DOI: 10.1055/s-00000084

Synthesis

eFirst

Publication Date: 04 March 2026

Paper

  • Verma, Aman; Chaudhary, Gyanendra; Manna, Bappa; Devi, Mahima; Yadav, Vivek Kumar; Prabhakar, Amit; Verma, Deepti:

    AgNO3/K2S2O8-Promoted Decarboxylative Oxyphosphorylation of Cinnamic Acids: A Mild Synthesis of β-Ketophosphonates

    Image for article: AgNO<sub>3</sub>/K<sub>2</sub>S<sub>2</sub>O<sub>8</sub>-Promoted Decarboxylative Oxyphosphorylation of Cinnamic Acids: A Mild Synthesis of β-Ketophosphonates
    Supplementary Material (DOC)

    • Publication Date: 03 March 2026

    Paper

  • Bertha, Ferenc; Porcs-Makkay, Márta; Halász, Judit; Németh, Gábor; Horváth, Simon; Nyerges, Miklós; Rojas, Anne; Ortuno, Jean-Claude; Pusztai, Gyöngyvér; Garádi, Zsófia; Simig, Gyula; Volk, Balázs:

    Pyrrolo[2,3-h]tetrahydroisoquinoline Derivatives Exhibiting Mixed Dopaminergic D3 > D2 and Serotoninergic 5-HT6 Affinity

    Image for article: Pyrrolo[2,3-<i>h</i>]tetrahydroisoquinoline Derivatives Exhibiting Mixed Dopaminergic D<sub>3</sub> &gt; D<sub>2</sub> and Serotoninergic 5-HT<sub>6</sub> Affinity
    Supplementary Material (PDF)

    • Paper

  • Torabi, Sara; Jamshidi, Mahdi; Senff, David; Martens, Maximilian; Hilt, Gerhard:

    The Iodination of Strongly Electron-Deficient Arenes under Electrochemical Conditions with I2 and Catalytic Amounts of Chloride Anions

    Image for article: The Iodination of Strongly Electron-Deficient Arenes under Electrochemical Conditions with I<sub>2</sub> and Catalytic Amounts of Chloride Anions
    Supplementary Material (PDF)

    • Publication Date: 02 March 2026

    Paper

  • Deng, Linbei; Cai, Ying; Qian, Jiasheng; Tao, Min; Liu, Jianbo:

    Synthesis of α-Secondary Carbon Fluorine Amides via Successive Acylation and Fluorination of Schiff Bases: A Modification Strategy for Oxalyl Amides

    Image for article: Synthesis of α-Secondary Carbon Fluorine Amides via Successive Acylation and Fluorination of Schiff Bases: A Modification Strategy for Oxalyl Amides
    Supplementary Material (PDF)

    • Paper

  • Gutala, Phaneendra; Badarla, Venkata Krishna Rao; Reddy, Lekkala Amarnath; Nariyam, Sekhar Munaswamy; Guntaka, Naveen Reddy; Gousia, Achugatla; Bhosale, Sachin Shahaji:

    A Novel and Scalable Synthesis of Anlotinib Dihydrochloride via Titanium-Catalyzed Kulinkovich–Szymoniak Cyclopropanation

    Image for article: A Novel and Scalable Synthesis of Anlotinib Dihydrochloride via Titanium-Catalyzed Kulinkovich–Szymoniak Cyclopropanation
    Supplementary Material (PDF)

    • Paper > Published as part of the Special Topic 22nd International Symposium on Organometallic Chemistry Directed Towards Organic Synthesis (OMCOS-22)

  • Liu, Xiangrong; Moon, Hye Won; Cornella, Josep:

    Reduction of Nitroarenes to Anilines with an Air-Stable Bismuth Catalyst

    Image for article: Reduction of Nitroarenes to Anilines with an Air-Stable Bismuth Catalyst
    Supplementary Material (PDF)

    • Publication Date: 26 February 2026

    Paper > Published as part of 22nd International Symposium on Organometallic Chemistry Directed Towards Organic Synthesis (OMCOS-22)

  • Kondo, Keisuke; Shizukuishi, Naoki; Kubota, Koji; Ito, Hajime:

    Sodium-Lump-Mediated Mechanochemical Deprotection of Benzyl-Derived Groups

    Image for article: Sodium-Lump-Mediated Mechanochemical Deprotection of Benzyl-Derived Groups

    • Publication Date: 19 February 2026

    Short Review > Published as part of the Special Topic Dedicated to Thieme Chemistry Journal Awardees

  • Zhang, Peiqi; Quan, Yangjian:

    Synthesis of C3B Four-membered Rings

    Image for article: Synthesis of C<sub>3</sub>B Four-membered Rings

    • Publication Date: 17 February 2026

    Paper

  • Bicic, Sergiu; Oestreich, Martin:

    Photoredox-Catalyzed Transfer Thiobenzoyloxylation of Styrenes Using Oxime-Based Surrogates

    Image for article: Photoredox-Catalyzed Transfer Thiobenzoyloxylation of Styrenes Using Oxime-Based Surrogates
    Supplementary Material (PDF)

    • Short Review

  • Xiong, Wenzhang; Wang, Rui; Liu, Wenbo H.:

    Recent Progress in the Synthesis and Application of 2-Acylaziridines

    Image for article: Recent Progress in the Synthesis and Application of 2-Acylaziridines

    • Publication Date: 13 February 2026

    Paper

  • Joardar, Suman Kumar; Rao, G. Prabhakar; Soumya, Jakkani; Dey, Soumen; Kundu, Mrinalkanti; Kundu, Taraknath:

    Nickel-Catalyzed 8-Aminoimidazo[1,2-a]pyridine-Assisted C(sp2)–H Alkynylation of (Hetero)arenes via an Inverse Sonogashira Strategy Suitable for Late-Stage Modification

    Image for article: Nickel-Catalyzed 8-Aminoimidazo[1,2-<i>a</i>]pyridine-Assisted C(sp<sup>2</sup>)–H Alkynylation of (Hetero)arenes via an Inverse Sonogashira Strategy Suitable for Late-Stage Modification
    Supplementary Material (PDF)

    • Short Review

  • Park, Yong Sun:

    Catalytic 1,2-Elimination: A Novel Asymmetric Approach

    Image for article: Catalytic 1,2-Elimination: A Novel Asymmetric Approach

    • Publication Date: 11 February 2026

    Paper > Published as part of the Special Issue dedicated to Prof. Franziska Schoenebeck, recipient of the 2025 Dr. Margaret Faul Women in Chemistry Award

  • Josephitis, Celena; McNally, Andrew:

    Selective Reductions of Complex Pyridines via NTf-Pyridinium Salts

    Image for article: Selective Reductions of Complex Pyridines via NTf-Pyridinium Salts
    Supplementary Material (PDF)

    • Paper

  • Li, Lu-Ting; Huang, Xiao-Cheng; Yao, Zhixiang; Su, Hui; Yang, Yuexin:

    Synthesis of 4-Sulfenyl-Isocoumarins via Thio-Annulation of 2-Alkynyl-benzonate with RSCl: In Situ Preparation using Disulfides and HCl/HNO3

    Image for article: Synthesis of 4-Sulfenyl-Isocoumarins via Thio-Annulation of 2-Alkynyl-benzonate with RSCl: In Situ Preparation using Disulfides and HCl/HNO<sub>3</sub>
    Supplementary Material (PDF)

    • Paper

  • Vaishya, Vartika; Verma, Abhishek Kumar; Pilania, Meenakshi:

    Rational Design, Synthesis, and in silico Bio-efficacy of Triazole-Clubbed Chalcone Hybrids

    Image for article: Rational Design, Synthesis, and in silico Bio-efficacy of Triazole-Clubbed Chalcone Hybrids
    Supplementary Material (PDF)

    • Short Review > Published as part of the Special Topic 22nd International Symposium on Organometallic Chemistry Directed Towards Organic Synthesis (OMCOS-22)

  • Fujii, Ikuya; Shintani, Ryo:

    1,n-Metal Migrations Mediated by 3d Transition Metals

    Image for article: 1,<i>n</i>-Metal Migrations Mediated by 3d Transition Metals

    • Publication Date: 04 February 2026

    Short Review

  • Xu, Jiahao; Liang, Mengjia; Wei, Liwen; Yang, Xing:

    Catalytic Asymmetric Construction of Medium-Sized Ring Systems with Single Axial or Inherent Chiral Element

    Image for article: Catalytic Asymmetric Construction of Medium-Sized Ring Systems with Single Axial or Inherent Chiral Element

    • Publication Date: 02 February 2026

    Paper

  • Benedix, Lars; Mross, David; Hiersemann, Martin:

    Synthetic Access to Indolo[2,3-d]tropone-Derived Tolanes and Synthesis of Indolo[2,3-d]tropolones

    Image for article: Synthetic Access to Indolo[2,3-<i>d</i>]tropone-Derived Tolanes and Synthesis of Indolo[2,3-<i>d</i>]tropolones
    Supplementary Material (PDF)

    • Publication Date: 30 January 2026

    Paper

  • Charles, Johana; Le Borgne, Marc; Verel, Ema; Guillon, Jean; Pinaud, Noël; Gast, Alexander; Jose, Joachim; Marminon, Christelle:

    Synthesis of Indeno[1,2-b]indole-9,10-diones: Toward a One-Pot, Two-Step Reaction

    Image for article: Synthesis of Indeno[1,2-<i>b</i>]indole-9,10-diones: Toward a One-Pot, Two-Step Reaction
    Supplementary Material (PDF)

    • Review

  • Tariq, Sobia; Haider, Arsalan; Yu, Qian; Chen, Jun; Bai, Xueling; Zhang, Runtong; Ma, Baode:

    Recent Advances on Asymmetric Synthesis of Benzofused Six-Membered Oxygen-Containing Heterocycles (2020–2025)

    Image for article: Recent Advances on Asymmetric Synthesis of Benzofused Six-Membered Oxygen-Containing Heterocycles (2020–2025)
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