DOI: 10.1055/s-00000131

Synfacts

Issue 01 · Volume 13 · January 2017 DOI: 10.1055/s-006-33134

Synform

A1
Zanda, Matteo: SYNFORM ISSUE 2017/01

Synthesis of Natural Products and Potential Drugs

z0001
All PDFs of this category
0001
Synthesis of an Atropisomeric HIV Integrase Inhibitor
0002
Synthesis of UM171
0003
Synthesis of (±)-Atropurpuran
0004
Enantioselective Synthesis of Efavirenz
0005
Synthesis of (–)-Cyclosmenospongine
0006
Synthesis of (±)-Morphine
0007
Synthesis of Swinholide A
0008
Manufacturing Route to Avibactam
0009
Synthesis of Tofogliflozin Hydrate
0010
Crystallization-Induced Dynamic Resolution of a Dibenzoazepinone
0011
α-Arylation of Malonate Derivatives via Oxidative Catalysis
0012
Synthesis of (–)-Englerin A
0013
Synthesis of (+)-Hinckdentine A
0014
Synthesis of Nisoxetine
0015
Synthesis of Araiosamines
0016
Synthesis of VPC01091
0017
Synthesis of Amino-Carbasugars

Synthesis of Heterocycles

z0019
All PDFs of this category
0019
Synthesis of 3,3-Diaryloxetanes from Oxetanols by a Friedel–Crafts Reaction
0020
Selective Functionalization of Pyridines via Their Phosphonium Salts
0021
Synthesis of Epoxides by a Darzens Reaction and Vicarious Nucleophilic Substitution
0022
Ytterbium(III)-Catalyzed Synthesis of Epiminodibenzo[b,f][1,5]diazocines
0023
Synthesis of Pyrrolidines, Pyrroles, and Carbazoles by Iridium Catalysis
0024
Enantiospecific Access to Bicyclic Morpholines and Piperazines
0025
Rhodium(III)-Catalyzed Synthesis of Benzo[a]carbazoles
0026
Synthesis of Azetidines by Ring Opening and Closing of Cyclopropanes
0027
Synthesis of Substituted Pyrroles from α-Iminodiazoacetates
0028
Enantioselective Synthesis of Spirooxindole 2H-Azirines
0029
Photochemical [2+2]-Cycloaddition Route to Enantiomerically Pure Oxetins
0030
Synthesis of Polyfunctional Pyrrolidines, Pyrrolines, and Thioxopyrrolidines

Synthesis of Materials and Unnatural Products

z0031
All PDFs of this category
0031
One-Pot, Why Not?
0032
Two Tastes of Propargyl Acetates
0033
Dancing with Sulfur
0034
Mutant Nanographenes
0035
An Approach to Zigzag Carbon Nanobelts
0036
Function by Switching: Heterodiazocines
0037
A Trophy for BOPHYs
0038
Two N-Tosyl Hydrazones Joined Together by the Hand of Sulfur
0039
Alkyne Metathesis Macrocyclization and Copper-Free Click Reactions
0040
One ‘S’tone, Two Bird‘S’
0041
Supercharged Snowflake
0042
Reversible Dimerization and Polymerization of a Janus Diradical

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z0043
All PDFs of this category
0043
Palladium-Catalyzed Asymmetric Synthesis of α,α-Disubstituted Allylic N-Arylamines
0044
Magnesium-Catalyzed Desymmetrization of meso-Aziridines with Hydroxylamines
0045
Cyclohexenylamines and Cyclohexenols by Rhodium-Catalyzed Cycloaddition
0046
Silver-Catalyzed Enantioselective Nitroso Aldol Reaction of Nitrosoarenes
0047
Palladium-Catalyzed Asymmetric Alkenylation of Trisubstituted Alkenols
0048
Rhodium-Catalyzed Conjugate Addition Towards Chiral Thioflavanones
0049
Zinc(II)-Catalyzed Asymmetric Aza-Friedel–Crafts Reaction of Ketimines
0050
Nickel-Catalyzed Asymmetric Allenyl Claisen Rearrangement
0051
Gold-Catalyzed Tandem Cycloisomerization/Hydrogenation
0052
Asymmetric Allylic Alkylation Towards Dihydrocoumarins and Isochromanones
0053
Palladium-Catalyzed Asymmetric Synthesis of Indolines by C(sp3)–H Arylation
0054
New Chiral Cyclic Sulfinamide–Olefin Ligands for Asymmetric 1,4-Additions
0055
Asymmetric Iridium(I)-Catalyzed Diene Hydrohydroxymethylation
0056
Rhodium Pincer Complex Catalyzed Direct Alkynylation of Ketones
0057
Copper(I)–NHC Catalyst for the Stereo-selective Semihydrogenation of Alkynes
0058
Enantioselective Palladium-Catalyzed Synthesis of 3-Indolyl Methanamines
0059
Nickel-Catalyzed Synthesis of Thiochromanyl-Spirooxindoles
0060
Ruthenium/Palladium Dual-Metal Catalysis for Oxindole Synthesis
0061
Enantioselective Rhodium-Catalyzed Arylation Generating Triarylmethanes
0062
Iridium-Catalyzed Asymmetric γ-Alkynylation of α,β-Unsaturated Amides
0063
Nickel(0)-Catalyzed Stereoselective Synthesis of Vinylcyclopropanes
0064
Enantioselective Silver-Catalyzed [3+2] Cycloaddition
0065
Asymmetric Synthesis of β-Hydroxy α-Amino Acid Derivatives
0066
Copper-Catalyzed Ring Opening of Cyclopropanes with Inversion
0067
Rhodium(II)-Catalyzed Asymmetric Cyclopropanation
0068
Oxidative Fragmentation Follows an Asymmetric Hydrogenation
0069
Iridium-Catalyzed Asymmetric Reduction of Pyridinium Salts
0070
Asymmetric Allenylation of Sulfonylimines Catalyzed by Rhodium

Metal-Mediated Synthesis

z0071
All PDFs of this category
0071
Ring-Forming Thioboration of C–C π-Bonds
0072
Synthesis of α-Trifluoromethylated Ketones
0073
Synthesis of β-Boryl-α-Aminosilanes
0074
Synthesis of α-Sila Benzamides
0075
Aldol Reactions of Azetidin-2-one
0076
Asymmetric Catalysis of Indoles and Dihydroisoquinolines via Allylboration
0077
Rhodium(I)-Catalyzed Coupling with Arylboronic Acids
0078
Catalytic Hydroboration of Nitriles and Imines
0079
Cobalt-Catalyzed C(sp2)–H Borylation
0080
Nucleophilic Tetrafluoroethylation
0081
C–O Bond Activation
0082
ortho-C–H Functionalization
0083
Diaryl Ketones by Nickel Catalysis
0084
Suzuki–Miyaura Cross-Coupling of Amides via Cooperative Catalysis
0085
C–F Bond Activation

Organo- and Biocatalysis

z0087
All PDFs of this category
0087
Allylboration of Aldehydes by Immobilized TRIP
0088
Asymmetric Oxidative Dearomatization/Oxa–Michael Addition Sequence
0089
Catalytic Asymmetric Aminoalkynylation of Arenes
0090
Regiodivergent Chlorination of Phenols Controlled by a Lewis Base Catalyst
0091
Regioisomeric Fluorolactonization via Hypervalent Iodine Catalysis
0092
Electrostatically Enhanced Phosphoric Acids in Brønsted Acid Catalysis
0093
Enantioselective Aza–Sakurai Cyclization
0094
Organocatalytic Asymmetric Vinylogous Prins Cyclization
0095
Enantioselective Catalytic Thioacetalization of Aldehydes

Polymer-Supported Synthesis

z0097
All PDFs of this category
0097
Conversion of Arylboronic Acids into Phenols with Biogenic Cu2O Nanoparticles
0098
Photocatalytic Click Chemistry with Copper Oxide Doped Semiconductors
0099
Spirocyclization of Alkyne-Tethered Aromatics with Silver Nitrate/Silica
0100
In–Co(Porphyrin) Metal–Organic Framework Catalyzed Hydration of Terminal Alkynes
0101
Olefin Metathesis with Metal–Organic Framework Adsorbed Ruthenium Complexes
0102
Nanoorganocatalyst for the Synthesis of 2-Amino-4H-chromene-3-carbonitriles
0103
Olefin Hydrogenation with Mesoporous Silica-Supported Pd–Fe Nanoreactors
0104
Copper-Catalyzed Synthesis of 2-Aryl-1-imidazo[1,2-a]pyridin-3-ylethane-1,2-diones
0105
Thiol-Grafted Cellulose Paper for Copper-Catalyzed Click Reactions
0106
Supported Copper Catalyst for N-Arylation Reactions and Click Chemistry
0107
Palladium Nanoparticle Catalyzed Hydrogenation of Quinolines and Quinoxalines
0108
Synthesis of 1-Amidoalkyl-2-naphthols with Graphene Oxide
0109
Sulfoximinocarbonylation of Aryl Halides with Palladium/Carbon
0110
Decarboxylative Arylation and Carbonylative C–C Coupling with Copper Nanoparticles
0111
FeCl3/SiO2-Catalyzed Condensation of 1,2-Diaminobenzenes with β-Keto Carbonyls
0112
Tetrahydropyranylation of Alcohols Catalyzed by an Acidic Ionic Liquid
0113
Hydroamination of Alkynes with Gold Nanoparticles/Titania