DOI: 10.1055/s-00000175

Arzneimittelforschung

Ausgabe 02 · Volume 56 · Februar 2006 DOI: 10.1055/s-002-22597

CNS-active Drugs · Hypnotics · Psychotropics · Sedatives

  • 59
    Almeida, Susana; Filipe, Augusto; Almeida, Ana; Antonijoan, Rosa; García-Gea, Consuelo; Gich, Ignasi; Barbanoj, Manuel; Caturla, Maria Cruz:

    Comparative Study on the Bioequivalence of Two Different Gabapentin Formulations

    • Lipid Reducers

  • 64
    Bradamante, Vlasta; Krnić, Žarka; Zrinski, Renata; Konjevoda, Paško; Reiner, Željko:

    Changes in Butyrylcholinesterase Activity and Serum Lipids after Oxprenolol and Glibenclamide Treatments in Non-diabetic Rats

    • Lipidsenker

  • 70
    Almeida, Susana; Filipe, Augusto; Almeida, Ana; Gich, Ignasi; Antonijoan, Rosa; Puntes, Montserrat; Barbanoj, Manuel; Caturla, Maria Cruz:

    Comparative Study on the Bioequivalence of Two Formulations of Pravastatin

    • Antiallergic Drugs · Antiasthmatics · Antitussives · Bronchodilators · Bronchosecretogogues · Mucolytics

  • 76
    Zimmer, Guido; Bernhörster, Markus; Pilz, Patrizius; Schuchmann-Fix, Jutta; Hüggelmeier, Rolf; Blüm, Nicole; Libertus, Herman:

    Mononuclear Cell Membranes: Stabilization by Reproterol and Cromoglycate, Destabilization by Fenoterol and Salbutamol

    • Antiosteoporotic Drugs · Chondroprotective Drugs

  • 84
    Almeida, Susana; Almeida, Ana; Filipe, Augusto; Penedo, Clarisse; Rocha, Alexandre; Lainesse, Audrey; Vallée, François:

    In vitro Disintegration and Dissolution and in vivo Bioequivalence of Two Alendronate Once-weekly Formulations

    • Antioxidants

  • 90
    Kurcer, Zehra; Iraz, Mustafa; Kelesyilmaz, Nedim; Kilic, Nermin; Olmez, Ercument:

    Beneficial Effects of Melatonin on Diaphragmatic Contractility and Fatigability in Escherichia coli Endotoxemic Rats

    • Antibiotics · Antiviral Drugs · Chemotherapeutics · Cytostatics

  • 96
    Bijev, Atanas:

    Synthesis and Preliminary Screening of Carbohydrazides and Hydrazones of Pyrrole Derivatives as Potential Tuberculostatics

  • 104
    Lotfy, Abeya A. M.; Ghanem, Lobna Y.; Shennawy, Amal M.; Gomaa, Nadia A.; El Said, Hamda H.:

    Assessment of the Toxicity of Artemisia inculta Extract on the Bone Marrow of Mice Infected with Schistosomiasis

    • Special Themes

  • 108
    Liedtke, Rainer K.:

    Pharmacological Concept for Topical Synergistic Analgesia of Peripheral Neuromuscular Pain

    • Book Reviews

  • 115

    Book Reviews

    • Preface

  • 117

    Unmet Challenges in HIV Therapy and Potential of Stampidine

    • Stampidine

  • 121
    Uckun, Fatih M.:

    Stampidine as a Novel Nucleoside Reverse Transcriptase Inhibitor with Potent Anti-HIV Activity

  • 136
    DuMez, Darin; Venkatachalam, Taracad K.; Uckun, Fatih M.:

    Large-Scale Synthesis and Formulation of GMP-Grade Stampidine, a New Anti-HIV Agent

  • 152
    Venkatachalam, Taracad K.; Qazi, Sanjive; Uckun, Fatih M.:

    Synthesis, Separation and Anti-HIV Activity of Distereoisomers of N-[p-(4-Bromophenyl)-2',3'-didehydro-3'-deoxy-5'-thymidylyl]-L-alanine Methyl Ester (Stampidine)

  • 159
    D'Cruz, Osmond J.; Erbeck, Douglas; Uckun, Fatih M.:

    Developmental Safety Profile of the Anti-HIV Agent Stampidine in Rabbits

  • 167
    Venkatachalam, Taracad K.; Qazi, Sanjive; Uckun, Fatih M.:

    Site-Specific Enzymatic Activation of the Anti-HIV Agent Stampidine

  • 176
    Uckun, Fatih M.; Waurzyniak, Barbara; Tibbles, Heather; Venkatachalam, Taracad K.; Erbeck, Doug:

    In vivo Pharmacokinetics and Toxicity Profile of the Anti-HIV Agent Stampidine in Dogs and Feline Immunodeficiency Virus-infected Cats

  • 193
    Uckun, Fatih M.; Venkatachalam, Taracad K.; Qazi, Sanjive:

    Potency of Stampidine Against Multi-Nucleoside Reverse Transcriptase Inhibitor Resistant Human Immunodeficiency Viruses