DOI: 10.1055/s-00000131

Synfacts

Issue 03 · Volume 14 · March 2018 DOI: 10.1055/s-008-39015

Synform

A31
Zanda, Matteo: SYNFORM ISSUE 2018/03

Synthesis of Natural Products and Potential Drugs

z0221
All PDFs of this category
0221
Concise Synthesis of the Alkaloid (±)-Aspergilline A
0222
Synthesis of a CXCR Antagonist
0223
Synthesis of a PCSK9 Inhibitor
0224
Synthesis of (±)-Maoecrystal P
0225
Synthesis of APD371
0226
Synthesis of (+)-Bryostatin 8
0227
Syntheses of Scaparvins B, C, and D
0228
Synthesis of Phomoidride D
0229
Synthesis of HIV-1 Protease Inhibitors
0230
Synthesis of Tropifexor
0231
Synthesis of Stemoamide-Type Alkaloids
0232
Synthesis of a Noradrenaline Reuptake Inhibitor

Synthesis of Heterocycles

z0233
All PDFs of this category
0233
Synthesis of Fused Indoles from Sulfonamides
0234
One-Pot Rhodium-Catalyzed Synthesis of Highly Substituted Quinolines
0235
Rhodium-Catalyzed Annulation of N-Methoxy-amides: Synthesis of Isoquinolones
0236
Copper-Catalyzed Synthesis of Fluorinated 2,2-Disubstituted Indolin-3-ones
0237
Continuous-Flow Electrosynthesis of Benzothiazoles and Thiazolopyridines
0238
Synthesis of Pyrrolidinones and Piperidinones by Using a Chiral Ammonia Equivalent
0239
Difluoromethoxylation of N-Heteroaromatics
0240
Rhodium(II)-Catalyzed Annulation Route to 5H-Pyrazino[2,3-b]indoles
0241
Synthesis of Fluoropyrrolidines by [3+2] Cycloaddition
0242
Cyclopentaquinolines by Palladium-Catalyzed Reaction of 2-Vinylanilines with Alkynes
0243
Enantioselective Synthesis of Heterocycle-Fused β-Lactones
0244
Hexafluoroisopropanol as a Solvent for Halogenation of (Het)aromatics
0245
Stereoselective Synthesis of Cyclic Ethers by Reductive Cyclization of Alkynols

Synthesis of Materials and Unnatural Products

z0247
All PDFs of this category
0247
Cage Compounds Sprout New Rings
0248
Metal-Free Phosphination with Diphenylphosphine Oxide
0249
Aminomethylation of Fullerene C60 with 1,3,5-Perhydrotriazines
0250
The Longest 1D Nanographene
0251
A New Twist on Acene Synthesis
0252
An ‘I’ for an ‘N’ to Obtain Acridines and Carbazoles
0253
Zipping Up Alkyl Chains to Obtain Conjugated Double Bonds
0254
Chains and Zincs Excite Me: Poly[n]catenane Success
0255
Giant, Nanographene-Substituted Phosphines
0256
One-Pot Synthesis of A2A1B1B2 Type Tetra-block Quaterpolymer
0257
Divergent Synthesis of Tetraphenylmethane Dendrimers
0258
Azulene’s D–A Structure for Optoelectronic Materials

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z0259
All PDFs of this category
0259
Enantioselective Cycloaddition of Cyclopropylcarboxamides to Alkynes
0260
Gold-Catalyzed Stereoselective Synthesis of Indolines and Oxindoles
0261
Stereoselective Synthesis of Trisubstituted Alkenes via Intermolecular Olefin Metathesis
0262
Palladium-Catalyzed Asymmetric α-Allylation of β-Keto Esters
0263
Isobenzofuranone Formation through Redox Allylation of Phthalaldehydes
0264
Asymmetric Allylation of Glycine Imino Esters and Glycine Amides
0265
Rhodium-Catalyzed Hydrogenation of Enol Esters
0266
Copper Hydride Catalyzed Enantioselective Synthesis of β-Chiral Aldehydes
0267
Enantioselective Synthesis of Allylic Silanes via Nickel-Catalyzed Reductive Cross-Coupling
0268
Zinc-Catalyzed Stereoselective Direct Vinylogous Mannich Reaction
0269
Synthesis of 2H-Azirines with a Tetrasubstituted Stereocenter
0270
Asymmetric Synthesis of Dihydroimidazoquinazolinones
0271
Asymmetric Diastereodivergent Synthesis of Spirocyclopropane Oxindoles
0272
Novel Chiral Bifunctional Phosphine-Carboxylate Ligands
0273
Copper-Catalyzed Asymmetric Borylation of β-Amidoacrylates
0274
Iridium-Catalyzed Fluorination of Allylic Trichloroacetimidates
0275
Rhodium-Catalyzed Asymmetric Addition of N-Hydroxyphthalimide to Allenes
0276
Copper-Catalyzed Stereoselective Cyclopropanation of 2-Vinylindoles
0277
Enantioselective Synthesis of syn-α-Amino β-Hydroxy Esters
0278
Linear C-Allylation by Iridium-Catalyzed N-Allylation and Aza-Cope Rearrangement
0279
Cobalt-Catalyzed Enantioselective Negishi Coupling of α-Bromo Esters and Arylzincs
0280
Rhodium-Catalyzed Enantioselective Synthesis of Propargyl Amides
0281
Cyclopropanation of Alkenylboronates with Ethyl Diazoacetate
0282
Nickel-Catalyzed Diastereoselective Arylboration of Unactivated Alkenes
0283
Copper-Catalyzed Enantioselective Synthesis of 1,2-Amino Tertiary Alcohols
0284
Rhodium-Catalyzed Enantioselective 1,2-Addition of Aldimines
0285
Binuclear Nickel Complex-Catalyzed Enantioselective Mannich Reaction
0286
Ruthenium-Catalyzed Asymmetric Transfer Hydrogenation of Chiral Sulfinylimines
0287
Palladium-Catalyzed Redox-Relay Heck Reaction of 4H-Chromenes
0288
Palladium-Catalyzed Enantioselective Synthesis of 3,4-Dihydroquinolin-2-ones

Metal-Mediated Synthesis

z0290
All PDFs of this category
0289
Highly Versatile Transmetalation Switch
0290
Nickel-Catalyzed Acylation of Aliphatic Amides
0291
Nickel-Catalyzed Cross-Coupling of Tertiary Sulfones
0292
Highly Stereoselective Cyclopropanation of Polyalkene Substrates
0293
Highly Efficient Copper-Catalyzed Perfluoroalkylation of Aryl Boronic Acids
0294
Ring Contraction of 1,5-Diazacyclo­octatetraenes to Pyridines
0295
SuFEx Chemistry of SOF4 with Organolithium Nucleophiles
0296
Dual Catalysis for the Cross-Coupling of Aryl(trialkyl)silanes
0297
Borylation of Aryl Sulfonium Salts
0298
Controlled Tandem Isomerization of o-Lith-iated Aryl Benzyl Ethers in Continuous Flow
0299
Innovative Synthesis of 1,2-Disubstituted Planar-Chiral Ferrocene Derivatives
0300
Novel Palladium Precatalyst for Cross-Coupling Reactions of Aryl Esters
0301
Lithiation and Electrophilic Quench of Tetrahydroquinolines
0302
Synthesis of 2,3-Diarylquinolines via Trapping of the Vinyl Metal Intermediate
0303
Mechanistic Studies of Four-Component Coupling Reactions

Organo- and Biocatalysis

z0305
All PDFs of this category
0305
Whole-Cell-Catalyzed Carbenoid B–H Insertion
0306
Diazaphosphenium Triflate Catalyzed Hydroboration of Pyridines
0307
Defluoroalkylation of Electron-Deficient Trifluoromethylarenes with Alkenes
0308
Dynamic Kinetic Resolution of Aliphatic Aldehydes by Biocatalytic Amination
0309
Asymmetric Aminalization by Cation-Binding Catalysis
0310
Chiral Brønsted Acid Catalyzed Enantioselective Tandem Cyclization
0311
Unnatural Amino Acid Ester Catalyzed Formal Synthesis of (+)-Pancracine
0312
Synthesis of Chiral Acyclic Pyrimidine Nucleosides
0313
Asymmetric Synthesis of 1,5-Diesters by Mukaiyama–Michael Reaction
0314
Photocatalytic Aerobic Phosphatation of Simple Olefins

Polymer-Supported Synthesis

z0315
All PDFs of this category
0315
Magnetic Pd- and CuO-Catalyzed Regioselective Direct Arylation of Anilides
0316
Catalytic Unsymmetrical Hantzsch Reaction and Knoevenagel Condensation
0317
Semihydrogenation of Alkynes on a Nanoporous Palladium Catalyst
0318
Hydrogenolysis of Allylic Alcohols on a Titania-Supported Palladium Catalyst
0319
Co2Rh2/C-Catalyzed Reductive Amination of Aldehydes with Nitrobenzenes
0320
Alcohol Protection–Deprotection Catalyzed by Fe3O4-Supported Silica Sulfuric Acid
0321
One-Pot Diazotization–Iodination of Anilines by Polymer-Supported Nitrite
0322
Acceptorless Dehydrogenation by Using an Iron-Based Nanocatalyst
0323
Hydrogenation of Phenols to Cyclohexanones on Pd/Titanate Nanosheets
0324
Nanocomposite Catalyst for the Aerobic Oxidation of Primary Alcohols
0325
Catalytic Applications of Metal Nanoparticles in a Covalent Organic Framework
0326
Dehydrogenative Coupling Using a Cobalt-Modified Carbon Nanotube Catalyst
0327
Suzuki–Miyaura Cross-Coupling of 9-Chloroacridines
0328
Aryl C–H Olefination on Ag1Pd1 Nanoparticles–Reduced Graphene Oxide
0329
Nickel-Catalyzed One-Pot Synthesis of Polyhydroquinolines
0330
Magnetic Cobalt Nanocatalyst for Cross-Coupling Reactions