DOI: 10.1055/s-00000084

Synthesis

Issue 02 · Volume 54 · January 2022 DOI: 10.1055/s-012-52652

table of contents

  • V

    Linked PDF of Table of Contents

    • review

  • 217
    Larionova, Natalia A.; Shestopalov, Anatoliy M.; Rodinovskaya, Lyudmila A.; Zubarev, Andrey A.:

    Synthesis of Biologically Active Heterocycles via a Domino Sequence Involving an SN2/Thorpe–Ziegler Reaction Step

    Image for article: Synthesis of Biologically Active Heterocycles via a Domino Sequence Involving an S<sub>N</sub>2/Thorpe–Ziegler Reaction Step

    • short review

  • 246
    Wei, Baosheng; Knochel, Paul:

    Recent Advances in Cross-Couplings of Functionalized Organozinc Reagents

    Image for article: Recent Advances in Cross-Couplings of Functionalized Organozinc Reagents
  • 255
    Oroz, Paula; Avenoza, Alberto; Busto, Jesús H.; Corzana, Francisco; Zurbano, María M.; Peregrina, Jesús M.:

    Strategies for the Synthesis of Selenocysteine Derivatives

    Image for article: Strategies for the Synthesis of Selenocysteine Derivatives
  • 271
    Glueck, David S.:

    Asymmetric Synthesis of P-Stereogenic Secondary Phosphine ­Oxides (SPOs)

    Image for article: Asymmetric Synthesis of P-Stereogenic Secondary Phosphine ­Oxides (SPOs)
  • 281
    Zhang, Yong; Sun, Wenxuan; Li, Chao:

    Nickel-Catalyzed Paired Electrochemical Cross-Coupling of Aryl Halides with Nucleophiles

    Image for article: Nickel-Catalyzed Paired Electrochemical Cross-Coupling of Aryl Halides with Nucleophiles
  • 295
    Fokin, Igor; Kuessner, Kai-Thorben; Siewert, Inke:

    Transition Metal Complex Catalyzed Photo- and Electrochemical (De)hydrogenations Involving C=O and C=N Bonds

    Image for article: Transition Metal Complex Catalyzed Photo- and Electrochemical (De)hydrogenations Involving C=O and C=N Bonds
    Supporting Information (PDF)
  • 315
    Feng, Yanping; Ye, Xiajuan; Huang, Dayun; Guo, Sheng-rong:

    α-Csp3–H Bond Functionalization of Simple Ethers in Radical Reactions

    Image for article: α-Csp<sup>3</sup>–H Bond Functionalization of Simple Ethers in Radical Reactions

    • feature

  • 334
    Beckers, Igor; O’Rourke, Galahad; De Vos, Dirk:

    Late-Stage C–H Arylation of Azepinoindole via Pd/Cu Catalysis: A Step Efficient and Convergent Synthesis of Rucaparib

    Image for article: Late-Stage C–H Arylation of Azepinoindole via Pd/Cu Catalysis: A Step Efficient and Convergent Synthesis of Rucaparib
  • 341
    Chand-Thakuri, Pratibha; Alahakoon, Indunil; Liu, Daniel; Kapoor, Mohit; Kennedy, John F.; Jenkins, Kenneth W.; Rabon, Allison M.; Young, Michael C.:

    Native Amine-Directed ortho-C–H Halogenation and Acetoxylation /Condensation of Benzylamines

    Image for article: Native Amine-Directed <i>ortho</i>-C–H Halogenation and Acetoxylation /Condensation of Benzylamines
    Supporting Information (PDF)
  • 355
    El-Tunsi, Ashraf; Carter, Nicholas; Yeo, Song-Hee; Priest, Joshua D.; Choi, Anthony; Kobras, Carolin M.; Ndlovu, Soneni; Proietti Silvestri, Ilaria; Fenton, Andrew K.; Coldham, Iain:

    Kinetic Resolution by Lithiation: Highly Enantioselective Synthesis of Substituted Dihydrobenzoxazines and Tetrahydroquinoxalines

    Image for article: Kinetic Resolution by Lithiation: Highly Enantioselective Synthesis of Substituted Dihydrobenzoxazines and Tetrahydroquinoxalines
    Supporting Information (PDF)
  • 369
    Tatevosyan, Stepan S.; Kotovshchikov, Yury N.; Latyshev, Gennadij V.; Lukashev, Nikolay V.; Beletskaya, Irina P.:

    Facile Access to Triazole-Fused 3,1-Benzoxazines Enabled by Metal-Free Base-Promoted Intramolecular C–O Coupling

    Image for article: Facile Access to Triazole-Fused 3,1-Benzoxazines Enabled by Metal-Free Base-Promoted Intramolecular C–O Coupling
    Supporting Information (PDF)

    • psp

  • 378
    Janicki, Ignacy; Kiełbasiński, Piotr:

    A Straightforward, Purification-Free Procedure for the Synthesis of Ando and Still–Gennari Type Phosphonates

    Image for article: A Straightforward, Purification-Free Procedure for the Synthesis of Ando and Still–Gennari Type Phosphonates
    Supporting Information (PDF)

    • paper

  • 383
    Islam, Md. Rafikul; Nishinaga, Tohru; Hirabayashi, Kazunori; Shimizu, Toshio; Sugiura, Ken-ichi:

    Oxidative Intramolecular C–C Bond Formation Reactions of 1,2-Diarylbenzenes: Syntheses of Highly Conjugated Double-Bridged Polycyclic Aromatic Hydrocarbons

    Image for article: Oxidative Intramolecular C–C Bond Formation Reactions of 1,2-Diarylbenzenes: Syntheses of Highly Conjugated Double-Bridged Polycyclic Aromatic Hydrocarbons
    Supporting Information (PDF)
  • 393
    Ghora, Santanu; Sreenivasulu, Chinnabattigalla; Satyanarayana, Gedu:

    A Domino Heck Coupling–Cyclization–Dehydrogenative Strategy for the One-Pot Synthesis of Quinolines

    Image for article: A Domino Heck Coupling–Cyclization–Dehydrogenative Strategy for the One-Pot Synthesis of Quinolines
    Supporting Information (PDF)
  • 403
    Wu, Weilong; Jing, Yongkang; Zhang, Deyi; Yan, Xianghe; Liang, Rong; Lu, Zhiqiang; Ji, Baoming:

    Palladium-Catalyzed Butoxycarbonylation of Polybromo(hetero)arenes: A Practical Method for the Preparation of (Hetero)arenepolycarboxylates and -carboxylic Acids

    Image for article: Palladium-Catalyzed Butoxycarbonylation of Polybromo(hetero)arenes: A Practical Method for the Preparation of (Hetero)arenepolycarboxylates and -carboxylic Acids
    Supporting Information (PDF)
  • 411
    Zhang, Dongke; Zhang, Jingran; Li, Xiaoxian; Yu, Zhenyang; Li, Yadong; Sun, Fengxia; Du, Yunfei:

    Intramolecular Chalcogenylation of Isooxazolines Mediated by PhICl2 and Diorganyl Disulfides or Diselenides

    Image for article: Intramolecular Chalcogenylation of Isooxazolines Mediated by PhICl<sub>2</sub> and Diorganyl Disulfides or Diselenides
    Supporting Information (PDF)
  • 421
    Zhou, Likai; Jia, Kuiyong; Liu, Xigong; Liu, Lei:

    Enantioselective Transfer Hydrogenation of Oxocarbenium Ions Enables Asymmetric Access to α-Substituted 1,3-Dihydroisobenzofurans

    Image for article: Enantioselective Transfer Hydrogenation of Oxocarbenium Ions Enables Asymmetric Access to α-Substituted 1,3-Dihydroisobenzofurans
    Supporting Information (PDF)
  • 429
    Zhou, Wei; Yao, Lan; Liu, Yongxiurong; Shen, Lichun; Chen, Jie; Deng, Hongmei; Shao, Min; Zhang, Hui; Tang, Xiaojun; Cao, Weiguo:

    A Catalyst-Free Synthesis of Fused Perfluoroalkylated 2,3-Dihydroisoxazoles via Oxa-Michael-Aldol Annulation

    Image for article: A Catalyst-Free Synthesis of Fused Perfluoroalkylated 2,3-Dihydroisoxazoles via Oxa-Michael-Aldol Annulation
    Supporting Information (PDF)
  • 439
    Mittersteiner, Mateus; Aquino, Estefania C.; Budragchaa, Tuvshinjargal; Wessjohann, Ludger A.; Bonacorso, Helio G.; Martins, Marcos A. P.; Zanatta, Nilo:

    Synthesis of Methylene-Bridged Trifluoromethyl Azoles Using 5-(1,2,3-Triazol-1-yl)enones

    Image for article: Synthesis of Methylene-Bridged Trifluoromethyl Azoles Using 5-(1,2,3-Triazol-1-yl)enones
    Supporting Information (PDF)
  • 451
    Brahmachari, Goutam; Mandal, Mullicka; Karmakar, Indrajit:

    Facile and Straightforward Synthesis of Racemic Version of Substituted 3-[3-(2-Hydroxyphenyl)-3-oxo-1-arylpropyl]-4-hydroxycoumarins: Easy Access to a Series of Biorelevant Warfarin Analogues

    Image for article: Facile and Straightforward Synthesis of Racemic Version of Substituted 3-[3-(2-Hydroxyphenyl)-3-oxo-1-arylpropyl]-4-hydroxycoumarins: Easy Access to a Series of Biorelevant Warfarin Analogues
    Supporting Information (PDF)
  • 465
    Heinemann, Maximilian J. B.; Voigt, Thomas; Menche, Dirk:

    Dihydroxylation Studies of Isoquinolinones: Synthesis of the EF-Ring of Lysolipin I

    Image for article: Dihydroxylation Studies of Isoquinolinones: Synthesis of the EF-Ring of Lysolipin I
    Supporting Information (PDF)
  • 475
    Xia, Xu-Ling; Zhu, Qi-Long; Chen, Jin-Quan; Shi, Zhen; Dong, Zhi-Bing:

    Synthesis of Aryl Dithiocarbamates from Tetramethylthiuram Monosulfide (TMTM) and Aryl Boronic Acids: Copper-Catalyzed Construction of C(sp2)–S Bonds

    Image for article: Synthesis of Aryl Dithiocarbamates from Tetramethylthiuram Monosulfide (TMTM) and Aryl Boronic Acids: Copper-Catalyzed Construction of C(sp<sup>2</sup>)–S Bonds
    Supporting Information (PDF)
  • 483
    Fuchiya, Asuka; Miyamura, Takuya; Nariki, Haruna; Noda, Shizuki; Makiyama, Kouhei; Sonoda, Motohiro; Tanimori, Shinji:

    A Facile Synthesis of 2-Aminobenzoxazines Based on Iodine­Catalyzed Desulfurative Cyclization

    Image for article: A Facile Synthesis of 2-Aminobenzoxazines Based on Iodine­Catalyzed Desulfurative Cyclization
    Supporting Information (PDF)
  • 490
    He, Jing; Wei, Yueting; Li, Xuezhen; Dai, Bin; Liu, Ping:

    Tetrabutylammonium Iodide Mediated Sulfenylation of Poly­substituted 1H-Pyrazol-5-amines with Arylsulfonyl Hydrazides

    Image for article: Tetrabutylammonium Iodide Mediated Sulfenylation of Poly­substituted 1<i>H</i>-Pyrazol-5-amines with Arylsulfonyl Hydrazides
    Supporting Information (PDF)
  • 499
    Ma, Yan-Hua; Meng, Fan-Xiao; Wang, Ruo-Nan; Fan, Ya-Xin; Su, Qing-Qiang; Du, Ji-Yuan:

    Diastereoselective Palladium-Catalyzed [4+1] Cycloadditions of 4-Vinyl-1,4-dihydro-2H-3,1-benzoxazin-2-ones with In Situ Formed Carbenes

    Image for article: Diastereoselective Palladium-Catalyzed [4+1] Cycloadditions of 4-Vinyl-1,4-dihydro-2<i>H</i>-3,1-benzoxazin-2-ones with In Situ Formed Carbenes
    Supporting Information (PDF)
  • 506
    Krylov, Igor B.; Paveliev, Stanislav A.; Budnikov, Alexander S.; Segida, Oleg O.; Merkulova, Valentina M.; Vil’, Vera A.; Nikishin, Gennady I.; Terent’ev, Alexander O.:

    Hidden Reactivity of Barbituric and Meldrum’s Acids: Atom-Efficient Free-Radical C–O Coupling with N-Hydroxy Compounds

    Image for article: Hidden Reactivity of Barbituric and Meldrum’s Acids: Atom-Efficient Free-Radical C–O Coupling with <i>N</i>-Hydroxy Compounds
    Supporting Information (PDF)