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Editorial

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A22

Zanda, Matteo:

SYNFORM ISSUE 2010/03

Full Text PDF (877 kb)

505

Qian, Zizheng; Baxendale, Ian R.; Ley, Steven V.:

A Flow Process Using Microreactors for the Preparation of a Quinolone Derivative as a Potent 5HT_1B Antagonist

Image for article: A Flow Process Using Microreactors
for the Preparation of a Quinolone Derivative as a Potent
5HT<SUB>1B</SUB> Antagonist

509

Silva, Eduarda M. P.; Pye, Richard J.; Cardin, Christine; Harwood, Laurence M.:

Probing a Biomimetic Approach to Mycaperoxide B: Hydroperoxidation Studies

514

Padwal, Jalindar; Lewis, William; Moody, Christopher J.:

Synthesis of the Reported Structure of Crassiflorone, a Pentacyclic Naphthoquinone Isolated from the African Ebony Diospyros crassiflora

Image for article: Synthesis of the Reported Structure
of Crassiflorone, a Pentacyclic Naphthoquinone Isolated
from the African Ebony <EM EMTYPE="ITALIC">Diospyros crassiflora</EM>

517

Chappell, David; Drew, Michael G. B.; Gibson, Shane; Harwood, Laurence M.; Russell, Andrew T.:

Formal Total Synthesis of (±)-Conduramine E Utilising the Bryce-Smith-Gilbert Photoamination Reaction

521

Keshipeddy, Santosh; Shi, Yu; Hnatiuk, Nathan; Morton, Martha; Yao, Xudong; Howell, Amy R.:

Design and Synthesis of an Activity-Based Probe Template for Protein Kinases

Supporting Information (PDF)

525

Sharma, Pallavi; Moses, John E.:

Photochemical Studies of the Tridachiahydropyrones in Seawater

529

Macleod, Fraser; Lang, Stuart; Murphy, John A.:

The 2-(2-Azidoethyl)cycloalkanone Strategy for Bridged Amides and Medium-Sized Cyclic Amine Derivatives in the Aubé-Schmidt Reaction

Image for article: The 2-(2-Azidoethyl)cycloalkanone
Strategy for Bridged Amides and Medium-Sized Cyclic Amine
Derivatives in the Aubé-Schmidt Reaction

Supporting Information (PDF)

535

Hameed, Abdul; Blake, Alexander J.; Hayes, Christopher J.:

An Enantioselective Formal Synthesis of (+)-Lactacystin from Hydroxymethyl Glutamic Acid (HMG)

539

Crosby, Stuart R.; Sessions, Richard B.; Willis, Christine L.:

Intermediates for the Synthesis of 4-Substituted Proline Derivatives

543

Clarke, Paul A.; Black, Richard J. G.; Iqbal, Mudassar:

Investigation of Transannelation Reactions Across a Cyclononene Ring

547

Goldring, William P. D.; Mann, John; Brockbank, Paul:

A Synthesis of (S)-(-)-Umbelactone and Related α,β-Butenolides

Image for article: A Synthesis of (<EM EMTYPE="ITALIC">S</EM>)-(-)-Umbelactone and Related α,β-Butenolides

Supporting Information (PDF)

551

Black, Richard J. G; Dungan, Victoria J.; Li, Rebecca Y. T.; Young, Philip G.; Jolliffe, Katrina A.:

A Cyclooligomerisation Approach to Backbone-Modified Cyclic Peptides Bearing Guanidinium Arms

Supporting Information (PDF)

555

Chattopadhyay, Shital K.; Singha, Sovan K:

Efficient Construction of the Carbon Skeleton of the Novel Polyoxazole-Based Cyclopeptide IB-01211 via a Biomimetic Macrocyclisation

Image for article: Efficient Construction of the
Carbon Skeleton of the Novel Polyoxazole-Based Cyclopeptide IB-01211
via a Biomimetic Macrocyclisation

559

Stockman, Robert A.; McDermott, Paul J.; Newton, Annabella F.; Magnus, Philip:

A Versatile Chiral Pyrrolidine Aldehyde Building-Block for Synthesis and Formal Synthesis of ent-Nakadomarin A

Image for article: A Versatile Chiral Pyrrolidine
Aldehyde Building-Block for Synthesis and Formal Synthesis of <EM EMTYPE="ITALIC">ent-</EM>Nakadomarin A

563

Wang, Lei; Liu, Junyang; Zhang, Hui; Xu, Zhengshuang; Ye, Tao:

Progress towards the Total Synthesis of Scytonemin A: Asymmetric Synthesis of (2S,3R,4R)-4-hydroxy-3-methylproline

Image for article: Progress towards the Total
Synthesis of Scytonemin A: Asymmetric Synthesis of (2<EM EMTYPE="ITALIC">S</EM>,3<EM EMTYPE="ITALIC">R</EM>,4<EM EMTYPE="ITALIC">R</EM>)-4-hydroxy-3-methylproline

Supporting Information (PDF)

567

Davies, Stephen G.; Hughes, Deri G.; Price, Paul D.; Roberts, Paul M.; Russell, Angela J.; Smith, Andrew D.; Thomson, James E.; Williams, Oliver M. H.:

Asymmetric Synthesis of Piperidines and Octahydroindolizines

571

Paterson, Ian; Rubenbauer, Philipp:

Synthetic Studies towards Iriomoteolide 1a: Stereocontrolled Construction of C1-C9 and C11-C23 Segments Using Lactate Aldol Chemistry

Image for article: Synthetic Studies towards Iriomoteolide
1a: Stereocontrolled Construction of C1-C9 and C11-C23
Segments Using Lactate Aldol Chemistry

575

Basar, Norazah; Donnelly, Sam; Liu, Hao; Thomas, Eric J.:

1,5-Stereocontrol in Bismuth-Mediated Reactions between Aldehydes and Allyl Bromides: Stereoselective Synthesis of Open-Chain all-syn- and anti, anti-1,3,5-Disposed Trimethylalkanes

Image for article: 1,5-Stereocontrol in Bismuth-Mediated
Reactions between Aldehydes and Allyl Bromides: Stereoselective
Synthesis of Open-Chain all-<EM EMTYPE="ITALIC">syn</EM>- and <EM EMTYPE="ITALIC">anti</EM>,<EM EMTYPE="ITALIC"> anti</EM>-1,3,5-Disposed
Trimethylalkanes

579

Killen, Jonathan C.; Leonard, John; Aggarwal, Varinder K.:

A Novel Asymmetric Azaspirocyclisation Using a Morita-Baylis-Hillman-Type Reaction

Supporting Information (PDF)

583

Winzar, Renee; Philips, Jessica; Kiefel, Milton J.:

A Simple Synthesis of C-8 Modified 2-Keto-3-deoxy-d-manno-octulosonic Acid (KDO) Derivatives

Image for article: A Simple Synthesis of C-8 Modified
2-Keto-3-deoxy-<EM EMTYPE="CAPS">d</EM>-<EM EMTYPE="ITALIC">manno</EM>-octulosonic
Acid (KDO) Derivatives

Supporting Information (PDF)

587

Garrido, Narciso M.; Rubia, Alfonso G.; Nieto, Carlos; Díez, David:

Potential of (2E,7E)-Nonadienedioates in Asymmetric Synthesis: Construction of Homopipecolic Acid and an Aminoester Building Block for Peptide Nucleic Acids

Image for article: Potential of (2<EM EMTYPE="ITALIC">E</EM>,7<EM EMTYPE="ITALIC">E</EM>)-Nonadienedioates
in Asymmetric Synthesis: Construction of Homopipecolic Acid and
an Aminoester Building Block for Peptide Nucleic Acids

591

Williams, David R.; Fu, Liangfeng:

Methodology for the Synthesis of Substituted 1,3-Oxazoles

595

Chapman, Helen A.; Herbal, Karim; Motherwell, William B.:

Studies towards the Taming of the ‘Carbocation’ in the Regioselective Ring Opening of Epoxides to Allylic Alcohols

599

Bray, Christopher D.; Olasoji, Joy:

A Total Synthesis of (+)-Bacillamide B

Supporting Information (PDF)

602

Beltrán-Rodil, Sandra; Edwards, Michael G.; Pugh, David. S.; Reid, Mark; Taylor, Richard J. K.:

The Preparation of Substituted Pyrazoles from β,β-Dibromo-enones by a Tandem Condensation/Suzuki-Miyaura Cross-Coupling Process

Image for article: The Preparation of Substituted
Pyrazoles from β,β-Dibromo-enones by a Tandem
Condensation/Suzuki-Miyaura Cross-Coupling Process

607

Roth, Stefanie; Thomas, Neil R.:

A Concise Route to l-Azidoamino Acids: l-Azidoalanine, l-Azidohomoalanine and l-Azidonorvaline

Image for article: A Concise Route to <EM EMTYPE="CAPS">l-</EM>Azidoamino Acids: <EM EMTYPE="CAPS">l-</EM>Azidoalanine, <EM EMTYPE="CAPS">l-</EM>Azidohomoalanine and <EM EMTYPE="CAPS">l-</EM>Azidonorvaline

610

Clark, Andrew J.; Fullaway, David R.; Murphy, Nicholas P.; Parekh, Hemal:

Copper(I) Halide Mediated Tandem 1,4-Aryl Migration-Oxidative Amidyl Radical Cyclisation of Bromosulfonamides

615

Brogan, Samantha; Carter, Neil B.; Lam, Hon Wai:

Copper-Bisphosphine-Initiated Pentafluorophenylation of Aldehydes and Ketones

Supporting Information (PDF)

618

Lygo, Barry; Beaumont, Douglas J.; Cooke, Jason W. B.; Hirst, David J.:

Synthesis of Brombyins II and III, Cyclostachines A and B, and Cyclopiperstachine, Plant-Derived Octahydronaphthalenes

623

North, Michael; Villuendas, Pedro:

Aluminium(salen) and Tetrabutylammonium Bromide Catalysed Synthesis of Cyclic Di- and Trithiocarbonates from Epoxides and Carbon Disulfide

Image for article: Aluminium(salen) and Tetrabutylammonium
Bromide Catalysed Synthesis of Cyclic Di- and Trithiocarbonates
from Epoxides and Carbon Disulfide

628

Knight, David W.; Proctor, Anthony J.; Clough, John M.:

New Regiospecific Catalytic Approaches to 4,5-Dihydroisoxazoles and 2,5-Dihydroisoxazoles from O-Propargylic Hydroxylamines

Image for article: New Regiospecific Catalytic
Approaches to 4,5-Dihydroisoxazoles and 2,5-Dihydroisoxazoles
from <EM EMTYPE="ITALIC">O</EM>-Propargylic Hydroxylamines

633

Denton, Ross M.; Scragg, James T.:

A Concise Synthesis of Dunnianol

636

Tang, Xiaoping; Rawson, Daniel; Woodward, Simon:

Direct Reaction of Aryl Iodides with Activated Aluminium Powder and Reactions of the Derived Aryl Sesquiiodides

639

Simpkins, Nigel S.; Taylor, James D.; Weller, Michael D.; Hayes, Christopher J.:

Synthesis of Nemorosone via a Difficult Bridgehead Substitution Reaction

644

Wipf, Peter; George, Kara M.:

Regioselective Palladium-Catalyzed Cross-Coupling Reactions of 2,4,7-Trichloroquinazoline

Supporting Information (PDF)

649

Kędzia, Jacek L.; Kerr, William J.; McPherson, Allan R.:

Regioselective Pauson-Khand Processes with Olefins Possessing Extended Phosphonates

654

Jones, Raymond C. F.; Choudhury, Abdul K.; Iley, James N.; Loizou, Georgia; Lumley, Christopher; McKee, Vickie:

New Methodologies for the Synthesis of 3-Acylpyridone Metabolites

659

Boto, Alicia; Hernández, Rosendo; Saavedra, Carlos J.:

One-Pot Conversion of α-Amino Acids into β-Amino Aldehydes or 2-Acetoxyazetidines: Application to the Synthesis of Modified Peptides

Image for article: One-Pot Conversion of α-Amino
Acids into β-Amino Aldehydes or 2-Acetoxyazetidines:
Application to the Synthesis of Modified Peptides

664

Sançon, Julien; Sweeney, J. B.:

Probing the Effect of Allylic Substitution on Cyclic Ammonium Ylid Rearrangements

667

Zhang, Kai; Gudipati, Venugopal; Curran, Dennis P.:

Fluorous Mixture Synthesis of Four Stereoisomers of the C21-C40 Fragment of Tetrafibricin

Supporting Information (PDF)

672

Stevenson, Brett; Lewis, William; Dowden, James:

Expedient Route to an Amine Precursor of Halichlorine and Pinnaic Acid from Nitrocyclopent-1-ene

Supporting Information (PDF)

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