Synthesis

Qin, Yang; Liu, Sheng; Shi, Shi-Liang: Transition-Metal-Free Cross-Coupling of Acetals and Grignard Reagents To Form Diarylmethyl Alkyl Ethers and Triarylmethanes

Khan, Farooq-Ahmad; Yaqoob, Sana; Qasim, Muhammad Wasim; Ali, Shujaat; Wang, Yan; Jiang, Zi-Hua: A Robust, Gram-Scale and High-Yield Synthesis of MDP Congeners for Activation of the NOD2 Receptor and Vaccine Adjuvantation

Chaskar, Sudhir P.; Honparkhe, Ramchandra; Aghao, Arvind K.; Thorat, Rakesh G.; Pramanik, Chinmoy: An Alternative Formal Synthesis of (S)-(+)-Vigabatrin

Chen, Yang; Li, Qiao-Yue; Xie, Xiao-Yan; Wang, Wei; Li, Dashan; Wang, Wen-Jing; Shao, Li-Dong: Construction of an Epoxy-lactone Moiety on the C/D Ring of Highly Oxygenated Triterpenes through a Modified SeO₂-Promoted Oxidative Cyclization

Varga, Petra Regina; Belovics, Alexandra; Karaghiosoff, Konstantin; Szabó, Rita; Bősze, Szilvia; Drahos, László; Keglevich, György: Efficient Synthesis of Diethyl, Dialkyl α-Hydroxy-propylenebisphosphonates and Related 5-Phosphonoyl-1,2-oxaphospholane 2-Oxides

Cui, Hai-Bo; Ma, Ting; Zhang, Ru-Yue; Shan, Jing; Wang, Zhong-Qiang; Bai, Mei; Chen, Yong-Zheng: Biocatalytic Synthesis of Chiral Benzylic Alcohols via Enantioselective Hydroxylation by a Self-Sufficient Cytochrome P450 from Deinococcus gobiensis

Kumar, Kankanala Naveen; Mhate, Mouzma; Ravichandiran, Velayutham; Swain, Sharada Prasanna: Bis(pinacoloto)diboron/4-Phenylpyridine System for One-Pot Photocatalyzed Borylation and Reduction of Aldehyde: Synthesis of Tavaborole in a Flow Reactor

Tintori, Guillaume; Jacob, Clément; Delsarte, Christine; Potié, François; Grimaud, Laurence; Vitale, Maxime; Echeverria, Pierre-Georges: Efficient and Scalable Synthesis of 6,6-Dimethyl-3-oxabicyclo [3.1.0]hexan-2-one through Organocatalyzed Desymmetrization and Chemoselective Reduction

Bera, Shyamal Kanti; Bhanja, Rosalin; Sahu, Chandan Chittapriya; Mal, Prasenjit: An Intramolecular Radical C–N Coupling by N-Iodosuccinimide

Nakahara, Yuichi; Endo, Yuta; Takahashi, Kazutoshi; Kawaguchi, Tomoko; Kato, Keisuke; Matsuda, Yutaka; Nagaki, Aiichiro: A Manufacturing Strategy Utilizing a Continuous-Mode Reactor toward Homogeneous PEGylated Bioconjugate Production

Ramu, Chennam; Kumaraguru, T.; Reddy, M. Sridhar; Rode, Haridas B.; Ghosh, Subhash; Reddy, Ch. Raji; Sudhakar, Gangarajula: Synthesis of Ledipasvir through a Late-Stage Cyclopropanation and Fluorination Process

Sunny, Steeva; Maingle, Mohit; Sheeba, Loddipalle; Pathan, Firojkhan Rajekhan; J., Gowri Sankar; Juloori, Harika; Gadewar, Sainath Ganesh; Seth, Kapileswar: Pd-Nanoparticles-Catalyzed C(sp²)–H Arylation for the Synthesis of Functionalized Heterocycles: Recent Progress and Prospects

Zhang, Fei; Zhou, Yong; Wang, Shuangqiang; Zhao, Yao; Wu, Xiaojin; Chen, Rizhi: Palladium-Loading Ceramic Catalytic Membrane Reactors for Mizoroki–Heck Reaction

Ohashi, Eisaku; Sahara, Naoto; Hirano, Yoichi; Hosoya, Masahiro; Takahashi, Yusaku; Tsuno, Naoki: An Effective Additive for Introducing the Triazole Unit of Ensitrelvir: Combination of LiCl and Et₃N to Easily Generate Lithium Triazinolate

Mahajan, Bhushan; Aand, Dnyaneshwar; Purwa, Mandeep; Mujawar, Taufiqueahmed; Ghosh, Subhash; Pabbaraja, Srihari; Singh, Ajay K.: Elements-Continuous-Flow Platform for Coupling Reactions and Anti-viral Daclatasvir API Synthesis

Adaoudi, Omaïma; Le Bescont, Julie; Bruneau-Voisine, Antoine; Evano, Gwilherm: Copper-Catalyzed Carbonylative Cross-Coupling of Alkyl Iodides with Alcohols and Sodium Hydroxide: Synthesis of Esters and Carboxylic Acids

Dash, Rupashri; Hota, Sudhir Kumar; Murarka, Sandip: Base-Promoted 1,6-Aza-Michael Addition of Azauracils to para-Quinone Methides

Algera, Russell F.; Davidson, Andrew; Herbert, David K.; Lian, Yajing; Liu, Fangfang; Liu, Yiyang; Nematalla, Asaad; Piper, Jared L.; Magano, Javier; Monfette, Sebastien; Nguyen, Bao; Raggon, Jeffrey W.; Rainville, Joseph P.; Rane, Anil; Tao, Yong; Wang, Ke; Yayla, Hatice G.: Exploratory Process Development of a Pulmonary Arterial Hypertension Clinical Compound via a Late-Stage Pd-Catalyzed Buchwald–Hartwig C–N Coupling

Das, Soumyadip; Chanda, Kaushik: One-Pot Telescopic Approach to Synthesize Disubstituted Benz­imidazoles in Deep Eutectic Solvent