DOI: 10.1055/s-00000084

Synthesis

Ausgabe 10 · Volume 2007 · Mai 2007 DOI: 10.1055/s-002-6704

review

  • 1439
    Domínguez de María, Pablo; García-Burgos, Carlos A.; Bargeman, Gerrald; van Gemert, Robert W.:

    Pig Liver Esterase (PLE) as Biocatalyst in Organic Synthesis: From Nature to Cloning and to Practical Applications

    Image for article: Pig Liver Esterase (PLE) as Biocatalyst in Organic Synthesis: From Nature to Cloning and to Practical Applications

    • short paper

  • 1453
    Kurz, Thomas; Thimann, Wolfgang; Geffken, Detlef:

    Synthesis of 3-Alkoxy-5,6-dihydro-4H-1,2,5-oxadiazines from Alkyl α-Aminohydroximates

    Image for article: Synthesis of 3-Alkoxy-5,6-dihydro-4<EM EMTYPE="BOLDITALIC">H</EM>-1,2,5-oxadiazines from Alkyl <EM EMTYPE="BOLD">α-</EM>Aminohydroximates
  • 1456
    Kuik, Árpád; Skoda-Földes, Rita; Jánosi, László; Kollár, László:

    Facile Synthesis of Unsymmetrical 1,n′-Disubstituted Ferrocenoyl Amino Acid Derivatives by Palladium-Catalyzed Aminocarbonylation

    Image for article: Facile Synthesis of Unsymmetrical 1,n′-Disubstituted Ferrocenoyl Amino Acid Derivatives by Palladium-Catalyzed Aminocarbonylation

    • paper

  • 1459
    Jiang, Yan; Zhou, Guo-Chuan; He, Guang-Li; He, Ling; Li, Ju-Lian; Zheng, Shi-Long:

    Ruthenium(II)-Porphyrin Catalyzed Selective N-Imidation of Aromatic Nitrogen Heterocycles

    Image for article: Ruthenium(II)-Porphyrin Catalyzed Selective N-Imidation of Aromatic Nitrogen Heterocycles
  • 1465
    Guan, Zheng-Hui; Zuo, Wei; Zhao, Lian-Biao; Ren, Zhi-Hui; Liang, Yong-Min:

    An Economical and Convenient Synthesis of Vinyl Sulfones

    Image for article: An Economical and Convenient Synthesis of Vinyl Sulfones
  • 1471
    Nery, Marcelo S.; Azevedo, Mariangela S.; Cardoso, Jari N.; Slana, Glaucia B. C.; Lopes, Rosangela S. C.; Lopes, Cláudio C.:

    A New Chemoselective Synthesis of Brombuterol

    Image for article: A New Chemoselective Synthesis of Brombuterol
  • 1475
    Paliakov, Ekaterina; Elleboe, Thomas; Boykin, David W.:

    New Synthons for the Preparation of Arylimidazolines and Tetrahydro­pyrimidine Analogues

    Image for article: New Synthons for the Preparation of Arylimidazolines and Tetrahydro­pyrimidine Analogues
  • 1481
    Thomas, James B.; Brieaddy, Lawrence E.; Boldt, Karl G.; Perretta, Carin; Carroll, F. Ivy:

    Synthesis and Resolution of the Benzomorphan-Based Kappa Opioid Agonist Bremazocine

    Image for article: Synthesis and Resolution of the Benzomorphan-Based Kappa Opioid Agonist Bremazocine
  • 1485
    Kumara Swamy, K. C.; Pavan Kumar, K. V. P.; Rama Suresh, R.; Satish Kumar, N.:

    Easy and Stereoselective Synthesis of Cyclopropyl-Substituted Phosphonates via α-Chlorophosphonates

    Image for article: Easy and Stereoselective Synthesis of Cyclopropyl-Substituted Phosphonates via α-Chlorophosphonates
  • 1491
    Tyrrell, Elizabeth; Hunie Tesfa, Kibur; Mann, Alastair; Singh, Kuldip:

    Enantioselective Alkynylation Reactions to Substituted Benzaldehyde and Salicylaldehyde Derivatives: The Effect of Substituents upon the Efficiency and Enantioselectivity

    Image for article: Enantioselective Alkynylation Reactions to Substituted Benzaldehyde and Salicylaldehyde Derivatives: The Effect of Substituents upon the Efficiency and Enantioselectivity
  • 1499
    Schobert, Rainer; Wicklein, André:

    Short Syntheses of (-)-(R)-Pyrrolam A and (1S)-1-Hydroxyindolizidin-3-one

    Image for article: Short Syntheses of (-)-<EM EMTYPE="BOLD">(</EM><EM EMTYPE="BOLDITALIC">R</EM><EM EMTYPE="BOLD">)</EM>-Pyrrolam A and (1<EM EMTYPE="BOLDITALIC">S</EM>)-1-Hydroxyindolizidin-3-one
  • 1503
    Kulik, Svetlana N.; Kobko, Alexander S.; Tolmachev, Andrey A.; Tverdokhlebov, Anton V.; Shishkin, Oleg V.; Chernega, Alexander N.:

    A New Approach to Pyrazino[2,1-b]quinazolines and Pyrazino[1,2-a]thi­eno[3,2-d]pyrimidines

    Image for article: A New Approach to Pyrazino[2,1-<EM EMTYPE="ITALIC">b</EM>]quinazolines and Pyrazino[1,2-<EM EMTYPE="ITALIC">a</EM>]thi­eno[3,2-<EM EMTYPE="ITALIC">d</EM>]pyrimidines
  • 1509
    Chandrasekhar, Srivari; Basu, Debjit; Raji Reddy, Ch.:

    Palladium-Catalyzed Reduction of N-(tert-Butoxycarbonyl)indoles by Polymethylhydrosiloxane

    Image for article: Palladium-Catalyzed Reduction of <EM EMTYPE="ITALIC">N</EM>-(<EM EMTYPE="ITALIC">tert</EM>-Butoxycarbonyl)indoles by Polymethylhydrosiloxane
  • 1513
    Alizadeh, Abdolhamid; Nematollahi, Davood; Hbibi, Davood; Hesari, Mahdi:

    Domino Oxidation-Michael Reactions of Catechols with Barbituric Acid Derivatives in Water: An Efficient Synthesis of Polycyclic Pyrimidinones

    Image for article: Domino Oxidation-Michael Reactions of Catechols with Barbituric Acid Derivatives in Water: An Efficient Synthesis of Polycyclic Pyrimidinones
  • 1517
    Woschek, Anna; Mahout, Marek; Mereiter, Kurt; Hammerschmidt, Friedrich:

    Synthesis of 2-Heptyl-1-hydroxy-4(1H)-quinolone - Unexpected Rearrangement of 4-(Alkoxycarbonyloxy)quinoline N-Oxides to 1-(Alkoxycarbonyloxy)-4(1H)-quinolones

    Image for article: Synthesis of 2-Heptyl-1-hydroxy-4(1<EM EMTYPE="ITALIC">H</EM>)-quinolone - Unexpected Rearrangement of 4-(Alkoxycarbonyloxy)quinoline <EM EMTYPE="ITALIC">N</EM>-Oxides to 1-(Alkoxycarbonyloxy)-4(1<EM EMTYPE="ITALIC">H</EM>)-quinolones
  • 1523
    Blair, Michael; Andrews, Philip C.; Fraser, Benjamin H.; Forsyth, Craig M.; Junk, Peter C.; Massi, Massimiliano; Tuck, Kellie L.:

    Facile Methods for the Separation of the cis- and trans-Diastereomers of Limonene­ 1,2-Oxide and Convenient Routes to Diequatorial and Diaxial 1,2-Diols

    Image for article: Facile Methods for the Separation of the <EM EMTYPE="ITALIC">cis</EM>- and <EM EMTYPE="ITALIC">trans</EM>-Diastereomers of Limonene­ 1,2-Oxide and Convenient Routes to Diequatorial and Diaxial 1,2-Diols
  • 1528
    Fukuhara, Tsuyoshi; Hasegawa, Chihiro; Hara, Shoji:

    A Facile Synthesis of Oxazolines, Thiazolines, and Imidazolines Using α,α-Difluoroalkylamines

    Image for article: A Facile Synthesis of Oxazolines, Thiazolines, and Imidazolines Using<EM EMTYPE="BOLD"> α,α-</EM>Difluoroalkylamines
  • 1535
    Tang, Shi; Li, Jin-Heng; Xie, Ye-Xiang; Wang, Nai-Xing:

    Halogenation of Indoles with Copper(II) Halides: Selective Synthesis of 2-Halo-, 3-Halo-, and 2,3-Dibromoindoles

    Image for article: Halogenation of Indoles with Copper(II) Halides: Selective Synthesis of 2-Halo-, 3-Halo-, and 2,3-Dibromoindoles
  • 1542
    Yoshida, Masanori; Osafune, Kanako; Hara, Shoji:

    Facile Synthesis of Iodonium Salts by Reaction of Organotrifluoroborates with p-Iodotoluene Difluoride

    Image for article: Facile Synthesis of Iodonium Salts by Reaction of Organotrifluoroborates with <EM EMTYPE="ITALIC">p</EM>-Iodotoluene Difluoride
  • 1547
    Sulima, Agnieszka; Folk, John; Jacobson, Arthur E.; Rice, Kenner C.:

    A New Approach to the Synthesis of the Nonpeptide NOP Receptor Antagonist J-113397

    Image for article: A New Approach to the Synthesis of the Nonpeptide NOP Receptor Antagonist J-113397
  • 1554
    Rybáčková, Markéta; Bělohradský, Martin; Holý, Petr; Pohl, Radek; Dekoj, Václav; Závada, Jiří:

    Synthesis of Highly Symmetrical Triptycene Tetra- and Hexacarboxylates

    Image for article: Synthesis of Highly Symmetrical Triptycene Tetra- and Hexacarboxylates
  • 1559
    Soley, Roger; Albericio, Fernando; Álvarez, Mercedes:

    Novel Synthesis of Arylethynyl Heterocycles

    Image for article: Novel Synthesis of Arylethynyl Heterocycles
  • 1566
    Prado, Soizic; Toum, Valérie; Saint-Joanis, Brigitte; Michel, Sylvie; Koch, Michel; Cole, Stewart T.; Tillequin, François; Janin, Yves L.:

    Antimycobacterial Benzofuro[3,2-f]chromenes from a 5-Bromochromen-6-ol

    Image for article: Antimycobacterial Benzofuro[3,2-<EM EMTYPE="ITALIC">f</EM>]chromenes from a 5-Bromochromen-6-ol
  • 1571
    Hesse, Stéphanie; Kirsch, Gilbert:

    Buchwald-Hartwig Amination of β-Chloroacroleins by Lactams and Heteroarylamines

    Image for article: Buchwald-Hartwig Amination of β-Chloroacroleins by Lactams and Heteroarylamines

    • feature article

  • 1576
    Restorp, Per; Dressel, Martina; Somfai, Peter:

    Synthesis of Functionalized Pyrrolidines by a Highly Stereoselective [3+2]-Annulation Reaction of N-Tosyl-α-Amino Aldehydes and 1,3-Bis(silyl)propenes

    Image for article: Synthesis of Functionalized Pyrrolidines by a Highly Stereoselective [3+2]-Annulation Reaction of <EM EMTYPE="ITALIC">N</EM>-Tosyl-α-Amino Aldehydes and 1,3-Bis(silyl)propenes

    • practical synthetic procedures

  • 1584
    Ward, Dale E.; Rasheed, M. Abdul; Gillis, H. Martin; Beye, Garrison E.; Jheengut, Vishal; Achonduh, George T.:

    Simple and Efficient Preparation of Reagents for Thiopyran Introduction:
    Methyl Tetrahydro-4-oxo-2H-thiopyran-3-carboxylate, Tetrahydro-4H-thiopyran-4-one, and 3,6-Dihydro-4-trimethylsilyloxy-2H-thiopyran

    Image for article: Simple and Efficient Preparation of Reagents for Thiopyran Introduction: <BR/>Methyl Tetrahydro-4-oxo-2<EM EMTYPE="ITALIC">H</EM>-thiopyran-3-carboxylate, Tetrahydro-4<EM EMTYPE="ITALIC">H</EM>-thiopyran-4-one, and 3,6-Dihydro-4-trimethylsilyloxy-2<EM EMTYPE="ITALIC">H</EM>-thiopyran
  • 1587
    Bandini, Marco; Eichholzer, Astrid; Tommasi, Simona; Umani-Ronchi, Achille:

    Practical Aspects in the Gram-Scale Synthesis of Chiral Diamino-Bithiophene ‘DAT2’ Ligand

    Image for article: Practical Aspects in the Gram-Scale Synthesis of Chiral Diamino-Bithiophene ‘DAT2’ Ligand

    • addenda and errata

  • e1
    Ward, Dale E.; Rasheed, M. Abdul; Gillis, H. Martin; Beye, Garrison E.; Jheengut, Vishal; Achonduh, George T.:

    Simple and Efficient Preparation of Reagents for Thiopyran Introduction: Methyl Tetrahydro-4-oxo-2H-thiopyran-3-carboxylate, Tetrahydro-4H-thiopyran-4-one, and 3,6-Dihydro-4-trimethylsilyloxy-2H-thiopyran