DOI: 10.1055/s-00000084

Synthesis

Issue 04 · Volume 51 · February 2019 DOI: 10.1055/s-009-42395

table of contents

  • V

    Linked PDF of Table of Contents

    • review

  • 787
    Trushkov, Igor V.; Uchuskin, Maxim G.; Abaev, Vladimir T.; Serdyuk, Olga V.:

    Indolylvinyl Ketones: Building Blocks for the Synthesis of Natural Products and Bioactive Compounds

    Image for article: Indolylvinyl Ketones: Building Blocks for the Synthesis of Natural Products and Bioactive Compounds

    • short review

  • 816
    Leonardi, Marco; Estévez, Verónica; Villacampa, Mercedes; Menéndez, J. Carlos:

    The Hantzsch Pyrrole Synthesis: Non-conventional Variations and Applications of a Neglected Classical Reaction

    Image for article: The Hantzsch Pyrrole Synthesis: Non-conventional Variations and Applications of a Neglected Classical Reaction
  • 829
    Palmieri, Alessandro; Petrini, Marino:

    Recent Advances in the Synthesis of Unsymmetrical Bisindolylmethane Derivatives

    Image for article: Recent Advances in the Synthesis of Unsymmetrical Bisindolylmethane Derivatives

    • psp

  • 842
    Morales-Chamorro, Maricela; Vázquez, Alfredo:

    A Facile Synthesis of N-Boc-azocan-5-one

    Image for article: A Facile Synthesis of <i>N</i>-Boc-azocan-5-one
    Supporting Information (PDF)

    • paper

  • 848
    Sokolov, Andriy; Golovach, Sergey; Kozlinsky, Ihor; Dolia, Krystyna; Tolmachev, Andrey A.; Kuchkovska, Yuliya; Grygorenko, Oleksandr O.:

    Diastereoselective Synthesis of Cyclic sp3-Enriched cis-β-Alkoxysulfonyl Chlorides

    Image for article: Diastereoselective Synthesis of Cyclic sp<sup>3</sup>-Enriched <i>cis</i>-β-Alkoxysulfonyl Chlorides
    Supporting Information (PDF)
  • 859
    Kim, Hyokwon; Zong, Kyukwan:

    A Convenient Synthesis of Benzo[1,2-b:6,5-b′:3,4-c′′]trithiophenes Starting from Thiophene

    Image for article: A Convenient Synthesis of Benzo[1,2-<i>b</i>:6,5-<i>b</i>′:3,4-<i>c</i>′′]trithiophenes Starting from Thiophene
  • 865
    Ndimba, A. Ngo; Roisnel, T.; Argouarch, G.; Lalli, C.:

    Harvesting New Chiral Phosphotriesters by Phosphorylation of BINOL and Parent Bis-phenols

    Image for article: Harvesting New Chiral Phosphotriesters by Phosphorylation of BINOL and Parent Bis-phenols
    Supporting Information (PDF)
  • 874
    Xue, Dengqi; Xue, Yijie; Yu, Haihua; Shao, Liming:

    Metal-Free Radical Cyclization of Vinyl Isocyanides with Alkanes: Synthesis of 1-Alkylisoquinolines

    Image for article: Metal-Free Radical Cyclization of Vinyl Isocyanides with Alkanes: Synthesis of 1-Alkylisoquinolines
    Supporting Information (PDF)
  • 885
    Kim, Sonhwan; Lee, Won Koo; Ha, Hyun-Joon:

    Asymmetric Synthesis of cis-5-(Aminomethyl)-3-(4-methoxy­phenyl)dihydrofuran-2(3H)-one

    Image for article: Asymmetric Synthesis of <i>cis</i>-5-(Aminomethyl)-3-(4-methoxy­phenyl)dihydrofuran-2(3<i>H</i>)-one
    Supporting Information (PDF)
  • 889
    Zhang, Xing; Du, Cong; Zhang, He; Li, Xiao-Cai; Wang, Yun-Long; Niu, Jun-Long; Song, Mao-Ping:

    Metal-Free Blue-Light-Mediated Cyclopropanation of Indoles by Aryl(diazo)acetates

    Image for article: Metal-Free Blue-Light-Mediated Cyclopropanation of Indoles by Aryl(diazo)acetates
    Supporting Information (PDF)
  • 899
    Zhu, Yuanyuan; Zhao, Shuang; Zhang, Minli; Song, Xixi; Chang, Junbiao:

    Diastereoselective Synthesis of Spirobarbiturate-Cyclopropanes through Organobase-Mediated Spirocyclopropanation of Barbiturate-Based Olefins with Benzyl Chlorides

    Image for article: Diastereoselective Synthesis of Spirobarbiturate-Cyclopropanes through Organobase-Mediated Spirocyclopropanation of Barbiturate-Based Olefins with Benzyl Chlorides
    Supporting Information (PDF)
  • 907
    Formánek, Bedřich; Šimek, Michal; Kamlar, Martin; Císařová, Ivana; Veselý, Jan:

    Organocatalytic Allylic Amination of Morita–Baylis–Hillman Carbonates­

    Image for article: Organocatalytic Allylic Amination of Morita–Baylis–Hillman Carbonates­
    Supporting Information (PDF)
  • 921
    Ramkumar, Rajagopal; Chandrasekaran, Srinivasan:

    Catalyst-Free, Metal-Free, and Chemoselective Transamidation of Activated Secondary Amides

    Image for article: Catalyst-Free, Metal-Free, and Chemoselective Transamidation of Activated Secondary Amides
    Supporting Information (PDF)
  • 933
    Lessi, Marco; Panattoni, Alessandro; Guglielmero, Luca; Minei, Pierpaolo; Bellina, Fabio:

    Imidazole-Fused Enediynes by Selective C5–C4 Alkynylations of 4,5-Dibromoimidazoles

    Image for article: Imidazole-Fused Enediynes by Selective C5–C4 Alkynylations of 4,5-Dibromoimidazoles
    Supporting Information (PDF)
  • 944
    Zheng, Xiu-An; Kong, Rui; Huang, Hua-Shan; Wei, Jing-Ying; Chen, Ji-Zong; Gong, Shan-Shan; Sun, Qi:

    Hafnium Triflate as a Highly Potent Catalyst for Regio- and Chemoselective­ Deprotection of Silyl Ethers

    Image for article: Hafnium Triflate as a Highly Potent Catalyst for Regio- and Chemoselective­ Deprotection of Silyl Ethers
    Supporting Information (PDF)
  • 953
    deLong, Mitchell A.; Sturdivant, Jill M.:

    Asymmetric Synthesis of Netarsudil: A New Therapeutic for Open-Angle Glaucoma

    Image for article: Asymmetric Synthesis of Netarsudil: A New Therapeutic for Open-Angle Glaucoma
    Supporting Information (PDF)
  • 960
    Parveen, Iram; Ahmed, Naseem:

    A Route to Highly Functionalized Stereospecific trans-Aminated Aurones from 3-Bromoflavones with Aniline and N-Phenylurea via a Domino Aza-Michael Ring Opening and Cyclization Reactions

    Image for article: A Route to Highly Functionalized Stereospecific <i>trans</i>-Aminated Aurones from 3-Bromoflavones with Aniline and <i>N</i>-Phenylurea via a Domino Aza-Michael Ring Opening and Cyclization Reactions
    Supporting Information (PDF)
  • 971
    Glachet, Thomas; Franck, Xavier; Reboul, Vincent:

    Late-Stage Sulfoximination: Improved Synthesis of the Anticancer Drug Candidate Atuveciclib

    Image for article: Late-Stage Sulfoximination: Improved Synthesis of the Anticancer Drug Candidate Atuveciclib
    Supporting Information (PDF)
  • 976
    Bartuschat, Amelie L.; Hegmann, Nina; Heinrich, Markus R.:

    Synthesis of Fmoc- and Boc-Protected (2S,5S)- and (2R,5R)-5-Aminomethylprolines

    Image for article: Synthesis of Fmoc- and Boc-Protected (2<i>S</i>,5<i>S</i>)- and (2<i>R</i>,5<i>R</i>)-5-Aminomethylprolines
    Supporting Information (PDF)