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Synthesis 1999; 1999(1): 138-144
DOI: 10.1055/s-1999-3681
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A Solid-Phase Synthesis of Functionalized 6-, 7- and 8-Membered Azacycles via Olefin Metathesis

Josef Pernerstorfer* , Matthias Schuster, Siegfried Blechert
  • *Institut für Organische Chemie der Technischen Universität, Straße des 17. Juni 135, D-10623 Berlin, Germany; Fax +49(30)31 42 36 19; E-mail: sibl@wap0105.chem.tu-berlin.de
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Publication Date:
31 December 1999 (online)

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A modular solid-phase synthesis of functionalized azacycles is described. The approach is based on a ring-closing metathesis to form heterocycles of different ring sizes. Furthermore, the epoxidation of the primarily formed cyclic double bond has been investigated.

metathesis - solid-phase synthesis - nitrogen heterocycles - epoxidation

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