DOI: 10.1055/s-00000131

Synfacts

Issue 01 · Volume 8 · January 2012 DOI: 10.1055/s-002-22508

Editorial

I
Editorial

Synform

A1
Zanda, Matteo: SYNFORM ISSUE 2012/01

Synthesis of Natural Products and Potential Drugs

z1
All PDFs of this category
0001
Synthesis of MK-7655
0002
Synthesis of Gelsemoxonine
0003
Synthesis of Pyripyropene A
0004
Synthesis of a PDE IVb Inhibitor
0005
Synthesis of Abamines
0006
Synthesis of Vaniprevir (MK-7009)
0007
Synthesis of (–)-Huperzine A
0008
Formal Synthesis of (–)-Indatraline
0009
Synthesis of Lonafarnib
0010
Synthesis of Florfenicol
0011
Synthesis of (+)-Yohimbine
0012
Synthesis of (±)-Dragmacidin E
0013
Synthesis of (±)-Hamayne
0014
Synthesis of (–)-8-Demethoxyrunanine and (–)-Cepharatines A, C and D
0015
Synthesis of (+)-Sertraline

Synthesis of Heterocycles

z17
All PDFs of this category
0017
Synthesis of Azabicyclo[3.1.1]heptane Derivatives from Cyclobutanones
0018
Ni-Catalyzed Cycloaddition Approach to Fused Pyridine Derivatives
0019
Phthalimide Synthesis via Oxidative Carbonylation of Benzamides
0020
[3+2]-Dipolar Cycloaddition Route to 2H-Indazoles
0021
Organocatalytic [3+2]-Cycloaddition Route to 1,2,3-Triazoles
0022
Pd-Catalyzed Cross-Coupling–Lactonization Route to Dibenzopyranones
0023
Concise Synthesis of Trifluoromethyl-Substituted Benzofuranols
0024
Quinolines and Tetrahydroquinolines via Pd(0)-Catalyzed C–H Bond Functionalization
0025
Intramolecular Heck-Type Synthesis of Piperideines and Pyridines
0026
Synthesis of 3,4-Diaryl-3-pyrrolin-2-ones from Pyrrole Weinreb Amides
0027
Pd-Catalyzed Synthesis of Furans from 1,3-Dicarbonyls and Propargylic Alcohols
0028
Mitsunobu-Based Synthesis of Four-Membered Cyclic Oxaphosphetanes
0029
Organocatalytic Enantioselective Synthesis of Functionalized Piperidines
0030
One-Pot Synthesis of Benzo[b]furans from Phenols and Bromoalkynes
0031
Stannous Chloride Mediated Synthesis of Spiroindolinone Quinazolines

Synthesis of Materials and Unnatural Products

z33
All PDFs of this category
0033
Polyenyne Cascade is Good as Gold
0034
An Efficient Route to Tetrathia[7]helicenes
0035
Taming 3,4-Dioxypyrroles
0036
Steric Strain Driven BODIPY Functionalization
0037
Switch the Light and the Carbenes!
0038
Supramolecular Russian Dolls by Self-Assembly
0039
Benzodipyrrolidone-Based Polymer: A New Donor–Acceptor Motif
0040
Simple Synthesis of Buckybowls
0041
Head-to-Tail-Type Oligothiophenes
0042
A ’Smart’ Polymer Disassembles in Near Infrared Light
0043
Coupling C,C-Diacetylenic Phosphaalkene this Way and that
0044
Unsymmetrical 9,10-Dihydro-9,10-dibora-anthracenes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z45
All PDFs of this category
0045
Asymmetric Conjugate Addition Catalyzed by a Nickel–Diamine Complex
0046
Gold-Catalyzed Diastereoselective Oxidative Cyclizations
0047
Palladium-Catalyzed Asymmetric Allyl–Allyl Cross-Coupling
0048
Yamamoto, Hisashi; Griffin, Kimberly: Cr(III)-Catalyzed AKR/ARO of Epoxides to β-Amino Alcohols
0049
Asymmetric Monofluoromethylation by Co-operative Organo- and Lewis Acid Catalysis
0050
Novel Carbohydrate-Derived Ligands for Asymmetric Transfer Hydrogenation
0051
Asymmetric Approach to Chiral Pyrogluta-mates with a Quaternary Stereocenter
0052
Rhodium-Catalyzed [2+2+2] Reaction of Ethynyl Ethers with Carbonyl Compounds
0053
Iridium-Catalyzed Asymmetric Hydrogenation with Proline-Based P,O Ligands
0054
Diastereoselective Cobalt-Catalyzed Multicomponent Couplings
0055
Ni-Catalyzed Asymmetric α-Arylation and Heteroarylation of Ketones
0056
Rhodium-Catalyzed Asymmetric Hydrogenation of Unsaturated Phosphonates
0057
Advances in Nazarov Cyclizations through Control of [1,2]-Migrations
0058
Palladium-Catalyzed Enantioselective Overman Rearrangement
0059
Cationic Palladium Catalyzed Stereoselective Synthesis of Aminoindenes
0060
Palladium-Catalyzed Stereoselective Transfer Hydrogenation of Alkynes
0061
Cyclometalated Complex Library for Transfer Hydrogenation
0062
Chiral Tetrahydroquinolines via an Aziridine Ring Opening/C–N Bond Formation Sequence
0063
Scandium-Catalyzed Electrophilic Addition of α-Diazoesters with Ketones
0064
New Cobalt Porphyrin Catalysts in Asymmetric Intramolecular Cyclopropanation
0065
Pyrrolines via SnCl4-Mediated [3+2] Cycloadditions of Cyclopropanes and Nitriles
0066
Enantioselective and Regioselective Indium-Catalyzed Addition of Pyrroles to Isatins
0067
Rhodium-Catalyzed 1:2 Coupling of Aldehydes with Allenes
0068
Lewis Base Catalyzed Enantioselective Hypervinylogous Aldol Reactions
0069
Yamamoto, Hisashi; Usanov, Dmitry L.: Trifluoromethylated Pyrrolidines via Cu-Mediated 1,3-Dipolar Cycloaddition
0070
Catalyst-Controlled Gold-Catalyzed Carbocyclizations
0071
Copper-Catalyzed Asymmetric Alkoxyamination
0072
Asymmetric Synthesis of Amino Acids by Dehydrogenative Coupling
0073
Regio- and Enantioselective Synthesis of Trifluoromethyl Allylic Amines

Metal-Mediated Synthesis

z75
All PDFs of this category
0075
Ag-Mediated C–H Trifluoromethylation of Aromatic Substrates
0076
Direct Hiyama Coupling of Enaminones With Triethoxy(aryl)silanes
0077
Boron–Ate Complexes as Chiral Nucleophiles for Asymmetric Synthesis
0078
Cu-Catalyzed Enantioselective Addition of Alkynes to Isochroman Acetals
0079
Selective Synthesis of Highly Substituted Isoquinolines
0080
Total Synthesis of (+)-Erogorgiaene Using Lithiation–Borylation Methodology
0081
Diastereoselective α-Trifluoromethylation of Carbonyl Compounds
0082
Aldehydes in Bifunctional Titanocene-Catalyzed Propargylic C–X Activations
0083
Knochel, Paul; Barl, Nadja M.: Scandium-Catalyzed Silylation of Aromatic C–H Bonds
0084
Direct Synthesis of Alkynylstannanes from Tributyltin Methoxide and Alkynes
0085
A New Method for the Synthesis of Difluoromethylated Aromatics
0086
Knochel, Paul; Sämann, Christoph: BiCl3-Catalyzed Synthesis of Alkoxy- and Acetoxysilanes from Chlorosilanes
0087
Knochel, Paul; Steib, Andreas K.: CoBr2-Catalyzed Direct Allylation of Alkyl Halides
0088
Chemo- and Regioselective Synthesis of Aluminoisoxazoles and Pyrazoles
0089
Enantioselective Preparation and Chemo-selective Coupling of 1,1-Diboronyls

Organo- and Biocatalysis

z91
All PDFs of this category
0091
NHC-Catalyzed Asymmetric Hydroacylation of Cyclopropenes
0092
SN2′–SN2 Sequence of Morita–Baylis–Hillman Adducts
0093
The Catalytic Asymmetric Fischer Indolization
0094
Enantioselective Protonation via an Enamine Intermediate
0095
Enantioselective Synthesis of α-Chiral 1,3-Azoles
0096
α-Arylation of Enals via Aminocatalysis
0097
Merging Organo- and Metal Catalysis
0098
Asymmetric Allylic Trifluoromethylation of Morita–Baylis–Hillman Adducts
0099
Stereoselective Addition of Azlactones to 3-Vinylindoles
0100
List, Benjamin; Wang, Qinggang: Conjugate Addition Catalyzed by a Recyclable C2-Symmetric Organocatalyst
0101
Michael Addition/Nitronate-Olefin Cycloaddition/Fragmentation Sequence

Polymer-Supported Synthesis

z103
All PDFs of this category
0103
One-Pot Tandem Reactions with a Bifunctional Solid Catalyst
0104
Preparation of 3,4-Dihydroquinoxalin-2-amines Catalyzed by Amberlyst-15
0105
CuII-MS4Å for Hydration of Nitriles into Amides
0106
Hydrogenation of Unprotected Indoles with Platinum Catalysts
0107
Hosomi–Sakurai Reaction with Silica Gel Supported Perchloric Acid
0108
Uozumi, Yasuhiro; Yamada, Yoichi M. A.; Ohno, Aya: Catalytic Aerobic Oxidation of Alcohols with Pd@PMO-IL
0109
Aerobic Oxidation of Alcohols with Au/MgCr-Hydrotalcite
0110
Uozumi, Yasuhiro; Hamasaka, Go: Synthesis of Quinolines from ArNO2 and Alcohols with Ir/TiO2-NCs
0111
Intermolecular Coupling of Alkynes with Acrylates Using Ru/CeO2
0112
Preparation of Benzimidazoles via Oxidation of Tertiary Amines
0113
Solvent-Free Hydrogenation and Suzuki–Miyaura Coupling Using Pd/C
0114
Hydrolysis of VX Using Solid-Supported Ammonium Fluorides
0115
Friedel–Crafts Addition of Indoles Using Graphite Oxide
0116
Synthesis of Hydroxy-1,2,3-Triazoles with Cu Nanoparticles on Activated Carbon in Water