DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 8 · August 2012 DOI: 10.1055/s-002-23511

Synform

  • A75

    SYNFORM ISSUE 2012/08

    • Synthesis of Natural Products and Potential Drugs

  • z811

    All PDFs of this category

  • 0811

    Synthesis of a CB1 Cannabinoid Receptor Antagonist

  • 0812

    Synthesis of (S)-Duloxetine

  • 0813

    Synthesis of (–)-Berkelic Acid

  • 0814

    Synthesis of Anominine and Tubingensin A

  • 0815

    Synthesis of a Telithromycin Analogue

  • 0816

    Synthesis of (–)-13-Oxyingenol and Its Natural Derivative

  • 0817

    Synthesis of a Glucosylceramide Synthase Inhibitor

  • 0818

    Synthesis of (+)-Gelsemine

  • 0819

    Synthesis of an Akt Kinase Inhibitor

  • 0820

    Synthesis of Pellasoren A

  • 0821

    Synthesis of (+)-Chimonanthine

  • 0822

    Synthesis of (R)-Ramatroban

  • 0823

    Synthesis of PF-00951966

  • 0824

    Synthesis of a Glucokinase Activator

  • 0825

    Synthesis of LY500307

  • 0826

    Synthesis of Doxercalciferol

  • 0827

    Synthesis of (–)-Mersicarpine

  • 0828

    Synthesis of AZD6906

    • Synthesis of Heterocycles

  • z829

    All PDFs of this category

  • 0829

    Au-Catalyzed Carbonyl Migration for the Synthesis of Azepinoindol-1-ones

  • 0830

    One-Pot Pd-Catalyzed Synthesis of Isoquinolines and Furo/Thienopyridines

  • 0831

    Synthesis of Isoquinolin-1(2H)-ones via Pd-Catalyzed Isocyanide Coupling

  • 0832

    Synthesis of Piperazine-2,5-diones via a Convenient Dieckmann Cyclization

  • 0833

    A Cu-Catalyzed Double C–N Coupling Approach to Cinnolines

  • 0834

    Functionalized Enantioenriched Dihydropyrans by [4+2] Cycloaddition

  • 0835

    DABCO-Mediated [4+2] Annulation Approach to 2,3-Dihydropyran-4-ones

  • 0836

    Selectivity in Palladium-Catalyzed Carboesterification – Amides versus Esters

  • 0837

    Synthesis of Benzofuro[3,2-d]pyrimidines from 3-Chlorochromones

  • 0838

    Synthesis and Suzuki Coupling of 2-Aryl-Trisubstituted Oxazoles

  • 0839

    Indoloazocines via a Sequential Ugi–Gold-Catalyzed Hydroarylation

  • 0840

    Polysubstituted Pyridines via Re-Catalyzed Alkyne Insertion

  • 0841

    Synthesis of 3-Carboxylated Indoles from 2-Ethynylanilines and CO2

  • 0842

    Iron-Catalyzed Substitution of Benzoxazoles and Benzothiazoles

  • 0843

    Palladium-Catalyzed Synthesis of Indoles via Oxidative C–H Activation

    • Synthesis of Materials and Unnatural Products

  • z845

    All PDFs of this category

  • 0845

    Polyethylene from Trimethylsulfoxonium Halide in Water

  • 0846

    Stabilized Heptacene for n-Type Materials

  • 0847

    Large Twisted Acenes

  • 0848

    Stable Boron–Boron Triple Bond

  • 0849

    Highly Flexible COT

  • 0850

    π-Conjugated Polycycle Containing Boron

  • 0851

    Zipping Oligo-Alkynes into Aromatic Ribbons

  • 0852

    Sensing Chirality of α-Hydroxyl Carboxylic Acids with a Fluorescent Polymer

  • 0853

    Activated Alumina Activates C–F Bonds: A New Route to PAHs

  • 0854

    Synthesis of New Types of Subporphyrins

  • 0855

    π-Expanded Diketopyrrolopyrrole Dyes

  • 0856

    Diastereoselective [2+2+2] Cycloisomerization in the Synthesis of Helicenes

    • Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

  • z857

    All PDFs of this category

  • 0857

    Palladium-Catalyzed Asymmetric Quaternary Stereocenter Formation

  • 0858

    Sc-Catalyzed Enantioselective Allylation of Isatins

  • 0859

    Rh-Catalyzed Addition of Arylboronic Acids to α,β-Unsaturated Sulfonyls

  • 0860

    Asymmetric, Titanium-Mediated Aldol-Type Enamide–Aldehyde Cyclization

  • 0861

    Copper-Catalyzed Highly Diastereoselective [3+3] Cycloaddition

  • 0862

    Rh-Catalyzed Amination of Tertiary Allylic Trichloroacetimidates

  • 0863

    Zinc–ProPhenol-Catalyzed Asymmetric Spirannulation of α-Hydroxyoxindoles

  • 0864

    Chiral Tin Dibromide Catalyzed Enantioselective N-Nitroso Aldol Reaction

  • 0865

    Asymmetric Allylic Alkylation of Pyrroles and 4,7-Dihydroindoles

  • 0866

    Asymmetric Epoxidations of Enones Mediated by Non-Heme Iron Catalysts

  • 0867

    Enantioselective Synthesis of Pyridylcarbinols

  • 0868

    Copper-Catalyzed Synthesis of Heterobicyclo[3.1.1]heptan-6-ones

  • 0869

    Iridium-Catalyzed Asymmetric Synthesis of syn-3-Fluoro-1-alcohols

  • 0870

    Rhodium-Catalyzed Cyclopropanation of Azido Alkenes

  • 0871

    Ru-Catalyzed Asymmetric Hydrogenation of Unsaturated β-Keto Esters

  • 0872

    Inversion of Chirality by Redox-Induced Catalyst Reconfiguration

  • 0873

    Palladium-Catalyzed Asymmetric Allylic Alkylation of Pyrroles

  • 0874

    Palladium-Catalyzed Asymmetric 6-endo Cyclization of Dienamides

  • 0875

    Au-Catalyzed Enantioselective Cope Rearrangement

  • 0876

    Ion-Paired Ligands for Palladium-Catalyzed Asymmetric Allylation

  • 0877

    Catalytic Hydrogenation for the Preparation of Alkyl Boron Compounds

  • 0878

    Multinuclear Cu-Catalyzed Asymmetric Conjugate Addition

  • 0879

    Pd-Catalyzed Asymmetric Synthesis of Indolines

  • 0880

    Palladium-Catalyzed Asymmetric Synthesis of Dibenzosiloles

  • 0881

    Ru-Catalyzed Enantioselective Addition of Amines to Styrenes

  • 0882

    Ni-Catalyzed Ring Opening of Cyclopropanes with Amines

  • 0883

    Scandium-Catalyzed Enantioselective Epoxidation of Chalcones

  • 0884

    Au(I)-Catalyzed Asymmetric Hydroamination of Racemic Allenes

  • 0885

    Cu-Catalyzed Reductive Coupling of Alkenylazaarenes with Ketones

    • Metal-Mediated Synthesis

  • z887

    All PDFs of this category

  • 0887

    Cu-Catalyzed/Ru-Photocatalyzed Trifluoromethylation of Boronic Acids

  • 0888

    Co-Catalyzed Asymmetric Addition of Acetylenes to Benzonorbornadienes

  • 0889

    Alkylmagnesium Reagents from Boron–Magnesium Exchange

  • 0890

    One-Pot Synthesis of 4-Aryl-N-methyl-1,2,3,4-tetrahydroisoquinolines

  • 0891

    β-Arylation of Ketones by a 1,4-Addition Sequence under Flow Conditions

  • 0892

    Asymmetric Ring Opening of Aziridines with Halides

  • 0893

    Amide-Forming Ligation of Acyltrifluoroborates and Hydroxylamines

  • 0894

    Novel Lewis Acid ATNP for Vinylogous Aldol Reactions

  • 0895

    Asymmetric Synthesis of Secondary Nitriles via Negishi Cross-Coupling

  • 0896

    Intramolecular Vinylation of Organolithiums

  • 0897

    Synthesis of Fluorinated Cyclopropanes

  • 0898

    Mes2Mg-Mediated Shapiro Reactions of Tosylhydrazones

  • 0899

    New Iron Thiolate Complexes for Cross-Coupling Reactions

  • 0900

    Synthesis of 1,4-Dihydropyridines and Pyridines out of N-Allyl Ynamides

  • 0901

    Ni-Catalyzed Alkylation of Purines and Benzimidazoles with Grignard Reagents

    • Organo- and Biocatalysis

  • z903

    All PDFs of this category

  • 0903

    Organocatalytic Approach to N−H Insertion Reactions

  • 0904

    Vinylogous Michael Addition Catalyzed by Cinchona Thiourea

  • 0905

    Catalytic Asymmetric 1,6-Addition of Alkyl Thiol to Cyclic Dienones

  • 0906

    Regiodivergent Asymmetric Allylic Alkylation

  • 0907

    Asymmetric Fluorination of Enamides

  • 0908

    α-Vinylation of Aldehydes via Combination of Copper and Aminocatalysis

  • 0909

    [4+2] Cycloaddition Catalyzed by Quinine-Derived Primary Amine

  • 0910

    Modified Cinchona Amine Catalyzed Epoxidation of 2-Cyclopentenones

  • 0911

    Catalytic Asymmetric Ring-Opening Reactions of Aziridines

  • 0912

    Enzymatic Reductive Amination of Diketones

    • Polymer-Supported Synthesis

  • z913

    All PDFs of this category

  • 0913

    Asymmetric Michael Addition of Aldehydes to Nitroalkenes Using JH-CPP

  • 0914

    Aerobic Oxidation of α-Hydroxy Ketones with CaO

  • 0915

    Epoxidation of Olefins with a Silica-Supported Peracid in Flowing scCO2

  • 0916

    Au/MoOx-Catalyzed Aerobic Oxidation of Alcohols

  • 0917

    A RuNPs-Based Supramolecular Hydrogel for Hydrogenation of Alkenes

  • 0918

    DMAP-Embedded Nanoporous Conjugated Polymer

  • 0919

    Asymmetric Hydrogenation of Ketones with Cp*RhTsDPEN-POSS

  • 0920

    Direct Synthesis of Vitamin K4 Using Bifunctional Heterogeneous Catalyst

  • 0921

    One-Pot Sonogashira–Click Coupling with a Cu-Pd MOF Catalyst

  • 0922

    Suzuki Coupling with Polymer-Supported Pd Nanoparticles in Water

  • 0923

    A3-Coupling Using TiO2-Supported Copper Nanoparticles

  • 0924

    Asymmetric Aldol Reaction with a Polymeric Organocatalyst

  • 0925

    Ring Opening of Epoxides Catalyzed by Graphene Oxide

  • 0926

    Hydration of Nitriles to Amides with Fe3O4@SiO2–Ru Catalyst

    • Addenda and Errata

  • 0927

    Synthesis of Acrivastine

  • 0927

    Ullmann Diaryl Etherification with Copper Fluorapatite

    • Erratum

  • 0927

    Synthesis of (+)-Scholarisine A