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Synthesis 2009(7): 1204-1208
DOI: 10.1055/s-0028-1088006
DOI: 10.1055/s-0028-1088006
PAPER
© Georg Thieme Verlag
Stuttgart ˙ New YorkMicrowave-Assisted Synthesis and Functionalization of Selenolopyrimidines
Weitere Informationen
Received
20 November 2008
Publikationsdatum:
06. März 2009 (online)
Publikationsverlauf
Publikationsdatum:
06. März 2009 (online)
Abstract
Microwave-assisted synthesis allowed efficient access to 4-chloroselenolo[3,2-d]pyrimidines in short times and very good yields. Some functionalizations by SNAr and palladium-catalyzed reactions are also reported.
Key words
selenium - pyrimidines - heterocycles - cyclizations - microwave-assisted reactions
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