Download PDF
Synlett 2000; 2000(9): 1257-1260
DOI: 10.1055/s-2000-7146
letter
© Georg Thieme Verlag, Rüdigerstr. 14, 70469 Stuttgart, Germany. All rights reserved. This journal, including all individual contributions and illustrations published therein, is legally protected by copyright for the duration of the copyright period. Any use, exploitation or commercialization outside the narrow limits set by copyright legislation, without the publisher's consent, is illegal and liable to criminal prosecution. This applies in particular to photostat reproduction, copying, cyclostyling, mimeographing or duplication of any kind, translating, preparation of microfilms, and electronic data processing and storage.

The Asymmetric Synthesis of β-Haloaryl-β-Amino Acid Derivatives

Steven D. Bull* , Stephen G. Davies, Santiago Delgado-Ballester, Garry Fenton, Peter M. Kelly, Andrew D. Smith
  • *The Dyson Perrins Laboratory, University of Oxford, South Parks Road, Oxford, UK, OX1 3QY
Further Information

Publication History

Publication Date:
31 December 2000 (online)

  PDF Download  Permissions and Reprints All articles of this category

Lithium N-benzyl-N-α-methyl-4-methoxybenzylamide is employed as a homochiral ammonia equivalent for the asymmetric synthesis of β-haloaryl-β-amino acid derivatives using a conjugate addition/oxidative deprotection strategy.

β-haloaryl β-amino acids - asymmetric synthesis - oxidative debenzylation - homochiral ammonia equivalent

      >