DOI: 10.1055/s-00000131

Synfacts

Ausgabe 07 · Volume 17 · Juli 2021 DOI: 10.1055/s-011-51189

Synform

  • A105

    SYNFORM ISSUE 2021/07

    • Synthesis of Natural Products and Potential Drugs

  • z0721

    All PDFs of this category

  • 0721

    Synthesis of (+)-Manginoid A and (–)-Manginoid C

  • 0722

    Synthesis of Sisunatovir

  • 0723

    Synthesis of β-Secretase Inhibitor NB-360

  • 0724

    Synthesis of 9,11-Secosteroids (+)-Pinnigorgiol B and (–)-Pinnigorgiol E

  • 0725

    Total Synthesis of (+)-Alstilobanine C, (+)-Undulifoline, and (−)-Alpneumine H

  • 0726

    Formal Synthesis of BMT-362265

  • 0727

    Synthesis of Tacalcitol

  • 0728

    Synthesis of (–)-Koumimine

  • 0729

    Total Synthesis of Perovskones and Hydrangenone

  • 0730

    Synthesis of AG-270

  • 0731

    Synthesis of P2X7 Receptor Antagonist Lu AF27139

  • 0732

    Synthesis of Emitasvir

  • 0733

    Synthesis of BPR1K871

  • 0734

    Formal Synthesis of Telmisartan

  • 0735

    Synthesis of Encequidar

  • 0736

    Total Synthesis of (±)-Dehydroxypycnidione

  • 0737

    Total Synthesis of (±)-Desacetylcolchicine and Formal Synthesis of (±)-Colchicine

    • Synthesis of Heterocycles

  • z0739

    All PDFs of this category

  • 0739

    One-Pot Stepwise Synthesis of γ-Lactams through Cycloadditions with Ketenes

  • 0740

    Palladium-Catalyzed Synthesis of Benzoxepines from Vinyl-Substituted Cyclopropanes and Salicylaldehydes

  • 0741

    Mild Regioselective Reduction of Pyridines to Dihydropyridines

  • 0742

    Rhenium-Mediated Synthesis of Five- and Six-Membered Nitrogen-Containing Heterocycles

  • 0743

    Sequential Palladium-Catalyzed Synthesis of Benzosultams

  • 0744

    Regioselective Synthesis of Indoles form Azoarenes or Azoxyarenes with Ketones

  • 0745

    Copper-Catalyzed Synthesis of Quinazolines and 1,2,4-Oxadiazoles

  • 0746

    Iridium-Photocatalyzed Synthesis of Bioactive Tetracyclic Nitrogen-Containing Products

  • 0747

    2-Pyridones from Enamides through Ni–Al Bimetallic Catalysis

  • 0748

    Synthesis of Functionalized Benzimidazoles through C(sp3)–H Amination/C–N Bond Cleavage

  • 0749

    Palladium-Catalyzed Synthesis of Enantiopure Eight-Membered Nitrogen Heterocycles

  • 0750

    One-Pot Construction of 2,3-Dialkyl-Substituted Quinazolinones from Secondary Amides and Isocyanate

  • 0751

    Iridium-Catalyzed Approach to Polycyclic Nitrogen-Containing Systems

  • 0752

    Selectfluor-Promoted Synthesis of Functionalized Isothiazolones

    • Synthesis of Materials and Unnatural Products

  • z0753

    All PDFs of this category

  • 0753

    Powerful Rotamers for Asymmetric Synthesis

  • 0754

    Inserting a Seventh Carbon into Perylene Bisimide

  • 0755

    Site-Selective Electrophilic Substitution of 9-Substituted Triptycenes

  • 0756

    Accessing Useful Quantities of CPP

  • 0757

    Carbons by the Barrel

  • 0758

    Efficient Six-Step Synthesis of peri-Heptacene

  • 0759

    Synthesis of β-Isoindigo Derivatives

  • 0760

    Elegant Ring Formation Aided by Iron

  • 0761

    One Step to Spiro Nation

  • 0762

    Selective Synthesis of Cyclo[9]pyrroles

  • 0763

    Falling into Place: Facile Access to Modular 2,6-Dicyanoanilines

  • 0764

    Silicon on the Run in a Gold-Catalyzed Cycloisomerization

    • Metals in Synthesis

  • z0765

    All PDFs of this category

  • 0765

    Nickel-Mediated C(sp3)–H Methylation via Photochemical Activation of Peroxides

  • 0766

    Switchable Selectivity in the Asymmetric Rhodium-Catalyzed Hydrothiolation of Cyclopropenes

  • 0767

    Ruthenium-Catalyzed Enantioselective Reductive Amination

  • 0768

    NiH-Catalyzed Hydroamidation of Alkynes with Dioxazolones

  • 0769

    Nickel-Catalyzed Site-Selective Heteroarylation of Cyclobutanols

  • 0770

    Synthesis of Indoles from N-Benzoyloxyallylamines and Iodoarenes by Palladium/Norbornene Catalysis

  • 0771

    Synthesis of Chiral Sulfones by Three-Component Radical Reaction

  • 0772

    Photocatalyzed Decarboxylation of Carboxylic Acids

  • 0773

    Iron-Catalyzed Oxidation of Olefins

  • 0774

    Alkylation and Alkenylation of Neopentylamine

  • 0775

    δ-Fluorination of N-Alkyl Sulfonamides

  • 0776

    Fluoroalkylative Reductive Coupling of Alkyl Bromides

  • 0777

    Dioxazolones as Nitrene Precursors under Iron Catalysis

  • 0778

    Photoredox and Nickel-Catalyzed Aminoarylation

  • 0779

    Preparation of Functionalized 1,3-Disbustituted BCBs

  • 0780

    Visible-Light Assisted Sulfonylation of (Hetero)Aryl Halides

  • 0781

    Dual-Ligand-Enabled Ruthenium-Catalyzed C–H Arylation of Buchwald Phosphine Ligands

  • 0782

    Manganese-Catalyzed Hydroboration of Unsaturated C=X Bonds

  • 0783

    Asymmetric, Light-Mediated Radical Sulfinyl-Smiles Rearrangement

  • 0784

    ortho-C–H Imidation of Benzaldehydes using a Transient Directing Group

  • 0785

    Nickel-Catalyzed Aldol Reactions

  • 0786

    Preparation of Polycyclic Lactams

  • 0787

    Asymmetric Synthesis of γ-Lactams by Palladium-Catalyzed Hydroesterificative Cyclization

  • 0788

    Synthesis of Nitrogen-Containing Terminal Alkyl Chlorides via Copper-Catalyzed Chloromethylazidation

  • 0789

    Synthesis of Fully Substituted Pyrroles from Imino Ethers and Enol Diazoacetates using Silver Catalysis

  • 0790

    1,4-Acetoxychlorination of Dienes: The Bäckvall Reaction

  • 0791

    Enantioselective Preparation of Propargylsilanes

  • 0792

    Incorporation of gem-Difluoroalkene Motifs via Regioselective C(sp3)–H Functionalization

    • Polymer-Supported Synthesis

  • z0793

    All PDFs of this category

  • 0793

    A Polymeric Bipyridyl Nickel Composite for C–H Arylation of Heteroarenes

  • 0794

    Suzuki–Miyaura Coupling with a Palladium-Complexed Azo Porous Organic Polymer

  • 0795

    Hydroaminomethylation of Alkenes Promoted by Ruthenium on TiO2

  • 0796

    Sulfonation of Enamides, Acrylamides, and Enones Photocatalyzed by Single-Atom Nickel on TiO2

  • 0797

    C–C Coupling of Nitriles with Arylboronic Acids Catalyzed by Mesoporous Silica-Tethered Platinum

  • 0798

    Photocatalytic Oxidative Amidation of Aldehydes with Magnetic Cadmium Sulfide Quantum Dots

  • 0799

    Catalytic Esterification of Amides by Using a Zirconium-Based Metal–Organic Framework

  • 0800

    Hydrogenation of Carbonyls, Nitriles, and Nitroarenes by Using Ni2P Nanoalloy Catalyst in Water

  • 0801

    Protection and Deprotection of Alcohols by Using a Zn Complex Supported on Magnetic Nanoparticles

  • 0802

    Tandem Asymmetric Michael/Transfer Hydrogenation by Using a Dual Rh-Incorporated Micelle Reactor

    • Organo- and Biocatalysis

  • z0803

    All PDFs of this category

  • 0803

    Heterofunctionalization of Arenes by Electrophotocatalysis

  • 0804

    Biosynthesis of Hirsutellones and Pyrrocidines through an exo-Selective Diels–Alder Cycloaddition

  • 0805

    Pyrrolidine Aminocatalytic Asymmetric [12+2] Cycloaddition toward Cycl[3.2.2]azines

  • 0806

    Activation of N-Heterocycles by Silylium Catalysis for C–C Bond Formation

  • 0807

    Catalytic (3+2) Annulation of Aminocyclopropane Monoesters and Indoles

  • 0808

    Organocatalytic, Visible-Light-Mediated Dicarboxylation with Carbon Dioxide via Anion Radicals

  • 0809

    Catalytic Asymmetric Stereospecific Substitutions of Racemic α-Aryl Aldehydes

  • 0810

    Catalytic Asymmetric α-Chlorination of Aldehydes

  • 0811

    Two Work Better Than One: Cooperative NHC and Photoredox Catalysis for Benzylic C–H Bond Acylation

    • Chemistry in Medicine and Biology

  • z0813

    All PDFs of this category

  • 0813

    Spirocyclic Ketone Construction via Semipinacol-Type Rearrangement

  • 0814

    Biphenyl Imidazopyridines as a New Scaffold for PD-L1 Inhibitors

  • 0815

    Synthesis and Application of the 3-Phosphonofluoresceins

  • 0816

    Selective Cannabinoid Type 2 Receptor Antagonists

  • 0817

    Watching RNA Do Its Job

  • 0818

    Site-Selective LYTACs for Targeted Protein Degradation

  • 0819

    Scalable Synthesis of Opioids Enabled by a Palladium-Catalyzed Dearomative Arylation

  • 0820

    Small-Molecule Inhibitor of an RNA-Modifying Enzyme for Acute Myeloid Leukemia Treatment

  • 0821

    Late-Stage Alkylation of Purine Nucleoside at the C6 Position

  • 0822

    Utorubicin: A Novel Anthracycline Cancer Prodrug

  • 0823

    Next-Generation Macrolide Antibiotics

  • 0824

    Stereostructure–Activity Studies of Spirooliganin

    • Peptide Chemistry

  • z0825

    All PDFs of this category

  • 0825

    Palladium-Catalyzed Olefination of Oxazole-Containing Peptides

  • 0826

    Oxidative Peptide Bond Formation of 2-(Aminomethyl)malononitriles

  • 0827

    Copper-Catalyzed Synthesis of Bulky Amides and Peptides

  • 0828

    Hypervalent-Iodine-Mediated Peptide-Bond Formation to Synthesize Hindered Peptides

  • 0829

    Nickel-Catalyzed Synthesis of β-Amino Acid Derivatives

  • 0830

    Synthesis of Isoquinolone-Containing Amino Acids by Rhodium-Catalyzed C–H Annulation

  • 0831

    Palladium-Catalyzed δ-C(sp3)–H Arylation of Amino Acids

  • 0832

    Petasis Reaction for the Synthesis of Unnatural Amino Acids

  • 0833

    Synthesis of N-Unprotected α-Amino Acid Methyl Esters

  • 0834

    Photoredox-Catalyzed Synthesis of γ-Amino Acid Derivatives

    • Flow Chemistry

  • z0835

    All PDFs of this category

  • 0835

    N-Arylation of Amino Acid Esters using a Pd(OH)2 Packed-Bed Reactor

  • 0836

    Bromine–Sodium Exchange and Directed Metalations in Continuous Flow

  • 0837

    Synthesis of Fluorinated Tertiary Alcohol Derivatives under Visible-Light Irradiation

  • 0838

    Ru-promoted Photooxidative C–H Functionalization of Isoquinolines in a Microflow Reactor

  • 0839

    Precise Control of cis−trans Isomerization of α-Anionic Stilbenes under Flow Conditions