DOI: 10.1055/s-00000083

Synlett

Issue 01 · Volume 27 · January 2016 DOI: 10.1055/s-005-30663

editorial

  • I

    Editorial

    • synform

  • A1
    Zanda, Matteo:

    SYNFORM ISSUE 2016/01

    • letter

  • 1
    Lewis, Frank W.; Harwood, Laurence M.; Hudson, Michael J.; Núñez, Ana; Galán, Hitos; Espartero, Amparo G.:

    Synthesis and Evaluation of a Novel Hydrophilic 6,6′-Bis(1,2,4-triazin-3-yl)-2,2′-bipyridine Ligand for Separating Actinide(III) from Lanthanide(III)

    Image for article: Synthesis and Evaluation of a Novel Hydrophilic 6,6′-Bis(1,2,4-triazin-3-yl)-2,2′-bipyridine Ligand for Separating Actinide(III) from Lanthanide(III)
    Supporting Information (PDF)
  • 6
    Armstrong, Roly J.; D’Ascenzio, Melissa; Smith, Martin D.:

    Cation-Directed Enantioselective N-Functionalization of Pyrroles

    Image for article: Cation-Directed Enantioselective N-Functionalization of Pyrroles
    Supporting Information (PDF)
  • 11
    Bisterfeld, Carolin; Küberl, Irene; Dick, Markus; Pietruszka, Jörg:

    A Fluorogenic Screening for Enantio- and Diastereoselectivity of 2-Deoxy-d-ribose-5-phosphate Aldolases

    Image for article: A Fluorogenic Screening for Enantio- and Diastereoselectivity of 2-Deoxy-<sc>d</sc>-ribose-5-phosphate Aldolases
    Supporting Information (PDF)
  • 17
    Al-Ani, Widad; Shankland, Kenneth; Cobb, Alexander J. A.:

    Asymmetric Organocatalytic Synthesis of Cyclopentane γ-Nitroketones

    Image for article: Asymmetric Organocatalytic Synthesis of Cyclopentane γ-Nitroketones
  • 21
    Robertson, Gerard P.; Farley, Alistair J. M.; Dixon, Darren J.:

    Bifunctional Iminophosphorane Catalyzed Enantioselective Ketimine Phospha-Mannich Reaction

    Image for article: Bifunctional Iminophosphorane Catalyzed Enantioselective Ketimine Phospha-Mannich Reaction
    Open Access
    Supporting Information (PDF)
  • 25
    Verhoog, Stefan; Pfeifer, Lukas; Khotavivattana, Tanatorn; Calderwood, Samuel; Collier, Thomas Lee; Wheelhouse, Katherine; Tredwell, Matthew; Gouverneur, Véronique:

    Silver-Mediated 18F-Labeling of Aryl-CF3 and Aryl-CHF2 with 18F-Fluoride

    Image for article: Silver-Mediated <sup>18</sup>F-Labeling of Aryl-CF<sub>3</sub> and Aryl-CHF<sub>2</sub> with <sup>18</sup>F-Fluoride
    Supporting Information (PDF)
  • 29
    Kim, Yo-Han; Han, Jusung; Jung, Byeong Yeon; Baek, Heeyoel; Yamada, Yoichi M. A.; Uozumi, Yasuhiro; Lee, Yoon-Sik:

    Production of Valuable Esters from Oleic Acid with a Porous Polymeric Acid Catalyst without Water Removal

    Image for article: Production of Valuable Esters from Oleic Acid with a Porous Polymeric Acid Catalyst without Water Removal
    Supporting Information (PDF)
  • 33
    Rota, Filippo; Benhamou, Laure; Sheppard, Tom D.:

    Asymmetric Synthesis of Secondary Alcohols and 1,2-Disubstituted Epoxides via Organocatalytic Sulfenylation

    Image for article: Asymmetric Synthesis of Secondary Alcohols and 1,2-Disubstituted Epoxides via Organocatalytic Sulfenylation
    Supporting Information (PDF)
  • 37
    Blunt, Christopher E.; Nawrat, Christopher C.; LeBozec, Lucille; Liutkus, Mantas; Liu, Yang; Lewis, William; Moody, Christopher J.:

    Oxidative Routes to the Heterocyclic Cores of Benzothiazole Natural Products

    Image for article: Oxidative Routes to the Heterocyclic Cores of Benzothiazole Natural Products
    Supporting Information (PDF)
  • 41
    Anderson, James C.; Rundell, Christopher D.:

    Stereoselective Synthesis of Densely Substituted Tetrahydroquinolines by a Conjugate Addition Nitro-Mannich Reaction with Carbon Nucleophiles

    Image for article: Stereoselective Synthesis of Densely Substituted Tetrahydroquinolines by a Conjugate Addition Nitro-Mannich Reaction with Carbon Nucleophiles
    Supporting Information (PDF)
  • 45
    Broadley, Kenneth J.; Buffat, Maxime G. P.; Davies, Robin H.; Thomas, Eric J.:

    A Stereoselective Synthesis of a 3,4,5-Substituted Piperidine of Interest as a Selective Muscarinic (M1) Receptor Agonist

    Image for article: A Stereoselective Synthesis of a 3,4,5-Substituted Piperidine of Interest as a Selective Muscarinic (M<sub>1</sub>) Receptor Agonist
    Supporting Information (PDF)
  • 51
    Buckley, Benjamin R.; Figueres, Maria M. P.; Khan, Amna N.; Heaney, Harry:

    A New Simplified Protocol for Copper(I) Alkyne–Azide Cycloaddition Reactions Using Low Substoichiometric Amounts of Copper(II) Precatalysts in Methanol

    Image for article: A New Simplified Protocol for Copper(I) Alkyne–Azide Cycloaddition Reactions Using Low Substoichiometric Amounts of Copper(II) Precatalysts in Methanol
    Supporting Information (PDF)
  • 57
    Seiple, Ian B.; Hog, Daniel T.; Myers, Andrew G.:

    Practical Protocols for the Preparation of Highly Enantioenriched Silyl Ethers of (R)-3-Hydroxypentan-2-one, Building Blocks for the Synthesis of Macrolide Antibiotics

    Image for article: Practical Protocols for the Preparation of Highly Enantioenriched Silyl Ethers of (<i>R</i>)-3-Hydroxypentan-2-one, Building Blocks for the Synthesis of Macrolide Antibiotics
    Supporting Information (PDF)
  • 61
    Muhammad, Rehmani N.; Draffan, Alistair G.; Banwell, Martin G.; Willis, Anthony C.:

    A Second-Generation Chemoenzymatic Total Synthesis of Platencin

    Image for article: A Second-Generation Chemoenzymatic Total Synthesis of Platencin
    Supporting Information (PDF)
  • 67
    Honraedt, Aurélien; Gallagher, Timothy:

    Concise Entries to 4-Halo-2-pyridones and 3-Bromo-4-halo-2-pyridones

    Image for article: Concise Entries to 4-Halo-2-pyridones and 3-Bromo-4-halo-2-pyridones
    Supporting Information (PDF)
  • 70
    Osler, Jonathan D.; Unsworth, William P.; Taylor, Richard J. K.:

    Synthetic Studies towards the Africanane Sesquiterpenes via the Cope Rearrangement of gem-Dimethyl-Substituted Divinyl Cyclopropanes

    Image for article: Synthetic Studies towards the Africanane Sesquiterpenes via the Cope Rearrangement of <i>gem</i>-Dimethyl-Substituted Divinyl Cyclopropanes
    Supporting Information (PDF)
  • 75
    Sonneck, Marcel; Kuhrt, David; Kónya, Krisztina; Patonay, Tamás; Villinger, Alexander; Langer, Peter:

    Regioselective Suzuki–Miyaura Cross-Coupling Reactions of the Bis(triflate) of 1,4-Dihydroxy-9H-fluoren-9-one

    Image for article: Regioselective Suzuki–Miyaura Cross-Coupling Reactions of the Bis(triflate) of 1,4-Dihydroxy-9<i>H</i>-fluoren-9-one
  • 80
    Bulman Page, Philip C.; Buckley, Benjamin R.; Elliott, Claire; Chan, Yohan; Dreyfus, Nicolas; Marken, Frank:

    Chemoselective Oxidation of Sulfides to Sulfoxides with Urea–Hydrogen Peroxide Complex Catalysed by Diselenide

    Image for article: Chemoselective Oxidation of Sulfides to Sulfoxides with Urea–Hydrogen Peroxide Complex Catalysed by Diselenide
    Supporting Information (PDF)
  • 83
    Monteiro, Julia L.; Pieber, Bartholomäus; Corrêa, Arlene G.; Kappe, C. Oliver:

    Continuous Synthesis of Hydantoins: Intensifying the Bucherer–Bergs Reaction

    Image for article: Continuous Synthesis of Hydantoins: Intensifying the Bucherer–Bergs Reaction
    Supporting Information (PDF)
  • 88
    McPherson, Christopher G.; Livingstone, Keith; Jamieson, Craig; Simpson, Iain:

    Palladium-Catalyzed Synthesis of Aryl Amides through Silanoate-Mediated Hydrolysis of Nitriles

    Image for article: Palladium-Catalyzed Synthesis of Aryl Amides through Silanoate-Mediated Hydrolysis of Nitriles
    Supporting Information (PDF)
  • 93
    Bates, Roderick W.; Vilaivan, Tirayut; Apparao, Suryavanshi Padmakar; Ho, Tu Thanh:

    Synthesis of a Tetrahydrofuranyl β-Amino Acid for Peptide Nucleic Acid Construction

    Image for article: Synthesis of a Tetrahydrofuranyl β-Amino Acid for Peptide Nucleic Acid Construction
    Supporting Information (PDF)
  • 96
    Tietze, Lutz F.; Jackenkroll, Stefan; Ganapathy, Dhandapani; Reiner, Johannes R.:

    Formal Synthesis of (–)-Siccanin Using an Enantioselective Domino Wacker/Carbonylation/Methoxylation Reaction

    Image for article: Formal Synthesis of (–)-Siccanin Using an Enantioselective Domino Wacker/Carbonylation/Methoxylation Reaction
    Supporting Information (PDF)
  • 101
    Flegeau, Emmanuel Ferrer; Harrison, Jack M.; Willis, Michael C.:

    One-Pot Sulfonamide Synthesis Exploiting the Palladium-Catalyzed Sulfination of Aryl Iodides

    Image for article: One-Pot Sulfonamide Synthesis Exploiting the Palladium-Catalyzed Sulfination of Aryl Iodides
    Open Access
    Supporting Information (PDF)
  • 106
    Morgan, Kate F.; Doran, Robert; Croft, Rosemary A.; Hollingsworth, Ian A.; Bull, James A.:

    2-Sulfinyl Oxetanes: Synthesis, Stability and Reactivity

    Image for article: 2-Sulfinyl Oxetanes: Synthesis, Stability and Reactivity
    Supporting Information (PDF)
  • 111
    Cross, Paul W. C.; Herbert, John M.; Kerr, William J.; McNeill, Alan H.; Paterson, Laura C.:

    Isotopic Labelling of Functionalised Arenes Catalysed by Iridium(I) Species of the [(cod)Ir(NHC)(py)]PF6 Complex Class

    Image for article: Isotopic Labelling of Functionalised Arenes Catalysed by Iridium(I) Species of the [(cod)Ir(NHC)(py)]PF<sub>6</sub> Complex Class
  • 116
    Williamson, Alice E.; Ngouansavanh, Tifelle; Pace, Robert D. M.; Allen, Anna E.; Cuthbertson, James D.; Gaunt, Matthew J.:

    Rapid Generation of Complex Molecular Architectures by a Catalytic Enantioselective Dearomatization Strategy

    Image for article: Rapid Generation of Complex Molecular Architectures by a Catalytic Enantioselective Dearomatization Strategy
    Supporting Information (PDF)
  • 121
    Gregory, Mark; Catimel, Bruno; Yin, Meng-Xin; Condron, Melanie; Burgess, Antony W.; Holmes, Andrew B.:

    Synthesis of a Tethered myo-Inositol (1,3,4,5,6)Pentakisphosphate (IP5) Derivative as a Probe for Biological Studies

    Image for article: Synthesis of a Tethered <i>myo</i>-Inositol (1,3,4,5,6)Pentakisphosphate (IP5) Derivative as a Probe for Biological Studies
    Supporting Information (PDF)
  • 126
    Bulman Page, Philip C.; Farah, Mohamed M.; Buckley, Benjamin R.; Chan, Yohan; Blacker, A. John:

    Preparation of C2-Symmetric Biaryl Bisiminium Salts and Their Use as Organocatalysts for Asymmetric Epoxidation

    Image for article: Preparation of <i>C</i><sub>2</sub>-Symmetric Biaryl Bisiminium Salts and Their Use as Organocatalysts for Asymmetric Epoxidation
    Supporting Information (PDF)
  • 131
    Cranwell, Philippa B.; Russell, Andrew T.; Smith, Christopher D.:

    Methyl Hydrazinocarboxylate as a Practical Alternative to Hydrazine in the Wolff–Kishner Reaction

    Image for article: Methyl Hydrazinocarboxylate as a Practical Alternative to Hydrazine in the Wolff–Kishner Reaction
    Supporting Information (PDF)
  • 136
    Clemente-Tejeda, David; Zard, Samir Z.:

    O-Ethyl-S-(1,2,2,2-Tetrafluoroethyl)-Dithiocarbonate: A Convenient Reagent for the Generation and Capture of 1,2,2,2-Tetra­fluoroethyl Radicals

    Image for article: <i>O</i>-Ethyl-<i>S</i>-(1,2,2,2-Tetrafluoroethyl)-Dithiocarbonate: A Convenient Reagent for the Generation and Capture of 1,2,2,2-Tetra­fluoroethyl Radicals
    Supporting Information (PDF)
  • 141
    Nixon, Gemma L.; Billington, Helen; Kalindjian, S. Barret; Steiner, Alexander; O’Neil, Ian A.:

    Tripodal Tris-N-oxides: Synthesis and Hydrogen Bonding Capabilities

    Image for article: Tripodal Tris-<i>N</i>-oxides: Synthesis and Hydrogen Bonding Capabilities
    Supporting Information (PDF)
  • 146
    Watson, Emma L.; Ball, Anthony; Raw, Steven A.; Marsden, Stephen P.:

    Synthetic Studies on Psychotrimine: Palladium-Catalysed Arylation of 2-(N-Indolyl) Amides

    Image for article: Synthetic Studies on Psychotrimine: Palladium-Catalysed Arylation of 2-(<i>N</i>-Indolyl) Amides
  • 151
    Armstrong, Alan; Pullin, Robert D. C.; Scutt, James N.:

    Tertiary Amine Promoted Aziridination: Preparation of NH-Aziridines from Aliphatic α,β-Unsaturated Ketones

    Image for article: Tertiary Amine Promoted Aziridination: Preparation of NH-Aziridines from Aliphatic α,β-Unsaturated Ketones
    Supporting Information (PDF)
  • 156
    Kaib, Philip S. J.; List, Benjamin:

    Highly Acidic BINOL-Derived Phosphoramidimidates and their Application in the Brønsted Acid Catalyzed Synthesis of α-Tocopherol

    Image for article: Highly Acidic BINOL-Derived Phosphoramidimidates and their Application in the Brønsted Acid Catalyzed Synthesis of α-Tocopherol
    Supporting Information (PDF)
  • 159
    Baumann, Marcus; Baxendale, Ian R.:

    Continuous-Flow Synthesis of 2H-Azirines and Their Diastereoselective Transformation to Aziridines

    Image for article: Continuous-Flow Synthesis of 2<i>H</i>-Azirines and Their Diastereoselective Transformation to Aziridines
    Supporting Information (PDF)
  • 164
    O’Brien, Matthew; Cooper, Dennis:

    Continuous Flow Liquid–Liquid Separation Using a Computer-Vision Control System: The Bromination of Enaminones with N-Bromosuccinimide

    Image for article: Continuous Flow Liquid–Liquid Separation Using a Computer-Vision Control System: The Bromination of Enaminones with <i>N</i>-Bromosuccinimide
    Supporting Information (PDF)
  • 169
    Beadle, Jonathan D.; Powell, Nicola H.; Raubo, Piotr; Clarkson, Guy J.; Shipman, Michael:

    Synthesis of Oxetane- and Azetidine-Containing Spirocycles Related to the 2,5-Diketopiperazine Framework

    Image for article: Synthesis of Oxetane- and Azetidine-Containing Spirocycles Related to the 2,5-Diketopiperazine Framework
    Supporting Information (PDF)

    • errata

  • e1
    Al-Ani, Widad; Shankland, Kenneth; Cobb, Alexander J. A.:

    Asymmetric Organocatalytic Synthesis of Cyclopentane γ-Nitroketones

  • e2
    Williamson, Alice E.; Ngouansavanh, Tifelle; Pace, Robert D. M.; Allen, Anna E.; Cuthbertson, James D.; Gaunt, Matthew J.:

    Rapid Generation of Complex Molecular Architectures by a Catalytic Enantioselective Dearomatization Strategy