DOI: 10.1055/s-00000131

Synfacts

Issue 04 · Volume 2011 · April 2011 DOI: 10.1055/s-002-21773

Synform

  • A28

    SYNFORM ISSUE 2011/04

    • Synthesis of Natural Products and Potential Drugs

  • z349

    All PDFs of this category

  • 0349

    Syntheses of (±)-Hamigeran B and (±)-4-Bromohamigeran B

  • 0350

    Synthesis of the HIV Integrase Inhibitor Raltegravir Potassium

  • 0351

    Asymmetric Synthesis of 1,1-Diarylethane Drugs

  • 0352

    Synthesis of (-)-Sclerophytin A

  • 0353

    Synthesis of (+)-Lyconadin A

  • 0354

    Synthesis of Glycine Transporter Inhibitor GSK2137305

  • 0355

    Synthesis of Triple Reuptake Inhibitor GSK1360707F

  • 0356

    Biomimetic Synthesis of (±)-Rossinone B

  • 0357

    Formal Synthesis of (-)- and (+)-Phalarine

  • 0358

    Synthesis of MK-3281

  • 0359

    Synthesis of Three of the Cladiellins

  • 0360

    Synthesis of a p38 MAP Kinase Inhibitor

  • 0361

    Synthesis of Sintokamides A, B and E

    • Synthesis of Heterocycles

  • z363

    All PDFs of this category

  • 0363

    One-Pot Synthesis of Tetrahydroisoquinolines via Benzene Ring Annulation

  • 0364

    Palladium-Catalyzed Atom-Economical Synthesis of Pyrroles

  • 0365

    Organocatalytic Cascade Synthesis of Decahydroquinolines

  • 0366

    Synthesis of Imidazolin-5-ones by Thermolysis of α-Azido Esters

  • 0367

    Base-Mediated Synthesis of 4,5-Disub-stituted Furan-2(5H)-ones

  • 0368

    Synthesis of Pyrazoloisoquinolines via a Multicomponent Suzuki Reaction Sequence

  • 0369

    Synthesis of 1,3,5-Trisubstituted Hydantoin via a Three-Component Reaction

  • 0370

    Unexpected Products from the Biginelli Reactions of 3-Amino-1,2,4-triazole

  • 0371

    Synthesis of Furo[3,2-c]pyridinones via an Aza-Oxy-Carbanion Relay Strategy

  • 0372

    1,3-Dipolar Cycloaddition Route to 1,3-Benzodiazepinones

  • 0373

    Extending the Scope of the Biginelli Reaction Using Palladium Catalysis

  • 0374

    Rhodium(II)-Catalyzed Hydroamination of Propargylguanidines

  • 0375

    Sonogashira-Heteroannulative Route to Dihydroisobenzofurans

  • 0376

    Combined Ugi-Pictet-Spengler Synthesis of Polycyclic Ketopiperazines

  • 0377

    Oxidative Approach to Isoxazolines

    • Synthesis of Materials and Unnatural Products

  • z379

    All PDFs of this category

  • 0379

    Donor-Acceptor Type Fused Porphyrin-Perylene Monoimides

  • 0380

    Lights, Magnets, Action!

  • 0381

    New 7b-Arylfluoradenes

  • 0382

    A Chelating Diphosphane Ligand on a β-Cyclodextrin Backbone

  • 0383

    Twist with Twin Porphyrin

  • 0384

    New Precursor for Difluorocarbenes

  • 0385

    Click it!

  • 0386

    Cross-Coupling Made Easy

  • 0387

    [2,2]Paracyclophanes with New Bridges

  • 0388

    Photon-Quantitative Cyclization of Dithiazolylarylene

  • 0389

    Photoinduced Rearrangements of 3,3′-Bis(arylbenzofurans)

  • 0390

    Extended Porphyrins

  • 0391

    Ivyanes from Dendralenes

    • Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

  • z393

    All PDFs of this category

  • 0393

    Rhodium(I)-Catalyzed Asymmetric Desymmetrization by Retro-Allylation

  • 0394

    Calcium-Catalyzed Enantioselective Electrophilic Amination of Enamides

  • 0395

    Enantioselective Conjugated Addition of Vinylaluminums to Cyclic Enones

  • 0396

    [6+2] Cycloadditions between Cyclohepta-triene and Allenes

  • 0397

    Gold-Catalyzed Cyclopenta- and Cyclo-heptannulation

  • 0398

    Palladium-Catalyzed Synthesis of Alkynylcyclopropanes

  • 0399

    Rhodium(II)-Catalyzed Enantioselective C-H Functionalization of Indoles

  • 0400

    Regio- and Stereoselective Bromocyanation of Alkynes

  • 0401

    Direct Aldol Reaction Catalyzed by a Chiral Bifunctional Catalyst System

  • 0402

    Catalytic Asymmetric Hydroboration of α-Substituted Styrenyl Derivatives

  • 0403

    Brønsted Acid Differentiated Metal Catalysis by Kinetic Discrimination

  • 0404

    Desymmetrization of 2,2-Disubstituted
    1,3-Propanediols

  • 0405

    Asymmetric Rhodium-Catalyzed Hydrogenation of β-Amino Ketones

  • 0406

    Highly Regio- and Diastereoselective [3+2] Cycloadditions

  • 0407

    Cinchona-Derived Amino Phosphine Precatalysts for Cooperative Catalysis

  • 0408

    Chiral Aminotriazole Ligands in Ruthenium-Catalyzed Transfer Hydrogenation

  • 0409

    Catalytic Asymmetric Vinylogous and Bisvinylogous Aldol Reactions

  • 0410

    Highly Selective Aluminum-Catalyzed Oxidation of Cyclic Dithioacetals

  • 0411

    Enantioselective Addition of Pyrazolones to Dialkyl Azodicarboxylates

  • 0412

    Chiral Auxiliary Controlled Asymmetric Synthesis of Tertiary Alcohols

  • 0413

    Enantioselective Mukaiyama Aldol Reactions with Glyoxylates

  • 0414

    Asymmetric Ketone Hydrogenation Catalyzed by Copper-Phosphine Complexes

  • 0415

    Brønsted Acid Activated Palladium-Catalyzed Hydrogenation of Ketimines

  • 0416

    Synthesis of 1,3-Diols through Grignard Addition to Isopropenyl Acetate

  • 0417

    Asymmetric Ene and Aldol Reactions of Isatins, Diketones, and Keto Esters

  • 0418

    Sequential Addition of Nucleophiles to Bicyclic Isoxazololactams

  • 0419

    Iridium-Catalyzed Asymmetric Intramolecular Allylic Amidation

  • 0420

    Asymmetric Hydrogenation of Ketimines

    • Metal-Mediated Synthesis

  • z421

    All PDFs of this category

  • 0421

    Copper-Catalyzed Direct Sulfoximination

  • 0422

    Co-Catalyzed Cross-Coupling of C-H Bonds with Grignard Reagents

  • 0423

    Rh(III)-Catalyzed C-H Activation and Oxidative Coupling with Alkenes

  • 0424

    CuCl2-Mediated Cyclization of N-Alkoxy-ortho-alkynylbenzamides

  • 0425

    Pd-Catalyzed Oxidative Intramolecular C-H Coupling for Medium-Ring Synthesis

  • 0426

    Polysequential Synthesis of 2-Azaanthra-cenes from Ethynylbenzenes

  • 0427

    Iron-Mediated Tandem Annulation for the Synthesis of Various Chromenes

  • 0428

    Polarity Inversion of Ketones: Umpolung Reaction at the α-Position

  • 0429

    Palladium-Catalyzed One-Pot C-C and C-N Bond Formation by Dual C-H Activation

  • 0430

    Asymmetric Synthesis of 2-Aryl and 2-Vinyl Piperidines by Dynamic Resolution

  • 0431

    Copper(I)-Catalyzed Coupling of N-Tosyl-hydrazones with Terminal Alkynes

  • 0432

    Palladium-Catalyzed Cross-Coupling of Tosylhydrazones and Aryl Nonaflates

  • 0433

    Cobalt-Catalyzed ortho-Alkylation through Directed C-H Bond Activation

  • 0434

    Palladium-Catalyzed Synthesis of Functionalized Allylsilanes and Allylboronates

    • Organo- and Biocatalysis

  • z435

    All PDFs of this category

  • 0435

    Biocatalytic Formation of C-C Bonds

  • 0436

    Asymmetric Michael Addition-Lactonization of Carboxylic Acids

  • 0437

    NHC-Catalyzed Addition of Homoenolate Equivalents to Unsaturated Keto Esters

  • 0438

    Asymmetric α-Fluorination of Cyclic Ketones

  • 0439

    Internal Lewis Acid Activation of Ureas

  • 0440

    Indole Annulation via an Internal Redox Cascade

  • 0441

    Enantioselective Protonation by Cinchona Alkaloids via Phospha-Brook Rearrangement

  • 0442

    Dipeptide-Based Phosphine Catalyst for Cycloaddition of Allenes to Acrylates

  • 0443

    A Cascade Annulation of Enals and Dienones

  • 0444

    Dehydrative Condensation of Dicarboxylic Acids with Aminoboronic Acids

  • 0445

    Asymmetric Vinylogous Aldol Reactions of Furanones and α-Keto Esters

  • 0446

    NHC-Catalyzed Intermolecular Stetter Reaction with Asymmetric Protonation

  • 0447

    Solvent-Dependance in Organocatalyzed Diels-Alder Reactions

    • Polymer-Supported Synthesis

  • z449

    All PDFs of this category

  • 0449

    Flow Macrocyclization Using Copper Tubing

  • 0450

    Heck and Suzuki Reactions Using Supported Palladium Nanoparticles

  • 0451

    Alkylation with Alcohols Catalyzed by Ag/Mo Hybrid Metal

  • 0452

    Synthesis of Dihydropyrimidinones with PEG-Supported Thiourea Dioxide

  • 0453

    Asymmetric Cyclopropanation with [Cu(OTf)2(t-Bu2-DABox)][Pt]@Si

  • 0454

    Aldol and α-Amination Reactions with Proline-Functionalized Reactors

  • 0455

    Polystyrene-Supported Iodosylbenzene Sulfate as an Oxidizing Agent

  • 0456

    Mono-N-Alkylation of Anilines with R3N Using Pd/C under Microwave Irradiation

  • 0457

    Triazine-Based Polymer/Nano-Pd: Oxidation of Alcohols

  • 0458

    Carbonylative Suzuki-Miyaura Coupling Using PS-Pd-NHC

  • 0459

    Synthesis of α,β-Acetylenic Ketones with Polystyrene-Supported ZnBr2

  • 0460

    A Silica-Supported Imidazolium Salt for Nucleophilic Substitution in Water