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Synlett 1998; 1998(2): 180-182
DOI: 10.1055/s-1998-1597
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A Convenient Synthesis of Dialkyl [[2-(Bromomethyl)aziridin-1-yl]methyl]phosphonates, New Heterocyclic β-Azaphosphonates

Christian Stevens* , Aart Verbeke, Norbert De Kimpe
  • *Department of Organic Chemistry, Faculty of Agricultural and Applied Biological Sciences, University of Gent, Coupure Links 653, B-9000 Gent, Belgium; Fax 32-9-2 64 62 43; E-mail: Chris.Stevens@rug.ac.be
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Publication History

Publication Date:
31 December 2000 (online)

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Dialkyl [[2-(bromomethyl)aziridin-1-yl]methyl] phosphonates were prepared in good yield by a convenient procedure involving the reaction of 1,3,5-triallylhexahydro[1,3,5]triazine with dialkyl phosphites, subsequent bromination and final ring closure upon treatment with sodium borohydride in methanol.

azaphosphonates - aziridines - aziridinylmethyl phosphonates

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