DOI: 10.1055/s-00000131

Synfacts

Issue 10 · Volume 2009 · October 2009 DOI: 10.1055/s-002-20426

Synform

A59
Zanda, Matteo: SYNFORM ISSUE 2009/07

Synthesis of Natural Products and Potential Drugs

z1059
All PDFs of this category
1059
Jackson, K. L.; Henderson, J. A.; Motoyoshi, H.; Phillips, A. J.: Synthesis of Norhalichondrin B
1060
Davulcu, A. H.; McLeod, D. D.; Li, J.; Katipally, K.; Littke, A.; Doubleday, W.; Xu, Z.; McConlogue, C. W.; Lai, C. J.; Gleeson, M.; Schwinden, M.; Parsons Jr., R. L.: Synthesis of BMS-317180
1061
Fix-Stenzel, S. R.; Hayes, M. E.; Zhang, X.; Wallace, G. A.; Grongsaard, P.; Schaffter, L. M.; Hannick, S. M.; Franczyk, T. S.; Stoffel, R. H.; Cusack, K. P.: Synthesis of an S1P1 Agonist
1062
Ramharter, J.; Mulzer, J.: Synthesis of Valerenic Acid
1063
Taniguchi, T.; Zaimoku, H.; Ishibashi, H.: Formal Synthesis of Haouamine A
1064
Masuo, R.; Ohmori, K.; Hintermann, L.; Yoshida, S.; Suzuki, K.: Synthesis of FD-594 Aglycon
1065
Nicolaou, K. C.; Lim, Y. H.; Becker, J.: Synthesis of (+)-BE-43472B
1066
Yamada, K.-i.; Yamashita, M.; Sumiyoshi, T.; Nishimura, K.; Tomioka, K.: Total Synthesis of (-)-Lycorine
1067
Frebault, F.; Simpkins, N. S.; Fenwick, A.: Synthesis of ent-Malbrancheamide B
1068
Ko, H. M.; Lee, C. W.; Kwon, H. K.; Chung, H. S.; Choi, S. Y.; Chung, Y. K.; Lee, E.: Synthesis of (-)-Amphidinolide K
1069
Bilke, J. L.; Moore, S. P.; O’Brien, P.; Gilday, J.: Synthesis of (+)-L-733,060
1070
Wu, Y.-C.; Bernadat, G.; Masson, G.; Couturier, C.; Schlama, T.; Zhu, J.: Synthesis of Lemonomycinone Amide
1071
Morimoto, Y.; Okita, T.; Kambara, H.: Synthesis of (+)-Omaezakianol
1072
Kim, H. C.; Kang, S. H.: Synthesis of Azithromycin
1073
Imaoaka, T.; Iwamoto, O.; Noguchi, K.-i.; Nagasawa, K.: Synthesis of (+)-Dibromophakellin

Synthesis of Heterocycles

z1075
All PDFs of this category
1075
Roveda, J.-G.; Clavette, C.; Hunt, A. D.; Gorelsky, S. I.; Whipp, C. J.; Beauchemin, A. M.: Synthesis of Azacarbocycles via Hydroamination and Aminocarbonylation
1076
Mei, T.-S.; Wang, X.; Yu, J.-Q.: Synthesis of Indolines by Pd(II)-Catalyzed Amination of C-H Bond
1077
Henssler, J. T.; Matzger, A. J.: Synthesis of theThieno[3,2-b]thiophene and Thieno[3,2-b]furan Bare Ring Systems
1078
Zhu, W.; Mena, M.; Jnoff, E.; Sun, N.; Pasau, P.; Ghosez, L.: Synthesis of Piperidones by MCR
1079
Shintani, R.; Hayashi, S.-y.; Murakami, M.; Takeda, M.; Hayashi, T.: Stereoselective Synthesis of Spirooxindoles
1080
Yavari, I.; Souri, S.; Sirouspour, M.; Bayat, M. J.: Synthesis of Fused Quinoxalines and Benzoxazines
1081
Anary-Abbasinejad, M.; Poorhassan, E.; Hassanabadi, A.: Synthesis of 2,5-Dihydropyrroles from Acetylene Esters and α-Arylamino Ketones
1082
Reddy, G.; Kumar, P. A.; Anand, R. V.; Mukkanti, K.; Reddy, P. P.: Synthesis of Indolo [1,2,5]-Triazepines and [1,2,5]-Oxadiazines
1083
Chen, Z.; Ding, Q.; Yu, X.; Wu, J.: Cyclization/[3+2]-Cycloaddition Reaction of N′-(2-Alkynylbenzylidene) Hydrazides
1084
Watanabe, T.; Oishi, S.; Fujii, N.; Ohno, H.: Palladium-Catalyzed Direct One-Pot Synthesis of Carbazoles
1085
McQuaid, K. M.; Long, J. Z.; Sames, D.: Synthesis of Dihydrobenzopyrans via Hydride Transfer Cyclization
1086
Khlebnikov, V.; Patel, K.; Zhou, X.; Reddy, M. M.; Su, Z.; Chiacchia, F. S.; Hansen, H. C.: Efficient Synthesis of 2-Aryl-4H-pyrano[2,3-b]pyridine-4-ones
1087
Han, Z.-Y.; Xiao, H.; Chen, X.-H.; Gong, L.-Z.: Synthesis of Chiral Tetrahydroquinolines by Relay Catalysis
1088
Zhong, W.; Guo, B.; Lin, F.; Liu, Y.; Su, W.: Synthesis of Thiazolopyrimidinones under Solvent-Free Conditions
1089
Li, J.; Wang, D.; Zhang, Y.; Chen, B.: Synthesis of N-Unsubstituted 1,2,3-Triazoles by a One-Pot Reaction

Synthesis of Materials and Unnatural Products

z1091
All PDFs of this category
1091
Tanaka, M.; Rastogi, A.; Toepperwein, G. N.; Riggleman, R. A.; Felix, N. M.; de Pablo, J. J.; Ober, C. K.: Green Lithography
1092
Suzuki, S.; Takeda, T.; Kuratsu, M.; Kozaki, M.; Sato, K.; Shiomi, D.; Takui, T.; Okada, K.: Bis(Radical Cation) Pyrene Building Blocks
1093
Wakamiya, A.; Mori, K.; Araki, T.; Yamaguchi, S.: A New 14π-Electron Aromatic System
1094
Nishiuchi, T.; Kuwatani, Y.; Nishinaga, T.; Iyoda, M.: Thermochromism in Molecular Tweezers
1095
Wei, J.; Jia, X.; Yu, J.; Shi, X.; Zhang, C.; Chen, Z.: Trisannulation to a Thio-Bridged Triphenylene
1096
Zhang, H.; Karasawa, T.; Yamada, H.; Wakamiya, A.; Yamaguchi, S.: Synthesis of Conjugated Ladder Systems by a Reductive Double Cyclization
1097
Kim, S. M.; Park, J. H.; Kang, Y. K.; Chung, Y. K.: Gold-Catalyzed Formation of Functionalized Carbocyclic Cages
1098
Kálai, T.; Jekõ, J.; Hideg, K.: Electrocyclization Route to Isoindoline Nitroxides
1099
Peterson, J. J.; Simon, Y. C.; Coughlin, E. B.; Carter, K. R.: Blue-Emitting p-Carborane Linked Polyfluorene
1100
Yang, S. K.; Ambade, A. V.; Weck, M.: Polymers from Living ROMP and Metal Coordination
1101
Chebny, V. J.; Navale, T. S.; Shukla, R.; Lindeman, S. V.; Rathore, R.: Benzenoid Rings in Triptycene are Communicated
1102
Yamaguchi, I.; Mizoguchi, N.; Sato, M.: An Electron-Accepting Polyphenylene
1103
Mochida, K.; Shimizu, M.; Hiyama, T.: Intramolecular Coupling and Reorganization
1104
Zhai, L.; Shukla, R.; Rathore, R.: An Efficient Method for Oxidative C-C Bond Formation
1105
Postma, A.; Yan, Y.; Wang, Y.; Zelikin, A. N.; Tjipto, E.; Caruso, F.: Poly(dopamine) Shells

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1107
All PDFs of this category
1107
Hou, G.; Gosselin, F.; Li, W.; McWilliams, J. C.; Sun, Y.; Weisel, M.; O’Shea, P. D.; Chen, C.-y.; Davies, I. W.; Zhang, X.: Enantioselective Hydrogenation of N-H Imines
1108
Zhao, Y.-J.; Tan, L.-J. S.; Li, B.; Li, S.-M.; Loh, T.-P.: Indium Bromide Catalyzed Aziridinyl Polyene Cyclization
1109
Evans, P. A.; Clizbe, E. A.: Rhodium-Catalyzed Stereospecific Construction of Allylic Amines
1110
Ohmura, T.; Taniguchi, H.; Suginome, M.: Pd-Catalyzed Kinetic Resolution of 1-Alkyl-2-methylenecyclopropanes
1111
Yin, L.; Kanai, M.; Shibasaki, M.: Cu-Catalyzed Decarboxylative Asymmetric Mannich-Type Reaction
1112
Shen, W.-Y.; Li, Y.-Y.; Dong, Z.-R.; Gao, J.-X.: Ru-Catalyzed Asymmetric Transfer Hydrogenation of Heteroaromatic Ketones
1113
Weix, D. J.; Marković, D.; Ueda, M.; Hartwig, J. F.: Iridium-Catalyzed Allylation of Carbamates
1114
Chen, C.-G.; Hou, X.-L.; Pu, L.: Copper-Catalyzed Asymmetric Alkylation of Glycine Derivatives
1115
Mukhopadhyay, C.; Datta, A.; Butcher, R. J.: syn-Selective, Three-Component Mannich Reaction in Aqueous Media
1116
Taylor, A. M.; Altman, R. A.; Buchwald, S. L.: Pd-Catalyzed Asymmetric α-Arylation and α-Vinylation of Oxindoles
1117
Liu, W.; Chen, D.; Zhu, X.-Z.; Wan, X.-L.; Hou, X.-L.: Palladium-Catalyzed Asymmetric Cyclopropanation
1118
Vrieze, D. C.; Hoge, G. S.; Hoerter, P. Z.; Van Haitsma, J. T.; Samas, B. M.: Enantioselective Allylic Amination and Kinetic Resolution of Allylic Carbonates
1119
Yang, L.; Wang, D.-X.; Huang, Z.-T.; Wang, M.-X.: Cr-Catalyzed Intramolecular Addition of Tertiary Enamides to Ketones
1120
Van Nguyen, H.; Matsubara, R.; Kobayashi, S.: Aza-enolate Addition to Imines Catalyzed by Alkaline Earth Metals
1121
Itoh, J.; Han, S. B.; Krische, M. J.: Enantioselective Additions to Isatins under Transfer Hydrogenation Conditions
1122
Schindler, C. S.; Diethelm, S.; Carreira, E. M.: Unprecedented Reactivity in Nucleophilic Ring Opening of Oxabicycles
1123
Matsumoto, K.; Kubo, T.; Katsuki, T.: Enantioselective Epoxidation of cis-Alkenyl-silanes
1124
Selvakumar, S.; Sivasankaran, D.; Singh, V. K.: Asymmetric Henry Reaction Catalyzed by Diamine-Copper(II) Complex
1125
Sun, B.-F.; Hong, R.; Kang, Y.-B.; Deng, L.: Asymmetric Nucleophilic Epoxidation of Acyclic Trisubstituted Olefins
1126
Demizu, Y.; Moriyama, A.; Onomura, O.: Copper-Catalyzed Kinetic Resolution of rac-α-Hydroxyphosphonates
1127
Wilsily, A.; Lou, T.; Fillion, E.: Copper-Catalyzed Conjugate Addition of Dimethylzinc to Meldrum’s Acids
1128
Nicolaou, K. C.; Li, A.; Ellery, S. P.; Edmonds, D. J.: Rhodium-Catalyzed Asymmetric Enyne Cycloisomerization
1129
Davies, I. R.; Cheeseman, M.; Green, R.; Mahon, M. F.; Merritt, A.; Bull, S. D.: Highly Efficient Synthesis of Trisubstituted γ-Butyrolactones
1130
Rupnicki, L.; Saxena, A.; Lam, H. W.: Cu-Catalyzed Asymmetric Conjugate Reductions of 2-Alkenylheteroarenes
1131
Lassauque, N.; Franciò, G.; Leitner, W.: Lewis Acid Activated Ni-Catalyzed Asymmetric Hydrovinylation
1132
Kang, S. H.; Kang, Y. K.; Kim, D. Y.: Palladium-Catalyzed Conjugate Addition to Give Aspartic Acid Derivatives
1133
Zoute, L.; Kociok-Köhn, G.; Frost, C. G.: Asymmetric Synthesis of Functionalized Pyrrolizidinones
1134
Dutheuil, G.; Webster, M. P.; Worthington, P. A.; Aggarwal, V. K.: An Iterative Approach to the Total Synthesis of (+)-Faranal
1135
Han, Z.; Wang, Z.; Zhang, X.; Ding, K.: Iridium/SpinPHOX Complex Catalyzed Hydrogenation of Ketimines

Metal-Mediated Synthesis

z1137
All PDFs of this category
1137
Yoshikai, N.; Matsuda, H.; Nakamura, E.: New Hydroxyphosphine Ligands for Highly Efficient Kumada Coupling
1138
Shi, F.; Tse, M. K.; Cui, X.; Gördes, D.; Michalik, D.; Thurow, K.; Deng, Y.; Beller, M.: Alkylation of Sulfonamides with Alcohols
1139
Vechorkin, O.; Proust, V.; Hu, X.: Functional Group Tolerant Kumada-Corriu-Tamao Coupling
1140
Su, Y.; Jiao, N.: Selective Ligand-Free Palladium-Catalyzed Oxidative Heck Coupling
1141
Wommack, A. J.; Moebius, D. C.; Travis, A. L.; Kingsbury, J. S.: Sc(OTf)3-Catalyzed Carbon Insertion into Formyl C-H Bond of Aldehydes
1142
Larsson, P.-F.; Correa, A.; Carril, M.; Norrby, P.-O.; Bolm, C.: Ullmann-Type Couplings Using Part-Per-Million Catalyst Loadings
1143
Yao, B.; Liang, Z.; Niu, T.; Zhang, Y.: Synthesis of Ynamides via Iron-Catalyzed Amidation of Alkynyl Bromides
1144
Niu, J.; Guo, P.; Kang, J.; Li, Z.; Xu, J.; Hu, S.: Copper(I)-Catalyzed Efficient Arylation of Alcohols with Aryl Bromides
1145
Arshad, N.; Hashim, J.; Kappe, C. O.: Pd(0)/Cu(I)-Mediated Cross-Coupling of Cyclic Thioamides and Thioureas
1146
Kuninobu, Y.; Matsuki, T.; Takai, K.: Rhenium-Catalyzed Regioselective Alkylation of Phenols
1147
Wasa, M.; Engle, K. M.; Yu, J.-Q.: Pd(0)-Catalyzed Intermolecular Arylation of sp³ C-H Bonds
1148
Stephenson, N. A.; Zhu, J.; Gellman, S. H.; Stahl, S. S.: Zr(NMe2)4-Catalyzed Transamidation and Amide Metathesis Reactions
1149
Balamurugan, R.; Gudla, V.: Naphthalenes via Gold(III)-Catalyzed Addition of Aryl Alkynes to Ketones
1150
Neisius, N. M.; Plietker, B.: Atom-Economic Synthesis of 1,3-Dienes via Hydrovinylation of Internal Alkynes
1151
Weiner, B.; Baeza, A.; Jerphagnon, T.; Feringa, B. L.: Wacker Oxidation of Allylic Phthalimides: A Catalytic Route to β-Amino Acids

Organo- and Biocatalysis

z1153
All PDFs of this category
1153
Nagib, D. A.; Scott, M. E.; MacMillan, D. W. C.: Photoredox Organocatalysis: Asymmetric α-Perfluoroalkylation of Aldehydes
1154
Zhang, F.-L.; Xu, A.-W.; Gong, Y.-F.; Wei, M.-H.; Yang, X.-L.: Four-Component Cascade Reaction
1155
Dickmeiss, G.; De Sio, V.; Udmark, J.; Poulsen, T. B.; Marcos, V.; Jørgensen, K. A.: Desymmetrization of meso-Cyclopentanones
1156
Peterson, E. A.; Jacobsen, E. N.: Intermolecular Addition of Indoles to Cyclic N-Acyliminium Ions
1157
Li, L.; Ganesh, M.; Seidel, D.: Enantioselective Synthesis of syn-α,β-Diamino Acid Derivatives
1158
Weseliñski, Ł.; Stępniak, P.; Jurczak, J.: A New Family of Catalysts for 1,3-Dipolar Cycloadditions
1159
DiRocco, D. A.; Oberg, K. M.; Dalton, D. M.; Rovis, T.: Fluorine-Substitution Effect in Intermolecular Stetter Reactions
1160
Wadhwa, K.; Chintareddy, V. R.; Verkade, J. G.: Organocatalytic Substrate-Controlled Aldehyde Alkynylations
1161
Muratore, M. E.; Holloway, C. A.; Pilling, A. W.; Storer, R. I.; Trevitt, G.; Dixon, D. J.: Enantioselective N-Acyliminium Cyclization Cascade
1162
Sheng, Y.-F.; Gu, Q.; Zhang, A.-J.; You, S.-L.: Enantioselective Friedel-Crafts Alkylation Using Chiral Phosphoric Acid
1163
Wilson, J. E.; Casarez, A. D.; MacMillan, D. W. C.: Enantioselective α-Nitroalkylation of Aldehydes Using SOMO Catalysis
1164
Lu, H.-H.; Zhang, F.-G.; Meng, X.-G.; Duan, S.-W.; Xiao, W.-J.: Enantioselective Michael Addition Using a Cinchona Alkaloid Derived Catalyst
1165
Bencivenni, G.; Wu, L.-Y.; Mazzanti, A.; Giannichi, B.; Pesciaioli, F.; Song, M.-P.; Bartoli, G.; Melchiorre, P.: Construction of Spirocyclic Oxindoles by Aminocatalysis Cascades

Polymer-Supported Synthesis

z1167
All PDF of this category
1167
Mitsudome, T.; Mikami, Y.; Mori, H.; Arita, S.; Mizugaki, T.; Jitsukawa, K.; Kaneda, K.: Hydration of Nitriles to Amides with Supported Silver Nanoparticles
1168
Falini, G.; Gualandi, A.; Savoia, D.: Rhodium/Graphite for the Hydrogenation of Aromatic Compounds
1169
Wang, Y.; Sauer, D. R.; Djuric, S. W.: Synthesis of Guanidines with a Brominated Polymer
1170
Ibarguren, O.; Zakri, C.; Fouquet, E.; Felpin, F.-X.: In situ Generated Pd/C Catalyst for the Synthesis of Oxindoles via HRC
1171
Huang, X.; Cao, J.; Huang, J.: Solid-Phase Synthesis of Benzofused Tricycles
1172
Ito, S.; Yamaguchi, H.; Kubota, Y.; Asami, M.: Mukaiyama Aldol Reaction with Al-MCM-41
1173
Elias, S.; Vigalok, A.: Polypeptide-Based Pd Complex as Micellar Catalyst in Water
1174
Miura, H.; Wada, K.; Hosokawa, S.; Sai, M.; Kondo, T.; Inoue, M.: Cascade Transfer-Allylation and Isomerization with Ru/CeO2
1175
Jana, S.; Haldar, S.; Koner, S.: Suzuki-Miyaura and Stille Coupling Reactions with Pd(0)-MCM-41 Catalyst
1176
De Marco, R.; Di Gioia, M. L.; Leggio, A.; Liguori, A.; Viscomi, M. C.: Deprotection of the N-Nosyl Group with a Thiol Resin
1177
Chen, X.; Wang, L.; Liu, J.: Kumada-Tamao Coupling by Using an Immobilized Nickel Catalyst
1178
Kantam, M. L.; Yadav, J.; Laha, S.; Jha, S.: Synthesis of Propargylamines with Copper Ferrite Nanoparticles
1179
Yamada, Y. M. A.; Arakawa, T.; Hocke, H.; Uozumi, Y.: Aerobic Oxidation of Variety Alcohols in Water with ARP-Pt

Addenda and Errata

1180
Ir(I)-Catalyzed sp³ C-H Bond Alkenylation of Amides with Alkynes