DOI: 10.1055/s-00000084

Synthesis

Issue 02 · Volume 50 · January 2018 DOI: 10.1055/s-008-36797

review

193
Verbitskiy, Egor V.; Rusinov, Gennady L.; Chupakhin, Oleg N.; Charushin, Valery N.: Recent Advances in Direct C–H Functionalization of Pyrimidines
https://www.thieme-connect.de/media/synthesis/201802/i_e0545_ga_10-1055_s-0036-1589520.gif

short review

211
Ramesh, Perla; Suman, Devatha; Reddy, Koti Siva Nagi: Asymmetric Synthetic Strategies of (R)-(–)-Baclofen: An Antispastic Drug
https://www.thieme-connect.de/media/synthesis/201802/i_m0419_ga_10-1055_s-0036-1590938.jpg
227
Vorobyeva, Daria V.; Osipov, Sergey N.: Selective Synthesis of 2- and 7-Substituted Indole Derivatives via Chelation-Assisted Metallocarbenoid C–H Bond Functionalization
https://www.thieme-connect.de/media/synthesis/201802/i_m0544_ga_10-1055_s-0036-1591498.gif
241
Largeron, Martine; Nguyen, Khac Minh Huy: Recent Advances in the Synthesis of Benzimidazole Derivatives from the Oxidative Coupling of Primary Amines
https://www.thieme-connect.de/media/synthesis/201802/i_z0450_ga_10-1055_s-0036-1590915.gif

feature

254
Paul, Jérôme; Presset, Marc; Le Gall, Erwan; Léonel, Eric; Retailleau, Pascal: Insights into the Cobalt-Catalyzed Three-Component Coupling of Mixed Aromatic Organozinc Species, Carbonyl Compounds or Imines and Michael Acceptors: Synthetic and Mechanistic Aspects
https://www.thieme-connect.de/media/synthesis/201802/i_z0581_ga_10-1055_s-0036-1590957.gif
Supporting Information
267
Mancuso, Raffaella; Veltri, Lucia; Russo, Patrizio; Grasso, Giuseppe; Cuocci, Corrado; Romeo, Roberto; Gabriele, Bartolo: Palladium-Catalyzed Carbonylative Synthesis of Functionalized Benzimidazopyrimidinones
https://www.thieme-connect.de/media/synthesis/201802/i_z0629_ga_10-1055_s-0036-1591835.gif
Supporting Information

psp

278
Buonomo, Joseph A.; Eiden, Carter G.; Aldrich, Courtney C.: Scalable Synthesis of Hydrido-Disiloxanes from Silanes: A One-Pot Preparation of 1,3-Diphenyldisiloxane from Phenylsilane
https://www.thieme-connect.de/media/synthesis/201802/i_n0283_ga_10-1055_s-0036-1588580.jpg
Supporting Information

paper

282
Motoyama, Atsushi; Arai, Tomoki; Ikeuchi, Kazutada; Aki, Kazuya; Wakamori, Shinnosuke; Yamada, Hidetoshi: α-Selective Glycosylation of 3,6-O-o-Xylylene-Bridged Glucosyl Fluoride
https://www.thieme-connect.de/media/synthesis/201802/i_f0519_ga_10-1055_s-0036-1590927.gif
Supporting Information
295
Bian, Chen-Yu; Li, Dan; Shi, Qian; Mei, Guang-Jian; Shi, Feng: Brønsted Acid Catalyzed Dehydrative Nucleophilic Substitution of C3-Substituted 2-Indolylmethanols with Azlactones
https://www.thieme-connect.de/media/synthesis/201802/i_h0548_ga_10-1055_s-0036-1590929.gif
Supporting Information CIF File
303
Habenicht, Stefanie H.; Rohland, Philip; Reichel, Jeaninne; Biver, Tarita; Minei, Pierpaolo; Jakobi, Dörthe; Pucci, Andrea; Weiß, Dieter; Beckert, Rainer; Görls, Helmar: Small Molecules as Long-Wavelength Fluorophores: Push-Pull Substituted 4-Alkoxy-1,3-thiazoles
https://www.thieme-connect.de/media/synthesis/201802/i_t0448_ga_10-1055_s-0036-1588581.gif
Supporting Information
314
Trubitsõn, Dmitri; Žari, Sergei; Kaabel, Sandra; Kudrjashova, Marina; Kriis, Kadri; Järving, Ivar; Pehk, Tõnis; Kanger, Tõnis: Asymmetric Organocatalytic Cascade Synthesis of Tetrahydro­furanyl Spirooxindoles
https://www.thieme-connect.de/media/synthesis/201802/i_t0475_ga_10-1055_s-0036-1590918.gif
Supporting Information
323
Jafari, Ehsan; Kundu, Dipti S.; Chauhan, Pankaj; Gajulapalli, V. P. Reddy; von Essen, Carolina; Rissanen, Kari; Enders, Dieter: Organocatalytic Enantioselective Vinylogous Henry Reaction of 3,5-Dimethyl-4-nitroisoxazole with Trifluoromethyl Ketones
https://www.thieme-connect.de/media/synthesis/201802/i_z0579_ga_10-1055_s-0036-1590928.jpg
Supporting Information
330
Qiao, Guanyu; Zhang, Zhen; Huang, Baoliang; Zhu, Liu; Xiao, Fan; Zhang, Zhenhua: Palladium-Catalyzed One-Pot Synthesis of N-Sulfonyl, N-Phosphoryl, and N-Acyl Guanidines
https://www.thieme-connect.de/media/synthesis/201802/i_h0444_ga_10-1055_s-0036-1588576.gif
Supporting Information
341
Min, Xiangting; Liu, Jianhui; Dong, Yawen; Hussain, Mustafa: One-Pot Assembly towards ω-Substituted Arylbiurets from ­Aromatic Amines, Potassium Cyanate, and Glacial Acetic Acid
https://www.thieme-connect.de/media/synthesis/201802/i_h0446_ga_10-1055_s-0036-1590934.gif
Supporting Information
349
Miao, Maozhong; Xu, Huaping; Luo, Yi; Jin, Mengchao; Chen, Zhengkai; Xu, Jianfeng; Ren, Hongjun: Catalyst-Free Regioselective Nazarov Cyclization of Aryl Allenyl Ketones
https://www.thieme-connect.de/media/synthesis/201802/i_h0504_ga_10-1055_s-0036-1591487.gif
Supporting Information CIF File
361
Pardeshi, Sachin D.; Sathe, Pratima A.; Vadagaonkar, Kamlesh S.; Melone, Lucio; Chaskar, Atul C.: Copper-Catalyzed Simultaneous Activation of C–H and N–H Bonds: Three-Component One-Pot Cascade Synthesis of Multi­substituted Imidazoles
https://www.thieme-connect.de/media/synthesis/201802/i_z0357_ga_10-1055_s-0036-1588585.gif
Supporting Information
371
Petrini, Marino; Chiurchiù, Elena; Rossi, Federico V.; Palmieri, Alessandro: Oxidative Conversion of Sulfonyl Indoles into 3-Alkylidene-2-oxindoles under Flow Chemical Conditions
https://www.thieme-connect.de/media/synthesis/201802/i_z0490_ga_10-1055_s-0036-1588584.gif
Supporting Information
377
Shang, Xian-Xing; Vu, Huu-Manh; Li, Xu-Qin: One-Pot Synthesis of 2-Arylbenzoxazinones from 2-Arylindoles with (Diacetoxyiodo)benzene as the Sole Oxidant
https://www.thieme-connect.de/media/synthesis/201802/i_h0453_ga_10-1055_s-0036-1590933.gif
Supporting Information
384
Al-Zoubi, Raed M.; Ibdah, Abdellatif; Al-Jammal, Walid K.; Al-Zoubi, Mazhar S.; Almasalma, Ahmad A.; McDonald, Robert: Mild, Efficient, and Regioselective Synthesis of Diiodophenyl­boronic Acid Derivatives via Metal–Iodine Exchange of 5-Substituted 1,2,3-Triiodoarenes
https://www.thieme-connect.de/media/synthesis/201802/i_t0486_ga_10-1055_s-0036-1589114.gif
Supporting Information CIF File

errata

e1
Verbitskiy, Egor V.; Rusinov, Gennady L.; Chupakhin, Oleg N.; Charushin, Valery N.: Recent Advances in Direct C–H Functionalization of Pyrimidines