Synfacts

Issue 10 · October 2023

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A167
SYNFORM ISSUE 2023/10 FREE ACCESS

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Synthesis of Natural Products
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0955
Total Synthesis of (–)-Cephinoid P FREE ACCESS

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0956
Total Synthesis of (+)-Aspidospermidine

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0957
Synthesis of (–)-Eugenial C

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0958
Synthesis of (+)-Pleiocarpamine and (+)-Bipleiophylline

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0959
Synthesis of (–)-Polyavolensinol and (–)-Greenwaylactam A

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0960
Total Synthesis of (+)-Lancilactone C

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0961
Synthesis of (±)-Nominine FREE ACCESS

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Synthesis of Heterocycles
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0963
Cu-Mediated Cyclization to Form 1H-Indazoles

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0964
Synthesis of Highly Substituted BN-9,1-Naphthalenes from BN-Butafulvenes

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0965
Revalorization of Nitrous Oxide for Use as an Oxygen-Transfer Reagent

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0966
Cp*Co(III)-Catalyzed Synthesis of Isoquinolones via Regioselective [4+2] Annulation of N-Chlorobenzamides

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0967
Secondary Amines from Ammonia Surrogate – Aminopyridinium Salts

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0968
Application of Strained Heterocycles as Electrophiles in Ni/Ir-Catalyzed Cross-Couplings

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0969
Synthesis of Substituted 2-Oxabicyclo[2.1.1]hexanes via [2π+2σ] Cycloadditions with Bicyclobutanes FREE ACCESS

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0970
Mechanism-Driven Development of a Novel Amide Directing Group for Directed C–H Functionalization

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0971
Validation, Development and Execution of an Automated Protocol for C–C Cross-Couplings

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0972
Access to Spiro-oxetane Oxindoles via DBU-Catalyzed Activation of Allenoates

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0973
General, Direct Ni-Catalyzed Cross-Coupling of Tertiary Synthons with Heteroaryl Halides

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Synthesis of Materials and Unnatural Products
z0975
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0975
Introducing Double Bonds to Polyolefins via Retro-Diels–Alder Reaction FREE ACCESS

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0976
One-Pot Synthesis of Benzo[c]phenanthridines

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0977
Reactivity of 1,2,3-Triazines and the Oxides

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0978
Difunctionalization Applied to Polymerization

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0979
Stoichiometry-Controlled Boration of Terminal Alkynes

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0980
Phenols from [3+3] Cycloaddition

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0981
All-Fused Rubicene Dimers and Trimers

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0982
1,3-Dipolar Cycloaddition Involving Arenes

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0983
Hydrolytically Stable Molecular Cage

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0984
Benzo[a]aceanthrylene from [4+2] Cyclization

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0985
Large Circumacene with a Pentacene Center

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0986
Negatively Curved Nanocarbons with Heptagon Modules

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Metals in Synthesis
z0987
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0987
Silver(I)-Catalyzed Rearrangement of 1,4-Disubstituted Cubanes to 1,3- or 2,6-Disubstituted Cuneanes FREE ACCESS

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0988
Pd/Charcoal Catalyzed Reduction of Vinyl Geminal Diboronates

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0989
Copper-Catalyzed Difluoroalkylation of Silyl-Enol Ethers FREE ACCESS

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0990
Regioselective Three-Component Intermolecular Dialkylation of Styrenes Enabled by Nickel Catalysis

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0991
Enantioselective Three-Component Synthesis of Trifluoromethylated Propargylic Ethers and Anilines

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0992
Iridium-Catalyzed Atroposelective Synthesis of Silylated 2-Arylisoquinolines via C–H Activation

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0993
ε-exo-Alkylidene ε-Lactones Synthesis via Cooperative Gold/Zinc-Catalyzed 7-exo-dig Cyclization

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0994
Oxoamination of Terminal Alkenes under Visible-Light-Induced Ruthenium Catalysis

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0995
Iridium-Catalyzed Asymmetric Allylic Alkylation via 1,2-Boryl Migration and Dynamic Kinetic Resolution

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0996
Rh-Catalyzed Unsymmetrical Heterobiaryl Synthesis via a Dual C–H Activation Cross-Coupling Process

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0997
Rapid Construction of Carbazole Frameworks through Gold-Catalyzed Cyclizations and [3+2] Annulation

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0998
Iron-Catalyzed C(sp³)–H Phosphorylation Enabled by Photoinduced Ligand-to-Metal Charge Transfer

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0999
Photoinduced Copper-Catalyzed Borylation of Non-Activated Alkanes

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1000
Pd-Catalyzed Synthesis of Spirocyclohexaneindolenines from Bromoarene-Tethered Indoles and Alkynes

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1001
Bismuth-Catalyzed Decarboxylative Amination of α-Amino Alkyl Phthalimide Esters with N-Heterocycles

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1002
Palladium/Copper Bimetallic-Catalyzed Direct C–H Heteroarylation of N-Methylpyridinium Salts

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1003
Nickel/Photoredox-Catalyzed Thioesterification of Carboxylic Acids Enabled by Sensitized Electron Transfer

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1004
Cobalt-Catalyzed Reductive Coupling of Nitroarenes and Formaldehyde to N,N'-Diarylethane-1,2-diamines

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1005
Ag-Catalyzed Synthesis of Functionalized Benzo[d]azepines

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1006
Access to Azacycles by Cobalt-Catalyzed Asymmetric Cross-Electrophile Coupling

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1007
Ruthenium-Catalyzed Intramolecular Cycloaddition of Cyclopropenynes and Cyclopropendiynes

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1008
Negishi Cross-Coupling Using Cobalt

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1009
Rhodium-Catalyzed Borylative Cyclization of Enynes

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1010
Synthesis of α-Fluoro-β-Ketophosphonates through Rh-Catalyzed Hydration/C–F Bond Cleavage

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1011
Coupling of Ketyl and Alkyl Radicals Generated under Photoredox Cooperative NHC/Palladium Catalysis

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1012
Co-Catalyzed Three-Component 1,2-Dialkylation of Alkenes Using Novel Salt-Stabilized Alkylzinc Pivalates

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1013
Sequential Borane- and Pd-Catalyzed C3-Allylation of Pyridines via a DYKAT Process

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Polymer-Supported Synthesis
z1015
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1015
Hydrogenation of N-Heterocycles Using Frustrated Lewis Pairs Incorporated in NU-1000 MOF FREE ACCESS

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1016
Hydrogenation of Arenes by Cobalt Nanoparticles Supported on Biomass-Derived Carbons

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1017
Reduction of Nitroarenes to Azoxy-, Azo-, and Hydrazo Compounds Promoted by Bismuth Porphyrin MOF

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1018
Visible-Light-Induced Cyclization of N-Phenyl-benzothioamides Using β-Ketoenamine-Linked COF

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1019
Bifunctional Catalysts with Core–Shell Distributed ZrO₂/Co NPs for Hydrogenation–Formylation of Nitroarenes

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1020
Preparation of Silica-Gel-Supported Photocatalysts

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1021
Photochemical Synthesis of Benzimidazoles Promoted by Palladium-Decorated ZnO Nanosheets

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1022
Photocatalytic C–H Amination of Arenes by a Ruthenium Complex on Faujasite-Type Zeolite

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1023
Photocatalytic Aerobic Oxidations by a 2D Microporous Covalent Organic Framework

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1024
A COF-Supported Cd(II) Catalyst for Carboxylative Cyclization of CO₂ with Propargylamines

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1025
Photocatalytic Dehydrogenative [4+2] Annulation of Benzothioamides with Alkynes Using g-C₃N₄

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1026
Ni-Catalyzed C–C Bond Forming Cross-Coupling of Aryl/Alkyl Halides with a Quantum Dots Photocatalyst

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Organo- and Biocatalysis
z1027
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1027
Synthesis of Eight-Membered Carbocycles by (I)/I(III)-Catalyzed Diene Cyclization FREE ACCESS

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1028
Ene-Reductase Outcompetes Hydrogen Atom Transfer in Asymmetric Carbohydroxylation of Alkenes

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1029
Photoredox Catalysis Enables New Synthetic Route Toward Oxetanes

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1030
Cytochrome P450-Derived Ketone Synthase Enables Regioselective Aerobic Oxidation of Arylalkenes

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1031
Enantioselective Protio-Semipinacol Rearrangement of Vinyl Cyclopropanols

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1032
N-Triflyl Phosphoramide Catalyzed Atroposelective C–C Cross-Coupling of 1-Azonaphthalenes

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1033
Photosensitized O₂Permits a Versatile Cyclopropanation Reaction

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1034
Direct, Additive-Free Electrochemical Dehydrative Esterification of Carboxylic Acids and Alcohols

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Innovative Drug Discovery and Development
z1035
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1035
Stereoselective Robinson Annulation Enables Access to Potent and Selective Salvinorin Analogs FREE ACCESS

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1036
Converting DNA-Encoding Ligands into BRET Probes

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1037
Identifying the Risk of Formation of Nitrosamines and Other Potentially Mutagenic Impurities during API Manufacture Using In Silico Risk Assessment

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1038
A Pathway-Selective Photoswitch for Understanding Cannabinoid 2 Receptor

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1039
Late-Stage Aryl C–H Bond Cyclopropenylation with Cyclopropenium Cations

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1040
Optimization of Cyclic Peptide Hits to Identify Clinical KRAS-SOS1 PPI Inhibitor, LUNA18

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1041
Toward Improved On-Target Safety: Discovery of Potent, Short Half-Life Macrocyclic Inhibitors of Mcl-1 FREE ACCESS

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1042
Design and Synthesis of MK-8768: a Potent and Selective mGluR2 Negative Allosteric Modulator

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1043
Transition Metal-Free syn-Dihydroxylation via Interrupted Ozonolysis

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1044
Cubane and Cyclooctatetraene Used as Bioisosteres in Drug Development

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1045
Initiation of Fluorescence and Bioactivity Using UV Light Photocage on PI3K Inhibitor

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1046
Synthesis of N-Acylsulfonamide Derivates: New Sulfa Drug Analogues by Sulfo-Click Reaction

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1047
CF₂X, a New Halogen Bond Donor Motif with Potential in Drug Design

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1048
Amide Derivatization Through Amino Acid Insertion

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1049
para-Selective Functionalization of Pyridines

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Peptide Chemistry
z1051
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1051
Rh-Catalyzed Maleimidation of Trp-Including Peptides FREE ACCESS

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1052
One-Pot Enantioselective Synthesis of α‑Amino Acid Esters

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1053
Synthesis of Small Cyclic Peptides Containing N-Methyl and β-Amino Acids

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1054
Asymmetric Synthesis of α-Sulfinamido Trithioformates and Transformation to Peptides

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1055
Co-Catalyzed Enantioselective Hydrogenation to Form Indazole-Containing Amino Acids

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1056
Palladium-Catalyzed Late-Stage Functionalization of Phenylalanine and Phenylalanine Derived Peptides

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1057
Cu-Catalyzed Three-Component Coupling for the Synthesis of α-Aryl α-Amino Acid Derivatives

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1058
Macrocyclization of Oligopeptides via Introduction of a Hypervalent Iodine Reagent

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1059
Direct Catalytic Asymmetric Synthesis of α-Alkylated α,α-Disubstituted Amino Esters

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1060
Photocatalyzed C–H Functionalization of Trp-Including Peptides

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1061
Ring-Opening of Aziridine Carboxylates for the Synthesis of Tryptophan Derivatives FREE ACCESS

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Flow Chemistry
z1063
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1063
Atroposelective Dual Catalysis in Flow

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1064
A Continuous-Flow Electron-Poor-Arene Dearomatization via Photocatalyzed Cycloaddition

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