Synfacts

Issue 11 · November 2020

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Synthesis of MIDD0301

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Total Synthesis of (±)-Ginkgolide B FREE ACCESS

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Scalable Synthesis of Functionalized gem-Difluorocyclopropanes

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C–H Bond Functionalization of Alicyclic Amines

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Synthesis of 2-Formylpyrroles from Pyridinium Iodide Salts

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Synthesis and Derivatization of N-Trifluoromethylated Indoles

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Mild Regioselective Halogenation of Anilines, Anilides, and Indoles

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Pd-Catalyzed Asymmetric [8+2]-Dipolar Cycloadditions: Synthesis of Ten-Membered Ring Heterocycles

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Cobalt(III)-Catalyzed Synthesis of Isoquinolinones and Pyridinones by Annulative Vinylene Transfer

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Chiral N,O-Acetals by Asymmetric Hydrogenation of Cationic Intermediates

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Metal-Free [5+1]-Cycloaddition Route to Pyrazine 1-Oxides and Pyrazines

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Two-Step Synthesis of Functionalized Benzoxazoles

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A Missing Member of the Cycloarene Family: Quintulene

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Amide–Alkene Isosterism: Synthesis of Olefin-Containing Foldamers

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Getting the SuFEx Right for Sulfamides

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Reductively Aminate, Reuse, Recycle

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Insert COins Here

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Oxygen Chelation Makes it Exclusive: Fluorene-Based Spirocycles via Aryl Halide Cross-Coupling

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Oxidative Dealkylation Strategy toward Functionalized Phenalenones

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Synthesis of as-Indacenoterrylene, a C₇₀ Fragment with NIR absorption

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1297
Air- and Moisture-Tolerant Synthesis of Catechol Boronic Esters

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Suzuki–Miyaura to the Rescue! Expanding the Scope for Tetraarylethylene Synthesis

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1299
Sticking Together: Fused Porphyrins Deliver Protection against Photodegradation to Pentacenes

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1300
The Coronation of Naphthalene Diimides: π-Extended Helicenes by Oxidative Cyclization

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Metals in Synthesis
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Asymmetric γ-Borylation of Aliphatic Amides and Esters FREE ACCESS

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Gold-Catalyzed Carbene Transfer towards the C–H Functionalization of N-Heterocycles

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1303
Dynamic Kinetic Resolution Strategy for the Asymmetric Nickel-Catalyzed Capture of Transient Cyclic Allenes FREE ACCESS

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1304
Visible-Light-Promoted Copper-Catalyzed Difunctionalization of Alkenes with Iodoform

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1305
Chlorocarbonylation of Aryl (Pseudo)Halides via Pd-Catalysis

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Synthesis of δ- and ε-Lactones Through γ-C(sp³)–H Activation of β-Disubstituted Carboxylic Acids

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Ruthenium-Catalyzed Synthesis of Cyclic Tetrasubstituted Olefins

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Synthesis of Cyclopropanes by Double C–H Activation

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1309
Synthesis of C-Aryl Glycosides by Catellani Reaction

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1310
Intermolecular Pd-Catalyzed Carbofunctionalization of Internal Alkynes with trans-Selectivity

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1311
Rh-Catalyzed Three-Component Synthesis of α,α,α-Trisubstituted Esters by C(sp²)–C(sp³) Bond Cleavage

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Photocontrolled Hydroboration of α,β-Unsaturated Ketones

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gem-Hydrogenation of Internal Alkynes by Grubbs Metathesis

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Cobalt-Catalyzed Dienylation of Quinoline-N-Oxides: C8-Selective Alkenylation

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Synthesis of Benzylic Ketones through Electrochemical Oxidation of Aryl Alkenes

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Nickel-Catalyzed Hydroarylation of Alkenes

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Regioselective Alkyne Cyclotrimerization Enabled by Hemilability of Salen Ligand

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1323
Sulfinyl Nitrene Based Synthesis of Sulfoximines and Sulfonimidamides

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1324
Asymmetric Synthesis of α‑Alkylated Pyrrolidinones from Homoallylic Carbamoyl Chlorides

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1325
Carbon Dioxide and Ammonia as Cyanide Source in Nickel-Catalyzed Reductive Cyanation of Aryl Chlorides

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1326
Design of a Catalyst Suitable for Aryl Aminations at Room Temperature

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1327
Titanium-Catalyzed Asymmetric Pauson–Khand Type Reaction FREE ACCESS

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1328
Synthesis of Chiral Alkenylphosphine Oxides

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Polymer-Supported Synthesis
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1329
A Single-Atom Cobalt Catalyst Supported on SBA-15 for Hydrodeoxygenation and Hydrogenation FREE ACCESS

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Enantioselective Addition of Dialkylzinc to Aldehydes on a Heterogeneous Magnetic Nanoparticle Catalyst

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Photocatalytic C–C Bond Cleavage of Lignin Model Compounds on Silver-Doped Cadmium Sulfide NPs

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Oxidative Amine Coupling and Thioamide Cyclization with a Photocatalytic Covalent Organic Framework

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1333
Hydrodeoxygenation of 4-Hydroxyacetophenones on Immobilized Fe–Ru Bimetallic Nanoparticles

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1334
Synthesis of 2-Amino-3-cyano-4H-chromenes on Graphene Oxide-Supported Piperazine

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1335
Oxidation of Sugar Alcohols Catalyzed by a Polymeric N-Heterocyclic Carbene–Iridium Complex

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1336
Parts Per Million Pd/C-Catalyzed Reductive Aminations in an Aqueous Micellar Medium

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1337
Aerobic C–C Bond Cleavage of Vicinal Diols Promoted by Heterogeneous Carbon Nitride CN620

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1338
Graphite-Supported Cu–Ag Nanoparticle Catalysts for Oxidation and Chan–Lam Coupling

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Cyclopropanation of Olefines Catalyzed N-doped Graphene-Supported Iron Nanoparticles

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Organo- and Biocatalysis
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Chemoenzymatic Dynamic Kinetic Resolution at Normally Static Stereogenic Centers FREE ACCESS

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1342
TEMPO-Catalyzed Di- and Trifluoromethoxylation of Arenes

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1343
Enzyme-Dependent Oxygenation Permits Highly Selective Synthesis of Diterpenes

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1344
Synthesis of Complex Isoprenoid Scaffolds by a Monodomain Class II Terpene Cyclase

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1345
Thiourea-Stabilized Carboxylic Acids Permit [4+2] Cycloadditions of Acetals and (Bis)homoallylic Alcohols

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Organocatalytic Oxygen Reduction: Dicarbenium Ions as Catalysts

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Organic Photoredox Catalyzed Deoxyfluorination of Electron-Rich Arenes

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A Dual Organocatalytic Approach to Chiral S-Heterocycles

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Radical N-Heterocyclic Carbene Catalysis for the Synthesis of Hindered Alkyl Ketones from Aldehydes

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1350
Chiral Imidazole-Catalyzed Synthesis of Remdesivir through Dynamic Kinetic Resolution

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1351
Purely Organocatalytic C–H Insertion and Cyclopropanation Reactions with α-Diazo Esters

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A PROTAC for KRAS G12C Degradation FREE ACCESS

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PEARL-seq: A Workflow for Analyzing Small Molecule–RNA Interactions

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Macropinocytosis is Key to Peptidomimetic Uptake in Cancer Cells

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Natural Products in Drug Discovery

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Copper Sensing by Electrophile Activation

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Introducing Phosphorylation-Inducing Chimeric Small Molecules (PHICS)

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Total Synthetic Lankacidin Antibiotics

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A Mild and General Synthesis of Substituted Anilines

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A Tool to Observe Cellular Apposition

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One, Two, Three – Nucleosides

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Bioluminescence Seeing Red

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The First Contraceptive FREE ACCESS

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Pumping and Probing for the Optimal Dienophile

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Peptide Chemistry
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Palladium-Catalyzed C(sp³)–H Arylation of Peptides Assisted by Unmodified Asparagine FREE ACCESS

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1368
Ni-Catalyzed Decarboxylative Borylation toward α-Aminoboronates and Peptide-Boronic Acids

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1369
Synthesis of Peptides Containing α,α-Difluoro-β-amino Acids from α,α-Difluoro Lactams

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1370
Transamination for Synthesis of Unprotected Glycine Derivatives

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1371
Modification of Tryptophan by Using Triarylbismuthines and Copper(II) Acetate

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1372
Photoredox-Catalyzed Synthesis of α-Amino Acid Derivatives

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1373
Chiral Phosphoric Acid-Catalyzed Synthesis of α-Amino Acid Derivatives

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1374
Cooperative Catalysis for the Synthesis of β-Prolines

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1375
Synthesis of Cyclic Peptides by Palladium-Catalyzed Intramolecular C(sp³)–H Arylation

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1376
Photoinduced α-C(sp³)–H Functionalization of Amino Acids and Peptides

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Dipeptide Synthesis from S-2-Formyl-4-Nitrophenyl Thioesters and Amino Acid Salts FREE ACCESS

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1378
Decarboxylative Carbonylation of α-Amino Acids

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Flow Chemistry
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1379
Asymmetric C–H Functionalization in Flow by an Immobilized Rhodium Carboxylate Catalyst

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1380
Iodine–Lithium Exchange Reaction of Benzylic Iodides

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Iridium-Photocatalyzed Formation of Tetrahydroquinolines

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