DOI: 10.1055/s-00000084

Synthesis

Current Issue 04 · Volume 46 · February 2014 DOI: 10.1055/s-004-26400

review

403
Olszewski, Tomasz K.: Environmentally Benign Syntheses of α-Substituted Phosphonates: Preparation of α-Amino- and α-Hydroxyphosphonates in Water, in Ionic Liquids, and under­ Solvent-Free Conditions
https://www.thieme-connect.de/media/synthesis/201404/i_e0646_ga_10-1055_s-0033-1338588.gif

short review

430
Sidduri, Achyutharao; Tilley, Jefferson W.; Fotouhi, Nader: Functionalized Organozinc Reagents in Medicinal Chemistry: Discovery of Novel Drug Candidates
https://www.thieme-connect.de/media/synthesis/201404/i_m0805_ga_10-1055_s-0033-1338589.gif

practical synthetic procedures

445
Zajdlik, Adam; He, Zhi; St Denis, Jeffrey D.; Yudin, Andrei K.: Efficient Preparation of α-Aminoboronic Acid Derivatives via Boroalkyl Group Migration
https://www.thieme-connect.de/media/synthesis/201404/i_z0731_ga_10-1055_s-0033-1340502.gif

paper

455
Kawase, Yasushi; Yamagishi, Takehiro; Kato, Jun-ya; Kutsuma, Teruo; Kataoka, Tadashi; Iwakuma, Takeo; Yokomatsu, Tsutomu: Reductive Alkylation of Hydrazine Derivatives with α-Picoline-Borane and Its Applications to the Syntheses of Useful Compounds Related to Active Pharmaceutical­ Ingredients
https://www.thieme-connect.de/media/synthesis/201404/i_f0602_ga_10-1055_s-0033-1340484.gif
Supporting Information
465
Vuppalapati, Srinivasu V. N.; Xia, Likai; Edayadulla, Naushad; Lee, Yong Rok: Mild and Efficient One-Pot Synthesis of Diverse Flavanone Derivatives via an Organocatalyzed Mannich-Type Reaction
https://www.thieme-connect.de/media/synthesis/201404/i_f0705_ga_10-1055_s-0033-1340466.gif
Supporting Information
475
Kretschmer, Florian; Wild, Andreas; Hager, Martin D.; Schubert, Ulrich S.: Synthesis of a Rigid Tetrahedral Linker with Thioether End Groups
https://www.thieme-connect.de/media/synthesis/201404/i_t0708_ga_10-1055_s-0033-1340494.gif
Supporting Information
479
Banoth, Linga; Chandarrao, Bhukya; Pujala, Brahmam; Chakraborti, Asit K.; Banerjee, U. C.: Efficient Chemoenzymatic Synthesis of (RS)-, (R)-, and (S)-Bunitrolol
https://www.thieme-connect.de/media/synthesis/201404/i_z0620_ga_10-1055_s-0033-1340465.gif
Supporting Information
489
Gao, Hong; Sun, Jing; Yan, Chao-Guo: Povarov Reaction of β-Enamino Esters and Isatin-3-imines for Diastereoselective Synthesis of Spiro[indoline-3,2′-quinolines]
https://www.thieme-connect.de/media/synthesis/201404/i_f0691_ga_10-1055_s-0033-1340459.gif
Supporting Information
496
Miura, Takuya; Fujioka, Saki; Takemura, Naoto; Iwasaki, Hiroki; Ozeki, Minoru; Kojima, Naoto; Yamashita, Masayuki: Synthesis of 6-Substituted 3-(Alkoxycarbonyl)-5-aryl-α-pyrones
https://www.thieme-connect.de/media/synthesis/201404/i_f0692_ga_10-1055_s-0033-1338575.gif
Supporting Information
503
Han, Liuquan; Zhang, Bijun; Xiang, Changbin; Yan, Jie: One-Pot Synthesis of Isoxazolines from Aldehydes Catalyzed by Iodobenzene
https://www.thieme-connect.de/media/synthesis/201404/i_f0700_ga_10-1055_s-0033-1340464.gif
510
Hu, Manman; He, Xinwei; Niu, Zhiqiang; Yan, Zhenglei; Zhou, Fuyin; Shang, Yongjia: Synthesis of 3,4,5-Trisubstituted Isoxazoles by the 1,3-Dipolar Cycloaddition Reaction of α-Azido Acrylates and Aromatic Oximes
https://www.thieme-connect.de/media/synthesis/201404/i_h0695_ga_10-1055_s-0033-1340470.gif
Supporting Information
515
Smith, D. David; Gallagher, Audrey T.; Crowley, Vincent M.; Gergens, Wayne M.; Abel, Peter W.; Hulce, Martin: An Efficient Synthesis of 4(5)-Benzyl-l-histidines Employing Catalytic Transfer Hydrogenolysis at Elevated Temperatures
https://www.thieme-connect.de/media/synthesis/201404/i_m0680_ga_10-1055_s-0033-1340462.gif
Supporting Information
522
Nordmann, Jan; Müller, Thomas J. J.: Anilines as Substrates in Consecutive Four-Component Synthesis of Novel 1-Aryl-5-benzoyl-6-phenyl-3,4-dihydropyridin-2(1H)-ones
https://www.thieme-connect.de/media/synthesis/201404/i_t0661_ga_10-1055_s-0033-1338574.gif
Supporting Information
531
Gaitzsch, Jens; Rogachev, Victor; Zahel, Martin; Metz, Peter: Synthesis of m-Terphenyl Derivatives via Domino Diels–Alder/Retro-Diels–Alder Reaction of 1,3-Dienic δ-Sultones with Alkynes
https://www.thieme-connect.de/media/synthesis/201404/i_z0580_ga_10-1055_s-0033-1340346.gif
Supporting Information