DOI: 10.1055/s-00000131

Synfacts

Issue 01 · Volume 2005 · 2005 DOI: 10.1055/s-002-4363

Synthesis of Natural Products and Potential Drugs

0091
Enantioselective Synthesis of Stephacidin B
0092
Total Synthesis of (+)-Discodermolide via Asymmetric Crotylation
0093
Total Synthesis of (-)-Brasoside and (-)-Littoralisone
0094
Total Synthesis of (-)-α-Kainic Acid
0095
Total Synthesis of Rubrenolide
0096
Total Synthesis of Tirandalydigin
0097
Total Synthesis of Cribrostatin IV
0098
Total Synthesis of (+)-trans-195A
0099
Total Synthesis of Gymnocin-A
0100
Synthesis of ABT-100, a Farnesyl Transferase Inhibitor
0101
Synthesis of Discodermolide Using Solely Substrate-Based Stereocontrol
0102
Total Synthesis of (+)-Pseudodistomin D
0103
Total Synthesis of Stephacidin A
0104
Total Synthesis of Cryptophycin 3
0105
Synthesis of ()-Dibromophakellstatin

Synthesis of Heterocycles

0107
Enantioselective Pyrrolidine Synthesis
0108
Regio- and Stereoselective Synthesis of Structurally Diverse Polycyclic Indolyldiamines
0109
Regioselective Hydroamination for the Synthesis of Tricyclic Quinolines
0110
Synthesis of a Highly Strained Heterocycle Involving a Nitro Acetal to Aminal Rearrangement
0111
A Heterocyclic N-Oxide-Mediated Morita-Baylis-Hillman Reaction
0112
Tandem Cyclization of Allenenes to Tri- and Tetracyclic Heterocycles
0113
Palladium-Catalyzed Regioselective Direct C-2 and C-3 Functionalization of Indoles
0114
Synthesis of Aza-Stilbenes via an Ullmann C-N Coupling Reaction in Ionic Liquids
0115
Carbolithiation of Vinyl Pyridines as a Route to 7-Azaindoles
0116
Synthesis of Fused Indoles by Sequential Heck Reaction and N-Heteroannulation
0117
A Stereospecific Synthesis of Imidazolidin-2-ones from Aziridine-2-carboxylates and Isocyanates
0118
Ruthenium-Catalyzed Cyclization of Diols to Lactones
0119
Cycloaddition of Carbodiimides to Selenazetidines
0120
Enantioselective Synthesis of Tryptamines and Tetrahydro-β-carbolines
0121
Tetraorganosilicon Reagents for Cross-Coupling Reactions

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

0123
Enantioselective Fluorination and Chlorination of Compounds Capable of Two-Point Binding
0124
Enantioenriched α,β-Unsaturated Lactones via Vinylogous Mukaiyama Aldol
0125
Protic Functionality-Tolerant Decarboxylative Thioester syn-Aldol Reactions
0126
Vanadium-Catalyzed Enantioselective Epoxidation of Allylic Alcohols
0127
Sequential Catalytic Asymmetric Heck-Iminium Ion Cyclization
0128
Rhodium-Catalyzed Asymmetric 1,6-Addition of Aryl Zinc Reagents to Dienones
0129
Synthesis of Furans by the Pd-Catalyzed Oshima-Utimoto Reaction
0130
OsO4-Catalyzed Diastereoselective Formation of cis-Tetrahydrofurans
0131
Asymmetric Hydrogenation of tert-Alkyl Ketones
0132
Enantioselective Synthesis of 2-Aryl-4-piperidones
0133
Dual Ru(II)/Lipase-Catalyzed Dynamic Kinetic Resolution of Secondary Alcohols
0134
Enantioenriched Allylic Alcohols via sp-Carbon Coupling of Allenes
0135
Asymmetric Couplings of Ketenes with Aldehydes to Generate Enol Esters
0136
anti-1,2-Diols via a Ni-Catalyzed Reductive Coupling
0137
Catalytic, Enantioselective, Conjugate Alkyne Addition
0138
Enantioselective Diels-Alder Using a Bimetallic Catalyst
0139
Asymmetric Epoxidation of α,β-Unsaturated Esters With Yttrium-Biphenyldiol Complex
0140
Enantioselective Double C-H Activation of Dihydronaphthalenes
0141
Copper-Catalyzed Asymmetric Nitro-Mannich Reactions
0142
Sc(III)-Catalyzed Syn-Selective Enantioselective Carbonyl Ene Reactions
0143
N-(2-Hydroxyacetyl)pyrrole as an Ester Surrogate in Asymmetric Mannich Reactions
0144
Catalytic Enantioselective Fluorination of Oxindoles
0145
Pd-Catalyzed Asymmetric Allylation of Aldehydes using Allylic Alcohols
0146
Enantioselective Friedel-Crafts Alkylations of α,β-Unsaturated 2-Acyl Imidazoles
0147
Diastereoselective [2+2] Cyclizations

Metal-Mediated Synthesis

0149
Cyclopropanation and Carbonyl Olefination of Alkynylsilyldithianes via Titanium Alkynyl­-carbenes
0150
A Robust and Versatile Allyl- and Crotylboration with a Recyclable Auxiliary
0151
Ni(II)-Catalyzed Arylation of Diarylamines
0152
One-Pot Synthesis of Spiro-Cyclopropanes from Oxoallylsilanes
0153
Enantioselective Allylation of Hydrazones by Allylindium Complexes
0154
A New Synthesis of Amides from Imines, Acid Chlorides and Organostannanes
0155
Pd-Catalyzed Coupling of Arylboronic Esters with Carbamoyl Chlorides
0156
Multicomponent Reactions Based on Dilithio Ketone α,β-Dianions
0157
Ti-Catalyzed Reductive Coupling of Terpenic Allylic Halides
0158
Rh-Catalyzed Cross-Coupling Reactions and Arylation of Benzonitrile
0159
Directed Metalation and Cross-Coupling of N,N-Dialkyl Aryl O-Sulfamates
0160
Asymmetric Conjugate Addition of Arylalkynes to Nitroolefins
0161
Copper-Catalyzed Arylation of Sulfoximines with Arylboronic Acids
0162
Base-Promoted Dimerization of Terminal Epoxides
0163
BF3-Substituted 1,3-Dienes and Their Diels-Alder/Cross-Coupling Reactions

Organo- and Biocatalysis

0165
Chiral Brønsted Acid Catalyzed Hydrophosphonylation of Imines
0166
Proline-Based N-Oxides as Modular Chiral Catalysts for Allylation

Polymer-Supported Synthesis

0167
Immobilization of Bis(oxazolinyl)pyridines
0168
The First Solid-Phase Synthesis of Bis(oxazolinyl)pyridine Ligands
0169
‘Volatilizable’ Supports for High-Throughput Organic Synthesis
0170
Polymer-Supported Acetylating Agent for the Kinetic Resolution of Amines
0171
Solid Phase Synthesis of Small Heterocyclic Scaffolds
0172
Synthetic Procedure for Azidoalcohols Utilizing Polymer-Supported Reagent
0173
A Thermomorphic Polymeric Catalyst for Alcoholic Oxidation
0174
Solid Phase Synthesis of α,α-Disubstituted Amino Acid Derivatives
0175
Selective Monoarylation of Dibromoarenes with Polymeric Palladium Catalyst
0176
Proline Editing: A New Strategy for the Diversity-Oriented Peptide Synthesis
0177
Universal Strategy for the Immobilization of Chiral Dirhodium Catalysts
0178
Reversible Substrate Anchoring in Solid-Supported Organic Synthesis
0179
Asymmetric Reduction of Ketones Catalyzed by a Polymeric Chiral Ru Complex
0180
Asymmetric Diels-Alder Reaction Using a Polymer-Supported N-P Type Ligand
0181
PGA-Catalyzed Hydrolysis of Phenylacetic Hydrazides on a Solid Phase