DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 11 · September 2015 DOI: 10.1055/s-005-29987

Synform

  • A120

    SYNFORM ISSUE 2015/09

    • Synthesis of Natural Products and Potential Drugs

  • z897

    All PDFs of this category

  • 0897

    Total Synthesis of (–)-Jiadifenolide

  • 0898

    Synthesis of Phthioceranic Acid

  • 0899

    Synthesis of JAK2 Inhibitor BMS-911543

  • 0900

    Synthesis of Trichodermamides A, B, and C

  • 0901

    Synthesis of CJ-16,264

  • 0902

    Synthesis of Alisertib

  • 0903

    Total Synthesis of (–)-Amphidinolide P

  • 0904

    Synthesis of a Matrix Metalloproteinase Inhibitor

  • 0905

    Synthesis of (+)-Machaeriol B, (+)-Machaeriol D, (+)-Δ8-THC, and Analogues

  • 0906

    Synthesis of Chk1 Inhibitor GDC-0425

  • 0907

    Synthesis of (R)-Ruxolitinib

  • 0908

    Synthesis of BMS-191011

  • 0909

    Synthesis of Oridamycins A and B

  • 0910

    Chemoenzymatic Synthesis of a Rosuvastatin Building Block

    • Synthesis of Heterocycles

  • z911

    All PDFs of this category

  • 0911

    Synthesis of Isoxazolino Phenanthridines

  • 0912

    Morpholines and Spirocyclic Dihydrofurans from Oxetanyl N,O-Acetals

  • 0913

    Synthesis of Dihydro-1H-benzothiazolopyridines by NHC Catalysis

  • 0914

    Azaquinolizinium Salts by Ring-Closing Metathesis

  • 0915

    Formal Hydroamination of Alkenes with Nitro- and Heteroarenes

  • 0916

    Radical-Mediated Annulations of Benzene-Linked 1,n-Enynes

  • 0917

    Optimized Process Route to a Benzoxazepine-Derived Kinase Inhibitor

  • 0918

    Metal-Free Synthesis of Perfluorinated Oxindoles

  • 0919

    Selective Synthesis of 3- or 5-Substituted Aminopyrazoles

  • 0920

    7-Azaindoles via Rhodium(III)-Catalyzed C–H Activation–Annulative Coupling

  • 0921

    Aminodifluoromethylation of Unactivated Alkenes

  • 0922

    Stereodivergent Synthesis of Substituted Tetrahydrofurans

  • 0923

    Pyrroles and Oxazines via Cycloaddition of Borodienes with Nitrosoarenes

  • 0924

    A Radical Oxidative Annulation Route to Dihydrofurans and Indolizines

  • 0925

    Synthesis of Benzazoles Catalyzed by Sodium tert-Butoxide

    • Synthesis of Materials and Unnatural Products

  • z927

    All PDFs of this category

  • 0927

    New CN and CC Group-Transfer Reagents

  • 0928

    A Different Angle

  • 0929

    One Reagent, Three Reactions in One Pot

  • 0930

    Boron Goes Both Ways

  • 0931

    An All-Pnictogen Aromatic

  • 0932

    Organic Traps: Getting Hydrocarbons to Shine

  • 0933

    Two Rings to Rule Them All: Catenated Polyesters via Macrocycle Expansion

  • 0934

    A Greener Path to Bioplastics

  • 0935

    Cages Interlocked by Dynamic Metathesis

  • 0936

    Propellers with Nitrogen: New Propulsion towards 2D Polymers?

  • 0937

    A One-Step Synthesis of Chelating, Alpha-C2-Bridged Biphospholes

  • 0938

    A Scratch ‘n’ Shine Polymer

    • Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

  • z939

    All PDFs of this category

  • 0939

    Palladacycle-Catalyzed Highly Enantioselective Arylation of Sulfonylimines

  • 0940

    Rhodium-Catalyzed Asymmetric Construction of 3-Hydroxypiperidones

  • 0941

    Copper-Catalyzed Synthesis of Chiral Phosphine Boronates

  • 0942

    Iridium-Catalyzed Asymmetric Hydroalkynylation of Norbornadienes

  • 0943

    Allylic Alkylation of 3-Substituted Indoles

  • 0944

    Asymmetric Allylic Dearomatization of Pyrroles and Controllable Migration

  • 0945

    Enantioselective Copper-Catalyzed Synthesis of Lactones

  • 0946

    Enantioselective Hydroamination of Unactivated Internal Olefins

  • 0947

    Asymmetric Transformation of 3-Isothiocyanatooxindoles

  • 0948

    Copper-Catalyzed Desymmetrative Reaction Forming Chiral O-Heterocycles

  • 0949

    N,N′-Dioxide/Nickel(II)-Catalyzed Asymmetric Hetero-Diels–Alder Reaction

  • 0950

    Enantioselective Synthesis of Allenoates by Copper Catalysis

  • 0951

    Highly Efficient Asymmetric Palladium-Catalyzed Decarboxylative Allylic Alkylation

  • 0952

    Transfer Hydrogenation–Dynamic Kinetic Resolution of α-Alkoxy β-Keto Esters

  • 0953

    syn-Stereoselective Ring Opening of Oxabenzonorbornadienes

  • 0954

    Enantioselective Synthesis of Isoxazolines by 1,3-Dipolar Cycloaddition

  • 0955

    Regio- and Enantioselective Intermolecular Hydroamination of Alkynes

  • 0956

    Asymmetric Copper-Catalyzed Formal [4+3] Annulation of Cyclopropanes and Dienes

  • 0957

    Regio- and Enantioselective Redox Relay Heck Reactions

  • 0958

    Asymmetric 1,4-Addition Using a Chiral Phosphine–Olefin Ligand

  • 0959

    Cycloheptenes by a Gold-Catalyzed Tandem Alkoxylation–Claisen Rearrangement

  • 0960

    Asymmetric Hydrogenation of Fluorinated Pyrazol-5-ols

  • 0961

    Rhodium(I)-Catalyzed Enantioselective Cycloadditions

  • 0962

    Allyl–Allyl Cross-Coupling of Allylic Carbonates with (E)-1,3-Diarylpropenes

  • 0963

    Cinchona Alkaloid Amide/Zinc(II) Catalyzed Mannich Reaction of Ketimines

  • 0964

    Diastereoselective Synthesis of Chromane-4-ones

  • 0965

    Aliphatic α-Amino Acids by Rhodium-Catalyzed Asymmetric Hydrogenation

  • 0966

    Enantioselective Interrupted Feist–Bénary Reaction with Ynones

  • 0967

    Multicomponent Reaction for the Synthesis of γ-Oxo-β-amino Esters

    • Metal-Mediated Synthesis

  • z969

    All PDFs of this category

  • 0969

    Directed Iron-Catalyzed C–H Methylation

  • 0970

    Spirocyclization of α-Aminonitriles

  • 0971

    α-Alkylation of α-MIDA Boryl Aldehydes

  • 0972

    Mn(OAc)3-Mediated Aerobic Oxidative Decarboxylative Coupling

  • 0973

    Iridium-Catalyzed Borylation of Benzylic C–H Bonds

  • 0974

    Palladium-Catalyzed Monofluoromethylation of Arylboronic Esters

  • 0975

    Copper-Catalyzed Reductive Alkylation of 1,3-Dienes with Alkyl Fluorides

  • 0976

    Lithiation of Azobenzenes

  • 0977

    One-Pot Unsymmetrical Ketone Synthesis

  • 0978

    Asymmetric Arylation of Amino Acids

  • 0979

    Diastereoselective Formation of Alcohols

  • 0980

    Titanium(IV)-Mediated Amination of Aryl Methyl Ethers

  • 0981

    Copper Nitrate Mediated Synthesis of Isoxazolines

  • 0982

    Chemoselective Suzuki–Miyaura Cross-Coupling

  • 0983

    Perfluoroalkyl and -aryl Zinc Ate Complexes in Synthesis

    • Organo- and Biocatalysis

  • z985

    All PDFs of this category

  • 0985

    Highly Efficient and Enantioselective Silylation of Alcohols

  • 0986

    Amine-Catalyzed Conjugate Addition of Aldehydes to β-Tosyl Enones

  • 0987

    In Situ Generated N-tert-Butoxycarbonyl Imines for Mannich Reactions

  • 0988

    Organocatalytic Nazarov–Semipinacol Rearrangement Cascade

  • 0989

    Stereospecific Oxidative C–H Amination Catalyzed by Iodoarenes

  • 0990

    Asymmetric α-Cyanoalkylation of Aldehydes by Photoredox Organocatalysis

  • 0991

    Chiral Phosphoric Acid Catalyzed Nucleophilic α-Amination of Azoalkenes

  • 0992

    Asymmetric Conjugate Peroxidations of α,β-Unsaturated Aldehydes

  • 0993

    Enzymatic Oxidative Decarboxylation of Fatty Acids to 1-Alkenes

  • 0994

    Asymmetric Dearomatization of Pyridines

    • Polymer-Supported Synthesis

  • z995

    All PDFs of this category

  • 0995

    Chemoselective Hydrogenation of Aldehydes on Stable Gold Nanoparticles

  • 0996

    Polymer Foam Supported Palladium Nanoparticles for Suzuki Reactions

  • 0997

    Flow Reactors Using Hollow Fibers for Acid, Base, or Chiral Rhodium Catalysis

  • 0998

    Oxidative Condensation of Aldehydes and Amines by Using Gold Nanoparticles

  • 0999

    Synthesis of Imidazoles with TFE/SBA-15-Pr-SO3H

  • 1000

    C–N Bond Formation of Secondary Amines with Cobalt/Alumina Catalyst

  • 1001

    Development of a Silica-Supported Ruthenium Bipyridyl Photocatalyst

  • 1002

    N-Arylation of Amines with Arylboronic Acids Using Supported Copper

  • 1003

    Base-Free Copper Powder-Catalyzed Knoevenagel Condensation

  • 1004

    Oxidative Amidation of Alcohols on Iron(III) Hydroxide/Magnetite Nanoparticles

  • 1005

    Controlled Aromatic Nitration with a Poly-(4-vinylpyridine)–Nitrating Mixture Complex

  • 1006

    Continuous-Flow Hydrogenation with Supported Platinum Nanoparticles

  • 1007

    Cycloisomerization of Dipeptides by Using Supported Gold Nanoparticles

  • 1008

    Solid-Phase Synthesis of γ- and δ-Lactams via N-Acyliminium Ions

  • 1009

    Reductive Alkylation by Using Calcium Hydride and Palladium on Carbon

  • 1010

    Borylation of Alkyl Bromides by Using Copper(I) Oxide Nanoparticles on Carbon Black