DOI: 10.1055/s-00000084

Synthesis

eFirst

Publication Date: 28 October 2020

short review

Clapham, Margaret L.; Murphy, Emma C.; Douglas, Christopher J.: Synthesis and Crystal Engineering of Rubrene and Its Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0414_ga_10-1055_s-0040-1707316.jpg

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 27 October 2020

paper

Langhals, Heinz; Reichherzer, Susanne; Mayer, Peter; Polborn, Kurt: A Three-Step Synthesis of 1,7-Diazaperylene and Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0294_ga_10-1055_s-0040-1707293.jpg

short review

Gonay, Marie; Batisse, Chloé; Paquin, Jean-François: Recent Advances in the Synthesis of Acyl Fluorides
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0474_ga_10-1055_s-0040-1705951.gif

Publication Date: 26 October 2020

paper

Bouarfa, Salima; Bentabed-Ababsa, Ghenia; Erb, William; Picot, Laurent; Thiéry, Valérie; Roisnel, Thierry; Dorcet, Vincent; Mongin, Florence: Iodothiophenes and Related Compounds as Coupling Partners in Copper-Mediated N-Arylation of Anilines
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0426_ga_10-1055_s-0040-1706542.gif

special topic > Functional Organic Molecules

Mei, Peifeng; Kurosaki, Ryo; Matsumoto, Akinobu; Yamada, Hiroko; Aratani, Naoki: One-Pot Synthesis of a Cyclic Pyrene Octamer from Two Bifunctionalized Pyrene Monomers
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0439_ga_10-1055_s-0040-1705950.gif

Publication Date: 22 October 2020

paper

dos Santos, Beatriz F.; da Silva, Beatriz A. L.; de Oliveira, Aline R.; Sarragiotto, Maria H.; Rinaldi, Andrelson W.; Domingues, Nelson Luís C.: Palladium Nanoparticles Anchored on Magnesium Organosilicate: An Effective and Selective Catalyst for the Heck Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0350_ga_10-1055_s-0040-1705938.gif

Publication Date: 20 October 2020

review

Ponra, Sudipta; Boudet, Bernard; Phansavath, Phannarath; Ratovelomanana-Vidal, Virginie: Recent Developments in Transition-Metal-Catalyzed Asymmetric Hydrogenation of Enamides
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0371_ga_10-1055_s-0040-1705939.gif

Publication Date: 19 October 2020

short review

Saway, Jason; Salem, Zena M.; Badillo, Joseph J.: Recent Advances in Photoacid Catalysis for Organic Synthesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0412_ga_10-1055_s-0040-1705952.gif

Publication Date: 15 October 2020

paper

paper

Liu, Shuangrong; Wu, You; Ying, Zhimin; Luo, Feng; Chen, En; Chen, Wenteng; Yu, Yongping: Facile and Mild Access to Fluorescent Ladder-Type Indolo[3,2-a]carbazoles via Cascade Annulation
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0407_ga_10-1055_s-0040-1706473.gif

Publication Date: 14 October 2020

Publication Date: 13 October 2020

special topic > Recent Advances in Metal-Catalyzed Ring Construction

Publication Date: 12 October 2020

paper

Xiao, Jun-An; Cheng, Xiu-Liang; Meng, Ru-Fang; Qin, Xiao-Shi; Peng, Hai; Ren, Ji-Wei; Xie, Zhen-Zhen; Cui, Jian-Guo; Huang, Yan-Min: Straightforward Synthesis of 3-Selenocyanato-Substituted Chromones through Electrophilic Selenocyanation of Enaminones under Grinding Conditions
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0418_ga_10-1055_s-0040-1707315.gif

short review

Macchia, Antonio; Eitzinger, Andreas; Brière, Jean-François; Waser, Mario; Massa, Antonio: Asymmetric Synthesis of Isoxazol-5-ones and Isoxazolidin-5-ones
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0390_ga_10-1055_s-0040-1706483.gif

Publication Date: 08 October 2020

Publication Date: 07 October 2020

paper

Le Guen, Clothilde; Mazzah, Ahmed; Penhoat, Maël; Melnyk, Patricia; Rolando, Christian; Chausset-Boissarie, Laëtitia: Direct and Regioselective C(sp3)–H Bond Fluorination of 2-Alkylazaarenes with Selectfluor
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0377_ga_10-1055_s-0040-1706482.gif

Publication Date: 06 October 2020

paper

review

Molina Betancourt, Ricardo; Echeverria, Pierre-Georges; Ayad, Tahar; Phansavath, Phannarath; Ratovelomanana-Vidal, Virginie: Recent Progress and Applications of Transition-Metal-Catalyzed Asymmetric Hydrogenation and Transfer Hydrogenation of Ketones and Imines through Dynamic Kinetic Resolution
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0335_ga_10-1055_s-0040-1705918.gif

Publication Date: 05 October 2020

feature

Banert, Klaus; Heck, Manuel; Ihle, Andreas; Michael, Erik; Weber, Richard: Record-Breaking Steric Crowding in Trialkylamines Prepared by Oxidative Ring Opening
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0361_ga_10-1055_s-0040-1707294.jpg

paper

Tomilin, Denis N.; Sobenina, Lyubov N.; Ushakov, Igor A.; Trofimov, Boris A.: Highly Functionalized Pyrrolylpyridines from 2-(Acylethynyl)-pyrroles
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0302_ga_10-1055_s-0040-1706474.gif

review

Dimitrov, Ivaylo V.; Suonio, Elina E. K.: Syntheses of Analogues of Propofol: A Review
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0288_ga_10-1055_s-0040-1707287.gif

special topic > Functional Organic Molecules

special topic > Functional Organic Molecules > Functional Organic Molecules

Yan, Feng-Zhi; Shao, Yuan-Guang; Zhang, Zibin; Shen, Yan-Feng; Huang, Xue-Chun; Zhang, Pei-Ling; Li, Shijun: Synthesis of Catenanes from a BMP32C10-Based Cryptand Tuned by the Linkage Length of Paraquat Salts
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0428_ga_10-1055_s-0040-1707290.gif

Publication Date: 01 October 2020

Publication Date: 30 September 2020

short review

Chen, Tieqiao; Tan, Qihang; Liu, Xue; Liu, Long; Huang, Tianzeng; Han, Li-Biao: Phosphorylation of Carboxylic Acids and Their Derivatives with P(O)–H Compounds Forming P(O)–C Bonds
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0379_ga_10-1055_s-0040-1707286.gif

Publication Date: 29 September 2020

paper

Strelnikova, Julia O.; Rostovskii, Nikolai V.; Khoroshilova, Olesya V.; Khlebnikov, Alexander F.; Novikov, Mikhail S.: An Efficient Synthesis of Functionalized 2H-1,3,5-Oxadiazines via Metal-Carbenoid-Induced 1,2,4-Oxadiazole Ring Cleavage
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0194_ga_10-1055_s-0040-1707278.gif

Publication Date: 24 September 2020

paper

Liu, Teng; He, Chixian; Wang, Fan; Shen, Xiang; Li, Yongqin; Lang, Man; Li, Guijun; Huang, Chao; Cheng, Feixiang: Organocatalyzed [2+2] Cycloaddition Reactions between Quinone Imine Ketals and Allenoates
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0406_ga_10-1055_s-0040-1707292.gif

Publication Date: 23 September 2020

Publication Date: 22 September 2020

paper

paper

Inatomi, Saki; Takayanagi, Yuta; Watanabe, Kento; Toita, Akinori; Yamakoshi, Hiroyuki; Nakamura, Seiichi: Stereoselective 1,4-Addition of Primary Alcohols to γ-Alkoxy-α,β-unsaturated Esters
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0364_ga_10-1055_s-0040-1707274.gif

short review

Publication Date: 21 September 2020

Publication Date: 15 September 2020

short review

Carreras, Virginie; Tanbouza, Nour; Ollevier, Thierry: The Power of Iron Catalysis in Diazo Chemistry
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0353_ga_10-1055_s-0040-1707272.jpg

Publication Date: 11 September 2020

Publication Date: 08 September 2020

psp

Bhilare, Shatrughn; Kori, Santosh; Shet, Harshita; Balaram, Gundapally; Mahendar, Koosam; Sanghvi, Yogesh S.; Kapdi, Anant R.: Scale-Up of a Heck Alkenylation Reaction: Application to the Synthesis of an Amino-Modifier Nucleoside ‘Ruth Linker’
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0312_ga_10-1055_s-0040-1707260.gif

Publication Date: 02 September 2020

paper

Dibdalli, Yuvaraja; Faúndez, Rodrigo; Preite, Marcelo; Molins, Elies; Chávez, Ivonne; Amshumali, Mungalimane K.; Morales-Verdejo, Cesar; Manriquez, Juan M.: An Improved Synthesis of 3,6-Dihydro-as-indacene
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0320_ga_10-1055_s-0040-1707372.gif

Publication Date: 01 September 2020

paper

Rozhkova, Yuliya S.; Storozheva, Tatyana S.; Plekhanova, Irina V.; Gorbunov, Alexey A.; Smolyak, Andrej A.; Shklyaev, Yurii V.: Synthesis of Aminoalkyl-Functionalized 4-Arylquinolines from 2-(3,4-Dihydroisoquinolin-1-yl)anilines via the Friedländer Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0376_ga_10-1055_s-0040-1706424.gif

short review

Yu, Jie; Singh, Anoop S.; Yan, Guobing; Yu, Jian; Tiwari, Vinod K.: Recent Developments on Denitrogenative Functionalization of Benzotriazoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0342_ga_10-1055_s-0040-1707253.gif

Publication Date: 27 August 2020

paper

Zong, Zhijian; Wu, Ke; Jin, Liqun; Sun, Nan; Hu, Baoxiang; Shen, Zhenlu; Hu, Xinquan: Large-Scale Synthesis of 2-Chlorotetrahydroquinoline and 2-Chlorotetrahydroquinolin-8-one
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0316_ga_10-1055_s-0040-1707236.gif

Publication Date: 25 August 2020

short review

Filippov, Ilya P.; Titov, Gleb D.; Rostovskii, Nikolai V.: Recent Advances in Denitrogenative Reactions of Pyridotriazoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0305_ga_10-1055_s-0040-1707254.gif

short review

Muñoz-Molina, José María; Belderrain, Tomás R.; Pérez, Pedro J.: Recent Advances in Copper-Catalyzed Radical C–H Bond Activation Using N–F Reagents
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0317_ga_10-1055_s-0040-1707234.gif

Publication Date: 24 August 2020

Publication Date: 20 August 2020

paper

Casadia, Izamara; Daher, Thalita O.; Moura, Sidnei; Back, Davi F.; Faoro, Eliandro; Schwalm, Cristiane S.; Casagrande, Gleison A.; Paveglio, Guilherme C.; Pizzuti, Lucas: A Domino Reaction for the Synthesis of Novel 1,3-Dihydrofuro[3,4-c]pyridines from Pyridoxal and Ketones
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0354_ga_10-1055_s-0040-1706422.gif

Publication Date: 19 August 2020

short review

Khandelwal, Manisha; Ray, Sumit Kumar; Khangarot, Rama Kanwar: Syntheses and Applications of Singh’s Catalyst
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0263_ga_10-1055_s-0040-1707235.jpg

Publication Date: 18 August 2020

Publication Date: 17 August 2020

paper

Lan, Jin-Ping; Lu, Yi-Nan; Chen, Ke-Wei; Jiang, Fei; Gao, Feng; Zhang, Yu-Chen; Shi, Feng: Catalytic Asymmetric Substitution Reaction of 3-Substituted 2-Indolylmethanols with 2-Naphthols
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0318_ga_10-1055_s-0040-1707237.gif

paper

Tarui, Atsushi; Ueo, Masakazu; Morikawa, Marino; Tsuta, Masahiko; Iwasaki, Sumika; Morishita, Noriko; Karuo, Yukiko; Sato, Kazuyuki; Kawai, Kentaro; Omote, Masaaki: One-Pot Ring-Opening Peptide Synthesis Using α,α-Difluoro-β-Lactams
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0329_ga_10-1055_s-0040-1707238.gif

Publication Date: 12 August 2020

Publication Date: 11 August 2020

short review

Pang, Xiaobo; Peng, Xuejing; Shu, Xing-Zhong: Reductive Cross-Coupling of Vinyl Electrophiles
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0276_ga_10-1055_s-0040-1707342.jpg

Publication Date: 06 August 2020

paper

Fedotov, Victor V.; Ulomsky, Evgeny N.; Savateev, Konstantin V.; Mukhin, Evgeny M.; Gazizov, Denis A.; Gorbunov, Evgeny B.; Rusinov, Vladimir L.: A PASE Approach to the Synthesis of Benzimidazopurines as Polycondensed Purine Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0333_ga_10-1055_s-0040-1707228.gif

Publication Date: 05 August 2020

short review

Publication Date: 04 August 2020

paper

Zhang, Xiang-Zhi; Qiu, Zong-Wang; Wen, Gui-Hua; Ma, Ai-Jun; Bao, Peng-Jin; Du, Ji-Yuan; Xu, Xue-Tao; Feng, Na; Li, Bao Qiong: Synthesis of Pyrrolo[1,2-a]indoles via (3+2)-Annulations of (Aza)-para-Quinone Methides with Indoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0369_ga_10-1055_s-0040-1707348.gif

Publication Date: 03 August 2020

review

Markovič, Martin; Lopatka, Pavol; Gracza, Tibor; Koóš, Peter: Recent Applications of Continuous Flow in Homogeneous Palladium Catalysis
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0277_ga_10-1055_s-0040-1707212.gif

Publication Date: 27 July 2020

paper

Osyanin, Vitaly A.; Osipov, Dmitry V.; Melnikova, Irina V.; Korzhenko, Kirill S.; Semenova, Irina A.; Klimochkin, Yuri N.: Catalyst-Free Synthesis of Chromane-Type N,O-Acetals via Intramolecular Addition of Phenols to Enamines
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0037_ga_10-1055_s-0040-1707209.gif

Publication Date: 22 July 2020

Publication Date: 21 July 2020

Publication Date: 20 July 2020

special topic

Publication Date: 13 July 2020

Publication Date: 16 June 2020

Publication Date: 08 June 2020

special topic

Wei, Bin; Li, Ke-Wei; Wu, Yan-Chen; Tong, Shi-Qi; Song, Ren-Jie: Radical Strategy for the Transition-Metal-Catalyzed Synthesis of γ-Lactones: A Review
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0226_ga_10-1055_s-0040-1707835.jpg

Publication Date: 03 March 2020