Synlett 1995; 1995(10): 1061-1062
DOI: 10.1055/s-1995-5172
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Improved Synthesis of 1-Aryl-β-Carbolines

Brian E. Love* , Prasad S. Raje
  • *Department of Chemistry, Auburn University, Auburn, AL 36849, USA
Further Information

Publication History

Publication Date:
31 December 2000 (online)

A method for the preparation of 1-aryl-β-carbolines is reported which provides these compounds in three steps (starting from 1-phenylsulfonyl-3-vinylindole) in yields of 40-60%. This method circumvents the use of acidic conditions at all stages. Additionally, its use in the preparation of a natural product is reported.