DOI: 10.1055/s-00000084

Synthesis

Issue 20 · Volume 44 · October 2012 DOI: 10.1055/s-002-23872

review

  • 3109
    Silva, Eduarda M. P.; Silva, Artur M. S.:

    1,6-Conjugate Addition of Nucleophiles to α,β,γ,δ-Diunsaturated Systems

    Image for article: 1,6-Conjugate Addition of Nucleophiles to α,β,γ,δ-Diunsaturated Systems

    • feature article

  • 3129
    Zhu, Feng; Zhou, Feng; Cao, Zhong-Yan; Wang, Chao; Zhang, Yong-Xue; Wang, Cui-Hong; Zhou, Jian:

    A Facile Method for the Synthesis of 3-Substituted 3-(Alkylthio)oxindoles or 3-Alkoxyoxindoles

    Image for article: A Facile Method for the Synthesis of 3-Substituted 3-(Alkylthio)oxindoles or 3-Alkoxyoxindoles
    Supporting Information (PDF)

    • practical synthetic procedures

  • 3145
    Ichibakase, Tomonori; Nakajima, Makoto:

    Efficient Preparation of 1,3-Diol Derivatives with Three Contiguous Stereocenters by an Enantioselective Direct Aldol–Tishchenko Reaction

    Image for article: Efficient Preparation of 1,3-Diol Derivatives with Three Contiguous Stereocenters by an Enantioselective Direct Aldol–Tishchenko Reaction
  • 3152
    Bahnck, Kevin B.; Shavnya, Andrei; Tao, Yong; Lilley, Susan C.; Andrews, Melissa P.; Aspnes, Gary E.; Bernhardson, David J.; Bill, David R.; Bundesmann, Mark W.; Dow, Robert L.; Karki, Kapil; Le, Tung; Li, Qifang; Munchhof, Michael J.; Nematalla, Asaad; Nihlawi, Mohammed; Patel, Leena; Perreault, Christian; Waldo, Michael:

    Efficient Synthesis of 4-Amino-2-methoxy-7,8-dihydropyrido[4,3-d]pyrimidin-5-ones: Practical Access to a Novel Chemotype in the Development of DGAT-1 Inhibitors

    Image for article: Efficient Synthesis of 4-Amino-2-methoxy-7,8-dihydropyrido[4,3-<i>d</i>]pyrimidin-5-ones: Practical Access to a Novel Chemotype in the Development of DGAT-1 Inhibitors

    • short paper

  • 3158
    Chapyshev, Sergei V.; Chernyak, Alexander V.:

    Synthesis of 2,4,6-Triazidopyridine and Its 3,5-Diiodo Derivative

    Image for article: Synthesis of 2,4,6-Triazidopyridine and Its 3,5-Diiodo Derivative

    • paper

  • 3161
    Kim, Hyun-Soo; Lee, Sang-Jin; Choi, Boram; Yoon, Cheol Min:

    Heck Reaction of Baylis–Hillman Adducts with Iodobenzenes Using a Catalytic Amount of Pd/C under Solvent-Free Conditions

    Image for article: Heck Reaction of Baylis–Hillman Adducts with Iodobenzenes Using a Catalytic Amount of Pd/C under Solvent-Free Conditions
  • 3165
    Kim, Bong Chan; Park, Aeri; An, Ji Eun; Lee, Won Koo; Lee, Hee Bong; Shin, Hyunik:

    Highly Improved Copper-Mediated Michael Addition of Ethyl Bromodifluoroacetate in the Presence of Protic Additive

    Image for article: Highly Improved Copper-Mediated Michael Addition of Ethyl Bromodifluoroacetate in the Presence of Protic Additive
    Supporting Information (PDF)
  • 3171
    Gomi, Noriaki; Kouketsu, Akiyasu; Ohgiya, Tadaaki; Shibuya, Kimiyuki:

    A Practical Synthesis of (S)-tert-Butyl 3-Methyl-1,4-diazepane-1-carboxylate, the Key Intermediate of Rho–Kinase Inhibitor K-115

    Image for article: A Practical Synthesis of (<i>S</i>)-<i>tert</i>-Butyl 3-Methyl-1,4-diazepane-1-carboxylate, the Key Intermediate of Rho–Kinase Inhibitor K-115
  • 3179
    Nakano, Hayato; Kutsumura, Noriki; Saito, Takao:

    Functionalized Carbodiimide Mediated Synthesis of 2,3-Disubstituted Quinazolin-4(3H)-ones via the Tandem Strategy of C-Nucleophilic Addition and Intramolecular NH-Substitution Cyclization

    Image for article: Functionalized Carbodiimide Mediated Synthesis of 2,3-Disubstituted Quinazolin-4(3<i>H</i>)-ones via the Tandem Strategy of C-Nucleophilic Addition and Intramolecular NH-Substitution Cyclization
    Supporting Information (PDF)
  • 3185
    Periasamy, Mariappan; Sanjeevakumar, Nalluri; Obula Reddy, Polimera:

    Convenient Methods to Access Chiral Camphanyl Amine Derivatives by ­Sodium Borohydride Reduction of d-(–)-Camphorquinone Imines

    Image for article: Convenient Methods to Access Chiral Camphanyl Amine Derivatives by ­Sodium Borohydride Reduction of <sc>d</sc>-(–)-Camphorquinone Imines
    Supporting Information (PDF)
  • 3191
    Qin, Wenling; Long, Sha; Panunzio, Mauro; Bongini, Alessandro:

    Catalyst-Free Amidation of Trimethylsilyl Ketene Imines with Isocyanates

    Image for article: Catalyst-Free Amidation of Trimethylsilyl Ketene Imines with Isocyanates
  • 3197
    Murai, Toshiaki; Ezaka, Tatsuya; Kato, Shinzi:

    Synthesis of γ,δ-Unsaturated Selenoamides via the Seleno-Claisen Rearrangement of in situ Generated Allylic Vinyl Selenides from Selenoamides and Allylic Bromides­

    Image for article: Synthesis of γ,δ-Unsaturated Selenoamides via the Seleno-Claisen Rearrangement of in situ Generated Allylic Vinyl Selenides from Selenoamides and Allylic Bromides­
  • 3202
    Righi, Giuliana; Bovicelli, Paolo; Marucci, Cristina; Tirotta, Ilaria:

    BF3·OEt2/TMSN3 Mediated Regioselective Azidolysis of Vinylaziridines

    Image for article: BF<SUB>3</SUB>·OEt<SUB>2</SUB>/TMSN<SUB>3</SUB> Mediated Regioselective Azidolysis of Vinylaziridines
    Supporting Information (PDF)
  • 3209
    Lauber, Markus Boris; Fröhlich, Roland; Paradies, Jan:

    Development of Tartaric Acid Derived Hydrogen-Bond Donors

    Image for article: Development of Tartaric Acid Derived Hydrogen-Bond Donors
  • 3216
    Ibrahim, Mohamed A.; Blaise, Emilie; Lozach, Olivier; Szalata, Claude; Schmitt, Martine; El-Etrawy, Abd-Allah. S.; Elagawany, Mohamed; El-Feky, Said A.; Abdel-Samii, Zakaria K.; Meijer, Laurent; Bourguignon, Jean-Jacques; Bihel, Frédéric:

    Palladium-Catalyzed Synthesis of Substituted Pyrido[2,3-d]pyridazines at Positions 5 and 8

    Image for article: Palladium-Catalyzed Synthesis of Substituted Pyrido[2,3-<i>d</i>]pyridazines at Positions 5 and 8
    Supporting Information (PDF)
  • 3225
    Lu, Xiao; Altharawi, Ali; Hansen, Emily N.; Long, Timothy E.:

    Phase-Transfer Catalysts in the O-Alkylation of 2-Hydroxynaphthoquinones

    Image for article: Phase-Transfer Catalysts in the O-Alkylation of 2-Hydroxynaphthoquinones
  • 3231
    Seki, Masahiko:

    An Efficient C–H Arylation of a 5-Phenyl-1H-tetrazole Derivative: A Practical Synthesis of an Angiotensin II Receptor Blocker

    Image for article: An Efficient C–H Arylation of a 5-Phenyl-1<i>H</i>-tetrazole Derivative: A Practical Synthesis of an Angiotensin II Receptor Blocker
  • 3238
    Budragchaa, Tuvshinjargal; Roller, Alexander; Widhalm, Michael:

    Regio- and Stereoselective Approach to 1,4-Ditertiary Carbinols from Dimethyl Tartrate

    Image for article: Regio- and Stereoselective Approach to 1,4-Ditertiary Carbinols from Dimethyl Tartrate