DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 10 · August 2014 DOI: 10.1055/s-004-27375

Synform

A101
Zanda, Matteo: SYNFORM ISSUE 2014/08

Synthesis of Natural Products and Potential Drugs

z779
All PDFs of this category
0779
Total Synthesis of (–)-Citrinalin B and (–)-Cyclopiamine B
0780
Total Syntheses of Hyperforin and Papuaforins A–C
0781
Biomimetic Synthesis of (±)-Dictazole B by Irradiation with Artificial Sunlight
0782
Synthesis of GPR40 Agonist AM-4668
0783
Synthesis of MK-8742
0784
Total Synthesis of (±)-Vaticanol A
0785
Synthesis of (±)-Merochlorin B
0786
Synthesis of an HDM2 Inhibitor
0787
Synthesis of (±)-Jiadifenolide
0788
Synthesis of Vernakalant
0789
Synthesis of (±)-Lundurine A and B

Synthesis of Heterocycles

z791
All PDFs of this category
0791
Pyrrolo- and Pyrazolopiperidines by Stereoselective Organocatalysis
0792
Synthesis of Benzofuro[2,3-c]pyridines
0793
Multicomponent Synthesis of Thiazepines
0794
Synthesis of 3-Substituted Isoxazole Derivatives Using Copper(II) Nitrate
0795
Synthesis of Dihydropyrroles via Sequential Heck–Suzuki Reaction
0796
Asymmetric Synthesis of 1,3-Oxathiolan-5-ones
0797
Synthesis of Polysubstituted Benzofurans from 2-Alkynylphenols
0798
Three-Component Synthesis of Fully Substituted Pyrazoles
0799
Pyridoquinazolinones by Palladium-Catalyzed C–H Bond Activation
0800
Copper-Mediated Synthesis of Fused Cyclopropylpyrrolidines
0801
Three-Step Synthesis of 3-Phosphonopyrroles via Hydroamination
0802
Regioselective Synthesis of Linear and Angular Pyridoquinazolones
0803
Michael Addition–Reductive Lactamization Route to 5-Alkyl-5-aryl-γ-lactams
0804
Isoquinolines by Manganese-Catalyzed Annulation of Aryl Imines with Alkynes
0805
Synthesis of Perfluoroalkyl Pyrroles and Thiophenes from Cyclopropanes

Synthesis of Materials and Unnatural Products

z807
All PDFs of this category
0807
A Treasure Trove of Tetraphenylenes
0808
Constructing Novel Polymer Architecture through a 1,4-Rhodium Migration
0809
Poly(o-arylene)s from [2.2.1]Oxabicyclic Alkenes as Monomers
0810
A Heptagon-Infused Pentacene
0811
The Right Writhe
0812
Mild Method for a Furan-Based o-Quinodimethane
0813
Efficient Transannular Cyclization via Dearomatization
0814
1,2,4,5-Tetrakis(trimethylsilyl)benzene as a 1,4-Benzdiyne Equivalent
0815
Cu(I) or Ni(0) = [4+2]: Naphthols from Cycloaddition Catalyzed by Base Metals
0816
Sulfonyl Compounds From Organozincs and Sulfonyl Halides via Copper(I)
0817
Two Sides to this Story: All-cis-1,2,4,5-tetrafluoro-3-arylcyclohexanes
0818
At Last, a Recyclable High-Performance Thermoset

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z819
All PDFs of this category
0819
Iridium-Catalyzed Asymmetric Dearomatization of Pyridines and Pyrazines
0820
Palladium-Catalyzed Asymmetric Allylic Dearomatization of Pyrroles
0821
Catalytic Asymmetric Aminations of 3-Bromooxindoles with Indolines
0822
Rhodium-Catalyzed Asymmetric Ring Expansion of Cyclobutanols
0823
Asymmetric Hydrogenation of Maleic Acid Diesters by Iridium Catalysis
0824
Asymmetric Alkynylation of Aldehydes Catalyzed by Ar-BINMOL-Phos/Zn
0825
Rhodium-Catalyzed Asymmetric Cycloisomerization of 1,6-Enynes
0826
Formal 1,2-Insertion of Rh(II) Azavinyl Carbenes into Formamides
0827
Asymmetric Intermolecular Allylic Alkylation Catalyzed by Palladium
0828
Asymmetric Ring Opening of Oxabenzonorbornadienes with Amines
0829
Catalytic Activity of New Ruthenium Complexes in the Mukaiyama Aldol Reaction
0830
Asymmetric Palladium-Catalyzed Amination of Allenyl Phosphates
0831
Enantioselective C–H Alkylation of Ferrocenes
0832
Palladium-Catalyzed Asymmetric Hydrogenation of Indoles
0833
Rhodium-Catalyzed Enantioselective β-Lactone Synthesis via C–H Activation
0834
Copper-Catalyzed Enantioselective Mannich Reaction of Cyclic Aldimines
0835
Lewis Acid/Brønsted Base Catalyzed Michael Addition to Thioamides
0836
A Bidentate Amide for the Silver-Mediated Enantioselective Direct Aldol Reaction
0837
Rhodium-Catalyzed Asymmetric Addition to Ketimines
0838
Copper-Catalyzed Asymmetric Intramolecular [3+2] Annulation
0839
Copper-Catalyzed Enantioselective Silylation of N-Sulfonylimines
0840
NHC–Copper(I)-Catalyzed Addition of Silicon Nucleophiles to Aldimines
0841
Chiral α-Hydroxy-β-Keto Esters via Asymmetric Carbonyl-Ene Reactions
0842
Rhodium-Catalyzed Asymmetric Hydrogenation of Acrylosulfones
0843
Asymmetric Synthesis of Vicinal Amino Alcohols by Rhodium Catalysis
0844
Iron(II)-Catalyzed Diastereoselective Intramolecular Aminofluorination
0845
Synthesis of Chiral Cyclopropylphosphonates by Ru(II)-Catalysis
0846
Silver-Catalyzed [3+2] Cyclization of α-Imino Esters with Isocyanoacetate
0847
Tertiary Vinylglycols via Palladium-Mediated Asymmetric Decarboxylative Cycloaddition
0848
Stereoselective Synthesis of Oxo-Heterocycles via Rhenium Catalysis

Metal-Mediated Synthesis

z849
All PDFs of this category
0849
Stereoselective Synthesis of syn-Homoallylic Alcohols
0850
Selective Lithiation of Azobenzenes
0851
Synthesis of Amino Cyclopentadienes
0852
One-Pot Allylation–Hydrostannation Sequence
0853
Synthesis of 5-Fluorinated Naphthols
0854
Tandem Carbannulation of Blaise Reaction Intermediates
0855
Trimerization of 2-Bromophenylboronic Esters via Metal-Bound Arynes
0856
Additions of Chloromethyllithium Carbenoid to Cyclic Enones
0857
Reductive Coupling of Aryl Iodides with CF3CH2I in the Presence of Copper
0858
Cross-Coupling of 2-Azidoarylboron Pinacolate Esters with Vinyl Triflates
0859
Directed ortho Metalation of Naphthyl-2-carbamates
0860
Three-Component Couplings of Imines/ Nitriles, Grignard Reagents and THF
0861
Cooperative Iron/Copper Catalysis: Borylation of Aryl Bromides
0862
Iron-Catalyzed Cross-Coupling Reactions of Non-Activated Alkyl Halides

Organo- and Biocatalysis

z863
All PDFs of this category
0863
Organocatalytic Atroposelective Synthesis of Axially Chiral Biaryls
0864
Asymmetric Three-Component Strecker Reaction Catalyzed by Disulfonimide
0865
Adjacent All-Carbon Quaternary Stereocenters via Nazarov Cyclization
0866
Enzyme Microtuning for the Synthesis of β-Blocker Precursors
0867
Chemoselective N-Heterocyclic Carbene Catalyzed Cross-Benzoin Reactions
0868
Chiral Phosphoric Acid Catalyzed Aza-Petasis–Ferrier Rearrangement
0869
Phase-Transfer-Catalyzed Nucleophilic Arylation of 3-Aryloxindoles
0870
HYDRA – Towards ppm-Level Asymmetric Organocatalysis
0871
Organocatalytic Oxidative Annulation of Benzamides with Alkynes
0872
Imidazolium-Based Organic–Inorganic Silica for Asymmetric Michael Additions
0873
Activation of Carboxylic Acids by Heterodimer Formation
0874
Enantioselective Iodolactonization by Cooperative Activation
0875
Phosphoric Acid Catalyzed Transfer Hydrogenation of Ethyl Ketimines

Polymer-Supported Synthesis

z877
All PDFs of this category
0877
Ligand-Controlled Copper-Catalyzed Oxidation of Benzylamines with Oxygen
0878
The Suzuki–Miyaura Coupling with a Polymeric Palladacycle Catalyst
0879
Alcoholysis and Hydrolysis of Silane Using PPX Nanotube Immobilized Gold
0880
Oxidative Hydroxylation of Arylboronic Acids Using CuFe2O4 NPs
0881
A Polymer-Supported Copper Complex for Asymmetric Henry Reaction
0882
Controlled Reduction of Alkynes with CO/H2O Using Au/HSA-TiO2
0883
Asymmetric Allylation of Ketones Using a Titanium–BINOLate Complex
0884
Borylation, Silylation, and Dehydrogenation Using Bipyridyl-Containing MOFs
0885
Hydrogenation of Amino Acids with Rh–MoOx/SiO2
0886
Imidazolium Salt Stabilized Palladium Nanoparticles for Cross-Couplings
0887
The Suzuki–Miyaura Cross-Coupling of Heteroaromatics Using Pd0-AmP-MCF
0888
Solid-Phase Synthesis of Anagrelide Sulfonyl Analogues
0889
Enantioselective Aldol Reactions Using a PS-Supported Threonine Derivative
0890
Reduction of Nitrobenzenes Using Dendrimer-Encapsulated [Rh5(CO)15]–
0891
Photocatalytic Aerobic Oxidation of Amines to Imines