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Synlett 2001; 2001(3): 0388-0390
DOI: 10.1055/s-2001-11384
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Readily Prepared Resin-Bound Thioimidates as Reagents for the Synthesis of Amidines

Antonella Ursini* , Monica Delpogetto, Giuseppe Guercio, Alcide Perboni, Tino Rossi
  • *GlaxoWellcome S.p.A. Chemical Development Department, Via A. Fleming 4, 37135 Verona, Italy; E-mail: au4438@GlaxoWellcome.co.uk
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Publikationsdatum:
31. Dezember 2001 (online)

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The use of commercially available resins to prepare novel and stable polymer supported thioimidates was investigated. Polymer supported thioimidates were found to enable acetamidine formation in a convenient manner, with a significantly easier work-up than solution-phase reactions.

amine - acetamidine - scale-up - solid-phase synthesis - polymers