DOI: 10.1055/s-00000131

Synfacts

Issue 10 · Volume 12 · October 2016 DOI: 10.1055/s-006-32474

Synform

A143
Zanda, Matteo: SYNFORM ISSUE 2016/10

Synthesis of Natural Products and Potential Drugs

z999
All PDFs of this category
0999
Synthesis of (+)-Notoamides F, I, and R and (–)-Sclerotiamide
1000
Syntheses and Structure Elucidation of Juglocombins A and B, and Juglorescein
1001
Synthesis of Vismodegib through meta-Selective Nitration of Arenes
1002
Synthesis of Exochomine
1003
Synthesis of (+)-Psiguadial B
1004
Synthesis of an αVβ6 Antagonist
1005
Synthesis of MK-8876
1006
Synthesis of (–)-Oseltamivir
1007
Highly Efficient Synthesis of (−)-Maoecrystal V
1008
Synthesis of MK-8718
1009
Synthesis of AS-3201 (Ranirestat)
1010
C–H Arylation of Heterocyclic N-Oxides: Application to SB222200
1011
Syntheses of (+)-Javaberine A, (+)-Javaberine B, and (–)-Latifolian A
1012
Synthesis of Palbociclib
1013
Syntheses of Hyperjapones A–E, and Hyperjaponols A and C

Synthesis of Heterocycles

z1015
All PDFs of this category
1015
Photocatalytic Azolylation of (Het)arenes
1016
C2-Alkylation of Pyridine N-Oxides with 1,1-Diborylalkanes
1017
Photoredox-Catalyzed Aryl Aminations with Ligand-Free Nickel(II) Salts
1018
Rhodium(III)-Catalyzed C–H Activation Route to 1H-Isoindoles
1019
Cobalt-Catalyzed Cross-Coupling Route to Homoallylic Alcohols and Amines
1020
Enantioselective Synthesis of Pyrrolidines by Aminotrifluoromethylation of Alkenes
1021
Directed Decarboxylative Cross-Coupling Route to Piperidines and Pyrrolidines
1022
Synthesis of Perfluorinated Isochromene Derivatives by Ring Expansion
1023
Synthesis of 3-Aminofurans from 1,2,3-Triazoles and Propargylic Alcohols
1024
Sulfonated β-Cyclodextrin-Catalyzed Synthesis of Imidazopyridinamines
1025
Gold-Catalyzed Synthesis of 1,5-Benzodiazepines
1026
Synthesis of Fused and Spiro Dihydrobenzofurans
1027
Synthesis of Isoquinolones and Isocoumarins by a Suzuki–Miyaura Coupling

Synthesis of Materials and Unnatural Products

z1029
All PDFs of this category
1029
Nitrogen Analogues of Polycyclic Aromatic Hydrocarbons
1030
Transition-Metal-Free Sulfoximidation with Hypervalent Iodine(III)
1031
Enantiospecific Reduction Leads to P-Stereogenic Synthons
1032
Introducing an Apical Anchor Group
1033
A Halogen Party
1034
Hydrogen-Bond Anionic Polymerization with Alkoxide and Thiourea
1035
Four-State Nanoswitch Controls Two-Step Sequential Catalysis
1036
Synthetic Route to Thiophene-Based Double Helical Oligomers
1037
Helical ortho-Arylene Foldamers
1038
N-Arylation of Iminodibenzyls and Iminostilbenes
1039
Nitrogen Heterocycles through Migratory Ring Expansion of Metalated Ureas
1040
Biazulene Diimide as a New Building Block for Organic Materials

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1041
All PDFs of this category
1041
Convenient Reagent for the Copper-Catalyzed Asymmetric Methyl 1,4-Addition Reaction
1042
Catalytic Asymmetric Henry Reaction
1043
Asymmetric Allylic Amination
1044
A Palladium-Catalyzed Dearomatization for the Synthesis of Polycyclic Indoles
1045
Asymmetric 1,4-Addition by Chiral Nanoparticle/Lewis Acid Catalysts
1046
Synthesis of Enantioenriched Arylglycines via Dynamic Kinetic Resolution
1047
Palladium-Catalyzed Asymmetric C–O Bond Cleavage of α-Acyloxy Ketones
1048
Highly Asymmetric Hydrogenation of Cyclic Enamides by Iridium Catalysis
1049
Palladium-Catalyzed Asymmetric Synthesis of α-Arylglycines
1050
Stereoselective Annulation by Palladium/Phosphine–Thiourea Catalysis
1051
Asymmetric Synthesis of Silylated Indanols by Nickel Catalysis
1052
Iridium-Catalyzed Enantioselective Hydrogenation of Pyridinium Bromides
1053
Copper-Catalyzed Asymmetric Conjugate Addition of α,β-Unsaturated Carbonyls
1054
Rhodium-Catalyzed Asymmetric Addition to N-Sulfonylimines
1055
Cobalt-Catalyzed Stereoselective Three-Component C–H Bond Addition
1056
Enantioselective Heck Reaction Leading to S- and P-Stereogenic Heterocycles
1057
Enantioselective Rhodium-Catalyzed Arylation of Aldehydes
1058
Synthesis of Tetrahydro-γ-Carbolines by [3+3] Cycloaddition
1059
Synthesis of Chiral Tertiary Alcohols by Asymmetric Cyanosilylation
1060
Asymmetric Copper-Catalyzed Etherification of Propargylic Esters
1061
Enantioselective Hydrogenation by a Supramolecular Chiral Catalyst
1062
Diastereoselective Synthesis of Amino Acids with a Quaternary Stereocenter
1063
Diastereoselective Copper-Catalyzed Cyanation and Diborylation of Allenes
1064
Ruthenium-Catalyzed Asymmetric Intermolecular Cyclopropanation Reaction
1065
Enantioselective Intermolecular Hydroalkoxylation of Allenes and Alkynes
1066
C2-Symmetric Bis-sulfinamide Ligands for the Asymmetric Rh-Catalyzed Conjugate Addition
1067
Palladium-Catalyzed Dearomative Reaction of Furans Towards Spirooxindoles
1068
Asymmetric Hydrogenation of Seven-Membered C=N-Containing Heterocycles

Metal-Mediated Synthesis

z1069
All PDFs of this category
1069
Addition of Organotrifluoroborates to Arylated Cyclopropyl Ketones
1070
Iron-Catalyzed Cycloisomerization/Cross-Coupling Cascade
1071
Aromatic Hydroxylation and Amination through Deprotonative Cupration
1072
Borylation of 2-Pyridones
1073
Carbonylative Coupling of Grignard Reagents
1074
Catalytic Difluoromethylation of Aryl Halogenides
1075
Enantioselective Allyl–Allyl Coupling between Boronates and Phosphates
1076
Ring Opening of 2-Alkylenecyclobutanones
1077
Boron Conjugate Addition Reactions
1078
Enantioselective Addition of Boronated Allylcopper Derivatives
1079
Ligand Coupling Reactions of Chiral Sulfoxides
1080
Coupling of Secondary and Tertiary Boronic Esters
1081
Photoredox-Mediated C–H Alkylation of N-Heteroarenes
1082
Preparation of Homoallylic Alcohols in Flow and Batch
1083
Enantioselective Conjugate Alkynylation of β-Aryl-β-trifluoromethyl Enones

Organo- and Biocatalysis

z1085
All PDFs of this category
1085
Catalytic Asymmetric Geminal Difluorination of β-Substituted Styrenes
1086
Asymmetric Mannich Reaction of Aliphatic N-Boc Imines
1087
Biocatalytic Asymmetric Synthesis of Bulky Amines
1088
Indolinecarboxylate-Catalyzed Enantio-selective oxa-Pictet–Spengler Reaction
1089
Chiral Pyridoxamine Catalyzed Transamination of α-Keto Acids
1090
Ser-His is Not a Microprotease
1091
Catalytic Cyanotritylation of Aldehydes
1092
Imidophosphate-Catalyzed Enantioselective Oxa-Pictet−Spengler Reaction
1093
Hydrogen-Bonding Catalysis with Tetraalkylammonium Salts
1094
Vanadium Chloroperoxidase Catalyzed Aza-Achmatowicz Reaction

Polymer-Supported Synthesis

z1095
All PDFs of this category
1095
Flow Reactions in a Palladium/Carbon-Packed Bed Reactor
1096
Aqueous Oxidation of Sugars on Hydrotalcite-Supported Gold Nanoparticles
1097
Asymmetric Michael and Aldol Reactions with a Supported Chiral Diamine
1098
Palladium/γ-Alumina-Catalyzed Amidation of Esters with Formamides
1099
Controlled Hydrogenation of Alkynes with Nickel Nanoparticles on an Ionic Liquid
1100
Asymmetric Michael Reaction on a Polystyrene-Supported Organocatalyst
1101
Cyanation of Enones on Polystyrene-Supported Ammonium Fluoride
1102
Suzuki–Miyaura Coupling on Palladium/Mesoporous Silica Microspheres in Water
1103
Synthesis of 3-(Aminoalkyl)indoles on Silver/Silver–Nickel Alloy Nanoparticles
1104
Hβ Zeolite Catalyzed Tandem Alkyne Hydration/Aldol Condensation
1105
Friedel–Crafts Acylation with a Polymer-Supported Indium(III) Catalyst
1106
Suzuki–Miyaura Coupling with Palladium Nanoparticles on Activated Carbon
1107
Photoreduction of Nitroarenes on Palladium/Silica
1108
Magnetic Zirconia Nanoparticle Catalyzed Trimethylsilylation of Alcohols
1109
Synthesis of 1,2,3-Triazoles on Cuttlebone-Supported Copper(II) Chloride
1110
Pt Nanoparticle/Polystyrene Catalyzed Indole Synthesis by Aerobic Oxidation

Erratum

1111
Liao, S.; Leutzsch, M.; Monaco, M. R.; List, B.: Organocatalytic Transformation of Epoxides into Thiiranes