Palladium-Catalyzed Intramolecular Direct Arylation for Phosphorus Heterocycle Synthesis

Abstract

A palladium-catalyzed intramolecular direct arylation of bromo-substituted phosphine oxides is reported for the synthesis of phosphorus-containing heterocycles with good to excellent yields (78–98%)

Key words

C–H activation - direct arylation - palladium - phosphorus heterocycles

• References


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