DOI: 10.1055/s-00000084

Synthesis

Issue 11 · Volume 2003 · August 2003 DOI: 10.1055/s-002-2719

editorial

  • I

    Editorial

    • paper

  • 1639
    Lennon, Ian C.; Pilkington, Christopher J.:

    The Application of Asymmetric Hydrogenation for the Manufacture of Pharmaceutical­ Intermediates: The Need for Catalyst Diversity

    Image for article: The Application of Asymmetric Hydrogenation for the Manufacture of Pharmaceutical­ Intermediates: The Need for Catalyst Diversity
  • 1643
    Miller, Joseph A.; Dankwardt, John W.; Penney, Jonathan M.:

    Nickel Catalyzed Cross-Coupling and Amination Reactions of Aryl Nitriles

    Image for article: Nickel Catalyzed Cross-Coupling and Amination Reactions of Aryl Nitriles
  • 1649
    Nettekoven, Matthias; Püllmann, Bernd; Schmitt, Sébastien:

    Synthetic Access to 2-Amido-5-aryl-8-methoxy-triazolopyridine and 2-Amido-5-morpholino-8-methoxy-triazolopyridine Derivatives as Potential Inhibitors of the Adenosine Receptor Subtypes

    Image for article: Synthetic Access to 2-Amido-5-aryl-8-methoxy-triazolopyridine and 2-Amido-5-morpholino-8-methoxy-triazolopyridine Derivatives as Potential Inhibitors of the Adenosine Receptor Subtypes
  • 1653
    Florjancic, Alan S.; Sheppard, George S.:

    A Practical Synthesis of α-Amino Ketones via Aryllithium Addition to N-Boc-α-Amino Acids

    Image for article: A Practical Synthesis of α-Amino Ketones via Aryllithium Addition to <EM EMTYPE="ITALIC">N</EM>-Boc-α-Amino Acids
  • 1657
    Wu, George; Huang, Mingsheng; Richards, Monique; Poirier, Marc; Wen, Xin; Draper, Richard W.:

    Novel ZnX2-Modulated Pd/C and Pt/C Catalysts for Chemoselective Hydrogenation and Hydrogenolysis of Halogen-Substituted Nitroarenes, Alkenes, Benzyl Ethers, and Aromatic Ketones

    Image for article: Novel ZnX<SUB>2</SUB>-Modulated Pd/C and Pt/C Catalysts for Chemoselective Hydrogenation and Hydrogenolysis of Halogen-Substituted Nitroarenes, Alkenes, Benzyl Ethers, and Aromatic Ketones
  • 1661
    Kudzma, Linas V.:

    Synthesis of Substituted Indoles and Carbazoles from 2-Fluorophenyl Imines

    Image for article: Synthesis of Substituted Indoles and Carbazoles from 2-Fluorophenyl Imines
  • 1667
    Hinterding, Klaus; Cottens, Sylvain; Albert, Rainer; Zecri, Frederic; Buehlmayer, Peter; Spanka, Carsten; Brinkmann, Volker; Nussbaumer, Peter; Ettmayer, Peter; Hoegenauer, Klemens; Gray, Nathanael; Pan, Shifeng:

    Synthesis of Chiral Analogues of FTY720 and its Phosphate

    Image for article: Synthesis of Chiral Analogues of FTY720 and its Phosphate
  • 1671
    Kuzmich, Daniel; Mulrooney, Carol:

    Synthesis of 2-Aryl-1-hydroxyazaindoles and 2-Arylazaindoles via Oxidation of o-Hydroxyaminostyrylpyridines

    Image for article: Synthesis of 2-Aryl-1-hydroxyazaindoles and 2-Arylazaindoles via Oxidation of <EM EMTYPE="ITALIC">o-</EM>Hydroxyaminostyrylpyridines
  • 1679
    Blaser, Hans-Ulrich; Burkhardt, Stephan; Kirner, Hans Jürg; Mössner, Tanja; Studer, Martin:

    Ethyl 2,4-Dioxo-4-phenylbutyrate: A Versatile Intermediate for the Large-Scale Preparation of Enantiomerically Pure α-Hydroxy and α-Amino Acid Esters

    Image for article: Ethyl 2,4-Dioxo-4-phenylbutyrate: A Versatile Intermediate for the Large-Scale Preparation of Enantiomerically Pure α-Hydroxy and α-Amino Acid Esters
  • 1683
    Beaulieu, Pierre L.; Haché, Bruno; von Moos, Elisabeth:

    A Practical Oxone®-Mediated, High-Throughput, Solution-Phase Synthesis of Benzimidazoles from 1,2-Phenylenediamines and Aldehydes and its Application to Preparative Scale Synthesis

    Image for article: A Practical Oxone®-Mediated, High-Throughput, Solution-Phase Synthesis of Benzimidazoles from 1,2-Phenylenediamines and Aldehydes and its Application to Preparative Scale Synthesis
  • 1693
    Caron, Stéphane; Do, Nga M.; Arpin, Patrice; Larivée, Alexandre:

    Enantioselective Addition of a Trifluoromethyl Anion to Aryl Ketones and Aldehydes

    Image for article: Enantioselective Addition of a Trifluoromethyl Anion to Aryl Ketones and Aldehydes
  • 1699
    Geiwiz, J.; Goetschi, E.; Hebeisen, P.:

    Concise Synthesis of Cyclothialidine Analogues with Ring Sizes from 12 to 15: Novel Macrocyclization Protocol Involving Reductive Thiolation

    Image for article: Concise Synthesis of Cyclothialidine Analogues with Ring Sizes from 12 to 15: Novel Macrocyclization Protocol Involving Reductive Thiolation
  • 1705
    Liu, Ligong:

    Enantioselective Synthesis of Protoberberine Alkaloids via (-)-Sparteine-mediated Asymmetric Condensation-Cyclisation of o-Toluamide Anions with 3,4-Dihydroisoquinolines

    Image for article: Enantioselective Synthesis of Protoberberine Alkaloids via (-)-Sparteine-mediated Asymmetric Condensation-Cyclisation of <EM EMTYPE="ITALIC">o</EM>-Toluamide Anions with 3,4-Dihydroisoquinolines
  • 1707
    Grieder, Alfred; Thomas, Andrew W.:

    A Concise Building Block Approach to a Diverse Multi-Arrayed Library of the Circumdatin Family of Natural Products

    Image for article: A Concise Building Block Approach to a Diverse Multi-Arrayed Library of the Circumdatin Family of Natural Products
  • 1712
    Berger, Dan M.; Birnberg, Gary; DeMorin, Frenel; Dutia, Minu; Powell, Dennis; Wang, Yanong D.:

    Regioselective Synthesis of a Potent Src Kinase Inhibitor: 4-(2,4-Dichloro-5-methoxyphenylamino)-7-methoxy-8-(2-morpholin-4-ylethoxy)benzo[g]quinoline-3-carbonitrile

    Image for article: Regioselective Synthesis of a Potent Src Kinase Inhibitor: 4-(2,4-Dichloro-5-methoxyphenylamino)-7-methoxy-8-(2-morpholin-4-ylethoxy)benzo[<EM EMTYPE="ITALIC">g</EM>]quinoline-3-carbonitrile
  • 1717
    Pei, Yazhong; Carroll, Amy K.; Anderson, Christen M.; Moos, Walter H.; Ghosh, Soumitra S.:

    Design and Combinatorial Synthesis of N-Acyl Iminodiacetic Acids as Bongkrekic Acid Analogues for the Inhibition of Adenine Nucleotide Translocase

    Image for article: Design and Combinatorial Synthesis of <EM EMTYPE="ITALIC">N</EM>-Acyl Iminodiacetic Acids as Bongkrekic Acid Analogues for the Inhibition of Adenine Nucleotide Translocase
  • 1722
    Andrews, David M.; Borthwick, Alan D.; Chaignot, Helene; Jones, Paul S.; Robinson, J. Ed; Shah, Pritom; Slater, Martin J.; Upton, Richard J.:

    Pyrrolidine-5,5-trans-lactams 3. Alternative Regiochemical Outcome of the Acyl-Iminium Coupling Reaction.

    Image for article: Pyrrolidine-5,5-<EM EMTYPE="ITALIC">trans</EM>-lactams 3. Alternative Regiochemical Outcome of the Acyl-Iminium Coupling Reaction.
  • 1727
    Singer, Robert A.; Caron, Stephane; McDermott, Ruth E.; Arpin, Patrice; Do, Nga M.:

    Alternative Biarylphosphines for Use in the Palladium-Catalyzed Amination of Aryl Halides

    Image for article: Alternative Biarylphosphines for Use in the Palladium-Catalyzed Amination of Aryl Halides
  • 1732
    Hu, X. Eric; Kim, Nick K.; Grinius, Leo; Morris, Charles M.; Wallace, Cynthia D.; Mieling, Glen E.; Demuth, Thomas P.:

    Synthesis of (5S)-Tricyclic Penems as Novel and Potent Inhibitors of Bacterial Signal Peptidases

    Image for article: Synthesis of (5<EM EMTYPE="ITALIC">S</EM>)-Tricyclic Penems as Novel and Potent Inhibitors of Bacterial Signal Peptidases
  • 1739
    Graveleau, Nadège; Masquelin, Thierry:

    Solid-Phase Synthesis of Pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-diones

    Image for article: Solid-Phase Synthesis of Pyrimido[4,5-<EM EMTYPE="ITALIC">d</EM>]pyrimidine-2,4(1<EM EMTYPE="ITALIC">H</EM>,3<EM EMTYPE="ITALIC">H</EM>)-diones

    • synthesis alerts

  • 1744
    Kocienski, P. J.:

    Synthesis Alerts 11/03

    • book review

  • 1752
    Laali, Kenneth K.:

    Ionic Liquids in Synthesis