DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 20 · September 2024 DOI: 10.1055/s-014-60079

Synform

  • A135

    SYNFORM ISSUE 2024/09

    • Synthesis of Natural Products

  • z0895

    All PDFs of this category

  • 0895

    Total Synthesis of (+)-Dihydropleurotinic Acid

  • 0896

    Synthesis of (+)-Enteropeptin A

  • 0897

    Total Synthesis of Sealutomicin C

  • 0898

    Total Synthesis of (+)-Alstrostine G

  • 0899

    Total Synthesis of (+)-Lirionol

  • 0900

    Total Synthesis of (–)-Cyclopamine

  • 0901

    First Synthesis of (±)-Retigeranic Acid

    • Synthesis of Heterocycles

  • z0903

    All PDFs of this category

  • 0903

    Bench-Stable Azabicyclo[2.1.1] Piperazinium Salt as a Versatile Synthetic Intermediate

  • 0904

    Enzyme-Catalyzed Access to Spiro-Oxazolidinones

  • 0905

    Photocatalyzed Enantioselective Access to Oxetanes

  • 0906

    Synthesis of 2,3-Dihydrofuro[3,2-c]quinolines via Acid-Mediated Condensation

  • 0907

    Versatile, Photochemical Approach to 2-Azanorbornanes

  • 0908

    Carboxylic-Acid-Directed Cyclization of N-Protected ω-Amino Acids

  • 0909

    Light-Mediated Deoxygenative Hydroalkylation of Olefins

  • 0910

    Hectogram Scale Synthesis of Key Prostaglandin Synthesis Intermediate

  • 0911

    Regioselective Difluoromethylation of Pyridines through Oxazino-pyridine Intermediates

  • 0912

    Synthesis of 2,3-Diaroylquinolines via Copper-Catalyzed [4+1+1] Annulation

  • 0913

    Modular Copper-Mediated Synthesis of Imidazolidines and Imidazolidinones

  • 0914

    Three-Component Photochemical Construction of Trisubstituted Oxazoles

  • 0915

    General Methodology for the α-Alkylation of Cyclic Ketones

  • 0916

    Same Substrates, Different Products: Regiodivergent Cycloaddition Pathways to 1,2,3- and 1,3,4-Triazoles

    • Synthesis of Materials and Unnatural Products

  • z0917

    All PDFs of this category

  • 0917

    Enantioselective Syntheses of π-Extended Carbohelicenes

  • 0918

    Spiro-Conjugated Chiral Radical Cations

  • 0919

    Nucleophilic Perfluoroalkylation Facilitated by 4-Pyridylthioether

  • 0920

    Backbone-Editing with Polyesters and Polyurethanes

  • 0921

    Triple Suzuki–Miyaura Arylation via Cyclic Iodonium Salts

  • 0922

    Joining Carborane with Arenes

  • 0923

    ‘Click’ Polymerization of Acetal-thiol

  • 0924

    Cyclic Polymers with Ultrahigh Molar Mass

  • 0925

    ‘Cage of Cages’

  • 0926

    Kinetic Resolution Polymerization

  • 0927

    Single-Atom Skeletal Editing: Turning N into C

  • 0928

    Isolable Secondary Carbon Radical

    • Metals in Synthesis

  • z0929

    All PDFs of this category

  • 0929

    Nickel- and Photocatalytic Enantioselective Alkylation of α-Amino C(sp3)–H Bonds

  • 0930

    Atroposelective Reductive Coupling of Two ortho-Substituted Aryl Halides under Nickel Catalysis

  • 0931

    Synthesis of Oximes by Nickel-Catalyzed Coupling of Nitrates with Organohalides

  • 0932

    Palladium-Catalyzed Cascade Reaction to Fused Isoindolinones

  • 0933

    Chromium-Catalyzed Enantioselective Addition of α-Chlorinated Esters and Amides to Aldehydes

  • 0934

    Nickel-Catalyzed Cine-Substitution of Enolates

  • 0935

    Enantioselective Synthesis of Highly Decorated Pyrrolidines Through a Zinc-Catalyzed [3+2] Reaction

  • 0936

    Synthesis of Chiral Allylic Alcohols by Enantioselective Alkenylation of Aldehydes Under Cobalt Catalysis

  • 0937

    Dearomative 1,2-Hydroamination of Nonactivated Arenes via Copper–Hydride Catalysis

  • 0938

    Synthesis of Anilines by Ruthenium/η5-Phenoxo-Catalyzed Condensation of Phenols and Amines

  • 0939

    Asymmetric Arylation of Enone Diesters Enabled by Synergistic Copper Catalysis

  • 0940

    Selective Palladium Visible Light Catalyzed Ether/Esterification of Allylic C–H Bonds

  • 0941

    Gold-Catalyzed Electrophilic Cyclopropenylation of Terminal Alkynes and Vinyl Boronic Acids

  • 0942

    Nickel-Catalyzed α-anti-Hydroarylation of Arylpropiolic Acids and Arylboronic Acids

  • 0943

    Asymmetric Aminooxygenation of 1,3-Dienes Enabled by Copper Catalysis

  • 0944

    Copper-Catalyzed Borylative Cyclization of Unactivated Vinylcyclopropanes

  • 0945

    Palladium-Catalyzed Chain-Walking of Alkynyl Alcohols to α,β-Unsaturated Carbonyls

  • 0946

    Asymmetric β-Arylation of Aliphatic Alcohols by Merging Relay Catalysis and Dynamic Kinetic Resolution

  • 0947

    Palladium-Catalyzed Spirocyclopropanation of gem-Difluoroalkenes

  • 0948

    Enantioselective Rhodium-Catalyzed N2-Allylation of Indazoles with Dienyl Allylic Alcohols

  • 0949

    Iridium-Catalyzed Allylation of Bis(alkenyl)boronates to Access Enantioenriched Tertiary Allylic Boronic Esters

  • 0950

    Separation by Isomerization: Kinetic Resolution of N-Allylic Pyrazoles under Photoexcited Copper Catalysis

  • 0951

    Semipinacol Rearrangement of Allylic Alcohols under Dual Photoredox and Cobalt Catalysis

  • 0952

    Decarboxylative C(sp3)–O Coupling Enabled by an Iron Ligand-to-Metal Charge Transfer

  • 0953

    Nickel/Photoredox-Catalyzed C(sp3)–H Alkenylation

  • 0954

    Dearomative Carbonylative trans-1,2-Difunctionali-zation of Arenes via Chromium–Arene Complexes

  • 0955

    Synthesis of anti-1,3-Diols: The Evans–Tishchenko Reaction

    • Polymer-Supported Synthesis

  • z0957

    All PDFs of this category

  • 0957

    Pd Nanoclusters Supported on N-Doped Carbon Spheres for Hydrogenation of Phenols and Benzoic Acids

  • 0958

    Hydrogenation of Arenes at Room Temperature under 1 atm of Hydrogen Gas by Rh-Pd/C or Rh-Pt

  • 0959

    Selective Hydrogenation of Aldehydes and Ketones under Syngas Using Au NPs Supported on CeO2

  • 0960

    Solvent-Free Aerobic Oxidation of C(sp3)–H by a Carbon- and PdO-Doped Nb2O5 Photocatalyst

  • 0961

    Hydrogenation of Dinitroarenes Catalyzed by Pt Clusters on a Graphene Shell with a Diamond Core

  • 0962

    Photocatalytic Thio/Selenocyanation of Indoles Using Lead-Free Cs2AgBiBr6 Double Perovskite MCs

  • 0963

    Nickel-Catalyzed C(sp2)–S Cross-Coupling with mpg-CN under Blue LED Irradiation

  • 0964

    Dehydrogenative Silacyclization with a Porous Polymer-Supported Iridium Catalyst

  • 0965

    Catalytic Transfer Hydrogenation of Carbonyls by SILP-Supported Manganese Nanoparticles

  • 0966

    Enantioselective [2+2] Cross-Photocycloaddition Using a Homochiral Metal–Organic Cage Reactor

  • 0967

    Photocatalytic Oxidative Bromination of Arenes by Al2O3-Supported Perylenetetracarboxylic Dianhydride

    • Organo- and Biocatalysis

  • z0969

    All PDFs of this category

  • 0969

    Photocalatytic C–H Alkylation Enabled by a Zwitterionic Acridinium Amidate Catalyst

  • 0970

    Asymmetric Synthesis of Seven-Membered N-Heterocycles and Carbocycles

  • 0971

    Alcohol-Directed Functionalization of Remote C–H Bonds

  • 0972

    Organocatalytic Asymmetric Epoxidation of Alkenyl Aza-Heteroarenes

  • 0973

    Consecutive Photoinduced Electron Transfer Enables Asymmetric [3+2] Cycloadditions

  • 0974

    Confined Acid Catalyzes the Enantioselective Hydroamination of Non-Activated Olefins

  • 0975

    Solid-State Preorganization Enables Highly-Selective [2+2] Cycloaddition towards Truxillates

  • 0976

    Organophotocatalytic Method for Synthesis of α-Amino Bicycloalkanes – Pharmaceutically Relevant Molecules

  • 0977

    Synergistic Catalytic Asymmetric Decarboxylation of β-Keto Acids with Acyclic α-Arylenamides

  • 0978

    Photoorganocatalytic Reduction of Esters to Alcohols

    • Innovative Drug Discovery and Development

  • z0979

    All PDFs of this category

  • 0979

    Synthesis and Medicinal Chemistry of Veragranine Alkaloids

  • 0980

    Functionalization of Oxetanes with C/N/O/S Nucleophiles – Convenient Access to Carbonyl Isosteres

  • 0981

    High-Throughput Access to Libraries of N-Acylsulfamide Derivatives, a Bioisostere of Carboxylic Acids

  • 0982

    Amination of Arenes Using Blue Light and Lewis Acids

  • 0983

    Vinylpyridine Based Covalent EGFR Inhibitors

  • 0984

    Photochemical Conversion of Pyridines into Diazepines, Pyrazolines and Pyrazoles

  • 0985

    Divergent Synthesis of 2- and 3-Azabicyclo[3.1.1]heptenes as Bioisosteres of Pyridines

  • 0986

    Development of the Photoresponsive Drug via Caging Triarylimidazoles

  • 0987

    An Eight-Step Total Syntheses of Clausenawallines A and E are Enabled by High-Throughput Experimentation

  • 0988

    HRO761: a First-in-Class Non-Covalent WRN Inhibitor with Synthetic Lethality in MSI Cancers

  • 0989

    A Modified Arbuzov–Michaelis Reaction for Chemoselective Alkylations

  • 0990

    New Method for the Highly Enantioselective Synthesis of cis-Hydrobenzofurans and cis-Hydroindoles

  • 0991

    Synthesis of a Selective Co-factor to Investigate Methyltransferase Activity

  • 0992

    Subcellular Uncaging of H2S and Drug with NIR Light

  • 0993

    Diverse Synthesis of C‑Glycosides by Stereoselective Ni-Catalyzed Carboboration of Glycals

  • 0994

    Expanding Chemical Space One Carbocycle at a Time

    • Peptide Chemistry

  • z0995

    All PDFs of this category

  • 0995

    N-Methylated Peptide Synthesis Using Flow Chemistry

  • 0996

    α,α-Disubstituted Unnatural Amino Acid Synthesis Using Photochemical Carboxylation

  • 0997

    Chiral Phenanthroline-Potassium-Catalyzed Synthesis of Axially Chiral Biaryl δ-Amino Acid Derivatives

  • 0998

    Utilizing Cyclen Installation as an Efficient Strategy for Macrocyclization and Multifunctionality of Peptides

  • 0999

    Synthesis of Proline Derivatives via [1,2]-Stevens Rearrangement of Azetidinium Salts

  • 1000

    Synthesis of Unprotected α-Tertiary Amino Acids Using Synergistic Photoenzymatic Catalysis

  • 1001

    Macrocyclic Thiazol(in)e Peptide Synthesis from Peptide Nitriles Using a Biocompatible Strategy

  • 1002

    Electrochemical Modification of Tryptophan and Tryptophan-Containing Peptides

  • 1003

    Tertiary Amine Catalyzed Late-Stage Tryptophan Allylation of Peptides

  • 1004

    Synthesis of Functionalized Diketopiperazines

  • 1005

    Photocatalyzed Synthesis of Unnatural α-Amino Acids

  • 1006

    Asymmetric Synthesis of α,α-Disubstituted α-Amino Acid Esters via Tsuji–Trost Allylation

  • 1007

    O-Hydroxybenzenesulfonyl Chloride Mediated Peptide Synthesis

    • Flow Chemistry

  • z1009

    All PDFs of this category

  • 1009

    Photocatalyst-, Oxidant-, Additive-Free Nitrosylation Using Continuous Flow/Photochemical Conditions