Synthesis of a Novel Rhizobitoxine-Like Triazole-Containing Amino Acid
Received: 10 June 2016
Accepted after revision: 05 August 2016
18 August 2016 (eFirst)
The synthesis of the four stereoisomers of a new 1,2,3-triazole analogue of rhizobitoxine from serine is described. The key step is a Huisgen 1,3-dipolar cycloaddition on an ethynylglycine synthon.