Cross-Coupling of Benzyl Phosphates with Arylboronic Acids

doi:10.1055/s-2005-921724

Subscribe to RSS

Please copy the URL and add it into your RSS Feed Reader.

https://www.thieme-connect.de/rss/thieme/en/10.1055-s-00000131.xml

Share / Bookmark

Facebook Linkedin Weibo

Download PDF

Synfacts 2006(1): 0062-0062
DOI: 10.1055/s-2005-921724

Metal-Mediated Synthesis

Cross-Coupling of Benzyl Phosphates with Arylboronic Acids

Contributor(s): Paul Knochel, Andrei Gavryushin
M. McLaughlin*
Merck Research Laboratories, Rahway, US

Further Information

Publication History

Publication Date:
16 December 2005 (online)

Permissions and Reprints

Significance

An interesting approach for the formation of diarylmethanes from easily available arylboronic acids is described. The protocol is simple and excellent tolerance of functional groups can be expected. Also, a practical method for the synthesis of benzylic diethyl phosphates is described.