Synthesis

Issue 11 · August 2003

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1639
Lennon, Ian C.; Pilkington, Christopher J.: The Application of Asymmetric Hydrogenation for the Manufacture of Pharmaceutical Intermediates: The Need for Catalyst Diversity

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1643
Miller, Joseph A.; Dankwardt, John W.; Penney, Jonathan M.: Nickel Catalyzed Cross-Coupling and Amination Reactions of Aryl Nitriles

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1649
Nettekoven, Matthias; Püllmann, Bernd; Schmitt, Sébastien: Synthetic Access to 2-Amido-5-aryl-8-methoxy-triazolopyridine and 2-Amido-5-morpholino-8-methoxy-triazolopyridine Derivatives as Potential Inhibitors of the Adenosine Receptor Subtypes

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1653
Florjancic, Alan S.; Sheppard, George S.: A Practical Synthesis of α-Amino Ketones via Aryllithium Addition to N-Boc-α-Amino Acids

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1657
Wu, George; Huang, Mingsheng; Richards, Monique; Poirier, Marc; Wen, Xin; Draper, Richard W.: Novel ZnX₂-Modulated Pd/C and Pt/C Catalysts for Chemoselective Hydrogenation and Hydrogenolysis of Halogen-Substituted Nitroarenes, Alkenes, Benzyl Ethers, and Aromatic Ketones

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1661
Kudzma, Linas V.: Synthesis of Substituted Indoles and Carbazoles from 2-Fluorophenyl Imines

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1667
Hinterding, Klaus; Cottens, Sylvain; Albert, Rainer; Zecri, Frederic; Buehlmayer, Peter; Spanka, Carsten; Brinkmann, Volker; Nussbaumer, Peter; Ettmayer, Peter; Hoegenauer, Klemens; Gray, Nathanael; Pan, Shifeng: Synthesis of Chiral Analogues of FTY720 and its Phosphate

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1671
Kuzmich, Daniel; Mulrooney, Carol: Synthesis of 2-Aryl-1-hydroxyazaindoles and 2-Arylazaindoles via Oxidation of o-Hydroxyaminostyrylpyridines

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1679
Blaser, Hans-Ulrich; Burkhardt, Stephan; Kirner, Hans Jürg; Mössner, Tanja; Studer, Martin: Ethyl 2,4-Dioxo-4-phenylbutyrate: A Versatile Intermediate for the Large-Scale Preparation of Enantiomerically Pure α-Hydroxy and α-Amino Acid Esters

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1683
Beaulieu, Pierre L.; Haché, Bruno; von Moos, Elisabeth: A Practical Oxone®-Mediated, High-Throughput, Solution-Phase Synthesis of Benzimidazoles from 1,2-Phenylenediamines and Aldehydes and its Application to Preparative Scale Synthesis

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1693
Caron, Stéphane; Do, Nga M.; Arpin, Patrice; Larivée, Alexandre: Enantioselective Addition of a Trifluoromethyl Anion to Aryl Ketones and Aldehydes

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1699
Geiwiz, J.; Goetschi, E.; Hebeisen, P.: Concise Synthesis of Cyclothialidine Analogues with Ring Sizes from 12 to 15: Novel Macrocyclization Protocol Involving Reductive Thiolation

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1705
Liu, Ligong: Enantioselective Synthesis of Protoberberine Alkaloids via (-)-Sparteine-mediated Asymmetric Condensation-Cyclisation of o-Toluamide Anions with 3,4-Dihydroisoquinolines

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1707
Grieder, Alfred; Thomas, Andrew W.: A Concise Building Block Approach to a Diverse Multi-Arrayed Library of the Circumdatin Family of Natural Products

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1712
Berger, Dan M.; Birnberg, Gary; DeMorin, Frenel; Dutia, Minu; Powell, Dennis; Wang, Yanong D.: Regioselective Synthesis of a Potent Src Kinase Inhibitor: 4-(2,4-Dichloro-5-methoxyphenylamino)-7-methoxy-8-(2-morpholin-4-ylethoxy)benzo[g]quinoline-3-carbonitrile

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1717
Pei, Yazhong; Carroll, Amy K.; Anderson, Christen M.; Moos, Walter H.; Ghosh, Soumitra S.: Design and Combinatorial Synthesis of N-Acyl Iminodiacetic Acids as Bongkrekic Acid Analogues for the Inhibition of Adenine Nucleotide Translocase

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1722
Andrews, David M.; Borthwick, Alan D.; Chaignot, Helene; Jones, Paul S.; Robinson, J. Ed; Shah, Pritom; Slater, Martin J.; Upton, Richard J.: Pyrrolidine-5,5-trans-lactams 3. Alternative Regiochemical Outcome of the Acyl-Iminium Coupling Reaction.

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1727
Singer, Robert A.; Caron, Stephane; McDermott, Ruth E.; Arpin, Patrice; Do, Nga M.: Alternative Biarylphosphines for Use in the Palladium-Catalyzed Amination of Aryl Halides

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1732
Hu, X. Eric; Kim, Nick K.; Grinius, Leo; Morris, Charles M.; Wallace, Cynthia D.; Mieling, Glen E.; Demuth, Thomas P.: Synthesis of (5S)-Tricyclic Penems as Novel and Potent Inhibitors of Bacterial Signal Peptidases

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1739
Graveleau, Nadège; Masquelin, Thierry: Solid-Phase Synthesis of Pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-diones

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synthesis alerts
1744
Kocienski, P. J.: Synthesis Alerts 11/03 FREE ACCESS

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book review
1752
Laali, Kenneth K.: Ionic Liquids in Synthesis FREE ACCESS

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