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Synthesis 2013; 45(16): 2273-2279
DOI: 10.1055/s-0033-1339179
paper
© Georg Thieme Verlag Stuttgart · New York

Rapid Access to 10-(Cyclohexylimino)-7,9-diazaspiro[4.5]decane-6,8-dione Derivatives for HIV-1 Reverse Transcriptase Inhibition via Ruthenium-Catalyzed Ring-Closing Metathesis

Tongbo Zhang
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Shaotong Wu
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Yuanyuan Cao
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Yuhong Fu
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Ying Guo
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Liang Zhang
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Li Li
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Han Zhou
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Xiangyi Liu
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Chao Li
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Xiaowan Tang
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Zhili Zhang
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Chao Tian
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Xiaowei Wang*
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
,
Junyi Liu*
a   Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100191, P. R. of China   Email: xiaoweiwang@bjmu.edu.cn
b   The State Key Laboratory of Natural and Biomimetic Drugs, Peking University, Beijing 100191, P. R. of China   Fax: +86(10)82805203   Email: jyliu@bjmu.edu.cn
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