DOI: 10.1055/s-00000084

Synthesis

eFirst

Publication Date: 15 April 2021

Publication Date: 14 April 2021

Publication Date: 13 April 2021

paper

Obydennov, Dmitrii L.; Steben’kov, Vyacheslav D.; Obydennov, Konstantin L.; Usachev, Sergey A.; Moshkin, Vladimir S.; Sosnovskikh, Vyacheslav Y.: Reactions of 4-Pyrones with Azomethine Ylides as a Chemo­selective Method for the Construction of Multisubstituted Pyrano[2,3-c]pyrrolidines
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0065_ga_10-1055_s-0040-1706032.gif

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 12 April 2021

paper

special topic > Cycloadditions – Established and Novel Trends – in Celebration of the 70th Anniversary of the Nobel Prize Awarded to Otto Diels and Kurt Alder

Publication Date: 09 April 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 08 April 2021

paper

Gritzenco, Fabiane; Kazmierczak, Jean C.; Anjos, Thiago; Sperança, Adriane; Peixoto, Maura L. B.; Godoi, Marcelo; Ledebuhr, Kauane N. B.; Brüning, César Augusto; Zamin, Lauren L.; Godoi, Benhur: Base-Free Synthesis and Synthetic Applications of Novel 3-(Organochalcogenyl)prop-2-yn-1-yl Esters: Promising Anticancer Agents
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0111_ga_10-1055_a-1477-6470.gif

paper

Zhao, Fenghai; Singh, Thishana; Xiao, Yumei; Su, Wangcang; Yang, Dongyan; Jia, Changqing; Li, Jia-Qi; Qin, Zhaohai: Divergent Synthesis of Substituted Amino-1,2,4-triazole Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0077_ga_10-1055_a-1477-4630.gif

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 01 April 2021

paper

Shaw, Jessica L.; Austermuehle, Brad J.; Witte, Jordan M.; Dorsey, Timothy R.; Delach, Christina; Hamaker, Christopher G.; Hitchcock, Shawn R.: N-p-Toluenesulfinylimidazole: A New in situ Reagent for the Mild and Efficient Synthesis of p-Toluenesulfinate Alkyl Esters and Aryl Esters
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0119_ga_10-1055_a-1472-7578.gif

short review

short review

Publication Date: 31 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 30 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 29 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 26 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Ishida, Tamao; Zhang, Zhenzhong; Murayama, Haruno; Yamamoto, Eiji; Tokunaga, Makoto: C–H Bond Functionalization Using Pd- and Au-Supported Catalysts with Mechanistic Insights of the Active Species
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0140_ga_10-1055_a-1468-1455.jpg

Publication Date: 25 March 2021

short review

Zhang, Sheng; Findlater, Michael: Cobalt-Catalyzed Isomerization of Alkenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0052_ga_10-1055_a-1464-2524.gif

special topic > Bond Activation – in Honor of Prof. Shinji Murai

special topic > Bond Activation – in Honor of Prof. Shinji Murai

special topic > Special Issue dedicated to Prof. Sarah Reisman, recipient of the 2019 Dr. Margaret Faul Women in Chemistry Award

Wienhold, Sebastian; Fritz, Lukas; Judt, Tatjana; Hackl, Sabrina; Neubauer, Thomas; Sauerer, Bastian; Bach, Thorsten: Studies towards the Synthesis of (–)-Pulvomycin: Construction of the C12–C40 Segment by a Stereoselective Aldol Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0156_ga_10-1055_a-1464-2576.gif

Publication Date: 24 March 2021

short review

Publication Date: 22 March 2021

paper

Al-Zoubi, Raed M.; Altamimi, Reem M.; Al-Jammal, Walid K.; Shawakfeh, Khaled Q.; Al-Zoubi, Mazhar S.; Ferguson, Michael J.; Zarour, Ahmad; Yassin, Aksam; Al-Ansari, Abdulla: CuI-Catalyzed Ullmann-Type Coupling of Phenols and Thiophenols with 5-Substituted 1,2,3-Triiodobenzenes: Facile Synthesis of Mammary Carcinoma Inhibitor BTO-956 in One Step
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0021_ga_10-1055_a-1458-2980.gif

short review

Rehpenn, Andreas; Walter, Alexandra; Storch, Golo: Molecular Editing of Flavins for Catalysis
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0064_ga_10-1055_a-1458-2419.gif

Publication Date: 16 March 2021

paper

Zhou, Xin; Long, Qing; Li, Dongwei; Gao, Jingru; Sun, Qikai; Sun, Shaozi; Su, Yong; Wang, Peng; Peng, Wenjie; Li, Ming: Convergent Synthesis of Branched β-Glucan Tridecasaccharides Ready for Conjugation
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0073_ga_10-1055_a-1440-9386.gif

Publication Date: 15 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Akahori, Shuhei; Fujihara, Tetsuaki; Tsuji, Yasushi; Shinokubo, Hiroshi; Miyake, Yoshihiro: Synthesis of Tetrasilatetrathia[8]circulenes through C–I and C–H Silylation
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0107_ga_10-1055_a-1437-9917.gif

Publication Date: 12 March 2021

paper

Teramoto, Masahiro; Imoto, Mitsutaka; Takeda, Motonori; Mizuno, Takumi; Nomoto, Akihiro; Ogawa, Akiya: Sulfur-Promoted Redox Cyclization of 2,2′-Dinitrodiphenyl Disulfides and Benzylamines
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0078_ga_10-1055_a-1430-5100.gif

Publication Date: 11 March 2021

feature

short review

short review

Zhang, Qiaoling; Xi, Jufang; Ze, He; Qingle, Zeng: Syntheses and Transformations of Sulfinamides
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0023_ga_10-1055_a-1426-4744.gif

Publication Date: 10 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 08 March 2021

paper

Ulyankin, Evgeny B.; Kostyuchenko, Anastasia S.; Chernenko, Sergey A.; Bystrushkin, Mikhail O.; Samsonenko, Anna L.; Shatsauskas, Anton L.; Fisyuk, Alexander S.: A Simple and Efficient Synthesis of Fused Benzo[b]thiophene Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0038_ga_10-1055_a-1416-4924.gif

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 04 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Tang, Zhi; Tong, Zhou; Qiu, Renhua; Yin, Shuang-Feng; Kambe, Nobuaki: Recent Advances on Benzofuranones: Synthesis and Transformation via C–H Functionalization
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0039_ga_10-1055_a-1405-5761.gif

Publication Date: 03 March 2021

Publication Date: 02 March 2021

special topic > Special Issue dedicated to Prof. Sarah Reisman, recipient of the 2019 Dr. Margaret Faul Women in Chemistry Award

Ryan, Jonathon S.; Schindler, Corinna S.: Total Synthesis of Mycocyclosin and the Herqulines
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0034_ga_10-1055_a-1403-4312.gif

Publication Date: 26 February 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 24 February 2021

Publication Date: 23 February 2021

special topic > Special Issue dedicated to Prof. Sarah Reisman, recipient of the 2019 Dr. Margaret Faul Women in Chemistry Award

Lam, Heather; Abel-Snape, Xavier; Köllen, Martin F.; Lautens, Mark: Recent Advances in Transition-Metal-Free (4+3)-Annulations
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0520_ga_10-1055_s-0040-1706023.gif

Publication Date: 22 February 2021

paper

Gagnot, Glwadys; Legrand, Pierre; Tadros, Amira; Ezzahra Hibti, Fatima; Quatela, Alessia; Janin, Yves L.: On Pyridopyrazinol Chemistry: Synthesis of Chemiluminescent Substances
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0028_ga_10-1055_a-1396-8607.gif

paper

Schädel, Nicole; Icik, Esra; Martini, Maike; Altevogt, Luca; Ramming, Isabell; Greulich, Andreas; Baro, Angelika; Bilitewski, Ursula; Laschat, Sabine: Synthesis of Imidazole and Histidine-Derived Cross-Linkers as Analogues of GOLD and Desmosine
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0588_ga_10-1055_s-0040-1706144.gif

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Watanabe, Hikaru; Nakajima, Kazuki; Ekuni, Kento; Edagawa, Ryota; Akagi, Yuta; Okuda, Yasuhiro; Wakamatsu, Kan; Orita, Akihiro: Custom-Made Pyrene Photocatalyst-Promoted Desulfonylation of Arylethenyl Sulfones Using Green-Light-Emitting Diodes
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0005_ga_10-1055_s-0040-1706025.gif

Publication Date: 18 February 2021

feature

Shaaban, Saad; Li, Houhua; Merten, Christian; Antonchick, Andrey P.; Waldmann, Herbert: Rhodium(III)-Catalyzed Enantioselective Benzamidation of Cyclopropenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0629_ga_10-1055_s-0040-1706026.gif

short review

Pedrood, Keyvan; Montazer, Mohammad Nazari; Larijani, Bagher; Mahdavi, Mohammad: Recent Advances in the Synthesis of Heterocycles by the Aza-Wittig Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0643_ga_10-1055_a-1394-7511.gif

Publication Date: 15 February 2021

Publication Date: 11 February 2021

short review

Livingstone, Keith; Little, Gemma; Jamieson, Craig: Recent Advances in the Generation of Nitrilium Betaine 1,3-Dipoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0658_ga_10-1055_a-1389-1281.gif

Publication Date: 10 February 2021

Publication Date: 09 February 2021

paper

Schefzig, Luise; Kurzawa, Timon; Rancan, Giaime; Linder, Igor; Leisering, Stefan; Bera, Mrinal K.; Gart, Max; Zimmer, Reinhold; Reissig, Hans-Ulrich: Access to Highly Substituted Pyrimidine N-Oxides and 4-Acetoxymethyl-Substituted Pyrimidines via the LANCA Three-Component Reaction–Cyclocondensation Sequence
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0636_ga_10-1055_s-0040-1706020.gif

Publication Date: 08 February 2021

short review

Inoa, Joan; Dominici, Grecia; Eldabagh, Reem; Foley, Jonathan J.; Xing, Yalan: Synthetic Applications and Computational Perspectives on Eosin Y Induced Direct HAT Process
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0616_ga_10-1055_a-1385-9398.jpg

Publication Date: 05 February 2021

Publication Date: 01 February 2021

paper

Kuwabara, Motoi; Matsuo, Ami; Kamo, Shogo; Matsuzawa, Akinobu; Sugita, Kazuyuki: Stereoselective Convergent Synthesis of Carbon Skeleton of Cotylenin A Aglycone
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0631_ga_10-1055_s-0040-1706684.gif

Publication Date: 27 January 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 26 January 2021

Publication Date: 25 January 2021

Publication Date: 22 January 2021

Publication Date: 21 January 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 20 January 2021

Publication Date: 19 January 2021

paper

Chen, Jyun-Siao; Ke, Yi-Fan; Lin, Heng-Yan; Lin, Wesley; Yen, Wei-Chung; Wu, Hsin-Ru; Luo, Shun-Yuan: Development of a Novel Method for Trimethylsilylation of Saccharides­
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0542_ga_10-1055_s-0040-1705990.gif

Publication Date: 18 January 2021

errata

Srinivasulu, Vunnam; Al-Marzooq, Farah; Hamad, Mohamad; Khanfar, Monther A.; Ramanathan, Mani; Soares, Nelson C.; Al-Tel, Taleb H.: Sequencing Groebke–Blackburn–Bienaymé and Aza-Michael Addition Reactions: A Modular Strategy for Accessing a Diverse Collection of Constrained Benzoxazepine and Imidazopyrazine Systems

paper

Mityuk, Andrey P.; Hrebonkin, Andrii; Lebed, Pavlo S.; Grabchuk, Galyna P.; Volochnyuk, Dmitriy M.; Ryabukhin, Sergey V.: Efficient Route for the Synthesis of Diverse Heteroannelated 5-Cyanopyridines
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0627_ga_10-1055_a-1360-9852.gif

paper

Wang, Siqi; Filatov, Alexander S.; Lozovskiy, Stanislav V.; Shmakov, Stanislav V.; Khoroshilova, Olesya V.; Larina, Anna G.; Selivanov, Stanislav I.; Boitsov, Vitali M.; Stepakov, Alexander V.: Construction of Spiro[3-azabicyclo[3.1.0]hexanes] via 1,3-Dipolar Cycloaddition of 1,2-Diphenylcyclopropenes to Ninhydrin-Derived Azomethine Ylides
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0574_ga_10-1055_a-1360-9716.gif

short review

Publication Date: 15 January 2021

Publication Date: 14 January 2021

errata

Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)

review

Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0484_ga_10-1055_s-0040-1705983.gif

Publication Date: 13 January 2021

Publication Date: 11 January 2021

paper

Lisovenko, Natalya Yu.; Nasibullina, Ekaterina R.; Kharitonova, Svetlana S.; Myshkina, Olga A.: Simple Synthesis of Substituted 3-Hydroxyfuran-2(5H)-ones
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0541_ga_10-1055_s-0040-1705998.gif

paper

Yassine, Hasna; Bouali, Jamila; Oumessaoud, Asmaa; Ourhzif, El Mahdi; Hamri, Salha; Hafid, Abderrafia; Khouili, Mostafa; Pujol, Maria Dolors: Synthesis of New Dialkyl 2,2′-[Carbonylbis(azanediyl)]dibenzoates via Curtius Rearrangement
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0458_ga_10-1055_s-0040-1706643.gif

Publication Date: 08 January 2021

paper

Kotha, Sambasivarao; Pulletikurti, Sunil; Fatma, Ambareen; Dhangar, Gopal; Naidu, Gonna Somu: Synthesis of Polycycles and Oxacycles via Tandem Metathesis of endo-Norbornene Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0532_ga_10-1055_a-1348-4242.gif

Publication Date: 07 January 2021

Publication Date: 21 December 2020

Publication Date: 15 December 2020

special topic > Bond Activation – in Honor of Prof. Shinji Murai

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 07 December 2020

paper

Hsu, Ming-Hua; Kapoor, Mohit; Pradhan, Tapan Kumar; Tse, Man-Him; Chen, Hsin-Ya; Yan, Man-Jun; Cheng, Yu-Tsen; Lin, Yu-Cheng; Hsieh, Cheng-Ying; Liu, Ker-Yin; Han, Chien-Chung: Mild and Efficient Copper-Catalyzed Synthesis of Trisubstituted Pyrroles
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0501_ga_10-1055_a-1331-7346.gif

Publication Date: 03 December 2020

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Publication Date: 28 October 2020

special topic > Bond Activation – in Honor of Prof. Shinji Murai