz, Benjamin; Balkenhohl, Moritz; Knochel, Paul: Thiolation of Pyridine-2-sulfonamides using Magnesium Thiolates
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0439_ga_10-1055_s-0039-1690199.gif
Supporting Information

paper

Jiang, Gan; Lin, Yang; Cai, Mingzhong; Zhao, Hong: Recyclable Heterogeneous Copper(II)-Catalyzed Oxidative Cyclization of 2-Pyridine Ketone Hydrazones Towards [1,2,3]Triazolo[1,5-a]pyridines
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0326_ga_10-1055_s-0037-1610726.gif
Supporting Information

Publication Date: 30 August 2019

paper

Mendoza, Manuel; Eom, Ryan; Salas, Celeste; Haynes-Smith, Jeremy; Billingsley, Kelvin L.: The Synthesis and Biological Evaluation of Indolactam Alkaloids
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0395_ga_10-1055_s-0039-1690198.gif
Supporting Information

Publication Date: 29 August 2019

paper

Rodrigues, Shirley M. M.; Previdi, Daniel; Baviera, Giovanni S.; Matias, Alexandre A.; Donate, Paulo M.: Niobium Pentachloride Mediated (Hetero)aromatic Aldehyde Friedel–Crafts Hydroxyalkylation with Arenes: An Efficient Strategy to Synthesize Triarylmethanes
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0349_ga_10-1055_s-0037-1610727.gif
Supporting Information

Publication Date: 28 August 2019

paper

Chen, Yangfan; Wu, Di; Zhou, Jiawen; Wang, Yun; Huang, Jing; Xu, Xichen: Thermally Induced Intramolecular Benzannulation of Diazoacetoacetate Enones Tethered with Unactivated Alkynes: Synthesis of Substituted 6H-Benzo[c]chromenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0266_ga_10-1055_s-0039-1690191.gif
Supporting Information

paper

Dar’in, Dmitry; Kantin, Grigory; Krasavin, Mikhail: Practical Application of the Aqueous ‘Sulfonyl-Azide-Free’ (SAFE) Diazo Transfer Protocol to Less α-C–H Acidic Ketones and Esters
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0367_ga_10-1055_s-0039-1690613.gif
Supporting Information

paper

Murre, Aleksandra; Erkman, Kristin; Kaabel, Sandra; Järving, Ivar; Kanger, Tõnis: Diastereoselective [2,3]-Sigmatropic Rearrangement of N-Allyl Ammonium Ylides
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0257_ga_10-1055_s-0039-1690185.gif
Supporting Information

Publication Date: 26 August 2019

paper

Ghotekar, Ganesh S.; Mujahid, M.; Muthukrishnan, M.: Efficient Synthesis of Optically Active Neolignans Ligraminol D and E
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0352_ga_10-1055_s-0037-1611919.gif
Supporting Information

paper

Kotha, Sambasivarao; Keesari, Ramakrishna Reddy; Ansari, Saima: Synthesis of Aza-polyquinanes via Fischer Indolization and Ring-Rearrangement Metathesis as Key Steps
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0256_ga_10-1055_s-0039-1690179.jpg
Supporting Information CIF File

paper

Rey, Marine; Beaumont, Stéphane: Molybdenum-Mediated One-Pot Synthesis of Pyrazoles from Isoxazoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0415_ga_10-1055_s-0039-1690615.gif
Supporting Information

paper

Singh, Adesh Kumar; Venkatesh, Rapelly; Kandasamy, Jeyakumar: Palladium-Catalyzed One-Pot Stereospecific Synthesis of 2-Deoxy Aryl C-Glycosides from Glycals and Anilines in the Presence of tert-Butyl Nitrite
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0165_ga_10-1055_s-0037-1611916.gif
Supporting Information

short review

Zeidan, Nicolas; Lautens, Mark: Migratory Insertion Strategies for Dearomatization
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0431_ga_10-1055_s-0037-1611918.gif

Publication Date: 22 August 2019

paper

Huang, Shuai Shuai; Zheng, Zhan Jiang; Cui, Yu Ming; Xu, Zheng; Yang, Ke Fang; Xu, Li Wen: Convenient Synthesis of 2-(2,2-Difluoroethoxy)-6-(trifluoromethyl)-benzenesulfonyl Chloride, A Key Building Block of Penoxsulam
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0389_ga_10-1055_s-0039-1690617.gif
Supporting Information

paper

Li, Xing; Yan, Wenjing; Zhang, Rui; Chang, Honghong; Gao, Wenchao; Tian, Xiuping; Wei, Wenlong: Direct Synthesis of Nitrones via Transition-Metal-Free Ring-Opening of N-Tosylaziridines with the Nitrogen Atom of Various (E)-Aldoximes and (E)-Ketoximes
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0309_ga_10-1055_s-0039-1690186.gif
Supporting Information

Publication Date: 21 August 2019

paper

da Silva, Caren D. G.; Katla, Ramesh; dos Santos, Beatriz F.; Tavares Junior, José M. C.; Albuquerque, Tábata B.; Kupfer, Vicente L.; Rinaldi, Andrelson W.; Domingues, Nelson L. C.: Cobalt Used as a Novel and Reusable Catalyst: A New and One-Pot Synthesis of Isatin-Derived N,S-Acetals Using Substituted Isatins and Thiols
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0306_ga_10-1055_s-0037-1611913.gif
Supporting Information

paper

Loubidi, M.; Lorion, M.; El Hakmaoui, A.; Bernard, P.; Akssira, M.; Guillaumet, G.: One-Step Synthesis of 1H-Imidazo[1,5-a]imidazole Scaffolds and Access to their Polyheterocycles
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0139_ga_10-1055_s-0039-1690182.gif
Supporting Information

paper

Petko, Dina; Pounder, Austin; Tam, William: Ruthenium-Catalyzed [2+2+2] Bis-Homo-Diels–Alder Cycloadditions of 1,5-Cyclooctadiene with Alkynyl Phosphonates
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0399_ga_10-1055_s-0039-1690612.gif
Supporting Information

paper

Zhang, Lin-Lin; Li, Ya-Ting; Gao, Ting; Guo, Sha-Sha; Yang, Bei; Meng, Zi-Hui; Dai, Qi-Pu; Xu, Zhi-Bin; Wu, Qin-Pei: Efficient Synthesis of Diverse 5-Thio- or 5-Selenotriazoles: One-Pot Multicomponent Reaction from Elemental Sulfur or Selenium
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0277_ga_10-1055_s-0039-1690618.gif
Supporting Information

special topic

Milicevic Sephton, Selena; Zhou, Xiaoyun; Thompson, Stephen; Aigbirhio, Franklin I.: Preparation of the Serotonin Transporter PET Radiotracer 2-({2-[(Dimethylamino)methyl]phenyl}thio)-5-[18F]fluoroaniline (4-[18F]ADAM): Probing Synthetic and Radiosynthetic Methods
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0355_ga_10-1055_s-0039-1690522.gif
Supporting Information

Publication Date: 15 August 2019

paper

Rajeshkumar, Venkatachalam; Neelamegam, Chinnaraj; Anandan, Sambandam: An Expedient, Direct, Three-Component Approach for the Synthesis of 4-Thioarylpyrroles
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0171_ga_10-1055_s-0039-1690024.gif
Supporting Information

psp

Ashida, Yuya; Kondo, Shoichi; Arashiba, Kazuya; Kikuchi, Takamasa; Nakajima, Kazunari; Kakimoto, Seizo; Nishibayashi, Yoshiaki: A Practical Synthesis of Ammonia from Nitrogen Gas, Samarium Diiodide and Water Catalyzed by a Molybdenum–PCP Pincer Complex
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0353_ga_10-1055_s-0039-1690151.gif

Publication Date: 14 August 2019

paper

Evangelista, Tereza C. Santos; Lopéz, Óscar; Sydnes, Magne O.; Fernández-Bolaños, José G.; Ferreira, Sabrina Baptista; Lindbäck, Emil: Bicyclic 1-Azafagomine Derivatives: Synthesis and Glycosidase Inhibitory Testing
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0308_ga_10-1055_s-0039-1690019.gif
Supporting Information

paper

Jian, Junsheng; Wang, Zijia; Chen, Liuqing; Gu, Ying; Miao, Liqiong; Liu, Yueping; Zeng, Zhuo: A Straightforward Conversion of Activated Amides and Haloalkanes into Esters under Transition-Metal-Free Cs2CO3/DMAP Conditions
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0204_ga_10-1055_s-0039-1690178.gif
Supporting Information

paper

Wang, Rui-Xiang; Fang, Zhuang; Qiu, Guanyinsheng; Xie, Wenlin; Liu, Jin-Biao: Copper-Catalyzed 6-endo-dig O-Cyclization of 2-(But-3-en-1-yn-1-yl)benzamide
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0342_ga_10-1055_s-0039-1690155.gif
Supporting Information

Publication Date: 12 August 2019

paper

Aguilar, Abel A. Arroyo; Ledesma, Gabriela N.; Tirloni, Bárbara; Kaufman, Teodoro S.; Larghi, Enrique L.: Convergent First Total Synthesis of Melovinone: A Densely Substituted 3-Methoxy-4-quinolone Isolated from Melochia tomentosa L.
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0298_ga_10-1055_s-0039-1690164.gif
Supporting Information CIF File

paper

Chuprun, Sergey; Dar’in, Dmitry; Kantin, Grigory; Krasavin, Mikhail: [3+2]-Cycloaddition of α-Diazocarbonyl Compounds with Arenediazonium Salts Catalyzed by Silver Nitrate Delivers 2,5-Disubstituted Tetrazoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0354_ga_10-1055_s-0039-1690159.gif
Supporting Information

paper

Reinus, Brandon J.; Kerwin, Sean M.: N-Alkynyl Pyrrole Based Total Synthesis of Shensongine A
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0275_ga_10-1055_s-0037-1611904.gif
Supporting Information

short review

Li, Yuyang; Kluger, Ronald: Metal-Catalyzed Site-Selective Monoacylation of Diols in Aqueous Media
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0260_ga_10-1055_s-0037-1611907.gif

Publication Date: 08 August 2019

paper

Gao, Yejun; Chen, Rener; Ma, Yongmin: Synthesis of Asymmetrical 2,6-Diarylpyridines from Linear α,β,γ,δ-Unsaturated Ketones by Addition of Ammonium Formate Followed by Annulation
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0317_ga_10-1055_s-0037-1610725.gif
Supporting Information

paper

Majnooni, Sahar; Almansaf, Zainab; Tsuji, Miu; Khosropour, Ahmad R.; Zali-Boeini, Hassan; Beyzavi, M. Hassan: Straightforward and Expeditious One-Pot Tandem Synthesis of 3,5-Diaryl-1,2,4-Selenadiazoles from Aryl Nitriles
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0286_ga_10-1055_s-0039-1690126.gif
Supporting Information

paper

Vagkidis, Nikolaos; Brown, Alexander J.; Clarke, Paul A.: Evaluation of Amino Nitriles and an Amino Imidate as Organo­catalysts in Aldol Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0330_ga_10-1055_s-0039-1690150.gif
Supporting Information

paper

Wei, Song; Ouyang, Banlai; Deng, Zhihong; Yang, Qin; Peng, Yiyuan: Palladium-Catalyzed and Quinazoline-Directed C–H Selective Acetoxylation of 2-Arylquinazolines
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0282_ga_10-1055_s-0037-1611908.gif
Supporting Information

Publication Date: 07 August 2019

errata

Dank, Christian; Sanichar, Randy; Choo, Ken-Loon; Olsen, Madeline; Lautens, Mark: Recent Advances Towards Syntheses of Diterpenoid Alkaloids

paper

Chiassai, Leonardo; Ballesteros-Garrido, Rafael; Clares, Maria Paz; García-España, Enrique; Ballesteros, Rafael; Abarca, Belén: Combining Amines and 3-(2-Pyridyl)-[1,2,3]Triazolo[1,5-a]pyridine: An Easy Access to New Functional Polynitrogenated Ligands
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0287_ga_10-1055_s-0037-1611901.gif
Supporting Information

paper

Lu, Jianyu; Koldas, Serkan; Fan, Huafang; Desper, John; Day, Victor W.; Hua, Duy H.: A One-Pot Intramolecular Tandem Michael–Aldol Annulation Reaction for the Synthesis of Chiral Pentacyclic Terpenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0327_ga_10-1055_s-0039-1690521.gif
Supporting Information

Publication Date: 06 August 2019

paper

Bhatt, Ashish; Singh, Rajesh K.; Kant, Ravi; Sarma, Bhupendra K.: A Convenient Synthesis of 1,5-Fused 1,2,4-Triazoles from N-Arylamidines via Chloramine-T Mediated Intramolecular Oxidative N–N Bond Formation
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0223_ga_10-1055_s-0037-1611906.gif
Supporting Information

paper

Garrido, Amanda; Delaye, Pierre-Olivier; Quintin, François; Abarbri, Mohamed; Lameiras, Pedro; Gueiffier, Alain; Thibonnet, Jérôme; Petrignet, Julien: Direct Access to Highly Functionalised Benzimidazoles and Benzoxazoles from a Common Precursor
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0372_ga_10-1055_s-0039-1690153.gif
Supporting Information

Publication Date: 05 August 2019

paper

Wang, Yang; Zhao, Cun-Yuan; Wang, Yi-Ping; Zheng, Wen-Hua: Enantioselective Intramolecular Dearomative Lactonization of Naphthols Catalyzed by Planar Chiral Iodoarene
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0292_ga_10-1055_s-0037-1611902.gif
Supporting Information

review

Dank, Christian; Sanichar, Randy; Choo, Ken-Loon; Olsen, Madeline; Lautens, Mark: Recent Advances Towards Syntheses of Diterpenoid Alkaloids
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0341_ga_10-1055_s-0037-1611897.jpg

Publication Date: 01 August 2019

paper

Redon, Sébastien; Kosso, Anne Roly Obah; Broggi, Julie; Vanelle, Patrice: Metal-Free ipso-Selenocyanation of Arylboronic Acids Using Malononitrile and Selenium Dioxide
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0324_ga_10-1055_s-0039-1690013.gif
Supporting Information

paper

Siddiqui, Saher H.; Navuluri, Chandrasekhar; Charette, André B.: Enantioselective Synthesis of cis- and trans-Borocyclopropylmethanol: Simple Building Blocks To Access Heterocycle-Substituted Cyclopropylmethanols
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0358_ga_10-1055_s-0037-1611896.gif
Supporting Information

paper

Zhang, Xu; Cao, Wen-Bin; Xu, Xiao-Ping; Ji, Shun-Jun: Treatment of Olefinic Amides with NBS in Water: Synthesis of Monobromo- and Multibromobenzoxazines
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0244_ga_10-1055_s-0037-1610724.gif
Supporting Information

Publication Date: 31 July 2019

paper

Kamijo, Shin; Kamijo, Kaori; Murafuji, Toshihiro: Aryl Ketone Mediated Photoinduced Radical Coupling for the Alkylation­ of Benzazoles Employing Saturated Heterocyclic Compounds­
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0264_ga_10-1055_s-0037-1611895.gif
Supporting Information

short review

Rossignon, Alexandre; Bonifazi, Davide: O-Annulation Leading to Five-, Six-, and Seven-Membered Cyclic Diaryl Ethers Involving C–H Cleavage
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0237_ga_10-1055_s-0037-1611892.gif

Publication Date: 30 July 2019

paper

Cortón, Pablo; Novo, Paula; López-Sobrado, Vanesa; García, Marcos D.; Peinador, Carlos; Pazos, Elena: Solid-Phase Zincke Reaction for the Synthesis of Peptide-4,4′-bipyridinium Conjugates
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0303_ga_10-1055_s-0039-1690016.gif
Supporting Information

paper

Zhang, Min; Yang, Wenbo; Li, Kailu; Sun, Ke; Ding, Jianfen; Yang, Liuqing; Zhu, Chunyin: Facile Synthesis of Dispiroheterocycles through One-Pot [3+2] Cycloaddition, and Their Antiviral Activity
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0156_ga_10-1055_s-0037-1611900.gif
Supporting Information

special topic

Thompson, Stephen; Lee, So Jeong; Jackson, Isaac M.; Ichiishi, Naoko; Brooks, Allen F.; Sanford, Melanie S.; Scott, Peter J. H.: Synthesis of [18F]-γ-Fluoro-α,β-unsaturated Esters and Ketones via Vinylogous 18F-Fluorination of α-Diazoacetates with [18F]AgF
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0373_ga_10-1055_s-0039-1690012.jpg
Supporting Information

Publication Date: 29 July 2019

paper

Khaldoun, Khadidja; Safer, Abdelmounaim; Saidi-Besbes, Salima; Carboni, Bertrand; Le Guével, Rémy; Carreaux, François: An Efficient Solvent-Free Microwave-Assisted Synthesis of Cinnamamides by Amidation Reaction Using Phenylboronic Acid/Lewis Base Co-catalytic System
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0333_ga_10-1055_s-0039-1690132.gif
Supporting Information

paper

Wang, Shi-Meng; S. Alharbi, Njud; Qin, Hua-Li: Construction of Esters through Sulfuryl Fluoride (SO2F2) Mediated Dehydrative Coupling of Carboxylic Acids with Alcohols at Room Temperature
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0319_ga_10-1055_s-0039-1690017.gif
Supporting Information

review

Wu, Ronghai; Huang, Keke; Qiu, Guanyinsheng; Liu, Jin-Biao: Synthesis of Thioethers from Sulfonyl Chlorides, Sodium Sulfinates, and Sulfonyl Hydrazides
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0209_ga_10-1055_s-0039-1690015.jpg

Publication Date: 25 July 2019

paper

Almasalma, Ahmad A.; Mejía, Esteban: Allylic C–H Alkynylation via Copper-Photocatalyzed Cross-Dehydrogenative Coupling
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0252_ga_10-1055_s-0039-1690014.jpg
Supporting Information

Publication Date: 24 July 2019

paper

Reddy, Chada Raji; Warudikar, Kamalkishor; Latha, Bellamkonda: Facile Strategy to Access the Indolo[2,3-a]quinolizidine Framework: Synthetic Study on Tangutorine
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0295_ga_10-1055_s-0039-1690004.gif
Supporting Information

special topic

Pang, Jia Hao; Ong, Derek Yiren; Watanabe, Kohei; Takita, Ryo; Chiba, Shunsuke: Leaving Group Ability in Nucleophilic Aromatic Amination by Sodium Hydride–Lithium Iodide Composite
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0368_ga_10-1055_s-0039-1690010.gif
Supporting Information

Publication Date: 23 July 2019

special topic

Kitahara, Kazumasa; Mizutani, Haruna; Iwasa, Seiji; Shibatomi, Kazutaka: Asymmetric Synthesis of α-Chloro-α-halo Ketones by Decarboxylative Chlorination of α-Halo-β-ketocarboxylic Acids
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0320_ga_10-1055_s-0039-1690009.gif
Supporting Information

Publication Date: 16 July 2019

paper

Chen, Yaoyao; Li, Chengliang; Cui, Yongmei; Sun, Mingming; Jia, Xueshun; Li, Jian: Bu4NI-Catalyzed C–C Bond Cleavage and Oxidative Esterification of Allyl Alcohols with Toluene Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0247_ga_10-1055_s-0039-1690105.gif
Supporting Information

paper

Fonzo, Santiago; Vargas, Didier F.; Kaufman, Teodoro S.: A Ruthenium-Catalyzed C–H Activation Strategy as an Efficient Shortcut in the Total Synthesis of 6,8-Dimethoxy-1,3-dimethyl­isoquinoline
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0296_ga_10-1055_s-0037-1610720.gif
Supporting Information

paper

Munnuri, Sailu; Verma, Saumya; Chandra, Dinesh; Anugu, Raghunath Reddy; Falck, John R.; Jat, Jawahar L.: Cu(OTf)2-Catalyzed Beckmann Rearrangement of Ketones Using Hydroxylamine-O-sulfonic Acid (HOSA)
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0314_ga_10-1055_s-0039-1690005.gif
Supporting Information

Publication Date: 15 July 2019

paper

Chen, Weiqiang; Zhang, Yin-Lin; Li, Hui-Jing; Nan, Xiang; Liu, Ying; Wu, Yan-Chao: Synthesis of N-Sulfonyl- and N-Acylpyrroles via a Ring-Closing Metathesis/Dehydrogenation Tandem Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0322_ga_10-1055_s-0039-1690002.gif
Supporting Information

paper

Jung, Seunghee; Kawashima, Yuya; Noguchi, Takuya; Imai, Nobuyuki: Synthesis of Acetaminophen Analogues Containing α-Amino Acids and Fatty Acids for Inhibiting Hepatotoxicity
https://www.thieme-connect.de/media/synthesis/EFirst/i_s0321_ga_10-1055_s-0037-1611893.gif

paper

Shabalin, Dmitrii A.; Ivanova, Elena V.; Ushakov, Igor A.; Schmidt, Elena Yu.; Trofimov, Boris A.: Regioselective Synthesis of 2-Acylbutadienes from β,γ-Unsaturated Ketones
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0299_ga_10-1055_s-0039-1690003.jpg
Supporting Information

Publication Date: 11 July 2019

paper

Silm, Estelle; Kaabel, Sandra; Järving, Ivar; Kanger, Tõnis: Asymmetric Organocatalytic Michael Addition–Cyclisation Cascade of Cyclopentane-1,2-dione with Alkylidene Malononitriles
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0274_ga_10-1055_s-0039-1690484.gif
Supporting Information

paper

Yang, Bo; Zhang, Songlin: Highly γ-Regioselective 1,2-Addition of α,β-Unsaturated Oxime Ethers with Allylzinc Bromides: A Straightforward Approach for the Synthesis of Homoallylic Amines
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0193_ga_10-1055_s-0039-1690127.gif
Supporting Information

Publication Date: 10 July 2019

paper

Yepez, Gerardo; Poyil, Anurag Noonikara; Bugarin, Alejandro: Large-Scale Synthesis of Aniline Trimers in Different Oxidation States
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0278_ga_10-1055_s-0037-1611889.gif
Supporting Information

Publication Date: 09 July 2019

special topic

Dubost, Emmanuelle; Babin, Victor; Benoist, Florian; Hébert, Alexandra; Pigrée, Gilbert; Bouillon, Jean-Philippe; Fabis, Frédéric; Cailly, Thomas: Improvements of C–H Radio-Iodination of N-Acylsulfonamides toward Implementation in Clinics
https://www.thieme-connect.de/media/synthesis/EFirst/i_s0301_ga_10-1055_s-0037-1611884.gif
Supporting Information

special topic

Sarie, Jérôme C.; Neufeld, Jessica; Daniliuc, Constantin G.; Gilmour, Ryan: Willgerodt-Type Dichloro(aryl)-λ3-Iodanes: A Structural Study
https://www.thieme-connect.de/media/synthesis/EFirst/i_s0315_ga_10-1055_s-0037-1611886.gif
Supporting Information

Publication Date: 08 July 2019

paper

Golushko, Andrei; Dar’in, Dmitry; Kantin, Grigory; Guranova, Natalia; Vasilyev, Aleksander V.; Krasavin, Mikhail: Medicinally Relevant Modification of the Isoquinoline-1,3-dione Scaffold via Metal-Free Arylation and Fluorination of Diazo Homophthalimides­ in Brønsted Acids
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0276_ga_10-1055_s-0037-1611882.gif
Supporting Information

paper

Nagaraju, Tumula; Krishna, Palakodety Radha; Sridhar, Balasubramanian; Mangarao, Nakka: PhI(OAc)2-Mediated Regioselective Synthesis of 5-Guanidino-1,2,4-thiadiazoles and 1,2,4-Triazolo[1,5-a]pyridines via Oxidative N–S and N–N Bond Formation
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0101_ga_10-1055_s-0037-1611854.gif
Supporting Information CIF File

paper

Tarasova, Olga A.; Nedolya, Nina A.; Albanov, Alexander I.; Trofimov, Boris A.: Synthesis of 2-[(5-Amino-1H-pyrrol-2-yl)sulfanyl]acetic Acid Esters: One-Pot Assembly from Propargyl Amines, Isothiocyanates, and Alkyl­ 2-Bromoacetates
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0271_ga_10-1055_s-0037-1611883.gif
Supporting Information

Publication Date: 03 July 2019

paper

Makarov, Anton S.; Kekhvaeva, Anna E.; Chalikidi, Petrakis N.; Abaev, Vladimir T.; Trushkov, Igor V.; Uchuskin, Maxim G.: A Simple Synthesis of Densely Substituted Benzofurans by Domino Reaction of 2-Hydroxybenzyl Alcohols with 2-Substituted Furans
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0232_ga_10-1055_s-0039-1690000.gif
Supporting Information

special topic

Sutherland, Andrew: Radiohalogenation of Organic Compounds: Practical Considerations and Challenges for Molecular Imaging
https://www.thieme-connect.de/media/synthesis/EFirst/i_s0302_ga_10-1055_s-0037-1611885.jpg

Publication Date: 01 July 2019

review

Mittal, Rupali; Awasthi, Satish K.: Recent Advances in the Synthesis of 5-Substituted 1H-Tetrazoles: A Complete Survey (2013–2018)
https://www.thieme-connect.de/media/synthesis/EFirst/i_e0207_ga_10-1055_s-0037-1611863.gif

Publication Date: 26 June 2019

paper

Fatykhov, Ramil F.; Khalymbadzha, Igor A.; Chupakhin, Oleg N.; Charushin, Valery N.; Inyutina, Anna K.; Slepukhin, Pavel A.; Kartsev, Victor G.: 1-Nicotinoylbenzotriazole: A Convenient Tool for Site-Selective Protection of 5,7-Dihydroxycoumarins
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0173_ga_10-1055_s-0039-1690104.gif
Supporting Information CIF File

Publication Date: 19 June 2019

paper

Sakai, Takeo; Tatematsu, Toshiki; Fukuta, Ayumi; Kasai, Satomi; Hayashi, Kahori; Mori, Yuji: Benzyl Acetylcarbamate Potassium Salt (BENAC-K): A Simple Nucleophilic N-Acetamide Equivalent
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0289_ga_10-1055_s-0039-1690097.gif
Supporting Information

Publication Date: 18 June 2019

paper

Kobayashi, Eiji; Togo, Hideo: Facile One-Pot Transformation of Primary Alcohols into 3-Aryl- and 3-Alkyl-isoxazoles and -pyrazoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0261_ga_10-1055_s-0039-1690102.gif
Supporting Information

Publication Date: 28 May 2019

paper

Galván, Adriana; de la Cruz, Fabiola N.; Cruz, Francisco; Martínez, Merced; Gomez, Clarisa Villegas; Alcaraz, Yolanda; Domínguez, José Manuel; Delgado, Francisco; Vázquez, Miguel A.: Heterogeneous Catalysis with Basic Compounds to Achieve the Synthesis and C–N Cleavage of Azetidin-2-ones under Microwave Irradiation
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0136_ga_10-1055_s-0037-1611851.gif
Supporting Information