DOI: 10.1055/s-00000084

Synthesis

Ausgabe 22 · Volume 52 · November 2020 DOI: 10.1055/s-010-49660

table of contents

  • V

    Linked PDF of Table of Contents

    • review

  • 3295
    Grover, Nitika; Senge, Mathias O.:

    Synthetic Advances in the C–H Activation of Rigid Scaffold Molecules

    Image for article: Synthetic Advances in the C–H Activation of Rigid Scaffold Molecules

    • short review

  • 3326
    Yorimitsu, Hideki; Yoshimura, Aya; Misaki, Yohji:

    Catalytic C–H Arylation of Tetrathiafulvalenes for the Synthesis of Functional Materials

    Image for article: Catalytic C–H Arylation of Tetrathiafulvalenes for the Synthesis of Functional Materials
  • 3337
    Li, Dan; Chen, Xiaochao; Gao, Wei:

    Asymmetric Synthesis of C1-Chiral THIQs with Imines in Isoquinoline Rings

    Image for article: Asymmetric Synthesis of C<sub>1</sub>-Chiral THIQs with Imines in Isoquinoline Rings

    • feature

  • 3356
    Ivanov, Konstantin L.; Tukhtaev, Hamidulla B.; Tukhtaeva, Feruza O.; Bezzubov, Stanislav I.; Melnikov, Mikhail Ya.; Budynina, Ekaterina M.:

    One-Pot Synthesis of γ-Azidobutyronitriles and Their Intramolecular Cycloadditions

    Image for article: One-Pot Synthesis of γ-Azidobutyronitriles and Their Intramolecular Cycloadditions
    Supporting Information (PDF) CIF File (OTHER)

    • psp

  • 3374
    Delpe Acharige, Anjana; Neri, Raul; Hodgson, James; Bossmann, Stefan H.:

    A Catalyst-Free, Temperature-Driven One-Pot Synthesis of 1-Adamantylhydrazine Hydrochloride

    Image for article: A Catalyst-Free, Temperature-Driven One-Pot Synthesis of 1-Adamantylhydrazine Hydrochloride
    Supporting Information (PDF)

    • special topic

    Synthesis in Industry

  • 3378
    Maligres, Peter E.; Song, Zhiguo Jake; Strotman, Neil A.; Yin, Jinquin; Pei, Tao; Strotman, Hallena R.; Itoh, Tetsuji; Sherer, Edward C.; Humphrey, Guy R.:

    Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376

    Image for article: Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376
    Supporting Information (PDF)
  • 3389
    Toussaint, Frédéric C.; Defrance, Thierry; Decouvreur, Serge; Carly, Nicolas; Merschaert, Alain:

    Intensification of Free-Radical Racemization for a Non-activated Amine in a Continuous Flow Reactor

    Image for article: Intensification of Free-Radical Racemization for a Non-activated Amine in a Continuous Flow Reactor
  • 3397
    Wächtler, Andreas; Bremer, Matthias; Maillard, David; Mohr, Thomas:

    Controlling the All-trans Stereochemistry in Liquid Crystalline 4,4′-Dialkyl-[1,1′-bicyclohexyl] Compounds

    Image for article: Controlling the All-<i>trans</i> Stereochemistry in Liquid Crystalline 4,4′-Dialkyl-[1,1′-bicyclohexyl] Compounds
  • 3406
    Stumpf, Andreas; St-Jean, Frédéric; Lao, David; Cheng, Zhigang Ken; Angelaud, Remy; Gosselin, Francis:

    Practical Early Development Synthesis of Nav1.7 Inhibitor GDC-0310

    Image for article: Practical Early Development Synthesis of Nav1.7 Inhibitor GDC-0310
    Supporting Information (PDF)
  • 3415
    Chen, Chengsheng; Wu, Ling; Wang, Yuwen; Wu, Linglin; Zhang, Yongda:

    Copper-Catalyzed Asymmetric Hydroamination of Styrenes with pivZPhos as Ligand

    Image for article: Copper-Catalyzed Asymmetric Hydroamination of Styrenes with <i><sup>piv</sup></i>ZPhos as Ligand
    Supporting Information (PDF)

    • Synthesis in Industry

  • 3420
    Crawford, James J.; Liao, Daohong; Kolesnikov, Aleksandr; Lee, Wendy; Landry, Matthew L.:

    Synthesis of an Azabicyclo[3.1.0]hexanone-Containing Inhibitor of NF-κΒ Inducing Kinase via Catalytic C–H Activation

    Image for article: Synthesis of an Azabicyclo[3.1.0]hexanone-Containing Inhibitor of NF-κΒ Inducing Kinase via Catalytic C–H Activation
    Supporting Information (PDF)

    • paper

  • 3427
    Kolupaeva, Ekaterina V.; Ozeryanskii, Valery A.; Pozharskii, Alexander F.:

    N-Methylated 1,8-Diaminonaphthalenes as Bifunctional Nucleo­philes in Reactions with α,ω-Dihalogenoalkanes: A Facile Route to Heterocyclic and Double Proton Sponges

    Image for article: <i>N</i>-Methylated 1,8-Diaminonaphthalenes as Bifunctional Nucleo­philes in Reactions with α,ω-Dihalogenoalkanes: A Facile Route to Heterocyclic and Double Proton Sponges
    Supporting Information (PDF)
  • 3439
    Luo, Nianhua; Zhong, Yuhong; Liu, Ji-Tian; Ouyang, Lu; Luo, Renshi:

    An Efficient Hydration and Tandem Transfer Hydrogenation of Alkynes for the Synthesis of Alcohol in Water

    Image for article: An Efficient Hydration and Tandem Transfer Hydrogenation of Alkynes for the Synthesis of Alcohol in Water
    Supporting Information (PDF)
  • 3446
    Xie, Dengbing; Wang, Yiqiong; Yang, Bo; Zhang, Songlin:

    Neodymium-Promoted Highly Selective Carbon–Carbon Double Bond Formation of Ketones with Allyl Halides in the Presence of Diethyl Phosphite

    Image for article: Neodymium-Promoted Highly Selective Carbon–Carbon Double Bond Formation of Ketones with Allyl Halides in the Presence of Diethyl Phosphite
    Supporting Information (PDF)
  • 3452
    Liza, Umme Aiman; Sugiura, Ken-ichi:

    Functionalization of Bipyrenol: Potential Precursors for Advanced Chiral Molecules

    Image for article: Functionalization of Bipyrenol: Potential Precursors for Advanced Chiral Molecules
    Supporting Information (PDF)
  • 3461
    Nakamura, Itaru; Shiga, Keigo; Suzuki, Mao; Terada, Masahiro:

    Efficient Synthesis of O-tert-Propargylic Oximes via Nicholas Reaction

    Image for article: Efficient Synthesis of <i>O</i>-<i>tert</i>-Propargylic Oximes via Nicholas Reaction
    Supporting Information (PDF)
  • 3466
    Li, Qiao; Jin, Hongwei; Liu, Yunkui; Zhou, Bingwei:

    Nickel-Catalyzed Multicomponent Coupling Reaction of Alkyl Halides, Isocyanides and H2O: An Expedient Way to Access Alkyl Amides

    Image for article: Nickel-Catalyzed Multicomponent Coupling Reaction of Alkyl Halides, Isocyanides and H<sub>2</sub>O: An Expedient Way to Access Alkyl Amides
    Supporting Information (PDF)
  • 3473
    Bonilla-Reyes, Edgar; Sánchez-Carrillo, Adrian; Vázquez, Alfredo:

    Synthesis of l-Kynurenine and Homo-l-Kynurenine via an Aza-Fries Rearrangement

    Image for article: Synthesis of <sc>l</sc>-Kynurenine and Homo-<sc>l</sc>-Kynurenine via an Aza-Fries Rearrangement
    Supporting Information (PDF)
  • 3480
    Chavan, Subhash P.; Pawar, Ambaji A.; Patil, Niteen B.; Kadam, Appasaheb L.; Shinde, Shrikrishna S.:

    Scalable Synthesis of 3-Ethyl-4-methyl-1,5-dihydro-2H-pyrrol-2-one: An Important Building Block of the Antidiabetic Drug Glimepiride

    Image for article: Scalable Synthesis of 3-Ethyl-4-methyl-1,5-dihydro-2<i>H</i>-pyrrol-2-one: An Important Building Block of the Antidiabetic Drug Glimepiride
    Supporting Information (PDF)
  • 3485
    Arabadzhi, Svetlana S.; Zharkov, Mikhail N.; Kuchurov, Ilya V.; Zlotin, Sergei G.:

    Synthesis of Chiral N-Nitro-oxazolidin-2-ones and O-(β-Nitraminoalkyl) Carbamates in Liquefied 1,1,1,2-Tetrafluoroethane Medium

    Image for article: Synthesis of Chiral <i>N</i>-Nitro-oxazolidin-2-ones and <i>O</i>-(β-Nitraminoalkyl) Carbamates in Liquefied 1,1,1,2-Tetrafluoroethane Medium
    Supporting Information (PDF)

    • book review

  • 3492
    Lakhdar, Sami:

    Science of Synthesis: Photocatalysis in Organic Synthesis