DOI: 10.1055/s-00000084

Synthesis

eFirst

Publication Date: 18 September 2017

paper

Trubitsõn, Dmitri; Žari, Sergei; Kaabel, Sandra; Kudrjashova, Marina; Kriis, Kadri; Järving, Ivar; Pehk, Tõnis; Kanger, Tõnis: Asymmetric Organocatalytic Cascade Synthesis of Tetrahydro­furanyl Spirooxindoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0475_ga_10-1055_s-0036-1590918.gif
Supporting Information

Publication Date: 14 September 2017

paper

Linke, Jens; Bader, Natalia; Tellenbröker, Jörg; Kuck, Dietmar: Sixfold Peripheral Halogenation of Tribenzotriquinacenes: An Alternative Access to Useful TBTQ Building Blocks
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0468_ga_10-1055_s-0036-1589107.gif
Supporting Information

Publication Date: 13 September 2017

short review

Chen, Yue-Gang; Xu, Xue-Tao; Zhang, Kun; Li, Yi-Qian; Zhang, Li-Pu; Fang, Ping; Mei, Tian-Sheng: Transition-Metal-Catalyzed Carboxylation of Organic Halides and Their Surrogates with Carbon Dioxide
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0418_ga_10-1055_s-0036-1590908.gif

Publication Date: 12 September 2017

feature

López-Rodríguez, Alberto; Domínguez, Gema; Pérez-Castells, Javier: Synthesis of Novel Iminosugar Derivatives Based on a 2-Azabi­cyclo[4.1.0]heptane Skeleton
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0404_ga_10-1055_s-0036-1589109.gif
Supporting Information

paper

Ding, Weijie; Hu, Juan; Jin, Huile; Yu, Xiaochun; Wang, Shun: One-Pot Synthesis of α,β-Unsaturated Esters, Ketones, and Nitriles from Alcohols and Phosphonium Salts
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0451_ga_10-1055_s-0036-1590904.gif
Supporting Information

paper

Kaboudin, Babak; Donyavi, Atousa; Kazemi, Foad: Trichloroisocyanuric Acid as an Efficient Reagent for the Synthesis of Phosphoroamidates via Atherton–Todd Reaction under Base-Free Conditions
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0440_ga_10-1055_s-0036-1589111.gif
Supporting Information

paper

Rahil, Rima; Sengmany, Stéphane; Le Gall, Erwan; Léonel, Eric: Nickel-Catalyzed Electrochemical Reductive Homocouplings of Aryl and Heteroaryl Halides: A Useful Route to Symmetrical Biaryls
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0393_ga_10-1055_s-0036-1589100.gif
Supporting Information

short review

Kimura, Tsutomu: Recent Advances in Magnesium Carbenoid Chemistry
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0420_ga_10-1055_s-0036-1590894.gif

Publication Date: 07 September 2017

paper

Cimarelli, Cristina; Bordi, Samuele; Piermattei, Pamela; Pellei, Maura; Del Bello, Fabio; Marcantoni, Enrico: An Efficient Lewis Acid Catalyzed Povarov Reaction for the One-Pot Stereocontrolled Synthesis of Polyfunctionalized Tetrahydroquinolines­
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0457_ga_10-1055_s-0036-1589104.gif
Supporting Information

paper

Liu, Qiang; Chen, Xiang-Yu; Li, Sun; Vetica, Fabrizio; Raabe, Gerhard; Enders, Dieter: Two-Step Synthesis of α,β-Unsaturated γ-Amino Acid Esters via N-Heterocyclic Carbene Catalyzed [4+2] Cycloaddition of Enals and Nitroso Compounds
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0502_ga_10-1055_s-0036-1590901.gif
Supporting Information

paper

Quintard, Adrien; Roudier, Mylène; Rodriguez, Jean: Multicatalytic Enantioselective Borrowing Hydrogen δ-Lactonization Strategy from β-Keto Esters and Allylic Alcohols
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0399_ga_10-1055_s-0036-1588547.gif
Supporting Information

Publication Date: 06 September 2017

paper

Ajdačić, Vladimir; Nikolić, Andrea; Simić, Stefan; Manojlović, Dragan; Stojanović, Zoran; Nikodinovic-Runic, Jasmina; Opsenica, Igor M.: Decarbonylation of Aromatic Aldehydes and Dehalogenation of Aryl Halides Using Maghemite-Supported Palladium Catalyst
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0452_ga_10-1055_s-0036-1590892.gif
Supporting Information

paper

Wu, Mingshu; Jiang, Jie; Zhu, Zhongxiang; Wang, Qinghe; Kong, Dulin: One-Pot Catalyst-Free Domino Condensation/Intramolecular 1,3-Dipolar Cycloaddition: Highly Stereoselective Access to Phosphadihydrocoumarin-Fused N,N-Bicyclic Pyrazolidin-3-ones
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0438_ga_10-1055_s-0036-1590896.gif
Supporting Information CIF File

short review

Pankova, Alena S.; Kuznetsov, Mikhail A.: Recent Advances in the Chemistry of 2-Acylaziridines
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0411_ga_10-1055_s-0036-1590889.gif

Publication Date: 31 August 2017

paper

Rao, Vijay V.; Mirzadeh, Nedaossadat; Bhargava, Suresh; Likhar, Pravin R.: Highly Selective Approach to α-Iodoketones from Aminoalkynols with Iodine Monochloride
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0415_ga_10-1055_s-0036-1590897.gif
Supporting Information

Publication Date: 30 August 2017

paper

Benischke, Andreas D.; Desaintjean, Alexandre; Juli, Thomas; Cahiez, Gérard; Knochel, Paul: Nickel-Catalyzed Cross-Coupling of Functionalized Organo­manganese Reagents with Aryl and Heteroaryl Halides Promoted by 4-Fluorostyrene
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0482_ga_10-1055_s-0036-1589101.gif
Supporting Information

psp

Hamper, Bruce C.; Sullivan, Brendan T.; Rath, Nigam P.; Spilling, Christopher D.: A Practical Gram-Scale Synthesis of Acrylohydroxamic Acid
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0463_ga_10-1055_s-0036-1589103.gif
Supporting Information

short review

Pathipati, Stalin R.; van der Werf, Angela; Selander, Nicklas: Indium(III)-Catalyzed Transformations of Alkynes: Recent Advances in Carbo- and Heterocyclization Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0431_ga_10-1055_s-0036-1588555.gif

short review

Wang, Chuan: Electrophilic Ring Opening of Small Heterocycles
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0460_ga_10-1055_s-0036-1589102.gif

Publication Date: 29 August 2017

paper

Dey, Papiya; Chatterjee, Sucheta; Gamre, Sunita S.; Chattopadhyay, Subrata; Sharma, Anubha: An Enantioselective Synthesis of (5S,6R,11S,14R)-Acremodiol
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0303_ga_s10-1055_s-0036-1588557.gif
Supporting Information

Publication Date: 28 August 2017

paper

Demidoff, Felipe C.; de Souza, Fabrícia P.; Netto, Chaquip D.: Synthesis of Stilbene-Quinone Hybrids through Heck Reactions in PEG-400
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0336_ga_10-1055_s-0036-1589095.gif
Supporting Information

paper

Kaduskar, Rahul D.; Pinto, Andrea; Scaglioni, Leonardo; Musso, Loana; Dallavalle, Sabrina: Synthesis of the Tripeptide Antibiotic Resormycin
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0385_ga_10-1055_s-0036-1588553.gif
Supporting Information

paper

Tao, Sheng; Ji, Enhui; Shi, Lei; Liu, Ning; Xu, Liang; Dai, Bin: Copper-Catalyzed C–N Bond Exchange of N-Heterocyclic Substituents around Pyridine and Pyrimidine Cores
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0286_ga_10-1055_s-0036-1590893.gif
Supporting Information

paper

Zhou, Xiao-Yu; Chen, Xia; Wang, Liang-Guang: Recycled Pd/C-Catalyzed Heck Reaction of 2-Iodoanilines under Ligand-Free Conditions
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0423_ga_10-1055_s-0036-1590895.jpg
Supporting Information

short review

Gusarova, Nina K.; Chernysheva, Nataliya A.; Trofimov, Boris A.: Catalyst- and Solvent-Free Addition of the P–H Species to Alkenes and Alkynes: A Green Methodology for C–P Bond Formation
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0352_ga_10-1055_s-0036-1588542.gif

short review

Henry, Martyn C.; Mostafa, Mohamed A. B.; Sutherland, Andrew: Recent Advances in Transition-Metal-Catalyzed, Directed Aryl C–H/N–H Cross-Coupling Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0443_ga_10-1055_s-0036-1588536.gif

short review

Hu, Wen-Li; Hu, Xiang-Guo; Hunter, Luke: Recent Developments in the Deoxyfluorination of Alcohols and Phenols: New Reagents, Mechanistic Insights, and Applications
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0392_ga_10-1055_s-0036-1590881.gif

Publication Date: 25 August 2017

short review

Aziz, Jessy; Piguel, Sandrine: An Update on Direct C–H Bond Functionalization of Nitrogen-Containing Fused Heterocycles
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0426_ga_10-1055_s-0036-1590859.gif

Publication Date: 24 August 2017

paper

Bencke, Carlos E.; Marangoni, Mário A.; Camargo, Adriano F.; Fantinel, Cassio A.; Bonacorso, Helio G.; Martins, Marcos A. P.; Zanatta, Nilo: Synthesis of Penta-2,4-dienenitriles by the Horner–Wadsworth–Emmons Olefination of Enones
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0398_ga_10-1055_s-0036-1590871.gif
Supporting Information

paper

Castelló-Micó, Alicia; Knochel, Paul: Zincation and Magnesiation of Functionalized Silylated Cyano­hydrins Using TMP-Bases
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0478_ga_10-1055_s-0036-1590887.gif
Supporting Information

paper

Katla, Ramesh; Chowrasia, Rakhi; da Silva, Caren D. G.; de Oliveira, Aline R.; dos Santos, Beatriz F.; Domingues, Nelson L. C.: Recyclable [Ce(l-Pro)2]2 (Oxa) used as Heterogeneous Catalyst: One-Pot Synthesis of 2,3-Dihydroquinazolin-4(1H)-ones in Ethanol
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0378_ga_10-1055_s-0036-1590886.gif
Supporting Information

Publication Date: 23 August 2017

paper

Ellwart, Mario; Höfner, Georg; Gerwien, Aaron; Wanner, Klaus T.; Knochel, Paul: Synthesis and Bioactivity of Novel N-Benzylic and N-Phenethylic Ephedrine Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0428_ga_10-1055_s-0036-1588523.gif
Supporting Information

paper

Türtscher, Paul L.; Davis, Holly J.; Phipps, Robert J.: Palladium-Catalysed Cross-Coupling of Benzylammonium Salts with Boronic Acids under Mild Conditions
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0402_ga_10-1055_s-0036-1588548.gif
Supporting Information

short review

Zhao, Qun; Poisson, Thomas; Pannecoucke, Xavier; Besset, Tatiana: The Transient Directing Group Strategy: A New Trend in Transition-Metal-Catalyzed C–H Bond Functionalization
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0456_ga_10-1055_s-0036-1590878.gif

Publication Date: 22 August 2017

paper

Dong, Zhi-Bing; Wang, Ming; Zhu, Hui; Liu, Xing; Chang, Cai-Zhu: Base-Promoted Synthesis of O-Aryl/Alkyl N,N-Dimethylthiocarbamates Starting from Inexpensive and Environmentally Benign Disulfide
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0430_ga_10-1055_s-0036-1588545.gif
Supporting Information

paper

Matveeva, Maria D.; Borisova, Tatiana N.; Titov, Alexander A.; Anikina, Lada V.; Dyachenko, Svetlana V.; Astakhov, Grigorii S.; Varlamov, Alexey V.; Voskressensky, Leonid G.: Domino Reactions of 1-Aroyl-3,4-dihydroisoquinolines with α,β-Unsaturated Aldehydes
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0260_ga_10-1055_s-0036-1588486.gif
Supporting Information

paper

Ortega-Martínez, Aitor; Molina, Cynthia; Moreno-Cabrerizo, Cristina; Sansano, José M.; Nájera, Carmen: Synthesis of 3,3-Disubstituted 2-Oxindoles by Deacylative Alkylation of 3-Acetyl-2-oxindoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0386_ga_10-1055_s-0036-1590880.gif
Supporting Information

paper

Rathod, Jayant; Sharma, Brijesh M.; Mali, Pramod S.; Kumar, Pradeep: Tf2NH-Catalyzed 1,6-Conjugate Addition of Vinyl Azides with p-Quinone Methides: A Mild and Efficient Method for the Synthesis of β-Bis-Arylamides
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0227_ga_10-1055_s-0036-1588546.gif
Supporting Information

paper

Zhu, Hui; Liu, Xing; Chang, Cai-Zhu; Dong, Zhi-Bing: Copper-Catalyzed C–S Cross-Coupling Reaction: S-Arylation of Arylthioureas
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0413_ga_10-1055_s-0036-1590879.gif
Supporting Information

Publication Date: 16 August 2017

paper

Shi, Yubai; Li, Cheng; Ma, Shaohua; Zhang, Yin: Synthesis and Properties of Nitrogen-Containing Curved Heterosuperbenzene
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0327_ga_10-1055_s-0036-1590872.gif
Supporting Information CIF File

Publication Date: 14 August 2017

paper

Glachet, Thomas; Fache, Fabienne; Pelotier, Béatrice; Piva, Olivier: Desymmetrization of Hepta-1,6-dien-4-ol by a Highly Stereo­selective Tandem Prins–Ritter Cyclization: Access to New THP Acetamides
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0315_ga_10-1055_s-0036-1588521.gif
Supporting Information

Publication Date: 10 August 2017

paper

Drawanz, Bruna B.; Zimmer, Georgia C.; Rodrigues, Leticia V.; Nörnberg, Andressa B.; Hörner, Manfredo; Frizzo, Clarissa P.; Cunico, Wilson: 5,6,7,8-Tetrahydronaphthalen-1-amine as Precursor for Thiazolidi­nones and Benzothiazepinones: Synthesis and Atropisomeric Relationship
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0387_ga_10-1055_s-0036-1590866.gif
Supporting Information

paper

Shamim, Anwar; Vasconcelos, Stanley N. S.; de Oliveira, Isadora Maria; Reis, Joel S.; Pimenta, Daniel C.; Zukerman-Schpector, Julio; Stefani, Hélio A.: Synthesis of Glycosyl Azides and Their Applications Using CuAAC Click Chemistry to Generate Bis- and Tris(triazolyl)glycosyl Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0353_ga_10-1055_s-0036-1589090.gif
Supporting Information

Publication Date: 09 August 2017

paper

Abdiaj, Irini; Bottecchia, Cecilia; Alcazar, Jesus; Noёl, Timothy: Visible-Light-Induced Trifluoromethylation of Highly Functionalized Arenes and Heteroarenes in Continuous Flow
https://www.thieme-connect.de/media/synthesis/EFirst/i_e0382_ga_10-1055_s-0036-1588527.gif
Supporting Information

Publication Date: 07 August 2017

paper

Abel, Anton S.; Averin, Alexei D.; Buryak, Alexei K.; Savelyev, Evgenii N.; Orlinson, Boris S.; Novakov, Ivan A.; Beletskaya, Irina P.: The Palladium-Catalyzed Heteroarylation of Adamantylalkyl Amines with Dihalogenopyridines: Scope and Limitations
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0401_ga_10-1055_s-0036-1590860.gif
Supporting Information

special topic

Tokumaru, Kazuyuki; Bera, Kalisankar; Johnston, Jeffrey N.: 1,3,4-Oxadiazole and Heteroaromatic-Fused 1,2,4-Triazole Synthesis­ Using Diverted Umpolung Amide Synthesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0292_ga_10-1055_s-0036-1590802.gif
Supporting Information

Publication Date: 03 August 2017

paper

Rostami, Abed; Rostami, Amin; Ghaderi, Arash; Gholinejad, Mohammad; Gheisarzadeh, Sajedeh: Copper-Catalyzed C–S Bond Formation via the Cleavage of C–O Bonds in the Presence of S8 as the Sulfur Source
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0842_ga_10-1055_s-0036-1588508.gif
Supporting Information

Publication Date: 02 August 2017

paper

Adam, Rosa; Abarca, Belén; Ballesteros, Rafael: Synthesis of Novel Polyazinyl-Substituted Triazolopyridines from [1,2,3]Triazolo[1,5-a]pyridines
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0358_ga_10-1055_s-0036-1588525.gif
Supporting Information

paper

Feofanov, Mikhail N.; Anokhin, Maxim V.; Averin, Alexei D.; Beletskaya, Irina P.: The Friedel–Crafts Reaction of Indoles with Michael Acceptors Catalyzed by Magnesium and Calcium Salts
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0285_ga_10-1055_s-0036-1589068.gif
Supporting Information

paper

Jozeliūnaitė, Augustina; Striela, Romualdas; Labanauskas, Linas; Orentas, Edvinas: Practical Preparation of Octa- and Tetrabromoperylene Diimides and Derivatives Thereof
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0366_ga_10-1055_s-0036-1589088.gif
Supporting Information

paper

Krishna Reddy, Alavala Gopi; Satyanarayana, Gedu: Palladium-Catalyzed Copper-Free Sonogashira Coupling of 2-Bromoarylcarbonyls: Synthesis of Isobenzofurans via One-Pot Reductive Cyclization
https://www.thieme-connect.de/media/synthesis/EFirst/i_n0152_ga_10-1055_s-0036-1588513.gif
Supporting Information CIF File

paper

Zhang, Qian; Yuan, Jingwen; Yu, Mangfei; Zhang, Rui; Liang, Yongjiu; Huang, Peng; Dong, Dewen: Triflic Anhydride Promoted Intramolecular Cyclization of N-Aryl Cinnamides: Access to Polysubstituted Quinolin-2(1H)-ones
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0271_ga_10-1055_s-0036-1590821.gif
Supporting Information

Publication Date: 01 August 2017

paper

Gajulapalli, V. Pratap Reddy; Jafari, Ehsan; Kundu, Dipti S.; Mahajan, Suruchi; Peuronen, Anssi; Rissanen, Kari; Enders, Dieter: Organocatalytic Asymmetric Synthesis of 2,3′-Connected Bis-Indolinones by Mannich Reactions of N-Acetylindolin-3-ones with Isatin N-Boc Ketimines
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0371_ga_10-1055_s-0036-1590823.gif
Supporting Information

paper

Vetrichelvan, Muthalagu; Bokkala, Vijayabhaskar; Renganathan, Surendran; Mathur, Arvind; Rampulla, Richard; Gupta, Anuradha: A Short and Scalable Synthesis of Orthogonally Protected Bis(aminomethyl)malonic Acid: Access to Bioactive Macrocyclic Peptides
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0282_ga_10-1055_s-0036-1588505.gif
Supporting Information

Publication Date: 31 July 2017

paper

Raju, Selvam; Annamalai, Pratheepkumar; Chan, Fu-Wei; Tseng, Po-Yen; Chen, Po-Yen; Kuo, Ting-Shen; Chuang, Shih-Ching: Palladium-Catalyzed Regio- and Stereoselective Hydrosulfonation of Propiolate Esters
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0257_ga_10-1055_s-0036-1588501.gif
Supporting Information CIF File

special topic

Lessi, Marco; Panzetta, Gianmarco; Marianetti, Giulia; Bellina, Fabio: Improved Synthesis of Symmetrical 2,5-Diarylimidazoles by One-Pot Palladium-Catalyzed Direct Arylation Tailored on the Electronic Features of the Aryl Halide
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0347_ga_10-1055_s-0036-1589071.gif
Supporting Information

Publication Date: 27 July 2017

paper

da Silva, Erica C.; Yamakawa, Nathália C. G.; Dos Santos, Alcindo A.; Coelho, Fernando: Short and Diastereoselective Total Synthesis of the Polyhydroxylated Pyrrolidine LAB-1: A Potent α-Glycosidase Inhibitor
https://www.thieme-connect.de/media/synthesis/EFirst/i_m1645_ga_10-1055_s-0036-1590799.gif
Supporting Information

Publication Date: 26 July 2017

paper

Li, Sun; Chen, Xiang-Yu; Liu, Qiang; Peuronen, Anssi; Rissanen, Kari; Enders, Dieter: N-Heterocyclic Carbene-Catalyzed Activation of α-Chloroaldehydes: Asymmetric Synthesis of 5-Cyano-Substituted Dihydropyranones
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0422_ga_10-1055_s-0036-1588509.gif
Supporting Information

paper

Liu, Yi; Li, Zhi; Xie, Yichuan; He, Peng; Qiao, Junfei; Fan, Xinyuan; Du, Yuguo: Efficient One-Pot Synthesis of 2,4-Disubstituted Thiazoles and Dimeric Thiazoles Directly from Acyl Chlorides and β-Azido Disulfides
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0274_ga_10-1055_s-0036-1590810.gif
Supporting Information

Publication Date: 25 July 2017

paper

Han, Xiao-Dan; Ren, Chuan-Qing; Fu, Jian-Ping; Xiong, Wei; Wang, Hui-Bin; Dong, Xiao-Na; Ji, Jian-Wei; Hu, Ju-Wu: An Intramolecular Cycloaddition Approach to Construct Polysubstituted Pyrrolidones from Alkynyl Carboxamides and PTSA
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0178_ga_10-1055_s-0036-1588500.gif
Supporting Information

paper

Sun, Hongpeng; Xiao, Li; Li, Wei; Xie, Qiong; Shao, Liming: On-Water Silver(I)-Catalyzed Cycloisomerization of Acetylenic Free Amines/Amides towards 7-Azaindole/Indole/Isoquinolone Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0264_ga_10-1055_s-0036-1589072.gif
Supporting Information

paper

Wang, Hu; Tang, Meng: Aluminum Chloride Promoted Hantzsch Reaction of N-Tosylhydrazones
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0263_ga_10-1055_s-0036-1588496.gif
Supporting Information

paper

Wu, Xiaoyan; Xue, Lu; Luo, Shilong; Jia, Shiqi; Ao, Jun; Qin, Wenling: K2S2O8-Activated Friedel–Crafts Type Alkylation of Indoles with α-Amido Sulfones
https://www.thieme-connect.de/media/synthesis/EFirst/i_h0266_ga_10-1055_s-0036-1589073.jpg

paper

Yoshioka, Eito; Goto, Yuya; Minato, Ikko; Miyabe, Hideto: Aqueous-Medium Selective Modification of Cysteine and Related Thiols with Tricyclic Oxygen-Heterocycles
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0337_ga_10-1055_s-0036-1588497.gif
Supporting Information

Publication Date: 20 July 2017

paper

Denisova, Alexandra O.; Tokunova, Yulia A.; Fateev, Ilja V.; Breslav, Alexandra A.; Leonov, Vladimir N.; Dorofeeva, Elena V.; Lutonina, Olga I.; Muzyka, Inessa S.; Esipov, Roman S.; Kayushin, Alexey L.; Konstantinova, Irina D.; Miroshnikov, Anatoly I.; Stepchenko, Vladimir A.; Mikhailopulo, Igor A.: The Chemoenzymatic Synthesis of 2-Chloro- and 2-Fluorocordycepins
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0220_ga_10-1055_s-0036-1590804.gif
Supporting Information

paper

Doan, Bao Nguyen Do; Tan, Xin Yi; Ang, Chin May; Bates, Roderick W.: Synthesis of (±)-γ-Lycorane by Using an Intramolecular Friedel–Crafts Reaction
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0284_ga_10-1055_s-0036-1589067.gif
Supporting Information

paper

Kaneko, Yuki; Wakamori, Shinnosuke; Ikeuchi, Kazutada; Ohara, Kenya; Tanaka, Takashi; Yamada, Hidetoshi: Total Synthesis of Lagerstannin C: Follow-up of the Khanbabaee’s Synthesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0296_ga_10-1055_s-0036-1588477.gif
Supporting Information

Publication Date: 05 July 2017

paper

Porwal, Digvijay; Oestreich, Martin: B(C6F5)3-Catalyzed Reduction of Sulfoxides and Sulfones to Sulfides with Hydrosilanes
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0361_ga_10-1055_s-0036-1588476.gif
Supporting Information

special topic

Yu, Zhao; Bo, Tang; Aiying, Guan; Weiwei, Wang; Zhenhua, Zhang; Mingan, Wang: Synthesis and Fungicidal Activity of (E)-5-[1-(4-Phenyl-2-oxo-1-oxaspiro[4.5]dec-3-en-3-yl)ethylidene]-2-aminoimidazolin-4-one Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0247_ga_10-1055_s-0036-1588463.gif

Publication Date: 27 June 2017

special topic

Shang, Xiao-Jie; Liu, Zhong-Quan: A Catalyzed Aerobic Intramolecular C–O Bond Formation: Facile Access to Ring-Fused Dihydrobenzoxazine Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0242_ga_10-1055_s-0036-1588465.gif
Supporting Information

Publication Date: 26 June 2017

special topic

Skonieczny, Kamil; Jaźwiński, Jarosław; Gryko, Daniel T.: The Synthesis of Imidazo[1,2-f]phenanthridines, Phenanthro-[9,10-d]imidazoles, and Phenanthro[9′,10′:4,5]imidazo[1,2-f]-phenanthridines via Intramolecular Oxidative Aromatic Coupling
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0239_ga_10-1055_s-0036-1589053.gif
Supporting Information

Publication Date: 20 June 2017

special topic

Sabat, Nazarii; Smoleń, Sabina; Nauš, Petr; Perlíková, Pavla; Cebová, Magdaléna; Poštová Slavětínská, Lenka; Hocek, Michal: Synthesis of 2,6-Substituted 7-(Het)aryl-7-deazapurine Nucleobases (2,4-Disubstituted 5-(Het)aryl-pyrrolo[2,3-d]pyrimidines)
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0206_ga_10-1055_s-0036-1588443.gif
Supporting Information

Publication Date: 12 June 2017

special topic

Couly, Florence; Dubouilh-Benard, Carole; Besson, Thierry; Fruit, Corinne: Late-Stage C–H Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one Backbone: Synthesis of an Array of Potential Kinase Inhibitors
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0132_ga_10-1055_s-0036-1588434.gif
Supporting Information

Publication Date: 29 May 2017

special topic

Pinet, Sandra; Liautard, Virginie; Debiais, Mégane; Pucheault, Mathieu: Radical Metal-Free Borylation of Aryl Iodides
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0180_ga_10-1055_s-0036-1588431.gif
Supporting Information

special topic

Saito, Hayate; Nogi, Keisuke; Yorimitsu, Hideki: Palladium-Catalyzed Double Borylation of Diaryl Sulfoxides with Diboron
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0217_ga_10-1055_s-0036-1588848.gif
Supporting Information

Publication Date: 15 May 2017

special topic

Takenouchi, Yuta; Ito, Hajime: Copper(I)-Catalyzed Boryl Substitution of Allyl Aminals: Selective Synthesis of Linear γ-Aminoallylboronates
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0078_ga_10-1055_s-0036-1588802.gif
Supporting Information

Publication Date: 08 May 2017

feature

Eastabrook, Andrew S.; Sperry, Jonathan: Synthetic Access to 3,5,7-Trisubstituted Indoles Enabled by Iridium­-Catalyzed C–H Borylation
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0155_ga_10-1055_s-0036-1589018.gif
Supporting Information

Publication Date: 03 May 2017

special topic

Jang, Won Jun; Han, Jung Tae; Yun, Jaesook: NHC-Copper-Catalyzed Tandem Hydrocupration and Allylation of Alkenyl Boronates
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0138_ga_10-1055_s-0036-1588811.gif
Supporting Information

special topic

Zhang, Xiaojuan; Han, Xiuling; Hu, Zhiyong; Lu, Xiyan: Synthesis of Substituted Piperidines via Cationic Palladium(II)-Catalyzed Reductive Coupling of N-Tosyl-Tethered Alkynones
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0141_ga_10-1055_s-0036-1588803.gif
Supporting Information

Publication Date: 02 March 2017

special topic

Miura, Wataru; Hirano, Koji; Miura, Masahiro: Iridium-Catalyzed Site-Selective C–H Borylation of 2-Pyridones
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0044_ga_10-1055_s-0036-1588735.gif
Supporting Information