DOI: 10.1055/s-00000084

Synthesis

eFirst

Publication Date: 23 February 2021

special topic > Special Issue dedicated to Prof. Sarah Reisman, recipient of the 2019 Dr. Margaret Faul Women in Chemistry Award

Lam, Heather; Abel-Snape, Xavier; Köllen, Martin F.; Lautens, Mark: Recent Advances in Transition-Metal-Free (4+3)-Annulations
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0520_ga_10-1055_s-0040-1706023.gif

Publication Date: 22 February 2021

paper

Schädel, Nicole; Icik, Esra; Martini, Maike; Altevogt, Luca; Ramming, Isabell; Greulich, Andreas; Baro, Angelika; Bilitewski, Ursula; Laschat, Sabine: Synthesis of Imidazole and Histidine-Derived Cross-Linkers as Analogues of GOLD and Desmosine
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0588_ga_10-1055_s-0040-1706144.gif

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Watanabe, Hikaru; Nakajima, Kazuki; Ekuni, Kento; Edagawa, Ryota; Akagi, Yuta; Okuda, Yasuhiro; Wakamatsu, Kan; Orita, Akihiro: Custom-Made Pyrene Photocatalyst-Promoted Desulfonylation of Arylethenyl Sulfones Using Green-Light-Emitting Diodes
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0005_ga_10-1055_s-0040-1706025.gif

Publication Date: 18 February 2021

feature

Shaaban, Saad; Li, Houhua; Merten, Christian; Antonchick, Andrey P.; Waldmann, Herbert: Rhodium(III)-Catalyzed Enantioselective Benzamidation of Cyclopropenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0629_ga_10-1055_s-0040-1706026.gif

Publication Date: 15 February 2021

Publication Date: 10 February 2021

Publication Date: 09 February 2021

paper

Schefzig, Luise; Kurzawa, Timon; Rancan, Giaime; Linder, Igor; Leisering, Stefan; Bera, Mrinal K.; Gart, Max; Zimmer, Reinhold; Reissig, Hans-Ulrich: Access to Highly Substituted Pyrimidine N-Oxides and 4-Acetoxymethyl-Substituted Pyrimidines via the LANCA Three-Component Reaction–Cyclocondensation Sequence
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0636_ga_10-1055_s-0040-1706020.gif

Publication Date: 08 February 2021

Publication Date: 01 February 2021

paper

Kuwabara, Motoi; Matsuo, Ami; Kamo, Shogo; Matsuzawa, Akinobu; Sugita, Kazuyuki: Stereoselective Convergent Synthesis of Carbon Skeleton of Cotylenin A Aglycone
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0631_ga_10-1055_s-0040-1706684.gif

Publication Date: 28 January 2021

short review

Walther, Melanie; Kipke, Waldemar; Schultzke, Sven; Ghosh, Souvik; Staubitz, Anne: Modification of Azobenzenes by Cross-Coupling Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0528_ga_10-1055_s-0040-1705999.gif

Publication Date: 27 January 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 26 January 2021

Publication Date: 25 January 2021

Publication Date: 22 January 2021

Publication Date: 21 January 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 20 January 2021

Publication Date: 19 January 2021

paper

Chen, Jyun-Siao; Ke, Yi-Fan; Lin, Heng-Yan; Lin, Wesley; Yen, Wei-Chung; Wu, Hsin-Ru; Luo, Shun-Yuan: Development of a Novel Method for Trimethylsilylation of Saccharides­
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0542_ga_10-1055_s-0040-1705990.gif

Publication Date: 18 January 2021

errata

Srinivasulu, Vunnam; Al-Marzooq, Farah; Hamad, Mohamad; Khanfar, Monther A.; Ramanathan, Mani; Soares, Nelson C.; Al-Tel, Taleb H.: Sequencing Groebke–Blackburn–Bienaymé and Aza-Michael Addition Reactions: A Modular Strategy for Accessing a Diverse Collection of Constrained Benzoxazepine and Imidazopyrazine Systems

paper

Mityuk, Andrey P.; Hrebonkin, Andrii; Lebed, Pavlo S.; Grabchuk, Galyna P.; Volochnyuk, Dmitriy M.; Ryabukhin, Sergey V.: Efficient Route for the Synthesis of Diverse Heteroannelated 5-Cyanopyridines
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0627_ga_10-1055_a-1360-9852.gif

paper

Wang, Siqi; Filatov, Alexander S.; Lozovskiy, Stanislav V.; Shmakov, Stanislav V.; Khoroshilova, Olesya V.; Larina, Anna G.; Selivanov, Stanislav I.; Boitsov, Vitali M.; Stepakov, Alexander V.: Construction of Spiro[3-azabicyclo[3.1.0]hexanes] via 1,3-Dipolar Cycloaddition of 1,2-Diphenylcyclopropenes to Ninhydrin-Derived Azomethine Ylides
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0574_ga_10-1055_a-1360-9716.gif

short review

Publication Date: 15 January 2021

Publication Date: 14 January 2021

errata

Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)

review

Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0484_ga_10-1055_s-0040-1705983.gif

Publication Date: 13 January 2021

Publication Date: 11 January 2021

feature

Pruteanu, Elena; Tappin, Nicholas D. C.; Gîrbu, Vladilena; Morarescu, Olga; Dénès, Fabrice; Kulciţki, Veaceslav; Renaud, Philippe: Forskolin Editing via Radical Iodo- and Hydroalkylation
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0561_ga_10-1055_s-0040-1706003.gif

paper

Lisovenko, Natalya Yu.; Nasibullina, Ekaterina R.; Kharitonova, Svetlana S.; Myshkina, Olga A.: Simple Synthesis of Substituted 3-Hydroxyfuran-2(5H)-ones
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0541_ga_10-1055_s-0040-1705998.gif

paper

Yassine, Hasna; Bouali, Jamila; Oumessaoud, Asmaa; Ourhzif, El Mahdi; Hamri, Salha; Hafid, Abderrafia; Khouili, Mostafa; Pujol, Maria Dolors: Synthesis of New Dialkyl 2,2′-[Carbonylbis(azanediyl)]dibenzoates via Curtius Rearrangement
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0458_ga_10-1055_s-0040-1706643.gif

Publication Date: 08 January 2021

paper

Kotha, Sambasivarao; Pulletikurti, Sunil; Fatma, Ambareen; Dhangar, Gopal; Naidu, Gonna Somu: Synthesis of Polycycles and Oxacycles via Tandem Metathesis of endo-Norbornene Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0532_ga_10-1055_a-1348-4242.gif

Publication Date: 07 January 2021

Publication Date: 04 January 2021

short review

Singh, Pushpinder; Batra, Aanchal; Singh, Kamal Nain; Mritunjay, Mritunjay: Transition-Metal-Free Strategies for the Synthesis of C-1 Aryl-Substituted Tetrahydroisoquinolines
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0570_ga_10-1055_a-1344-2074.jpg

Publication Date: 30 December 2020

Publication Date: 29 December 2020

paper

Klochkova, Anastasiia; Bubyrev, Andrey; Dar’in, Dmitry; Bakulina, Olga; Krasavin, Mikhail; Sokolov, Viktor: Straightforward Route to γ-Sultams via Novel Tandem SN/Michael Addition
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0566_ga_10-1055_a-1343-9451.gif

Publication Date: 28 December 2020

feature

Ikari, Yuta; Kaihara, Takahito; Goto, Shimpei; Bovenkerk, Marcel; Grenz, David C.; Esser, Birgit; Ferreira, Marli; Stachelek, Patrycja; Data, Przemyslaw; Yoshida, Takumu; Ikai, Tomoyuki; Tohnai, Norimitsu; Minakata, Satoshi; Takeda, Youhei: Peripherally Donor-Installed 7,8-Diaza[5]helicenes as a Platform for Helical Luminophores
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0613_ga_10-1055_a-1343-5810.gif

Publication Date: 21 December 2020

feature

Ponce, Marian Blanco; Parpart, Silvio; Villinger, Alexander; Rodríguez, Eugenio Torres; Ehlers, Peter; Langer, Peter: Synthesis of Pyrrolo[1,2-a][1,6]- and [1,8]naphthyridines by Alkyne-Carbonyl Metathesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0529_ga_10-1055_s-0040-1706105.gif

paper

Publication Date: 18 December 2020

short review

Publication Date: 17 December 2020

Publication Date: 15 December 2020

paper

Gurbanov, Rustam; Sokolov, Andriy; Golovach, Sergey; Melnykov, Kostiantyn; Dobrydnev, Alexey V.; Grygorenko, Oleksandr O.: Synthesis of sp3-Enriched β-Fluoro Sulfonyl Chlorides
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0036_ga_10-1055_s-0040-1706101.jpg

special topic > Bond Activation – in Honor of Prof. Shinji Murai

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 14 December 2020

Publication Date: 10 December 2020

paper

Kitamura, Kei; Kanagawa, Hinano; Ozakai, Chiharu; Nishimura, Taichi; Tokuda, Hayato; Tsunoda, Tetsuto; Kaku, Hiroto: Synthesis of the Common Monomeric Unit of Uroleuconaphins and Viridaphins via Hauser–Kraus Annulation
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0609_ga_10-1055_a-1334-6982.gif

paper

Sole, Roberto; Agostinis, Lodovico; Conca, Silvia; Gatto, Vanessa; Bardella, Noemi; Morandini, Andrea; Buranello, Chiara; Beghetto, Valentina: Synthesis of Amidation Agents and Their Reactivity in Condensation Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0576_ga_10-1055_a-1334-6916.gif

Publication Date: 08 December 2020

Publication Date: 07 December 2020

paper

Talavera-Alemán, Armando; Marrot, Jérome; Dagousset, Guillaume; Thomassigny, Christine: Synthesis of Nitrogen- and Oxygen-Containing Heterocycles by Prins Cyclization in Continuous Flow
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0476_ga_10-1055_s-0040-1705988.gif

Publication Date: 03 December 2020

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 02 December 2020

Publication Date: 30 November 2020

Publication Date: 26 November 2020

paper

Siera, Hannah; Semleit, Nina; Kreuzahler, Mathis; Wölper, Christoph; Haberhauer, Gebhard: Gold Catalysis of Non-Conjugated Haloacetylenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0402_ga_10-1055_s-0040-1706606.gif

Publication Date: 23 November 2020

Publication Date: 19 November 2020

Publication Date: 17 November 2020

Publication Date: 12 November 2020

paper

Jeminejs, Andris; Goliškina, Svetlana M.; Novosjolova, Irina; Stepanovs, Dmitrijs; Bizdēna, Ērika; Turks, Māris: Application of Azide-Tetrazole Tautomerism and Arylsulfanyl Group Dance in the Synthesis of Thiosubstituted Tetrazoloquinazolines
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0383_ga_10-1055_s-0040-1706568.gif

Publication Date: 11 November 2020

Publication Date: 10 November 2020

Publication Date: 05 November 2020

Publication Date: 04 November 2020

paper

Collin, Diego E.; Jackman, Edward H.; Jouandon, Nicolas; Sun, Wei; Light, Mark E.; Harrowven, David C.; Linclau, Bruno: Decagram Synthesis of Dimethyl 1,4-Cubanedicarboxylate Using Continuous-Flow Photochemistry
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0462_ga_10-1055_s-0040-1705964.jpg

Publication Date: 02 November 2020

Publication Date: 29 October 2020

paper

Ivanov, Konstantin L.; Melnikov, Mikhail Ya.; Budynina, Ekaterina M.: Reductive Knoevenagel Condensation with the Zn–AcOH System
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0283_ga_10-1055_s-0040-1705940.gif

Publication Date: 28 October 2020

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 26 October 2020

paper

Bouarfa, Salima; Bentabed-Ababsa, Ghenia; Erb, William; Picot, Laurent; Thiéry, Valérie; Roisnel, Thierry; Dorcet, Vincent; Mongin, Florence: Iodothiophenes and Related Compounds as Coupling Partners in Copper-Mediated N-Arylation of Anilines
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0426_ga_10-1055_s-0040-1706542.gif

Publication Date: 22 October 2020

paper

dos Santos, Beatriz F.; da Silva, Beatriz A. L.; de Oliveira, Aline R.; Sarragiotto, Maria H.; Rinaldi, Andrelson W.; Domingues, Nelson Luís C.: Palladium Nanoparticles Anchored on Magnesium Organosilicate: An Effective and Selective Catalyst for the Heck Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0350_ga_10-1055_s-0040-1705938.gif

Publication Date: 19 October 2020

Publication Date: 15 October 2020

paper