Synfacts

Issue 11 · November 2019

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A162
SYNFORM ISSUE 2019/11

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Synthesis of Natural Products and Potential Drugs
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Nanomolar Inhibitor of Trypanosoma brucei Trypanothione Reductase FREE ACCESS

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Total Synthesis of (±)-Atlanticone C

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Total Synthesis of Illisimonin A FREE ACCESS

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Artificial Intelligence Guides the Synthesis of SCH 47949

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Synthesis of the Immunosuppressant FR252921

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Synthesis of GSK2798745

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1221
Synthesis of (±)-Rhabdastrellic Acid A

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Total Synthesis of (–)-Himeradine A

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Synthesis of (+)-Jungermatrobrunin A

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1224
Synthesis of Antibacterial LpxC Inhibitors

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1225
Synthesis of Esketamine

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Synthesis of (±)-Isocomene FREE ACCESS

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1227
Synthesis of Omecamtiv Mecarbil

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Synthesis of Heterocycles
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1229
Copper-Catalyzed Synthesis of Di(het)arylamines

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1230
Synthesis of Enaminones and Thiazoles Using Iodonium Ylides as Carbene Equivalents

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1231
Cooperative Catalysis for the Asymmetric Synthesis of Piperidines

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1232
Selective C-2 Directed-Carbonylation of Indoles and Pyrroles

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1233
Synthesis of Substituted Morpholines by Fragmentation of Tetrazoles

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1234
Rhodium-Catalyzed Synthesis of 2‑Arylindoles from N‑Aryl-2-aminopyridines

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1235
Synthesis of Benzazepinones Involving an Unexpected Intramolecular Cyclization

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1236
Electrocatalytic Synthesis of Imidazo[1,5-a]quinoline-3-carbonitriles

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1237
Asymmetric Radical C–H Amination for the Synthesis of Azoles

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1238
Three-Component Assembly of 3,4-Dihydroquinazolines

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1239
Synthesis of Phosphinolines and Phosphepines

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1240
Buchwald–Hartwig Coupling of Piperidines with Hetaryl Bromides

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1241
Synthesis of 3-Phenylimidazo[1,2-a]pyridines by Annulation of Tetrazoles with Phenylacetylenes

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1242
Copper-Catalyzed Cyclization of Enaminones to Polycyclic N-Fused Indoles

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1243
An Illuminating Synthesis of Benzimidazoles

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Synthesis of Materials and Unnatural Products
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1245
Developing a Dye for Lysosome

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1246
Synthesis of a π-Conjugated Macrocyclic Oligofuran: The First of Many to Come

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1247
peri-Disubstituted Naphthalimides via Decarboxylative Arylation

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1248
Finally, Furfural Flourishes

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1249
Unmasked ‘Click Chemistry’

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1250
Proton Hole-in-One With TriQuinoline

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1251
Synthesis of Carbon-Skeleton-Like Molecules

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1252
Going Full Circle: From Linear to Cyclic pH-Responsive Water-Soluble Cyclic Polymer

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1253
Aryl Sulfones and Aryl Boronic Acids Make a Nice Couple

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1254
Ring-Opening Doors to Controlled Polymerization with Hydrogen-Bond-Driven Organocatalysis

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1255
Stepwise Synthesis of an Axially Chiral 1,1′-Biazulene and its π-Extended Derivative

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1256
Synthesis of Sumanene FREE ACCESS

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Metals in Synthesis
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1257
Palladium-Catalyzed Synthesis of Carboxylic Acids FREE ACCESS

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1258
Copper-Mediated Trifluoromethylation of Aryl Sulfonium Salts

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1259
Asymmetric C–H Alkylation of Fluoroarenes with Alkenes via Nickel/NHC Catalysis FREE ACCESS

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1260
C–H Acetoxylation of Carboxylic Acids

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1261
Reductive Dicarbofunctionalization of Alkenes

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1262
Zinc-Catalyzed Tandem Asymmetric Friedel–Crafts Alkylation/Michael Addition

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1263
Hydroalkylation of Terminal Alkynes with Primary or Secondary Alkyl Iodides

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1264
Synthesis of 2-Arylquinazolines via Visible-Light-Induced Benzylic C–H Functionalization

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1265
Enantioselective Allylic Substitution with Nucleophiles in Aqueous Solution under Iridium Catalysis

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1266
Catalytic Interrupted Click/Acylation Reactions

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1267
Enantioselective Preparation of Chiral Diamines

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1268
Base-Catalyzed Synthesis of Fully Substituted Silyl Enol Ethers

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1269
Photoredox/Nickel-Catalyzed C(sp³)–C(sp³) Cross-Coupling

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1270
Anti-Markovnikov Hydroamination and Hydroamidation of Allylic Alcohols through Iron Catalysis

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1271
Rhodium(III)-Catalyzed C–H Activation/Carbene Insertion/Lossen Rearrangement Sequence

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1272
Nickel-Catalyzed Asymmetric Reductive Heck Cyclization

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1273
Heteroaryl Thioether Directing Group in Oxidative Heck and C–H Functionalization Reactions

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1274
Enantioselective Benzylic Arylations

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1275
Photoreduction of Arenes and Heteroarenes

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1276
Decarbonylative Suzuki–Couplings of Amides

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1277
Ruthenium-Catalyzed Cross-Coupling of Anilines

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1278
Enantioselective Access to Tetrahydroquinoxalines through Relay Epoxide Opening/Amination of Alcohols

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1279
Photocatalysis: Asymmetric Intramolecular HAT in Photoexcited Catalyst–Substrate Complex

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1280
β-C(sp³)-Methylation of Alcohols

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1281
Preparation of β-Aminoboronates

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1282
Copper-Catalyzed Asymmetric Annulation of Carbenes to Access Enantioenriched 2,3-Dihydrobenzofurans

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1283
Palladium-Catalyzed C(sp³)–H Bond Activation of Phenylacetaldehydes

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1284
Palladium-Catalyzed Aerobic Oxidative C-H Arylation

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1285
The Hiyama–Denmark Cross-Coupling FREE ACCESS

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Polymer-Supported Synthesis
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1287
Zeolitic Imidazole Framework Encapsulated Copper Nanoparticles for Hydrogenation of Aldehydes FREE ACCESS

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1288
Transfer Hydrogenation of Unsaturated Compounds by Co NPs Encapsulated in N-doped Graphene

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1289
Copper-Catalyzed Oxidative Cyclization of Benzylamines with 1,3-Dicarbonyl Compounds

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1290
Controlled Reduction of Nitroarenes to Azo Compounds with Iron–Nitrogen Co-Doped Mesoporous Carbon

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1291
Rh-Catalyzed Asymmetric Arylation of α,β-Unsaturated Carbonyl Compounds, Nitroalkenes, or Imines

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1292
Hybrid Palladium Catalyst for Suzuki–Miyaura and Heck Reactions

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1293
Selective Deprotection of Benzyl Carbamates on Micellar Nickel–Palladium Nanoparticles in Water

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1294
Ruthenium-Photocatalyzed Aerobic Oxidation of Benzylic Halides and Cyclization of Tertiary Anilines

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1295
One-Pot Synthesis of 5-Substituted 1H-Tetrazoles on a Silica-Coated Fe₃O₄-Supported Copper(II) Complex

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1296
Oxidative Synthesis of Nitriles from Primary Alcohols and Ammonia Catalyzed by Cobalt Nanoparticles

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1297
Synthesis of Xanthene Derivatives by Using a Lewis Acidic Ionic Liquid Immobilized on Perlite NPs

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1298
Cerium(IV) Oxide-Catalyzed Direct Phenolysis of Amides

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Organo- and Biocatalysis
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1299
A Newly Designed Catalyst for Additive-Free Mitsunobu Reactions FREE ACCESS

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1300
Brønsted Acid Catalyzed Asymmetric House–Meinwald Rearrangement of p-Hydroxyphenyl Epoxides

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1301
Asymmetric Functionalization of C(sp³)–H Bonds in 2-Alkylindoles

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1302
NHC-Catalyzed Carboacylation of Alkenes

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1303
Lewis Base Catalyzed Enantioselective Sulfenoamination of Olefins

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1304
Asymmetric NHC-Catalyzed Rauhut–Currier Reaction of Weakly Electrophilic Bisenoates

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1305
Phosphenium Ion Catalyzed Enantioselective Reduction of Cyclic Imines

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1306
Asymmetric Phosphoric Acid Catalyzed Multi-Component Synthesis of Axially Chiral N-Arylindoles

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1307
N-Heterocyclic Carbene Catalyzed Stetter Reaction of Cyclic Enones

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1308
Organometallic Organocatalysts FREE ACCESS

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Chemistry in Medicine and Biology
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1309
Water-Soluble BODIPY Dyes for Voltage Imaging FREE ACCESS

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1310
Pre-Exposure Prophylaxis (PrEP) FREE ACCESS

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1311
Sign-Inversion in Photopharmacology

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1312
HPLC-Free Synthesis of Nucleoside Triphosphates

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1313
Targetable, Bright Small-Molecule Ca²⁺ Indicators

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1314
Macrocycle Library Synthesis through Thiol-to-Amine Cyclization

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1315
Membrane Probes for Super-Resolution Imaging of Plasma Membranes

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1316
Activatable Photosensitizers for Photodynamic Therapy

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1317
C–N Coupling of Aryl Thianthrenium Salts

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1318
An Aromatic Brønsted Acid Catalyst for the Direct Glycosylation of Amides

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1319
pH-Sensitive μ Opioid Receptor Agonists

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1320
Conformational Restricted Cyclopropanated Nucleoside Derivatives

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1321
SPiDER-Killer-βGal: A Photosensitizer for Targeted Cell Ablation with Single-Cell Resolution

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Peptide Chemistry
z1323
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1323
Synthesis of Cyclic and Bicyclic Peptides FREE ACCESS

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1324
Palladium-Catalyzed Conversion of Phenyl Aspartates into Ketones

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1325
Ruthenium-Catalyzed C–H Alkylation of Resin-Attached Tryptophan

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1326
Asymmetric Hydrogenation of β-Aminoacrylates to β-Amino Acid Derivatives

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1327
Palladium-Catalyzed Acylation of Phenylalanine-Containing Peptides

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1328
Palladium-Catalyzed Arylation of Sulfonamide-Containing Peptides

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1329
Synthesis of Diazirines from Amino Acids by Using Phenyliodonium Diacetate

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1330
Synthesis of Dehydroamino Acid Containing Peptides FREE ACCESS

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1331
Synthesis of Benzotriazole-Derived α-Amino Acids

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1332
Synthesis of Activated Amides and Directed C(sp³)–H Arylation

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1333
Peptide Nanoassemblies Promote Enantioselective Hydrogenation

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Flow Chemistry
z1335
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1335
Continuous Flow Electrochemical Oxidation of Alcohols

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1336
Functionalized Alkyllithium Reagents Towards Heterotelechelic Polymers

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1337
Radical-Based Late-Stage C−H ¹⁸F-Difluoromethylation of N-Heteroaromatics

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1338
Organocatalyzed Photooxygenation of β-Dicarbonyl Compounds in Flow Photomicroreactors

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1339
One-Step Synthesis of 2-Fluoroadenine in a Continuous Flow Operation

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