DOI: 10.1055/s-00000084

Synthesis

Issue 15 · Volume 57 · August 2025 DOI: 10.1055/s-015-62001

table of contents

  • V

    Linked PDF of Table of Contents

    • review

  • 2261
    Álvarez-Calero, José María; Horwitz, Matthew A.:

    Stereoselectivity Seems To Be the Hardest Word: Tracking the Evolution of Asymmetric API Syntheses from Medicinal Chemistry to Process Development

    Image for article: Stereoselectivity Seems To Be the Hardest Word: Tracking the Evolution of Asymmetric API Syntheses from Medicinal Chemistry to Process Development

    • short review

  • 2278
    Aida, Kazuhiro; Ota, Eisuke; Yamaguchi, Junichiro:

    Recent Advances in Single Electron Reduction Induced Ring Opening of N-Acyl Cyclic Amines

    Image for article: Recent Advances in Single Electron Reduction Induced Ring Opening of <i>N</i>-Acyl Cyclic Amines
  • 2289
    Ni, Qian; Chen, Yaqi; Ma, Yuanhong:

    Recent Progress in Base-Metal-Catalyzed Dearomative Reaction of N-Heteroarenes

    Image for article: Recent Progress in Base-Metal-Catalyzed Dearomative Reaction of <i>N</i>-Heteroarenes

    • feature

  • 2307
    Li, Zihan; Li, Yichao; Zhang, Ruihao; Wang, Yuhao; Wang, Yilong; Yi, Ziqi; Huang, Yiyong:

    Chiral Phosphoric Acid Catalyzed Cascade Asymmetric Allylboration/Oxa-Cyclization of Aldehydes for Access to Multisubstituted Tetrahydrofurans

    Image for article: Chiral Phosphoric Acid Catalyzed Cascade Asymmetric Allylboration/Oxa-Cyclization of Aldehydes for Access to Multisubstituted Tetrahydrofurans
    Supporting Information (PDF)

    • paper

    Bürgenstock Special Section 2023 – Future Stars in Organic Chemistry

  • 2320
    Gupta, Neha; Deng, Hao; Ding, Huanyu; Qiu, Zihang; Neumann, Constanze N.:

    Rh(II)-Catalyzed Synthesis of 1,3-Diols via 5-endo-trig Cyclization of Silyl Radicals

    Image for article: Rh(II)-Catalyzed Synthesis of 1,3-Diols via 5-<i>endo</i>-<i>trig</i> Cyclization of Silyl Radicals
    Open Access
    Supporting Information (PDF)
  • 2331
    Chen, Heng; Gurung, Sing R.; Li, Ling; Mancheno, Danny E.; Radtke, M. Alex; Ma, Zhou; Zhang, Zhi; Yang, Wuxing; Sun, Liang; Xie, Shiping:

    Development of an Efficient Synthesis toward a 4,4-Difluoropiperidine Intermediate Bearing a Pyridine N-Oxide Motif at the Carbon Stereocenter

    Image for article: Development of an Efficient Synthesis toward a 4,4-Difluoropiperidine Intermediate Bearing a Pyridine <i>N</i>-Oxide Motif at the Carbon Stereocenter
    Supporting Information (PDF)
  • 2337
    Zhang, Xiao-Yan; An, Yang; Liu, Zhou-Zhou; Fan, Ling-Tao:

    Claisen-Type Condensation of Ketones with Carboxylic Acids: Synthesis of α,α-Disubstituted β-Keto Carbonyl Compounds

    Image for article: Claisen-Type Condensation of Ketones with Carboxylic Acids: Synthesis of α,α-Disubstituted β-Keto Carbonyl Compounds
    Supporting Information (PDF) CIF File (OTHER)
  • 2345
    Sommer, Ava G.; Tung, Pinku; Mankad, Neal P.:

    Alkylation of Arylsulfonyl Cyanides To Form Alkyl Sulfones

    Image for article: Alkylation of Arylsulfonyl Cyanides To Form Alkyl Sulfones
    Supporting Information (PDF)
  • 2351
    Barabash, Oksana V.; Ostapiuk, Mary Y.; Kravets, Mykola; Obushak, Mykola D.; Schmidt, Andreas; Ostapiuk, Yurii V.:

    Pyrazol-3-yldiazonium Salts as Key Reagents for C–C Bond Formation and Pyrazole-Containing Heterocycle Synthesis

    Image for article: Pyrazol-3-yldiazonium Salts as Key Reagents for C–C Bond Formation and Pyrazole-Containing Heterocycle Synthesis
    Supporting Information (PDF)
  • 2363
    Chaise, Samantha; Gacogne, Audrey; Garcin, Ilan; de Figueiredo, Renata Marcia; Campagne, Jean-Marc; Legrand, Baptiste; Maillard, Ludovic T.:

    Expanding the Scope of Azole-Based γ-Amino Acids – Synthesis and Structural Diversity

    Image for article: Expanding the Scope of Azole-Based γ-Amino Acids – Synthesis and Structural Diversity
    Supporting Information (PDF)
  • 2373
    Annapurna, Sasikala Cheemalapati Venkata; Rao, Srinivas Talasila; Bathini, Pavan Kumar; Gaddameedhi, Prashanth Reddy; Komati, Shravan Kumar; Manda, Amarendhar; Nahide, Pradip D.; Reddy, B Ramalinga; Madhra, Mukesh Kumar; Annapragada, Ratnamala; Bandichhor, Rakeshwar:

    Quality by Design Driven Improved Process of Abiraterone Acetate

    Image for article: Quality by Design Driven Improved Process of Abiraterone Acetate
    Supporting Information (PDF)
  • 2391
    Novák, Tamás T.; Turczel, Gábor; Hornyánszky, Gábor; Szabó, Pál T.; Kiss, Loránd; Fustero, Santos; Nonn, Melinda:

    Fluorinative Difunctionalization of a Cyclooctene-Fused β-Lactam and Cyclooctene-Fused β-Amino Esters

    Image for article: Fluorinative Difunctionalization of a Cyclooctene-Fused β-Lactam and Cyclooctene-Fused β-Amino Esters
    Supporting Information (PDF)