DOI: 10.1055/s-00000131

Synfacts

Ausgabe 04 · Volume 17 · April 2021 DOI: 10.1055/s-011-50572

Synform

  • A49

    SYNFORM ISSUE 2021/04

    • Synthesis of Natural Products and Potential Drugs

  • z0363

    All PDFs of this category

  • 0363

    Total Synthesis of (+)-Peniciketal A

  • 0364

    Total Synthesis of (+)-Mycinolide IV

  • 0365

    Synthesis of PF-07059013

  • 0366

    Synthesis of ent-Plagiochianin B

  • 0367

    Synthesis of (–)-Dehydrocostus Lactone

  • 0368

    Synthesis of Eldecalcitol

  • 0369

    Synthesis of PF-06843195

  • 0370

    Synthesis of DS79932728

  • 0371

    Synthesis of Ceralasertib

  • 0372

    Synthesis of (–)-Euonyminol

  • 0373

    Total Synthesis of (±)-Longifolene

  • 0374

    Total Synthesis of (+)-Punicafolin and (+)-Macaranganin

    • Synthesis of Heterocycles

  • z0375

    All PDFs of this category

  • 0375

    Rhodium(III)-Catalyzed C–H Activation/Annulation To Form Isoquinolone Scaffolds

  • 0376

    Chiral Phosphoric Acid Catalyzed Enantioselective Synthesis of 8-Azabicyclo[4.3.1]decanes

  • 0377

    Preparation of Imidazolidine-2-ones from N-Benzoyloxyureas by C–H Amination

  • 0378

    Nickel/Copper-Catalyzed Amidation of 2-Iodoglycals to Access Glycosamine Analogues

  • 0379

    Palladium-Catalyzed Synthesis of Azepines from Pyrrolidines

  • 0380

    Three-Component Approach to Indoles

  • 0381

    Synthesis of N-Fused Hetarenes from Alkenes

  • 0382

    N-Containing Bicyclic Heterocycles by Annulation of 2H-Azirines with 2-Chloropyridine Derivatives

  • 0383

    Et3N-Direct Cycloaddition of Allenoates with Acceptor Diazo-Compounds

  • 0384

    Diastereoselective Synthesis of 2,3-Dihydrofurans from Silver Allenes

  • 0385

    Synthesis of Enantiomerically Enriched Chiral 1-Pyrrolines

    • Synthesis of Materials and Unnatural Products

  • z0387

    All PDFs of this category

  • 0387

    From Saddles to Helices

  • 0388

    Easy as 1,2,3,4-Tetrasubstituted Benzenes

  • 0389

    An Expedient Approach to a Zigzag Carbon Nanobelt

  • 0390

    Stereospecific Synthesis of Pyrene-Fused [5]Helicenes

  • 0391

    Flip-Flopping Nanohoops

  • 0392

    BRB, Looking for Aromaticity

  • 0393

    Easy as 8π

  • 0394

    Efficient Synthesis of azahelicenes through Imine-Based Mallory Cyclization

  • 0395

    Alternative Retrosynthetic Approach towards Synthesis of Nile Red Analogues

  • 0396

    Facile Functionalization of 6-Aryl-2,20-bipyridines

  • 0397

    No Resolution Necessary

  • 0398

    Novel Synthesis of Piperidinium-Functionalized Polyethylene for Alkaline Anion Exchange Membranes

    • Metals in Synthesis

  • z0399

    All PDFs of this category

  • 0399

    Iron-Catalyzed Asymmetric Carboazidation of Styrenes

  • 0400

    Diastereoselective Synthesis of (Spiro)Indanones by Nickel-Catalyzed Reductive Cyclization

  • 0401

    Acyl Chlorides as Dual Source of Carbon Nucleophile and Carbon Monoxide

  • 0402

    Enantioselective Nickel Hydride Catalyzed Cross Coupling of Alkyl Electrophiles

  • 0403

    Pd(0)-Catalyzed, Stereoselective Intermolecular Cycloaddition: Towards Substituted Cyclopentanes

  • 0404

    α-Arylation of Ketones with Nitroarenes

  • 0405

    Asymmetric Hydroarylation of N-Acyl Enamines

  • 0406

    4-Thiooxazole Synthesis and Sulfanyl–Lithium Exchange

  • 0407

    Palladium-Catalyzed Z-Selective Dienylations

  • 0408

    Silver-Catalyzed Heteroarylation of Aliphatic Alcohols in Water

  • 0409

    Site-Selective Silver-Catalyzed C−H Bond Deuteration of Five-Membered Heterocycles

  • 0410

    Chiral Aldehydes from Cycloproyplacetylenes via Palladium/Organo Dual-Catalysis

  • 0411

    Pd-Catalyzed Enantioselective Carbohalogenation Employing a H-Bonding Driven Reductive Elimination

  • 0412

    Palladium-Catalyzed C–H Addition to Nitriles: α-Iminol Rearrangement

  • 0413

    Scandium-Catalyzed Asymmetric Homologation of Ketones using α-diazo Esters

  • 0414

    Photoredox Catalysis: Decarboxylative Cross-Coupling of Nitrones with α‑Amino Acids

  • 0415

    Enantio- and Diastereoselective Conjugate Addition of Borylalkenes to α,β-Unsaturated Diesters

  • 0416

    Asymmetric Heck–Matsuda Reaction for the Preparation of β-Chiral Ketones

  • 0417

    Enantioselective Sulfimidation of Pyridones and Quinolones via Silver Catalysis

  • 0418

    Copper-Catalyzed Asymmetric Alkylamination of Unactivated Alkenes Generating β-Lactams

  • 0419

    Generation of Secondary and Tertiary Alcohols via Anaerobic Mukaiyama-Type Hydration

  • 0420

    meta-Selective C–H Functionalization of Phenols

  • 0421

    Palladium-Catalyzed Carbonylation of 1,3-Dienes

  • 0422

    Asymmetric Synthesis of 4-Aryl-3,4-dihydrocoumarins by Palladium-Catalyzed Hydroesterification

  • 0423

    Hydrofuctionalization of Styrene via a Photoredox Process Catalyzed by a Decatungstate Complex

  • 0424

    Nickel-Catalyzed Enantioselective Hydroalkylation of Enecarbamates

  • 0425

    Copper-Catalyzed Enantioselective Vinylogous Aldol Reaction of Allylazaarenes

  • 0426

    Asymmetric Conjugate Addition of 1,1-Diborylmethane

  • 0427

    Directed ortho-Lithiation of Benzamides

    • Polymer-Supported Synthesis

  • z0429

    All PDFs of this category

  • 0429

    Synthesis of Alkynylcyclopentenols on a Foam-Supported Palladium Catalyst

  • 0430

    Dehydrogenative Condensation of Anilines with Dioles on Platinum/Alumina

  • 0431

    One-Step Deoxydehydration–Transfer Hydrogenation of Sugar Acids with a Pt–Re Oxide Catalyst

  • 0432

    Supported Cobalt Phosphide Nanoalloy Catalysts for Hydrogenation of Furfurals

  • 0433

    Synthesis of Spiro-4-thiazolidinones on a Porous Polymeric Ionic Liquid Containing Co3O4

  • 0434

    Hydrocarboxylation of Alkenes Catalyzed by Rhodium Supported on Porous Organic Polymer

  • 0435

    Heterogeneous Gold-Nanoparticle-Catalyzed Stille Coupling of Benzylic Bromides and Allylstannanes

  • 0436

    Cobalt-Catalyzed Reductive Alkylation of Nitriles with Aldehydes or Ketones

  • 0437

    Selective Oxidation of Alcohols with TEMPO Supported on Hollow Porous Aromatic Frameworks

  • 0438

    Gold/Titania-Catalyzed Borylation of Allylic, Propargylic, and Benzylic Esters

    • Organo- and Biocatalysis

  • z0439

    All PDFs of this category

  • 0439

    Photoenzymatic Intermolecular Hydroalkylation of Alkenes

  • 0440

    Asymmetric Photoredox Dearomatization of Indoles by Neutral α-Amino Radicals

  • 0441

    Photoenzymatic Reduction of α,β-Unsaturated Amides with Ene-Reductases

  • 0442

    BINOL-Derived Photoswitchable Phase-Transfer Catalysts

  • 0443

    Synthesis of a Chiral Pentafluorinated Isopropyl Group by Aryl Iodide Catalyzed Difluorination of Styrenes

  • 0444

    N-Fluorosulfonyl Carbamate and Organoiodine Catalysis: Vicinal Heterodifunctionalization of Olefins

  • 0445

    Synergistic Dual Organocatalysis for Highly Selective Michael Additions

  • 0446

    Catalytic Asymmetric Chloroamidation of Allylic Amides

  • 0447

    High Lewis Acidity of Bidentate Iodine(III)-Based Halogen-Bond Donors

  • 0448

    Photocatalytic Minisci Alkylation of Azaarenes

  • 0449

    Room-Temperature Carbon Isotope Exchange of Carboxylic Acids Through Photoredox Catalysis

    • Chemistry in Medicine and Biology

  • z0451

    All PDFs of this category

  • 0451

    Sucrose Analogues for Real-Time Imaging of Intracellular Plant Metabolism

  • 0452

    Total Synthesis of Cephalosporin C

  • 0453

    Optical Control of the Cannabinoid Receptor 2

  • 0454

    Novel Prodrugs for Targeted Cancer Therapy

  • 0455

    Light-Induced Cell Cycle Arrest and Apoptosis

  • 0456

    A Potent Preclinical Plasmodium Proteasome Inhibitor

  • 0457

    Modular Chemoenzymatic Synthesis of GE81112 B1

  • 0458

    Diversity-Focused Semisynthesis of Polyether Ionophores with New Antibacterial Selectivity

  • 0459

    Evaluation of C2−C2′ Bond Stereochemistry Influence on Cytotoxicity of (–)-Lomaiviticin A

    • Peptide Chemistry

  • z0461

    All PDFs of this category

  • 0461

    Ball-Milling Strategy for Epimerization-Free Peptide Synthesis

  • 0462

    Rhodium-Catalyzed Synthesis of β2/γ2/δ2-Amino Acid Derivatives

  • 0463

    Synthesis of All-Alkyl α-Tertiary Amino Acid Derivatives under Visible-Light Irradiation

  • 0464

    β-Seleno-α-Amino Acids Synthesis by Seleno-Michael Additions to Bicyclic Dehydroalanine

  • 0465

    Photocatalyzed Modification for Tryptophane-Containing Peptides

  • 0466

    Triflic Acid Catalyzed N–H Insertion Reaction for the Synthesis Unnatural α-Amino Esters

  • 0467

    Synergistic Brønsted Acid/Photoredox Catalysis for the Synthesis of α-Amino Acids

  • 0468

    Rhodium-Catalyzed Formation of Proline Analogues

  • 0469

    Peptide Bond Formation by Using 2-Pyridyl Thio Esters

    • Flow Chemistry

  • z0471

    All PDFs of this category

  • 0471

    Halogen–Lithium Exchange on Isothiocyanate-Substituted Aryl Halides

  • 0472

    Safer Handling of Diazomethane through Continuous Generation and Consumption

  • 0473

    Oxidative Debenzylation of Protected Carbohydrates under Flow Conditions

  • 0474

    Synthesis of Aminoimidazo Heterocycles under Flow Conditions

  • 0475

    Generation and Use of Lithiated 1-Azabicyclo[1.1.0]butanes in Flow Microreactors

  • 0476

    Selective Oxidation of Alcohols under Flow Conditions