Synfacts

Issue 10 · October 2021

Recommend Journal

Synform
A157
SYNFORM ISSUE 2021/10
FREE ACCESS

PDF (1900 kb)
Synthesis of Natural Products and Potential Drugs
z1071
All PDFs of this category

PDF (445 kb)
1071
Synthesis of Sotorasib
FREE ACCESS

HTML

PDF (131 kb)
1072
Synthesis of (+)-Davisinol

HTML

PDF (80 kb)
1073
Synthesis of (–)-Talatisamine and (–)-Liljestrandisine
FREE ACCESS

HTML

PDF (130 kb)
1074
Synthesis of Anti-Malarial MMV390048

HTML

PDF (80 kb)
1075
Total Synthesis (+)-Pepluanol A

HTML

PDF (93 kb)
1076
Synthesis of Pemigatinib

HTML

PDF (80 kb)
1077
Total Synthesis of (+)-Ambiguine G

HTML

PDF (91 kb)
1078
Synthesis of (+)-Mannolide C

HTML

PDF (91 kb)
1079
Total Synthesis of (+)-Prostratin

HTML

PDF (96 kb)
1080
Synthesis of (±)-Pentacycloanammoxic Acid Methyl Ester
FREE ACCESS

HTML

PDF (141 kb)
Synthesis of Heterocycles
z1081
All PDFs of this category

PDF (223 kb)
1081
Synthesis of Silazacycles from the Elusive 3-Silaazetidine

HTML

PDF (92 kb)
1082
Synthesis of 2,1-Benzisoxazoles via Decyanative Cyclization

HTML

PDF (75 kb)
1083
Direct Preparation of N-Substituted Pyrazoles from Primary Aliphatic or Aromatic Amines

HTML

PDF (83 kb)
1084
Dithioesters as Thiocarbonyl Precursors in Thorpe–Ziegler-Type Cyclization

HTML

PDF (80 kb)
1085
Regiospecific Three-Component Synthesis of 2-Aminothiophenes

HTML

PDF (91 kb)
1086
Rh-Catalyzed Synthesis of Thienoacenes from Thiophenes

HTML

PDF (95 kb)
1087
Direct C–H Functionalization of N-Heteroaromatics with Cyclic Ethers

HTML

PDF (74 kb)
Synthesis of Materials and Unnatural Products
z1089
All PDFs of this category

PDF (301 kb)
1089
Dendritic Donor for Good π-Stacking

HTML

PDF (94 kb)
1090
A Tetrathia[8]circulene–Azaborine Fusion

HTML

PDF (79 kb)
1091
Living Helix

HTML

PDF (69 kb)
1092
Synthesis of Stereogenic Fluoroborate as a Fluorophore with an Increased Stokes Shift

HTML

PDF (71 kb)
1093
Nitrogen Incorporation in a Nanographene through Direct Oxidative Cyclization

HTML

PDF (80 kb)
1094
A Benzene- Bridged Bismacrocycle

HTML

PDF (73 kb)
1095
Metal-Free Oxidative Decarboxylative Coupling

HTML

PDF (72 kb)
1096
Easy Access to a Nitrogen- Doped Aromatic Belt with a [6]Cycloparaphenylene Skeleton

HTML

PDF (77 kb)
1097
Efficient Synthesis of a Novel Benzo-Incorporated Smallest Expanded Calix[4]pyrrole

HTML

PDF (83 kb)
1098
A New Meta in meta-Halophenol Synthesis

HTML

PDF (97 kb)
1099
Thiolated Pillar[5]arene and Its Supramolecular-Complexation-Accelerated Dimerization

HTML

PDF (80 kb)
1100
Calix[3]-Type Macrocycles: The Missing Family Member

HTML

PDF (69 kb)
Metals in Synthesis
z1101
All PDFs of this category

PDF (673 kb)
1101
Denitrogenative Ring Shrinkage of Heterocycles
FREE ACCESS

HTML

PDF (137 kb)
1102
Synthesis of Chiral Cyclopropane-1-Carboxylates

HTML

PDF (81 kb)
1103
One-Pot α,α′-Difunctionalization of Cyclic Amines

HTML

PDF (83 kb)
1104
Trifluoroacetylation of Styrenes

HTML

PDF (81 kb)
1105
Copper-Catalyzed Arene Ring Cleavage

HTML

PDF (70 kb)
1106
Enantioselective Rhodium-Catalyzed Synthesis of Fluorinated Allenes

HTML

PDF (84 kb)
1107
Iron-Catalyzed Cross-Coupling of Propargyl Ethers with Grignard Reagents

HTML

PDF (86 kb)
1108
Stereoselective Synthesis of (E)-δ-Vinyl-Homoallylic Alcohols from α-Vinyl Allylboronate

HTML

PDF (104 kb)
1109
Preparation of Chiral Allylic Alcohols by Asymmetric Reduction of Substituted Cycloalkenones

HTML

PDF (85 kb)
1110
Vinylation of Aldehydes through Twofold C–H Functionalization

HTML

PDF (80 kb)
1111
Rhodium-Catalyzed Alkynylcyclopropanation of Alkenes Using Alkynylcycloheptatrienes

HTML

PDF (99 kb)
1112
Iridium-Catalyzed Alkenylation of Enamides

HTML

PDF (81 kb)
1113
Preparation of (Het)arylgermanes

HTML

PDF (72 kb)
1114
Palladium and Ammonium Halide Catalysis for Enantioselective [4+2] Annulations

HTML

PDF (85 kb)
1115
Enantio- and Diastereoselective Synthesis of Trifluoromethyl-Cyclopropylboronates

HTML

PDF (73 kb)
1116
Directed Nickel-Catalyzed Hydrofunctionalization of Alkenes

HTML

PDF (78 kb)
1117
Synthesis of gem-Difluorohomoallylic Alcohols by Reductive Defluorinative Coupling

HTML

PDF (90 kb)
1118
Palladium-Catalyzed Benzylic C(sp³)–H Carbonylative Arylation of Azaarylmethyl Amines

HTML

PDF (80 kb)
1119
Nickel-Catalyzed Ring-Opening Allylation of Cyclopropanols with Allylic Carbonates

HTML

PDF (78 kb)
1120
Rhodium-Catalyzed Stereoselective Synthesis of Enones and Enals from 2,3-Allenols and Organoboronic Acids
FREE ACCESS

HTML

PDF (119 kb)
1121
Copper-Catalyzed Amination of Secondary Alkyl Iodides

HTML

PDF (78 kb)
1122
Stereodivergent Aldehyde α-Allylation with 1,3-Dienes

HTML

PDF (93 kb)
1123
Palladium-Catalyzed Dearomatization of Nitroindoles

HTML

PDF (79 kb)
1124
Palladium-Catalyzed Carbonylative-Amination Reaction Generating Fluorinated β-Lactams

HTML

PDF (90 kb)
1125
Regiodivergent Hydroalkenylation of 1,6-Enynes with Acrylates and Alkenes

HTML

PDF (86 kb)
1126
Nickel-Catalyzed Cross-Coupling of α-Magnesiated Nitriles by Using a Benzonitrile Ligand

HTML

PDF (86 kb)
Polymer-Supported Synthesis
z1127
All PDFs of this category

PDF (314 kb)
1127
Selective Synthesis of Imines and Secondary Amines by Homocoupling of Primary Amines

HTML

PDF (77 kb)
1128
Cobalt-Catalyzed Synthesis of Tetrahydropyridine Derivatives and Oxidation of Benzylic Alcohols

HTML

PDF (103 kb)
1129
Zirconium Metal–Organic Framework Catalyzed Direct Amide-Bond Formation
FREE ACCESS

HTML

PDF (139 kb)
1130
Hydrogenation of Quinolines Catalyzed by Tungsten- Doped Cobalt Nanoparticles

HTML

PDF (74 kb)
1131
N-Alkylation of Amines with Aldehydes Catalyzed by a Graphene-Co-Shelled Ni/NiO@C Nanocatalyst

HTML

PDF (85 kb)
1132
Synthesis of Pyrans by a Zirconium-Catalyzed Three-Component Condensation

HTML

PDF (72 kb)
1133
Ruthenium-Catalyzed Transformations of 2,5-Hexanediones into Furans or Pyrrolidines

HTML

PDF (75 kb)
1134
Controlled Hydrogenation of Azoarenes to Hydrazoarenes on Palladium/Carbon

HTML

PDF (75 kb)
1135
Aerobic Oxidation of α-Diazo Esters Catalyzed by Charcoal-Supported Copper Nanoparticles

HTML

PDF (93 kb)
1136
Palladium-Catalyzed α-Arylation of Ketones in Water

HTML

PDF (93 kb)
Organo- and Biocatalysis
z1137
All PDFs of this category

PDF (350 kb)
1137
Biocatalytic Directed Cationic Cyclization Cascades toward Fragrance Ingredients
FREE ACCESS

HTML

PDF (154 kb)
1138
Carbon-Bonding Interaction Catalyst

HTML

PDF (73 kb)
1139
Organocatalytic Enantiodivergent Bromolactonizations

HTML

PDF (78 kb)
1140
Development of a Novel Chiral Framework: The SPHENOL Backbone

HTML

PDF (82 kb)
1141
Synthesis of Chiral Cyclazines by Aminocatalytic Stereoselective [8+2] Cycloaddition

HTML

PDF (90 kb)
1142
Protecting Group-Free Late-Stage S-Glycosylation of Peptides

HTML

PDF (86 kb)
1143
Visible-Light Photoredox-Catalytic Coupling of Aryl Chlorides via Radical Anions

HTML

PDF (76 kb)
1144
Organocatalytic Kinetic Resolution of Amido Tertiary Allylic Alcohols

HTML

PDF (81 kb)
1145
Cinchona-Alkaloid-Catalyzed Annulation Enables an Asymmetric Synthesis of Chiral Oxacycles

HTML

PDF (90 kb)
1146
Chiral Triazolium Salt-Catalyzed Asymmetric Cyanoalkylation of Electron-Deficient Olefins

HTML

PDF (88 kb)
Chemistry in Medicine and Biology
z1147
All PDFs of this category

PDF (484 kb)
1147
Aziridines Cross-Dimerize to Larger N-Heterocycles
FREE ACCESS

HTML

PDF (125 kb)
1148
Photocatalyzed Site-Selective Tyrosine Bioconjugation

HTML

PDF (89 kb)
1149
Doubly Caged Puromycin

HTML

PDF (178 kb)
1150
A Novel P(V)-Based Reagent for Asymmetric Synthesis of Thiophosphoramidates

HTML

PDF (85 kb)
1151
Eschenmoser Sulfide Contraction in the Synthesis of Kinase Inhibitors

HTML

PDF (79 kb)
1152
Gram-Scale Synthesis of Iboxamycin

HTML

PDF (77 kb)
1153
Optical Control of Phosphatidic Acid Signaling

HTML

PDF (80 kb)
1154
Beating Resistant Plasmodium Parasites with the Antimalarial MMV688533

HTML

PDF (92 kb)
1155
Potent and Selective Orphan GPCR Agonist for the Treatment of Schizophrenia

HTML

PDF (71 kb)
1156
Activity-Based Probe for Monitoring Ethylene

HTML

PDF (79 kb)
1157
Optical Control of Sodium Channels

HTML

PDF (82 kb)
1158
A Rigid Vitamin Diet: Allenic derivatives of Vitamin D

HTML

PDF (84 kb)
Peptide Chemistry
z1159
All PDFs of this category

PDF (383 kb)
1159
Organoboron-Catalyzed Synthesis of Serine- and Threonine-Derived Weinreb Amides

HTML

PDF (72 kb)
1160
Palladium-Catalyzed C–H Functionalization of Cyclic-Aminal-Protected Peptides

HTML

PDF (84 kb)
1161
Synthesis of Sulfonyl Fluoro Peptides by an Ugi Reaction
FREE ACCESS

HTML

PDF (120 kb)
1162
Unnatural Peptide Synthesis by Photochemical Acyl Radical Addition of Dehydroalanine

HTML

PDF (84 kb)
1163
Palladium-Catalyzed Modification of Aspartic Acid-Containing Peptides

HTML

PDF (74 kb)
1164
Electrochemical Synthesis of α-Amino Esters

HTML

PDF (88 kb)
1165
Enantioselective Synthesis of 2-Chloroaziridines

HTML

PDF (85 kb)
1166
Chiral Phosphoric Acid-Catalyzed Synthesis of α-Amino Esters

HTML

PDF (84 kb)
1167
Ruthenium-Catalyzed Dehydrogenative Amidation of Alcohols by Amines

HTML

PDF (67 kb)
1168
Unnatural α-Amino Acid Synthesis by Photoinduced Alkylation of Dehydroalanine

HTML

PDF (87 kb)
1169
Synthesis of a Side-Chain-Tethered Solid Support for Peptide Synthesis
FREE ACCESS

HTML

PDF (144 kb)
1170
Synthesis of γ-Oxo-α-Amino Acids by Iridium Catalysis

HTML

PDF (94 kb)
Flow Chemistry
z1171
All PDFs of this category

PDF (138 kb)
1171
Photocatalytic C(sp³)–H Heteroarylation in Flow

HTML

PDF (82 kb)
1172
Decarboxylation and Decarboxylative Deuteration of Carboxylic Acids by Using a Ag–Bi Hybrid Material

HTML

PDF (82 kb)
1173
A Fixed-Bed Approach for Wittig-Type Olefinations in Continuous Flow

HTML

PDF (69 kb)
1174
Ozone-Mediated Oxidation of Amines and Pyridines under Flow Conditions

HTML

PDF (71 kb)

Archive
Articles by Category
Free Sample Issue

Journal

More About This Journal
Synfacts Videos
Editorial Board
Editorial Office
Brochure

Authors

Instructions for Authors

Subscription

Subscription Information & Contacts
Institutional Licensing

Nobel Prize 2016

Instructions for Authors

Journals
Book Series
Login
Help
Portal
Return to Classic Website

German English

Thieme E-Books & E-Journals is a service of Georg Thieme Verlag and Thieme Medical Publishers, Inc.
© Georg Thieme Verlag KG

Imprint | Privacy policy statement

Your Current IP Address: 216.73.216.23