Synthesis

Publication Date: 15 April 2021

feature

Wata, Chisato; Hashimoto, Takuya: Organoiodine-Catalyzed Enantioselective Intramolecular Oxy­aminations of Alkenes with N-(Fluorosulfonyl)carbamate

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paper

Donges, Jonas; Hofmann, Sandra; Walter, Johannes C.; Reichertz, Julia; Brüggemann, Moritz; Frank, Andrea; Nubbemeyer, Udo: Synthesis of Optically Active N-(4-Hydroxynon-2-enyl)pyrrolidines: Key Building Blocks in the Total Synthesis of Streptomyces coelicolor Butanolide 5 (SCB-5) and Virginiae Butanolide A (VB-A)

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paper

Xu, Zhimin; Zheng, Yue; Tian, Lifang; Wang, Yahui: Synthesis of Bempedoic Acid through Electrochemical Decarboxylation of Dialkylated Malonic Acid

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Supporting Information

Publication Date: 14 April 2021

errata

Demidov, Maxim R.; Osyanin, Vitaly A.; Osipov, Dmitry V.; Klimochkin, Yuri N.: Oxidative Dimerization of 1Н-Benzo[f]chromenes: Synthesis of Benzannulated Analogues of Spirobiflavonoids Welwitschins E and F

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paper

Kumari, Arram Haritha; Kumar, Jangam Jagadesh; Krishna, Gamidi Rama; Reddy, Raju Jannapu: Nickel-Catalyzed Difunctionalization of Alkynyl Bromides with Thiosulfonates and N-Arylthio Succinimides: A Convenient Synthesis of 1,2-Thiosulfonylethenes and 1,1-Dithioethenes

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Publication Date: 13 April 2021

paper

Li, Hengyuan; Zhu, Chuanle: Dual Roles of TBHP-Enabled Regioselective Hydroetherification of (Trifluoromethyl)alkenes with Boronic Acids: Access to α-Trifluoromethyl β-Aryloxy Tertiary Alcohols

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paper

Obydennov, Dmitrii L.; Steben’kov, Vyacheslav D.; Obydennov, Konstantin L.; Usachev, Sergey A.; Moshkin, Vladimir S.; Sosnovskikh, Vyacheslav Y.: Reactions of 4-Pyrones with Azomethine Ylides as a Chemo­selective Method for the Construction of Multisubstituted Pyrano[2,3-c]pyrrolidines

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Vijaykumar, Muniyappa; Punji, Benudhar: Advances in Transition-Metal-Catalyzed C–H Bond Oxygenation of Amides

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Publication Date: 12 April 2021

paper

Wiredu, Bernard; Thapa, Mahendra; Hua, Sheen Y.; Desper, John; Hua, Duy H.: Synthesis of 2,24-Diene-12,13,15,16,34,35,37,38-octaphenyl[4.4]triphenylparacyclophane

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special topic > Cycloadditions – Established and Novel Trends – in Celebration of the 70th Anniversary of the Nobel Prize Awarded to Otto Diels and Kurt Alder

He, Jian; Liu, Qiang: Highly Efficient Visible-Light-Driven [2+2] Cycloaddition of Maleimides to Alkenes and Alkynes for the Synthesis of 3-Aza­bicyclo[3.2.0]heptane-Fused Scaffolds

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Publication Date: 09 April 2021

paper

Zhang, Yang; Liu, Yi; Du, Yuguo: First Total Synthesis of 27-Deoxylyngbyabellin A

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Supporting Information Primary Data

psp

Erb, William; Wen, Min; Roisnel, Thierry; Mongin, Florence: Synthesis of Ferrocenesulfonyl Chloride: Key Intermediate toward Ferrocenesulfonamides

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Supporting Information CIF File

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Maeda, Kyogo; Motokura, Ken: Recent Advances in Heterogeneous Ir Complex Catalysts for Aromatic C–H Borylation

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Publication Date: 08 April 2021

paper

Gritzenco, Fabiane; Kazmierczak, Jean C.; Anjos, Thiago; Sperança, Adriane; Peixoto, Maura L. B.; Godoi, Marcelo; Ledebuhr, Kauane N. B.; Brüning, César Augusto; Zamin, Lauren L.; Godoi, Benhur: Base-Free Synthesis and Synthetic Applications of Novel 3-(Organochalcogenyl)prop-2-yn-1-yl Esters: Promising Anticancer Agents

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paper

Lu, Xiuqiang; Chen, Guofen; Li, Fei: Synthesis of Diporphyrins by Oxidative Coupling with Pd(TFA)₂-Cu(OTf)₂ under Ball-Milling Conditions

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paper

Shelar, Santosh V.; Argade, Narshinha P.: Wittig Reactions of Maleimide-Derived Stabilized Ylides with Alkyl Pyruvates: Concise Approach to Methyl Ester of (±)-Chaetogline A

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paper

Zhao, Fenghai; Singh, Thishana; Xiao, Yumei; Su, Wangcang; Yang, Dongyan; Jia, Changqing; Li, Jia-Qi; Qin, Zhaohai: Divergent Synthesis of Substituted Amino-1,2,4-triazole Derivatives

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Yabe, Ryota; Ebe, Yusuke; Nishimura, Takahiro: Iridium-Catalyzed Direct C–H Allylation of Ketimines

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Publication Date: 01 April 2021

paper

Shaw, Jessica L.; Austermuehle, Brad J.; Witte, Jordan M.; Dorsey, Timothy R.; Delach, Christina; Hamaker, Christopher G.; Hitchcock, Shawn R.: N-p-Toluenesulfinylimidazole: A New in situ Reagent for the Mild and Efficient Synthesis of p-Toluenesulfinate Alkyl Esters and Aryl Esters

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short review

Majdecki, Maciej; Niedbała, Patryk; Tyszka-Gumkowska, Agata; Jurczak, Janusz: Assisted by Hydrogen-Bond Donors: Cinchona Quaternary Salts as Privileged Chiral Catalysts for Phase-Transfer Reactions

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short review

Youssef-Saliba, Sparta; Vallée, Yannick: Sulfur Amino Acids: From Prebiotic Chemistry to Biology and Vice Versa

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Publication Date: 31 March 2021

paper

Seki, Masahiko; Takahashi, Yusuke: Convergent Synthesis of Angiotensin II Receptor Blockers through C–H Arylation of 1-Benzyl-5-phenyl-1H-tetrazole with Functionalized Aryl Bromides

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Dalal, Arup; Babu, Srinivasarao Arulananda: Pd(II)-Catalyzed Directing-Group-Aided C–H Arylation and Alkylation of Pyrene Core: Synthesis of C1,C2- and C1,C10-Disubstituted Pyrene Motifs

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Kona, Chandrababu Naidu; Oku, Rikuto; Nishii, Yuji; Miura, Masahiro: Peri-Selective Direct Acylmethylation and Amidation of Naphthalene Derivatives Using Iridium and Rhodium Catalysts

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Publication Date: 30 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Oonishi, Yoshihiro; Sakamoto, Shunki; Agata, Shuya; Sato, Yoshihiro: Rhodium(I)-Catalyzed Enantioselective Cyclization of Enynes through Site-Selective C(sp³)–H Bond Activation Triggered by Formation of Rhodacycle

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Publication Date: 29 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Kiyosu, Yuuki; Tanaka, Shino; Okumura, Sota; Kiyokawa, Kensuke; Minakata, Satoshi: Synthesis of Fused Diaziridine Derivatives from Cyclic Secondary Amines by Utilizing N-Bromosulfonamides as an Aminating Reagent

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Morimoto, Tsumoru; Wang, Chuang; Tanimoto, Hiroki; Artok, Levent; Kakiuchi, Kiyomi: Rhodium(I)-Catalyzed CO-Gas-Free Arylative Dual-Carbonylation of Alkynes with Arylboronic Acids via the Formyl C–H Activation of Formaldehyde

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Publication Date: 26 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Ishida, Tamao; Zhang, Zhenzhong; Murayama, Haruno; Yamamoto, Eiji; Tokunaga, Makoto: C–H Bond Functionalization Using Pd- and Au-Supported Catalysts with Mechanistic Insights of the Active Species

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Publication Date: 25 March 2021

paper

Mitachi, Katsuhiko; Mingle, David; Kurosu, Michio: A Convenient Protecting Group for Uridine Ureido Nitrogen: (4,4′-Bisfluorophenyl)methoxymethyl Group

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short review

Zhang, Sheng; Findlater, Michael: Cobalt-Catalyzed Isomerization of Alkenes

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Pan, Feng-Feng; Guo, Peng; Huang, Xiaochuang; Shu, Xing-Zhong: Synthesis of Dibenzyls by Nickel-Catalyzed Homocoupling of Benzyl Alcohols

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Shimazumi, Ryoma; Morita, Kosuke; Yoshida, Tomoki; Yasui, Kosuke; Tobisu, Mamoru: Late-Stage Derivatization of Buflavine by Nickel-Catalyzed Direct Substitution of a Methoxy Group via C–O Bond Activation

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Supporting Information

special topic > Special Issue dedicated to Prof. Sarah Reisman, recipient of the 2019 Dr. Margaret Faul Women in Chemistry Award

Wienhold, Sebastian; Fritz, Lukas; Judt, Tatjana; Hackl, Sabrina; Neubauer, Thomas; Sauerer, Bastian; Bach, Thorsten: Studies towards the Synthesis of (–)-Pulvomycin: Construction of the C12–C40 Segment by a Stereoselective Aldol Reaction

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Supporting Information Primary Data

Publication Date: 24 March 2021

feature

Jia, Zongbin; Yang, Qi; Luo, Sanzhong: Photoredox-Mediated Asymmetric Cross-Dehydrogenative Coupling of Enones and Tertiary Amines by Chiral Primary Amine Catalysis

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Supporting Information

short review

Jurinic, Carla K.; Belladona, Andrei L.; Schumacher, Ricardo F.; Godoi, Benhur: Diorganyl Dichalcogenides and Copper/Iron Salts: Versatile Cyclization System To Achieve Carbo- and Heterocycles from Alkynes

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short review

Roche, Stéphane P.: In the Pursuit of (Ald)Imine Surrogates for the Direct Asymmetric Synthesis of Non-Proteinogenic α-Amino Acids

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Publication Date: 22 March 2021

paper

Al-Zoubi, Raed M.; Altamimi, Reem M.; Al-Jammal, Walid K.; Shawakfeh, Khaled Q.; Al-Zoubi, Mazhar S.; Ferguson, Michael J.; Zarour, Ahmad; Yassin, Aksam; Al-Ansari, Abdulla: CuI-Catalyzed Ullmann-Type Coupling of Phenols and Thiophenols with 5-Substituted 1,2,3-Triiodobenzenes: Facile Synthesis of Mammary Carcinoma Inhibitor BTO-956 in One Step

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Supporting Information CIF File

review

Mamedov, Vakhid A.; Zhukova, Nataliya A.: Recent Developments Towards Synthesis of (Het)arylbenzimidazoles

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short review

Rehpenn, Andreas; Walter, Alexandra; Storch, Golo: Molecular Editing of Flavins for Catalysis

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Publication Date: 16 March 2021

paper

Zhou, Xin; Long, Qing; Li, Dongwei; Gao, Jingru; Sun, Qikai; Sun, Shaozi; Su, Yong; Wang, Peng; Peng, Wenjie; Li, Ming: Convergent Synthesis of Branched β-Glucan Tridecasaccharides Ready for Conjugation

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Supporting Information

Publication Date: 15 March 2021

review

Bellina, Fabio: Real Metal-Free C–H Arylation of (Hetero)arenes: The Radical Way

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Akahori, Shuhei; Fujihara, Tetsuaki; Tsuji, Yasushi; Shinokubo, Hiroshi; Miyake, Yoshihiro: Synthesis of Tetrasilatetrathia[8]circulenes through C–I and C–H Silylation

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Supporting Information

Publication Date: 12 March 2021

paper

Teramoto, Masahiro; Imoto, Mitsutaka; Takeda, Motonori; Mizuno, Takumi; Nomoto, Akihiro; Ogawa, Akiya: Sulfur-Promoted Redox Cyclization of 2,2′-Dinitrodiphenyl Disulfides and Benzylamines

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Publication Date: 11 March 2021

feature

Lupi, Michela; Menichetti, Stefano; Stagnaro, Paola; Utzeri, Roberto; Viglianisi, Caterina: Thia-Bridged Triarylamine[4]helicene-Functionalized Polynorbor­nenes as Redox-Active pH-Sensitive Polymers

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Supporting Information

short review

Li, Qingjiang; Guo, Zhongwu: Enzymatic Synthesis of Glycosphingolipids: A Review

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short review

Rubtsov, Aleksandr E.; Malkov, Andrei V.: Recent Advances in the Synthesis of 2,2′-Bipyridines and Their Derivatives

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short review

Zhang, Qiaoling; Xi, Jufang; Ze, He; Qingle, Zeng: Syntheses and Transformations of Sulfinamides

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Publication Date: 10 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Kanyiva, Kyalo Stephen; Tang, King Hung Nigel; Wang, Jiarui; Shibata, Takanori: Palladium-Catalyzed sp³ C–H Benzoxylation of Alanine Derivatives Using Aldehydes under Ambient Conditions

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Supporting Information

Publication Date: 08 March 2021

paper

Ulyankin, Evgeny B.; Kostyuchenko, Anastasia S.; Chernenko, Sergey A.; Bystrushkin, Mikhail O.; Samsonenko, Anna L.; Shatsauskas, Anton L.; Fisyuk, Alexander S.: A Simple and Efficient Synthesis of Fused Benzo[b]thiophene Derivatives

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Inai, Yasuhito; Usuki, Yoshinosuke; Satoh, Tetsuya: Synthesis of Benzo-Fused Cyclic Compounds via Rhodium-Catalyzed Decarboxylative Coupling of Aromatic Carboxylic Acids with Alkynes

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Wan, Bin; Zhang, Yanghui: Synthesis of Unsymmetrically Substituted Tetraphenylenes through Palladium-Catalyzed C(sp²)–H Activation

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Publication Date: 04 March 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Tang, Zhi; Tong, Zhou; Qiu, Renhua; Yin, Shuang-Feng; Kambe, Nobuaki: Recent Advances on Benzofuranones: Synthesis and Transformation via C–H Functionalization

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Publication Date: 03 March 2021

paper

Gross, Benjamin M.; Oestreich, Martin: The Trityl Cation Embedded into a [7]Helicene-Like Backbone: Preparation and Application as a Lewis Acid Catalyst

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paper

Junk, Lukas; Papadopoulos, Emanuel; Kazmaier, Uli: Tryptophan N¹-Alkylation: Quick and Simple Access to Diversely Substituted Tryptophans

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Supporting Information

Publication Date: 02 March 2021

special topic > Special Issue dedicated to Prof. Sarah Reisman, recipient of the 2019 Dr. Margaret Faul Women in Chemistry Award

Ryan, Jonathon S.; Schindler, Corinna S.: Total Synthesis of Mycocyclosin and the Herqulines

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Publication Date: 26 February 2021

paper

Bin Shahari, Muhammad Syafiq; Junaid, Ahmad; Tiekink, Edward R. T.; Dolzhenko, Anton V.: A New One-Pot Three-Component Synthesis of 4-Aryl-6-cycloamino-1,3,5-triazin-2-amines under Microwave Irradiation

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Supporting Information

short review

Kahlert, Lukas; Schotte, Carsten; Cox, Russell J.: Total Mycosynthesis: Rational Bioconstruction and Bioengineering of Fungal Natural Products

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Gu, Zheng-Yang; Wu, Yang; Jin, Feng; Bao, Xiaoguang; Xia, Ji-Bao: Intermolecular C–H Amidation of Alkenes with Carbon Monoxide and Azides via Tandem Palladium Catalysis

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Supporting Information

Publication Date: 24 February 2021

paper

Yadav, Mangal S.; Singh, Sumt K.; Agrahari, Anand K.; Singh, Anoop S.; Tiwari, Vinod K.: N-Acylbenzotriazoles as Proficient Substrates for an Easy Access to Ureas, Acylureas, Carbamates, and Thiocarbamates via Curtius Rearrangement Using Diphenylphosphoryl Azide (DPPA) as Azide Donor

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Supporting Information

Publication Date: 23 February 2021

special topic > Special Issue dedicated to Prof. Sarah Reisman, recipient of the 2019 Dr. Margaret Faul Women in Chemistry Award

Lam, Heather; Abel-Snape, Xavier; Köllen, Martin F.; Lautens, Mark: Recent Advances in Transition-Metal-Free (4+3)-Annulations

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Publication Date: 22 February 2021

paper

Demidov, Maxim R.; Osyanin, Vitaly A.; Osipov, Dmitry V.; Klimochkin, Yuri N.: Oxidative Dimerization of 1Н-Benzo[f]chromenes: Synthesis of Benzannulated Analogues of Spirobiflavonoids Welwitschins E and F

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Supporting Information

paper

Deng, Si; Ouyang, Wenliang; Bai, Jiang; Song, Xian-Rong; Yang, Ruchun; Xiao, Qiang: Synthesis of Multibromo-Substituted Quinolines by NBS-Mediated Cascade Electrophilic Bromination/Cyclization of N-(3-Phenylprop-2-ynyl)anilines

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Supporting Information

paper

Gagnot, Glwadys; Legrand, Pierre; Tadros, Amira; Ezzahra Hibti, Fatima; Quatela, Alessia; Janin, Yves L.: On Pyridopyrazinol Chemistry: Synthesis of Chemiluminescent Substances

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Supporting Information

paper

Schädel, Nicole; Icik, Esra; Martini, Maike; Altevogt, Luca; Ramming, Isabell; Greulich, Andreas; Baro, Angelika; Bilitewski, Ursula; Laschat, Sabine: Synthesis of Imidazole and Histidine-Derived Cross-Linkers as Analogues of GOLD and Desmosine

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Supporting Information

review

Cullen, Stephen T. J.; Friestad, Gregory K.: Synthesis of Chiral Amines by C–C Bond Formation with Photoredox Catalysis

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special topic > Bond Activation – in Honor of Prof. Shinji Murai

Watanabe, Hikaru; Nakajima, Kazuki; Ekuni, Kento; Edagawa, Ryota; Akagi, Yuta; Okuda, Yasuhiro; Wakamatsu, Kan; Orita, Akihiro: Custom-Made Pyrene Photocatalyst-Promoted Desulfonylation of Arylethenyl Sulfones Using Green-Light-Emitting Diodes

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Supporting Information

Publication Date: 18 February 2021

feature

Li, Fusheng; Lin, Shuangjie; Li, Xiyu; Shi, Lei: Photocatalytic Generation of π-Allyltitanium Complexes from Butadiene via a Radical Strategy

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Supporting Information

feature

Shaaban, Saad; Li, Houhua; Merten, Christian; Antonchick, Andrey P.; Waldmann, Herbert: Rhodium(III)-Catalyzed Enantioselective Benzamidation of Cyclopropenes

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Supporting Information

paper

Li, Zhi; Fang, Mougui; Wu, Jingjing; Liu, Yunli; Liu, Yecheng; Wu, Fanhong: Efficient Monofluoroalkylation of Thiophenols or Phenols with α-Bromo-α-Fluoroketones under Mild Conditions

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Supporting Information

short review

Pedrood, Keyvan; Montazer, Mohammad Nazari; Larijani, Bagher; Mahdavi, Mohammad: Recent Advances in the Synthesis of Heterocycles by the Aza-Wittig Reaction

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Publication Date: 15 February 2021

paper

Zhang, Wenjie; Liu, Xueyan; Tian, Zhenfeng; Li, Hongji: Rh(III)-Catalyzed Olefination and Alkylation of Arenes with Maleimides: A Tunable Strategy for C(sp²)–H Functionalization

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Supporting Information CIF File

Publication Date: 11 February 2021

feature

Maximiano, Adrielle P.; Ramos, Giovana S.; Marques, Marcelo V.; Sá, Marcus M.: Functionalized Cyclopropanes as Versatile Intermediates for the Diversity-Oriented Synthesis of γ-Lactones, γ-Lactams and δ-Lactams

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Supporting Information

short review

Liu, Jiaming; Chen, Ming: 1,3-Bifunctional Nucleophilic Allylation Reagents: Preparative Methods and Synthetic Applications

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short review

Livingstone, Keith; Little, Gemma; Jamieson, Craig: Recent Advances in the Generation of Nitrilium Betaine 1,3-Dipoles

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Publication Date: 10 February 2021

paper

Saravanan, Velu; Mohanakrishnan, Arasambattu K.: Synthesis of Annulated Carbazoles via FeCl₃/SnCl₄‑Mediated Domino Reaction of Vinyl Ketone Tethered Bromomethylindoles with Arenes and Heteroarenes

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Supporting Information

Publication Date: 09 February 2021

paper

Schefzig, Luise; Kurzawa, Timon; Rancan, Giaime; Linder, Igor; Leisering, Stefan; Bera, Mrinal K.; Gart, Max; Zimmer, Reinhold; Reissig, Hans-Ulrich: Access to Highly Substituted Pyrimidine N-Oxides and 4-Acetoxymethyl-Substituted Pyrimidines via the LANCA Three-Component Reaction–Cyclocondensation Sequence

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Publication Date: 08 February 2021

paper

Avila-Melo, José Luis; Benavides, Adriana; Fuentes-Gutiérrez, Alfredo; Tamariz, Joaquín; Jiménez-Vázquez, Hugo A.: Total Synthesis of the Natural Carbazoles O-Demethylmurrayanine and Murrastanine A, and of a C4,C4′ Symmetric Murrastanine A Dimer from N-Phenyl-4,5-dimethylene-1,3-oxazolidin-2-one

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Supporting Information

paper

Yadav, Mamta; Jat, Ram Singh; Sarma, Bibek; Bhanuchandra, M.: 2-Pyridyl Sulfoxide Directed Pd(II)-Catalyzed C–H Olefination of Arenes with Molecular Oxygen as the Sole Oxidant

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Supporting Information

short review

Inoa, Joan; Dominici, Grecia; Eldabagh, Reem; Foley, Jonathan J.; Xing, Yalan: Synthetic Applications and Computational Perspectives on Eosin Y Induced Direct HAT Process

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Publication Date: 05 February 2021

paper

Pramanik, Sayan; Ray, Suman; Maity, Suvendu; Ghosh, Prasanta; Mukhopadhyay, Chhanda: Diastereoselective trans Cyclopropanation of 3-Alkylidene Oxindoles with In Situ Generated α-Diazo Carbonyls or α,β-Unsaturated Diazo Compounds

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Supporting Information CIF File

Publication Date: 01 February 2021

paper

Kuwabara, Motoi; Matsuo, Ami; Kamo, Shogo; Matsuzawa, Akinobu; Sugita, Kazuyuki: Stereoselective Convergent Synthesis of Carbon Skeleton of Cotylenin A Aglycone

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Supporting Information

Publication Date: 27 January 2021

paper

Peng, Jing; Hu, Ludan; Chen, Mu-Wang; Deng, Zhihong; Peng, Yiyuan: Synthesis of Difluoromethyl-Substituted Quinazolines through Selective Difluoromethylation

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Supporting Information

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Fukumoto, Yoshiya; Shiratani, Motohiro; Noguchi, Hikaru; Chatani, Naoto: Iridium-Catalyzed Direct Amidation of Imidazoles at the C-2 Position with Isocyanates in the Presence of Hydrosilanes Leading to Imidazole-2-Carboxamides

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Supporting Information

Publication Date: 26 January 2021

paper

He, Chang; Wang, Zijuan; Chen, Yitong; Zhang, Guolin; Yu, Yongping: Palladium(II)-Catalyzed C(sp)–C(sp²) Coupling: A Direct Approach to Multi-Substituted Pyrrolo[1,2-a]pyrazines

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Supporting Information

Publication Date: 25 January 2021

feature

Steinke, Tim; Wonner, Patrick; Engelage, Elric; Huber, Stefan M.: Catalytic Activation of a Carbon–Chloride Bond by Dicationic Tellurium-Based Chalcogen Bond Donors

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Supporting Information

paper

Khalili Foumeshi, Maryam; Ziyaei Halimehjani, Azim; Alaei, Ali; Klepetářová, Blanka; Beier, Petr: Tandem Alkylation/Michael Addition Reaction of Dithiocarbamic Acids with Alkyl γ-Bromocrotonates: Access to Functionalized 1,3-Thiazolidine-2-thiones

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short review

Zu, Bing; Guo, Yonghong; Ke, Jie; He, Chuan: Transient- and Native-Directing-Group-Enabled Enantioselective C–H Functionalization

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Publication Date: 22 January 2021

paper

Yavari, Issa; Sheikhi, Sara; Sheykhahmadi, Jamil; Taheri, Zohreh; Halvagar, Mohammad Reza: Ultrasound-Promoted Synthesis of Spirocyclopropanes from Switchable Starting Materials via Azomethine Ylide [3+2]-Cycloaddition

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short review

Neri, Raul; Bossmann, Stefan H.: Isoselenocyanates: Synthesis and Their Use for Preparing Selenium-Based Heterocycles

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Publication Date: 21 January 2021

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Yamamoto, Sonoka; Shibuya, Yushin; Suzuki, Toyoko; Okano, Kentaro; Horie, Masaki; Mori, Atsunori: One-Shot Deprotonative Metalation/Transmetalation/Polymerization of Halothiophenes Catalyzed by Nickel Complex for Polythiophene Synthesis

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Publication Date: 20 January 2021

paper

Majeed, Kashif; Liu, Bangjie; Zhou, Fengtao; Zhang, Qiuyu: Synthesis of 1,2,3-Triazole-Fused Indole Derivatives via Copper-Catalyzed Cascade Reaction

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Publication Date: 19 January 2021

paper

Chen, Jyun-Siao; Ke, Yi-Fan; Lin, Heng-Yan; Lin, Wesley; Yen, Wei-Chung; Wu, Hsin-Ru; Luo, Shun-Yuan: Development of a Novel Method for Trimethylsilylation of Saccharides­

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paper

Nazarian, Zohreh; Forsyth, Craig M.: A Cascade Process of Hydroxamates Renders 1,6-Dioxa-3,9-diazaspiro[4.4]nonane-2,8-diones

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Publication Date: 18 January 2021

errata

Srinivasulu, Vunnam; Al-Marzooq, Farah; Hamad, Mohamad; Khanfar, Monther A.; Ramanathan, Mani; Soares, Nelson C.; Al-Tel, Taleb H.: Sequencing Groebke–Blackburn–Bienaymé and Aza-Michael Addition Reactions: A Modular Strategy for Accessing a Diverse Collection of Constrained Benzoxazepine and Imidazopyrazine Systems

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paper

Gairola, Deepti; Peddinti, Rama Krishna: Methanesulfonic Acid Catalyzed Friedel–Crafts Reaction of Electron-Rich Arenes with N-Arylmaleimides: A Highly Efficient Metal-Free Route To Access 3-Arylsuccinimides

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paper

Mityuk, Andrey P.; Hrebonkin, Andrii; Lebed, Pavlo S.; Grabchuk, Galyna P.; Volochnyuk, Dmitriy M.; Ryabukhin, Sergey V.: Efficient Route for the Synthesis of Diverse Heteroannelated 5-Cyanopyridines

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paper

Wang, Siqi; Filatov, Alexander S.; Lozovskiy, Stanislav V.; Shmakov, Stanislav V.; Khoroshilova, Olesya V.; Larina, Anna G.; Selivanov, Stanislav I.; Boitsov, Vitali M.; Stepakov, Alexander V.: Construction of Spiro[3-azabicyclo[3.1.0]hexanes] via 1,3-Dipolar Cycloaddition of 1,2-Diphenylcyclopropenes to Ninhydrin-Derived Azomethine Ylides

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short review

Ashikari, Yosuke; Nagaki, Aiichiro: Homogeneous Catalyzed Aryl–Aryl Cross-Couplings in Flow

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Publication Date: 15 January 2021

paper

Zheng, Qiang; Boltjes, André; Dömling, Alexander: An Ugi Reaction/Intramolecular Cyclization/Oxidation Cascade towards Tetrazole-Linked Dibenzoxazepines

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Publication Date: 14 January 2021

errata

Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)

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review

Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)

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Publication Date: 13 January 2021

paper

You, Shengyong; Zhang, Rongli; Cai, Mingzhong: A Magnetically Recyclable Palladium-Catalyzed Formylation of Aryl Iodides with Formic Acid as CO Source: A Practical Access to Aromatic Aldehydes

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Publication Date: 11 January 2021

paper

Dziuba, Kamil; Frynas, Sławomir; Szwaczko, Katarzyna: Knoevenagel Condensation of Phosphinoylacetic Acids with Aldehydes: An Efficient One-Pot Strategy for the Synthesis of P-Functionalized Alkenyl Compounds

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paper

Lisovenko, Natalya Yu.; Nasibullina, Ekaterina R.; Kharitonova, Svetlana S.; Myshkina, Olga A.: Simple Synthesis of Substituted 3-Hydroxyfuran-2(5H)-ones

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paper

Yassine, Hasna; Bouali, Jamila; Oumessaoud, Asmaa; Ourhzif, El Mahdi; Hamri, Salha; Hafid, Abderrafia; Khouili, Mostafa; Pujol, Maria Dolors: Synthesis of New Dialkyl 2,2′-[Carbonylbis(azanediyl)]dibenzoates via Curtius Rearrangement

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paper

Yu, Haifeng; Wang, Kehua; Zhang, Xue; Wang, Wenju: Complementary and Regioselective Synthesis of Isomeric 3-[Isoxazol-3(or 5)-yl]indoles from β-Ethylthio-β-indolyl-α,β-unsaturated Ketones

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Publication Date: 08 January 2021

paper

Borisov, Denis D.; Chermashentsev, Grigorii R.; Novikov, Roman A.; Tomilov, Yury V.: Synthesis of Substituted β-Styrylmalonates by Sequential Isomerization of 2-Arylcyclopropane-1,1-dicarboxylates and (2-Arylethylidene)malonates

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paper

Budeev, Anton V.; Kantin, Grigory; Dar’in, Dmitry; Krasavin, Mikhail: Continued Exploration of Trifunctional Alkyl 4-Chloro-2-diazo-3-oxobutanoates: Streamlined Entry into [1,2,3]Triazolo[5,1-c][1,4]benzoxazines and [1,2,3]Triazolo[5,1-c][1,4]benzoxazepines

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paper

Kotha, Sambasivarao; Pulletikurti, Sunil; Fatma, Ambareen; Dhangar, Gopal; Naidu, Gonna Somu: Synthesis of Polycycles and Oxacycles via Tandem Metathesis of endo-Norbornene Derivatives

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Publication Date: 07 January 2021

paper

Glas, Carina; Wirawan, Ricky; Bracher, Franz: A Short Approach to N-Aryl-1,2,3,4-tetrahydroisoquinolines from N-(2-Bromobenzyl)anilines via a Reductive Amination/Palladium-Catalyzed Ethoxyvinylation/Reductive N-Alkylation Sequence

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paper

Srinivasulu, Vunnam; Al-Marzooq, Farah; Hamad, Mohamad; Khanfar, Monther A.; Ramanathan, Mani; Soares, Nelson C.; Al-Tel, Taleb H.: Sequencing Groebke–Blackburn–Bienaymé and Aza-Michael Addition Reactions: A Modular Strategy for Accessing a Diverse Collection of Constrained Benzoxazepine and Imidazopyrazine Systems

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Supporting Information

Publication Date: 21 December 2020

paper

Jurkowski, Kellsie; Bauer, Eike B.: Ferrocenium Ions as Catalysts: Decomposition Studies and Counteranion Influence on Catalytic Activity

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Publication Date: 15 December 2020

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Kawakami, Haruka; Nohira, Itsuki; Chatani, Naoto: Nickel-Catalyzed C–F/N–H Annulation of 2-(2-Fluoroaryl) N-Heteroaromatic Compounds with Alkynes: Activation of C–F Bonds

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Supporting Information CIF File

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Xu, Wengang; Wu, Mingbo; Yoshikai, Naohiko: Iron-Catalyzed Remote C–H Alkylation of 8-Amidoquinolines with Cycloalkanes

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Publication Date: 07 December 2020

paper

Hsu, Ming-Hua; Kapoor, Mohit; Pradhan, Tapan Kumar; Tse, Man-Him; Chen, Hsin-Ya; Yan, Man-Jun; Cheng, Yu-Tsen; Lin, Yu-Cheng; Hsieh, Cheng-Ying; Liu, Ker-Yin; Han, Chien-Chung: Mild and Efficient Copper-Catalyzed Synthesis of Trisubstituted Pyrroles

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Supporting Information CIF File

paper

Ji, Jiu-Jian; Zhu, Zhi-Qiang; Xie, Zong-Bo; Tang, Juan; Yuan, En; Le, Zhang-Gao: Highly Efficient Copper-Catalyzed Dehydrogenative Cross-Coupling of Azoles with α-Amino Carbonyl Compounds

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Publication Date: 03 December 2020

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Takahashi, Hiroto; Honjo, Yusaku; Shibata, Yu; Nagashima, Yuki; Tanaka, Ken: Dienylation of Unfunctionalized Arenes with 1,6-Diynes via Rhodium-Catalyzed Directing-Group-Free C–H Bond Activation

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Publication Date: 28 October 2020

special topic > Bond Activation – in Honor of Prof. Shinji Murai

Ishida, Naoyoshi; Iwamoto, Hiroaki; Sunagawa, Denise Eimi; Ohashi, Masato; Ogoshi, Sensuke: CsF-Catalyzed Fluoroacylation of Tetrafluoroethylene Using Acyl Fluorides for the Synthesis of Pentafluoroethyl Ketones

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