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Synthesis 1991; 1991(11): 993-995
DOI: 10.1055/s-1991-26626
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Coupling of Arylboronic Acids with a Partially Reduced Pyridine Derivative

David J. Wustrow* , Lawrence D. Wise
  • *Parke-Davis Pharmaceutical Research Division, Warner-Lambert Company, 2800 Plymouth Rd., Ann Arbor, MI 48106-1047, USA
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Publication Date:
29 April 2002 (online)

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tert-Butylcarbonyl 1,2,3,6-tetrahydro-4-[(trifluoromethyl)sulfonyloxy]pyridine-1-carboxylate (2) was prepared and underwent palladium-catalyzed coupling reactions with a variety of substituted arylboronic acids 3 to produce a series of tert-butyl-4-aryl-1,2,3, 6-tetrahydropyridine-1-carboxylates 4.

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