DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 15 · August 2019 DOI: 10.1055/s-009-43556

Synform

  • A113

    SYNFORM ISSUE 2019/08

    • Synthesis of Natural Products and Potential Drugs

  • z0833

    All PDFs of this category

  • 0833

    Synthesis of (+)-Longirabdiol, (–)-Longirabdolactone, and (–)-Effusin

  • 0834

    Synthesis of a PDE10A Inhibitor

  • 0835

    Synthesis of E2212

  • 0836

    Synthesis of Taselisib

  • 0837

    Synthesis of Taselisib

  • 0838

    Syntheses of (±)-Rhodomolleins XX and XXII

  • 0839

    Total Syntheses of (–)-Daphlongamine H and (–)-Isodaphlongamine H

  • 0840

    Total Synthesis of Englerins A and B

  • 0841

    Synthesis of (–)-7-Deacetoxyalcyonin Acetate

  • 0842

    Synthesis of a Renin Inhibitor

  • 0843

    Synthesis of a TAK-480 Fragment

  • 0844

    Synthesis of TAK-063

  • 0845

    Synthesis of (+)-Arborisidine

  • 0846

    Synthesis of Dolutegravir

  • 0847

    Synthesis of Dolutegravir

  • 0848

    Synthesis of an Edoxaban Fragment

  • 0849

    Synthesis of (+)-Principinol D

  • 0850

    Synthesis of Tofogliflozin

  • 0851

    Synthesis of BMS-986236

    • Synthesis of Heterocycles

  • z0853

    All PDFs of this category

  • 0853

    Synthesis of Two Azaborine Building Blocks

  • 0854

    Phosphonium-Salt-Catalyzed Synthesis of Fused Aziridines by an Aza-Darzens Reaction

  • 0855

    Chemoselective Demethylation of Methoxypyridines over Anisoles

  • 0856

    Catalytic Azole Acylation with Acyl Fluorides

  • 0857

    Acridone Synthesis by Double Amination of Dibromobenzophenones

  • 0858

    Enantioselective Catalytic Aryl-Alkenylation To Give Dihydrobenzofurans

  • 0859

    Synthesis of 1,2-Benzothiazine 1-Imines as New Heterocyclic Scaffolds

  • 0860

    Selective C–H Alkenylation of Isoxazoles

  • 0861

    Gold(III)-Catalyzed Synthesis of 4-Aminooxazoles

  • 0862

    Synthesis of 1,4-Benzothiazines by Iodide-Catalyzed Alkene Sulfenoamination

  • 0863

    Copper-Catalyzed Synthesis of 3,4-Dihydroquinazolines from Anthranils

  • 0864

    Silver-Catalyzed Synthesis of Trifluoromethylated Triazines and Pyridines

  • 0865

    Asymmetric Synthesis of Dihydrobenzofurans by an Organocatalytic [4+1] Cyclization

  • 0866

    DBU-Mediated Synthesis of Bicyclic Heterocycles

    • Synthesis of Materials and Unnatural Products

  • z0867

    All PDFs of this category

  • 0867

    A Prefix to SuFEx

  • 0868

    The Whole Kit and Caboodle: A Ferrocenyl Halogen Bonding Rotaxane for Electrochemical Bromide Sensing

  • 0869

    It takes Strained Alkynes to make Polycyclic Aromatic Hydrocarbons

  • 0870

    Forced into Antiaromaticity

  • 0871

    Tetrahydroquinoline-Fused Fullerenes

  • 0872

    (N-Phenylfluorenylidene)acridanes: Mechanochromic BAEs

  • 0873

    Organocopper Cross-Coupling for Crowded Environments

  • 0874

    Deep LUMO Level Diimide π-Electron Core

  • 0875

    Renewing the Synthesis of Sterically Hindered Phenanthrenes

  • 0876

    Studies of Polyarylether COFs

  • 0877

    Cranking out Functionalized Helicenes

  • 0878

    Unlocking a [2.2.2]Carbon Nanocage

    • Metals in Synthesis

  • z0879

    All PDFs of this category

  • 0879

    Diastereoselective [4+4] Cycloadditions

  • 0880

    Asymmetric Copper-Catalyzed Hydroamination of Enamines

  • 0881

    Iridium-Catalyzed Asymmetric Hydroalkynylation of Unactivated Alkenes

  • 0882

    Nickel-Catalyzed Amination of Phenols

  • 0883

    Mild Copper-Catalyzed N-Arylation of Sulfoximines

  • 0884

    Enantioselective Synthesis of Chiral Homoallylic Tertiary Alcohols through Copper Catalysis

  • 0885

    Dual Nickel/Photo-Catalyzed Esterification of Aryl Halides

  • 0886

    Nickel-Catalyzed Cyano-Borrowing Reaction Affording β-Cyano Ketones

  • 0887

    Cobalt-Catalyzed Aminocarbonylation of Alkyl Tosylates

  • 0888

    Synthesis of Chiral β-Nitroamides

  • 0889

    Enantioselective Synthesis of Tertiary α-Silyl Alcohols

  • 0890

    The Catalytic Kulinkovich Reaction

  • 0891

    Synthesis of Areneamides

  • 0892

    Intermolecular [2+2] Carbonyl–Olefin Photocycloadditions Enabled by a Copper(I)–Norbornene Complex

  • 0893

    Regioselective Palladium-Catalyzed C–H Iodination of Alkenes

  • 0894

    Amide Enolate Surrogates in Asymmetric Allylation Reactions

  • 0895

    Catalytic Preparation of Potassium Acyltrifluoroborates

  • 0896

    Amination of Triaryl Phophates

  • 0897

    Palladium-Catalyzed Dearomative Carboamination

  • 0898

    Counterion-Controlled Cobalt-Catalyzed Addition of Cyclopropanols to Oxabyciclic Alkenes

  • 0899

    Palladium-Catalyzed Enantioselective N‑Alkylation of Indoles

  • 0900

    Decarboxylative Alkylation

  • 0901

    Iodination/Cross-Coupling Cascade Reaction

  • 0902

    Radical-Driven Deoxygenation of Secondary Alcohols: The Barton–McCombie Reaction

  • 0903

    Nickel-Catalyzed Reaction of Umpolung Carbonyls and Alkyl Halides

  • 0904

    Ligand-Controlled Selection of Diastereoisomers in Asymmetric 1,3-Dipolar Cycloaddition

  • 0905

    Ruthenium-Catalyzed Transfer Hydrogenation of α-Acetamido Benzocyclic Ketones

  • 0906

    Intramolecular Asymmetric Hydroamination of Allenes

  • 0907

    Preparation of 2-Substituted Propenes

  • 0908

    Nickel/Manganese Dual-Catalyzed Hydroalkylation of Olefins

    • Polymer-Supported Synthesis

  • z0909

    All PDFs of this category

  • 0909

    Ion-Exchange-Resin-Supported Hydrogen Fluoride for Fluorination Reactions

  • 0910

    Michael Addition on a Squaramide-Decorated Covalent Organic Framework

  • 0911

    Aqueous Flow Hydroxycarbonylation on an Amphiphilic Polymer-Supported Pd Complex

  • 0912

    Transfer Hydrogenation of Aryl Ketones on Mesoporous Silica-Supported Nickel

  • 0913

    Buchwald–Hartwig Amination on NHC-Pd Immobilized on Wang Resin

  • 0914

    Couplings of Aryl Halides with Arylboronic Acids on Silica-Supported Nickel

  • 0915

    Palladium-Catalyzed Dehydrogenative Aromatization of Cyclic Amines

  • 0916

    Dehydrogenation of N-Heterocycles with Cobalt Nanocrystals on Carbon

  • 0917

    Suzuki–Miyaura Coupling on Aluminosilicate-Encapsulated Palladium Nanoparticles

  • 0918

    Benzylic C(sp3)–H Bond Oxidation Catalyzed by a Supported Manganese Complex

  • 0919

    Alumina-Supported Copper Oxide Hydrogenation Catalyst

  • 0920

    Hydroxylation of Alkyl Halides on an Aminopolystyrene-Supported Ionic Liquid

  • 0921

    Nickel-Catalyzed Cross-Coupling of Aryl Chlorides with Organolithiums

  • 0922

    Porous NiCo-Catalyzed Reduction of Nitroarenes with Ammonia Borane

    • Organo- and Biocatalysis

  • z0923

    All PDFs of this category

  • 0923

    Enzyme-Catalyzed Site-Selective C–H Amidation

  • 0924

    Chiral Phosphine Catalyzed Asymmetric Staudinger–aza-Wittig Reaction

  • 0925

    Photochemical Organocatalytic Borylation of Alkyl Halides and Sulfonates

  • 0926

    Benzothiophene-Catalyzed Oxidative Coupling of 2-Naphthols

  • 0927

    Benziodoxole-Catalyzed Anti-Markovnikov Hydroazidation of Olefins

  • 0928

    Organocatalytic Enantioselective Dichlorination of Cyclic Styrenes

  • 0929

    [4+2] Cycloaddition via NHC-Bound Aza-ortho-Quinone Methides

  • 0930

    Diazaphospholene-Catalyzed Reductive Ireland–Claisen Rearrangement

  • 0931

    Asymmetric Catalytic Transannular Morita–Baylis–Hillman Reaction

  • 0932

    A Bifunctional Catalyst Permits Atroposelective Aromatization

  • 0933

    Enantioselective Protonation of Disilyl Ketene Acetals with Water or Methanol

  • 0934

    Thiazolium Salt Catalyzed Asymmetric Benzoin Reaction

    • Chemistry in Medicine and Biology

  • z0935

    All PDFs of this category

  • 0935

    A Mitochondria-Targeting Calcium Dye

  • 0936

    Small-Molecule Inhibitors of CRISPR-Cas9

  • 0937

    In Vivo Imaging of Glucose Uptake

  • 0938

    Chemical Diversification of Pleuromutilin

  • 0939

    Highly Selective Insulin-Degrading Enzyme Inhibitors

  • 0940

    Selective α-Glycosidation of Sialic Acid

  • 0941

    Short Synthesis of the 3-Deazaguanosine RNA Building Block

  • 0942

    SCOTfluors: Small, Conjugatable, Orthogonal, and Tunable Fluorophores

  • 0943

    Photoactivated Fluxional Fluorophore Enables Extended Time-Lapse Microscopy

    • Peptide Chemistry

  • z0945

    All PDFs of this category

  • 0945

    Organcatalytic Transamination for the Synthesis of α-Amino Acids

  • 0946

    One-Pot Four-Component Strategy for Electrophilic Fluorination

  • 0947

    Site-Selective Reduction of Cyclosporine A by Borane Catalysis

  • 0948

    Palladium-Catalyzed β-C–H Arylation of N-Methylated Peptides

  • 0949

    Synthesis of Rigidified Cyclic Peptides by Ring-Closing Metathesis

  • 0950

    Azotide Ligands for Hetero-Diels–Alder Reactions

  • 0951

    Synthesis of N-Terminal Cysteinyl Thioesters

  • 0952

    Nickel-Catalyzed Synthesis of Amides from Methyl Esters

  • 0953

    Pd-Catalyzed Arylation of α-Amino Esters with Diaryliodonium Triflates

    • Flow Chemistry

  • z0955

    All PDFs of this category

  • 0955

    Continuous-Flow Preparation of Alkynylzinc and its Subsequent Cross-Coupling Reaction

  • 0956

    Continuous-Flow Electrochemical Oxidation with Hypervalent Iodine Reagents

  • 0957

    Syntheses of Sulfilimines and Sulfoximines in a Flow System

  • 0958

    Flow Synthesis of Vaborbactam

  • 0959

    Flow Synthesis of Ceramide d-erythro-CER[NDS]

  • 0960

    Synthesis of Sialic Acid Derivatives in a Continuous-Flow Enzymic Reactor

  • 0961

    Cascade Oxidation over Contiguous Dual Catalyst Beds in Continuous Flow

    • Erratum

  • 0962

    Iron-Catalyzed Synthesis of Fluoroalkylated 2H-Azirines from Alkynes

  • 0962

    Continuous-Flow, Michaelis−Arbuzov Rearrangement