Synthesis

Issue 06 · March 2017

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review
1131
Miyamura, Shin; Itami, Kenichiro; Yamaguchi, Junichiro:
Syntheses of Biologically Active 2-Arylcyclopropylamines

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short review
1150
Zhang, Min; Zhu, Chunyin; Ye, Long-Wu:
Recent Advances in Dual Visible Light Photoredox and Gold-Catalyzed Reactions

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1158
Lepori, Clément; Hannedouche, Jérôme:
First-Row Late Transition Metals for Catalytic (Formal) Hydroamination of Unactivated Alkenes

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1168
Comas-Barceló, Júlia; Harrity, Joseph P. A.:
Metal Acetylides in Cycloaddition Reactions

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1182
Grimaud, Laurence; Jutand, Anny:
Role of Fluoride Ions in Palladium-Catalyzed Cross-Coupling Reactions

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feature
1190
Jung, Eun-Kyung; Pilkington, Lisa I.; Barker, David:
Synthesis of Benzodioxane and Benzofuran Scaffolds Found in Neolignans via TMS Triflate Mediated Addition to 1,4-Benzodioxane Hemiacetals

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1206
Ábrahámi, Renáta A.; Kiss, Loránd; Fustero, Santos; Fülöp, Ferenc:
Functionalized Dialdehydes as Promising Scaffolds for Access to Heterocycles and β-Amino Acids: Synthesis of Fluorinated Piperidine and Azepane Derivatives

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paper
1214
Kazem-Rostami, Masoud:
Design and Synthesis of Ʌ-Shaped Photoswitchable Compounds Employing Tröger’s Base Scaffold

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1223
Garnier, Tony; Sakly, Randa; Danel, Mathieu; Chassaing, Stefan; Pale, Patrick:
Chan–Lam-Type C–N Cross-Coupling Reactions under Base- and Ligand-Free Cu^I-Zeolite Catalysis

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1231
Lizza, Joseph R.; Moura-Letts, Gustavo:
Solvent-Directed Epoxide Opening with Primary Amines for the Synthesis of β-Amino Alcohols

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1243
Bröhl, Nina Felicitas; Kundu, Dipti Sankar; Raabe, Gerhard; Enders, Dieter:
One-Pot Synthesis of 1-Substituted 1H-Isochromenes by Combining Brønsted Acid with Silver Catalysis
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1255
Shirinian, Valerii Z.; Kavun, Alexey M.; Lvov, Andrey G.; Zavarzin, Igor V.; Krayushkin, Michail M.:
Practical and Efficient Synthesis of Polyaryl(hetaryl)-Substituted Cyclohexenones and Salicylates

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1264
Jeong, Hyeonsu; Yadav, Nagendra Nath; Ha, Hyun-Joon:
Synthesis of Lacosamide (Vimpat) and Its Derivatives from Aziridine-(2R)-carboxylate

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1273
Chuang, Che-Ping; Chen, Ying-Yu; Chuang, Tsung-Han; Yang, Cheng-Hao:
Copper-Salt-Promoted Carbocyclization Reactions of α-Bromo-N-arylacylamides

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1285
Fujita, Keisuke; Nakagawa, Naoki; Sunahara, Kazuhiro; Ogura, Tadayuki; Okano, Kentaro; Mori, Atsunori:
A Step-Efficient Pathway to Chlorine-Functionalized Thiophene Oligomers by Palladium-Catalyzed Deprotonative Coupling of Chlorothiophenes

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1295
Yoshida, Masanori; Yano, Shohei; Hara, Shoji:
Asymmetric Allylation of 2-Oxocycloalkanecarboxylates

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1301
Okada, Iku; Fukuda, Takuya; Kuroda, Yu; Noguchi, Keiichi; Chiba, Kazuhiro; Kitano, Yoshikazu:
Direct Synthesis of Bis(alkylamino)maleonitriles from Alcohols and TMSCN with Bi(OTf)₃

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1307
Ma, Zhi-Wei; Liu, Xiao-Feng; Sun, Bin; Huang, Xian-Hui; Tao, Jing-Chao:
Chiral Primary Amine–Squaramide Catalyzed Highly Enantioselective Michael Addition of Isobutyraldehyde to Nitroolefins

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1315
González-Cardenete, Miguel A.; Zaragozá, Ramón J.:
A Short and Improved Synthesis of the Antiprotozoal Abietane Diterpenoid (–)-Sugikurojin A

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1319
Schettini, Rosaria; D’Amato, Assunta; De Riccardis, Francesco; Della Sala, Giorgio; Izzo, Irene:
Catalytic Alkylation of 2-Aryl-2-oxazoline-4-carboxylic Acid Esters Using Cyclopeptoids; Newly Designed Phase-Transfer Catalysts

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1327
Batool, Farhat; Emwas, Abdul-Hamid; Gao, Xin; Munawar, Munawar A.; Chotana, Ghayoor A.:
Synthesis and Suzuki Cross-Coupling Reactions of 2,6-Bis(trifluoromethyl)pyridine-4-boronic Acid Pinacol Ester

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1335
Zhu, Ranran; Wang, Yuntao; Liu, Jialin; Wang, Qing; Huang, Jianhui:
One-Pot Synthesis of Imidazolyl Isoquinolines under a Palladium-Catalyzed C–H Activation/Annulation (CHAA) Reaction

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1342
Zhang, Min; Zhao, Yun; Chen, Wanzhi:
Peroxide-Free Co(OAc)₂-Catalyzed Radical Addition of sp³ C–H Bonds to Alkynes

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1349
Li, Bin; Zheng, Jianxiong; Zeng, Weifeng; Li, Yibiao; Chen, Lu:
Efficient Ruthenium(II)-Catalyzed Direct Reductive Amination of Aldehydes under Mild Conditions Using Hydrosilane as the Reductant

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1356
Guo, Dong-Cai; Zhang, Chao; Li, Fei; Zhang, Fenghua; Yu, Fang; He, Yu-Peng:
Synthesis of Tricyclic Isoxazoles via Sequential [3+2] Dipolar Cycloaddition and Palladium-Catalyzed Intramolecular Arylation Reactions

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1371
Feng, Yue; Zhou, Wanjia; Sun, Ge; Liao, Peiqiu; Bi, Xihe; Li, Xingqi:
Highly Efficient Synthesis of N-Sulfonylamidines via Silver-Catalyzed or Metal-Free Thermally Promoted Denitrogenative Amination of N-Sulfonyl-1,2,3-triazoles

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1380
Zhang, Ting; Dai, Yifeng; Cheng, Siwei; Liu, Yongguo; Yang, Shaoxiang; Sun, Baoguo; Tian, Hongyu:
A Facile Method for the Sulfenyllactonization of Alkenoic Acids Using Dimethyl Sulfoxide Activated by Oxalyl Chloride

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1387
Buxaderas, Eduardo; Graziano-Mayer, Marilyn; Volpe, María Alicia; Radivoy, Gabriel:
Bimetallic Cu-Pd Nanoparticles Supported on Bio-silica as an Efficient Catalyst for Selective Aerobic Oxidation of Benzylic Alcohols

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1394
Perrey, David A.; Li, Jun-Xu; Zhang, Yanan:
Modified Synthesis of NOP Receptor Antagonist SB612111

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1401
Deb, Mohit L.; Borpatra, Paran J.; J. Saikia, Prakash; Baruah, Pranjal K.:
Base-Promoted Three-Component One-Pot Approach to 3-(α,α-Diarylmethyl)indoles via Arylation of 3-Indolylalcohols

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1410
Chavan, Subhash P.; Khatod, Harshali S.:
Application of Unusual Grignard Reaction for the Stereoselective Synthesis of Antidepressant Drug (R)-(–)-Venlafaxine

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